Eddy Sotelo

ResearcherID Loop profile ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 33

Top Venues

Journal of medicinal chemistry

Pharmaceutics

Molecules (Basel, Switzerland)

International journal of molecular sciences

Universidade de Santiago de Compostela

Universidade de Santiago de Compostela (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Universidade de Santiago de Compostela Jan 02 2011

Spain

Profesor Titular/Associate Professor :: Faculty of Pharmacy, Department of Organic Chemistry

Education History

Universidade de Santiago de Compostela Oct 01 1995 - May 05 2000

Spain

PHD :: Organic Chemistry

Publications

Francesca Intranuovo, Maria Majellaro, Francesco Mastropasqua, Pietro Delre, Francesca Serena Abatematteo, Giuseppe Felice Mangiatordi, Angela Stefanachi, Jose Brea, Maria Isabel Loza, Chiara Riganti, Alessia Ligresti, Poulami Kumar, Daniela Esposito, Luigia Cristino, Alessandro Nicois, Lucía González, Maria Grazia Perrone, Nicola Antonio Colabufo, Eddy Sotelo, Carmen Abate, Marialessandra Contino
N -Adamantyl-1-alkyl-4-oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as Fluorescent Probes to Detect Microglia Activation through the Imaging of Cannabinoid Receptor Subtype 2 (CB2R). Journal of medicinal chemistry (2024)
Miguel Pereira-Silva, Darío Miranda-Pastoriza, Luis Diaz-Gomez, Eddy Sotelo, Ana Cláudia Paiva Santos, Francisco Veiga, Angel Concheiro, Carmen Alvarez-Lorenzo
Gemcitabine-Vitamin E Prodrug-Loaded Micelles for Pancreatic Cancer Therapy. Pharmaceutics 16 (1) (2024)
Francesca Intranuovo, Maria Majellaro, Francesco Mastropasqua, Pietro Delre, Francesca Serena Abatematteo, Giuseppe Felice Mangiatordi, Angela Stefanachi, Jose Brea, Maria Isabel Loza, Chiara Riganti, Alessia Ligresti, Poulami Kumar, Daniela Esposito, Luigia Cristino, Alessandro Nicois, Lucía González, Maria Grazia Perrone, Nicola Antonio Colabufo, Eddy Sotelo, Carmen Abate, Marialessandra Contino
N -Adamantyl-1-alkyl-4-oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as Fluorescent Probes to Detect Microglia Activation through the Imaging of Cannabinoid Receptor Subtype 2 (CB2R). Journal of medicinal chemistry 67 (13) (2024)
Francesca Intranuovo, Maria Majellaro, Francesco Mastropasqua, Pietro Delre, Francesca Serena Abatematteo, Giuseppe Felice Mangiatordi, Angela Stefanachi, Jose Brea, Maria Isabel Loza, Chiara Riganti, Alessia Ligresti, Poulami Kumar, Daniela Esposito, Luigia Cristino, Alessandro Nicois, Lucía González, Maria Grazia Perrone, Nicola Antonio Colabufo, Eddy Sotelo, Carmen Abate, Marialessandra Contino
N -Adamantyl-1-alkyl-4-oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as Fluorescent Probes to Detect Microglia Activation through the Imaging of Cannabinoid Receptor Subtype 2 (CB2R). Journal of medicinal chemistry 67 (13) (2024)
Miguel Pereira-Silva, Darío Miranda-Pastoriza, Luis Diaz-Gomez, Eddy Sotelo, Ana Cláudia Paiva Santos, Francisco Veiga, Angel Concheiro, Carmen Alvarez-Lorenzo
Gemcitabine-Vitamin E Prodrug-Loaded Micelles for Pancreatic Cancer Therapy. Pharmaceutics 16 (1) (2024)
Miguel Pereira-Silva, Darío Miranda-Pastoriza, Luis Diaz-Gomez, Eddy Sotelo, Ana Cláudia Paiva Santos, Francisco Veiga, Angel Concheiro, Carmen Alvarez-Lorenzo
Gemcitabine-Vitamin E Prodrug-Loaded Micelles for Pancreatic Cancer Therapy. Pharmaceutics 16 (1) (2024)
Francesca Serena Abatematteo, Maria Majellaro, Bianca Montsch, Rubén Prieto-Díaz, Mauro Niso, Marialessandra Contino, Angela Stefanachi, Chiara Riganti, Giuseppe Felice Mangiatordi, Pietro Delre, Petra Heffeter, Eddy Sotelo, Carmen Abate
