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A selective WDR5 degrader inhibits acute myeloid leukemia in patient-derived mouse models.

Xufen YuDongxu LiJithesh KotturYudao ShenHuen Suk KimKwang-Su ParkYi-Hsuan TsaiWeida GongJun WangKyogo SuzukiJoel S ParkerLaura E HerringHusnu Ümit KaniskanLing CaiRinku JainJing LiuAneel K AggarwalGang Greg WangJian Jin
Published in: Science translational medicine (2021)
[Figure: see text].
Keyphrases
  • acute myeloid leukemia
  • mouse model
  • allogeneic hematopoietic stem cell transplantation
  • smoking cessation
  • acute lymphoblastic leukemia