Amaury E Fernández-Montalván (Amaury Fernández-Montalván)

ORCID

Publication Activity (10 Years)

Years Active: 2017-2020
Publications (10 Years): 9

Top Venues

Journal of medicinal chemistry

British journal of pharmacology

Drug metabolism and disposition: the biological fate of chemicals

ACS chemical biology

This page only lists publications with an associated author ORCID identifier.

Publications

Cornelius Trünkle, Christian Lechner, Daniel Korr, Léa Bouché, Naomi Barak, Amaury E Fernández-Montalván, Roderich D Süssmuth, Andreas Reichel
Concentration Dependence of the Unbound Partition Coefficient Kpuu and Its Application to Correct for Exposure-Related Discrepancies between Biochemical and Cellular Potency of KAT6A Inhibitors. Drug metabolism and disposition: the biological fate of chemicals 48 (7) (2020)
Volker Klaus Schulze, Ulrich Klar, Dirk Kosemund, Antje M Wengner, Gerhard Siemeister, Detlef Stöckigt, Roland Neuhaus, Philip Lienau, Benjamin Bader, Stefan Prechtl, Simon J Holton, Hans Briem, Tobias Marquardt, Hartmut Schirok, Rolf Jautelat, Rolf Bohlmann, Duy Nguyen, Amaury E Fernández-Montalván, Ulf Bömer, Uwe Eberspaecher, Michael Brüning, Olaf Döhr, Marian Raschke, Bertolt Kreft, Dominik Mumberg, Karl Ziegelbauer, Michael Brands, Franz von Nussbaum, Marcus Koppitz
Treating Cancer by Spindle Assembly Checkpoint Abrogation: Discovery of Two Clinical Candidates, BAY 1161909 and BAY 1217389, Targeting MPS1 Kinase. Journal of medicinal chemistry 63 (15) (2020)
Olaf Panknin, Andrea Wagenfeld, Wilhelm Bone, Eckhard Bender, Katrin Nowak-Reppel, Amaury E Fernández-Montalván, Reinhard Nubbemeyer, Stefan Bäurle, Sven Ring, Norbert Schmees, Olaf Prien, Martina Schäfer, Christian Friedrich, Thomas M Zollner, Andreas Steinmeyer, Thomas Mueller, Gernot Langer
Discovery and Characterization of BAY 1214784, an Orally Available Spiroindoline Derivative Acting as a Potent and Selective Antagonist of the Human Gonadotropin-Releasing Hormone Receptor as Proven in a First-In-Human Study in Postmenopausal Women. Journal of medicinal chemistry 63 (20) (2020)
Victoria Georgi, Alexey Dubrovskiy, Stephan Steigele, Amaury E Fernández-Montalván
Considerations for improved performance of competition association assays analysed with the Motulsky-Mahan's "kinetics of competitive binding" model. British journal of pharmacology 176 (24) (2019)
Reggie Bosma, Leigh A Stoddart, Victoria Georgi, Monica Bouzo-Lorenzo, Nick Bushby, Loretta Inkoom, Michael J Waring, Stephen J Briddon, Henry F Vischer, Robert J Sheppard, Amaury E Fernández-Montalván, Stephen J Hill, Rob Leurs
Probe dependency in the determination of ligand binding kinetics at a prototypical G protein-coupled receptor. Scientific reports 9 (1) (2019)
Gerhard Siemeister, Anne Mengel, Amaury E Fernández-Montalván, Wilhelm Bone, Jens Schröder, Sabine Zitzmann-Kolbe, Hans Briem, Stefan Prechtl, Simon J Holton, Ursula Mönning, Oliver von Ahsen, Sandra Johanssen, Arwed Cleve, Vera Pütter, Marion Hitchcock, Franz von Nussbaum, Michael Brands, Karl Ziegelbauer, Dominik Mumberg
Inhibition of BUB1 Kinase by BAY 1816032 Sensitizes Tumor Cells toward Taxanes, ATR, and PARP Inhibitors In Vitro and In Vivo. Clinical cancer research : an official journal of the American Association for Cancer Research 25 (4) (2018)
Victoria Georgi, Felix Schiele, Benedict-Tilman Berger, Andreas Steffen, Paula A Marin Zapata, Hans Briem, Stephan Menz, Cornelia Preusse, James D Vasta, Matthew B Robers, Michael Brands, Stefan Knapp, Amaury E Fernández-Montalván
Binding Kinetics Survey of the Drugged Kinome. Journal of the American Chemical Society 140 (46) (2018)
Wilhelmus E A de Witte, Joost W Versfelt, Maria Kuzikov, Solene Rolland, Victoria Georgi, Philip Gribbon, Sheraz Gul, Dymphy Huntjens, Piet Hein van der Graaf, Meindert Danhof, Amaury E Fernández-Montalván, Gesa Witt, Elizabeth C M De Lange
In vitro and in silico analysis of the effects of D2 receptor antagonist target binding kinetics on the cellular response to fluctuating dopamine concentrations. British journal of pharmacology 175 (21) (2018)
Amaury E Fernández-Montalván, Markus Berger, Benno Kuropka, Seong Joo Koo, Volker Badock, Joerg Weiske, Vera Puetter, Simon J Holton, Detlef Stöckigt, Antonius Ter Laak, Paolo A Centrella, Matthew A Clark, Christoph E Dumelin, Eric A Sigel, Holly H Soutter, Dawn M Troast, Ying Zhang, John W Cuozzo, Anthony D Keefe, Didier Roche, Vincent Rodeschini, Apirat Chaikuad, Laura Díaz-Sáez, James M Bennett, Oleg Fedorov, Kilian V M Huber, Jan Hübner, Hilmar Weinmann, Ingo V Hartung, Mátyás Gorjánácz
Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action. ACS chemical biology 12 (11) (2017)

Amaury E Fernández-Montalván.css-eqlu8i{font-size:small;padding-left:4px;} (Amaury Fernández-Montalván)

Publication Activity (10 Years)

Top Topics

Top Venues

Amaury E Fernández-Montalván (Amaury Fernández-Montalván)