Development of Fluorescent 4-[4-(3 H -Spiro[isobenzofuran-1,4'-piperidin]-1'-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based Techniques. Journal of medicinal chemistry 66 (6) (2023)
Gemma Navarro, Eddy Sotelo, Iu Raïch, María Isabel Loza, Jose Brea, Maria Majellaro
A Robust and Efficient FRET-Based Assay for Cannabinoid Receptor Ligands Discovery. Molecules (Basel, Switzerland) 28 (24) (2023)
Giovanni Graziano, Angela Stefanachi, Marialessandra Contino, Rubén Prieto-Díaz, Alessia Ligresti, Poulami Kumar, Antonio Scilimati, Eddy Sotelo, Francesco Leonetti
Multicomponent Reaction-Assisted Drug Discovery: A Time- and Cost-Effective Green Approach Speeding Up Identification and Optimization of Anticancer Drugs. International journal of molecular sciences 24 (7) (2023)
Francesca Serena Abatematteo, Maria Majellaro, Bianca Montsch, Rubén Prieto-Díaz, Mauro Niso, Marialessandra Contino, Angela Stefanachi, Chiara Riganti, Giuseppe Felice Mangiatordi, Pietro Delre, Petra Heffeter, Eddy Sotelo, Carmen Abate
Development of Fluorescent 4-[4-(3 H -Spiro[isobenzofuran-1,4'-piperidin]-1'-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based Techniques. Journal of medicinal chemistry (2023)
Gemma Navarro, Eddy Sotelo, Iu Raïch, María Isabel Loza, Jose Brea, Maria Majellaro
A Robust and Efficient FRET-Based Assay for Cannabinoid Receptor Ligands Discovery. Molecules (Basel, Switzerland) 28 (24) (2023)
Francesca Serena Abatematteo, Maria Majellaro, Bianca Montsch, Rubén Prieto-Díaz, Mauro Niso, Marialessandra Contino, Angela Stefanachi, Chiara Riganti, Giuseppe Felice Mangiatordi, Pietro Delre, Petra Heffeter, Eddy Sotelo, Carmen Abate
Development of Fluorescent 4-[4-(3 H -Spiro[isobenzofuran-1,4'-piperidin]-1'-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of σ Receptors via Fluorescence-Based Techniques. Journal of medicinal chemistry 66 (6) (2023)
Francesca Intranuovo, Leonardo Brunetti, Pietro DelRe, Giuseppe Felice Mangiatordi, Angela Stefanachi, Antonio Laghezza, Mauro Niso, Francesco Leonetti, Fulvio Loiodice, Alessia Ligresti, Magdalena Kostrzewa, Jose Brea, Maria Isabel Loza, Eddy Sotelo, Alessandro Tossi, Nicola Antonio Colabufo, Chiara Riganti, Carmen Abate, Marialessandra Contino
Development of N -(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. Journal of medicinal chemistry 66 (1) (2022)
Rubén Prieto-Díaz, Manuel González-Gómez, Hugo Fojo-Carballo, Jhonny Azuaje, Abdelaziz El Maatougui, Maria Majellaro, Maria Isabel Loza, Jose Brea, Víctor Fernández-Dueñas, M Rita Paleo, Alejandro Díaz-Holguín, Beatriz García-Pinel, Ana Mallo-Abreu, Juan C Estévez, Antonio Andújar-Arias, Xerardo García-Mera, Iria Gomez-Tourino, Francisco Ciruela, Cristian O Salas, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring the Effect of Halogenation in a Series of Potent and Selective A 2B Adenosine Receptor Antagonists. Journal of medicinal chemistry 66 (1) (2022)
Rubén Prieto-Díaz, Manuel González-Gómez, Hugo Fojo-Carballo, Jhonny Azuaje, Abdelaziz El Maatougui, Maria Majellaro, Maria Isabel Loza, Jose Brea, Víctor Fernández-Dueñas, M Rita Paleo, Alejandro Díaz-Holguín, Beatriz García-Pinel, Ana Mallo-Abreu, Juan C Estévez, Antonio Andújar-Arias, Xerardo García-Mera, Iria Gomez-Tourino, Francisco Ciruela, Cristian O Salas, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring the Effect of Halogenation in a Series of Potent and Selective A 2B Adenosine Receptor Antagonists. Journal of medicinal chemistry 66 (1) (2022)
Cristina Val, Carlos Rodríguez-García, Rubén Prieto-Díaz, Abel Crespo, Jhonny Azuaje, Carlos Carbajales, Maria Majellaro, Alejandro Díaz-Holguín, José M Brea, Maria Isabel Loza, Claudia Gioé-Gallo, Marialessandra Contino, Angela Stefanachi, Xerardo García-Mera, Juan C Estévez, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A 1 Antagonists. Journal of medicinal chemistry 65 (3) (2022)
Darío Miranda-Pastoriza, Rodrigo Bernárdez, Jhonny Azuaje, Rubén Prieto-Díaz, Maria Majellaro, Ashish V Tamhankar, Lucien Koenekoop, Alejandro González, Claudia Gioé-Gallo, Ana Mallo-Abreu, José Brea, Maria Isabel Loza, Aitor García-Rey, Xerardo García-Mera, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring Non-orthosteric Interactions with a Series of Potent and Selective A 3 Antagonists. ACS medicinal chemistry letters 13 (2) (2022)
Rubén Prieto-Díaz, Manuel González-Gómez, Hugo Fojo-Carballo, Jhonny Azuaje, Abdelaziz El Maatougui, Maria Majellaro, Maria Isabel Loza, Jose Brea, Víctor Fernández-Dueñas, M Rita Paleo, Alejandro Díaz-Holguín, Beatriz García-Pinel, Ana Mallo-Abreu, Juan C Estévez, Antonio Andújar-Arias, Xerardo García-Mera, Iria Gomez-Tourino, Francisco Ciruela, Cristian O Salas, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring the Effect of Halogenation in a Series of Potent and Selective A 2B Adenosine Receptor Antagonists. Journal of medicinal chemistry 66 (1) (2022)
Francesca Intranuovo, Leonardo Brunetti, Pietro DelRe, Giuseppe Felice Mangiatordi, Angela Stefanachi, Antonio Laghezza, Mauro Niso, Francesco Leonetti, Fulvio Loiodice, Alessia Ligresti, Magdalena Kostrzewa, Jose Brea, Maria Isabel Loza, Eddy Sotelo, Alessandro Tossi, Nicola Antonio Colabufo, Chiara Riganti, Carmen Abate, Marialessandra Contino
Development of N -(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. Journal of medicinal chemistry 66 (1) (2022)
Rubén Prieto-Díaz, Manuel González-Gómez, Hugo Fojo-Carballo, Jhonny Azuaje, Abdelaziz El Maatougui, Maria Majellaro, Maria Isabel Loza, Jose Brea, Víctor Fernández-Dueñas, M Rita Paleo, Alejandro Díaz-Holguín, Beatriz García-Pinel, Ana Mallo-Abreu, Juan C Estévez, Antonio Andújar-Arias, Xerardo García-Mera, Iria Gomez-Tourino, Francisco Ciruela, Cristian O Salas, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring the Effect of Halogenation in a Series of Potent and Selective A 2B Adenosine Receptor Antagonists. Journal of medicinal chemistry (2022)
Rubén Prieto-Díaz, Manuel González-Gómez, Hugo Fojo-Carballo, Jhonny Azuaje, Abdelaziz El Maatougui, Maria Majellaro, Maria Isabel Loza, Jose Brea, Víctor Fernández-Dueñas, M Rita Paleo, Alejandro Díaz-Holguín, Beatriz García-Pinel, Ana Mallo-Abreu, Juan C Estévez, Antonio Andújar-Arias, Xerardo García-Mera, Iria Gomez-Tourino, Francisco Ciruela, Cristian O Salas, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring the Effect of Halogenation in a Series of Potent and Selective A 2B Adenosine Receptor Antagonists. Journal of medicinal chemistry 66 (1) (2022)
Francesca Intranuovo, Leonardo Brunetti, Pietro DelRe, Giuseppe Felice Mangiatordi, Angela Stefanachi, Antonio Laghezza, Mauro Niso, Francesco Leonetti, Fulvio Loiodice, Alessia Ligresti, Magdalena Kostrzewa, Jose Brea, Maria Isabel Loza, Eddy Sotelo, Alessandro Tossi, Nicola Antonio Colabufo, Chiara Riganti, Carmen Abate, Marialessandra Contino
Development of N -(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. Journal of medicinal chemistry (2022)
Rubén Prieto-Díaz, Manuel González-Gómez, Hugo Fojo-Carballo, Jhonny Azuaje, Abdelaziz El Maatougui, Maria Majellaro, Maria Isabel Loza, Jose Brea, Víctor Fernández-Dueñas, M Rita Paleo, Alejandro Díaz-Holguín, Beatriz García-Pinel, Ana Mallo-Abreu, Juan C Estévez, Antonio Andújar-Arias, Xerardo García-Mera, Iria Gomez-Tourino, Francisco Ciruela, Cristian O Salas, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Exploring the Effect of Halogenation in a Series of Potent and Selective A 2B Adenosine Receptor Antagonists. Journal of medicinal chemistry 66 (1) (2022)
Francesca Intranuovo, Leonardo Brunetti, Pietro DelRe, Giuseppe Felice Mangiatordi, Angela Stefanachi, Antonio Laghezza, Mauro Niso, Francesco Leonetti, Fulvio Loiodice, Alessia Ligresti, Magdalena Kostrzewa, Jose Brea, Maria Isabel Loza, Eddy Sotelo, Alessandro Tossi, Nicola Antonio Colabufo, Chiara Riganti, Carmen Abate, Marialessandra Contino
Development of N -(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. Journal of medicinal chemistry 66 (1) (2022)
Ana Mallo-Abreu, Irene Reyes-Resina, Jhonny Azuaje, Rafael Franco, Aitor García-Rey, Maria Majellaro, Darío Miranda-Pastoriza, Xerardo García-Mera, Willem Jespers, Hugo Gutiérrez-de-Terán, Gemma Navarro, Eddy Sotelo
Potent and Subtype-Selective Dopamine D2 Receptor Biased Partial Agonists Discovered via an Ugi-Based Approach. Journal of medicinal chemistry 64 (12) (2021)
Ana Mallo-Abreu, Rubén Prieto-Díaz, Willem Jespers, Jhonny Azuaje, Maria Majellaro, Carmen Velando, Xerardo García-Mera, Olga Caamaño, José Brea, María I Loza, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists. Journal of medicinal chemistry 63 (14) (2020)
María Majellaro, Willem Jespers, Abel Crespo, María J Núñez, Silvia Novio, Jhonny Azuaje, Rubén Prieto-Díaz, Claudia Gioé, Belma Alispahic, José Brea, María I Loza, Manuel Freire-Garabal, Carlota Garcia-Santiago, Carlos Rodríguez-García, Xerardo García-Mera, Olga Caamaño, Christian Fernandez-Masaguer, F Javier Sardina, Angela Stefanachi, Abdelaziz El Maatougui, Ana Mallo-Abreu, Johan Åqvist, Hugo Gutiérrez-de-Terán, Eddy Sotelo
3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition. Journal of medicinal chemistry 64 (1) (2020)
Zuzana Jandova, Willem Jespers, Eddy Sotelo, Hugo Gutiérrez-de-Terán, Chris Oostenbrink
Free-Energy Calculations for Bioisosteric Modifications of A3 Adenosine Receptor Antagonists. International journal of molecular sciences 20 (14) (2019)
Ana Mallo-Abreu, María Majellaro, Willem Jespers, Jhonny Azuaje, Olga Caamaño, Xerardo García-Mera, José M Brea, María I Loza, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Trifluorinated Pyrimidine-Based A2B Antagonists: Optimization and Evidence of Stereospecific Recognition. Journal of medicinal chemistry 62 (20) (2019)
Jhonny Azuaje, Willem Jespers, Vicente Yaziji, Ana Mallo, María Majellaro, Olga Caamaño, María I Loza, María I Cadavid, José Brea, Johan Åqvist, Eddy Sotelo, Hugo Gutiérrez-de-Terán
Effect of Nitrogen Atom Substitution in A3 Adenosine Receptor Binding: N-(4,6-Diarylpyridin-2-yl)acetamides as Potent and Selective Antagonists. Journal of medicinal chemistry 60 (17) (2017)
Carlos Carbajales, Jhonny Azuaje, Ana Oliveira, María I Loza, José Brea, María I Cadavid, Christian F Masaguer, Xerardo García-Mera, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Enantiospecific Recognition at the A2B Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylates. Journal of medicinal chemistry 60 (8) (2017)
Carlos Carbajales, Jun-Ichi Sawada, Giovanni Marzaro, Eddy Sotelo, Luz Escalante, Antonio Sánchez-Díaz Marta, Xerardo García-Mera, Akira Asai, Alberto Coelho
Multicomponent Assembly of the Kinesin Spindle Protein Inhibitor CPUYJ039 and Analogues as Antimitotic Agents. ACS combinatorial science 19 (3) (2017)
Willem Jespers, Ana Oliveira, Rubén Prieto-Díaz, María Majellaro, Johan Åqvist, Eddy Sotelo, Hugo Gutiérrez-de-Terán
Structure-Based Design of Potent and Selective Ligands at the Four Adenosine Receptors. Molecules (Basel, Switzerland) 22 (11) (2017)

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Publication Activity (10 Years)

Top Topics

Top Venues

Eddy Sotelo