Milan Dejmek

Publication Activity (10 Years)

Years Active: 2021-2024
Publications (10 Years): 11

Top Topics

Acute Myeloid Leukemia

Bioinformatics Analysis

Respiratory Syndrome Coronavirus

Allogeneic Hematopoietic Stem Cell Transplantation

Top Venues

Beilstein journal of organic chemistry

Cancer research

RSC medicinal chemistry

Journal of medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Luca Julianna Tóth, Kateřina Krejčová, Milan Dejmek, Eva Žilecká, Blanka Klepetářová, Lenka Poštová Slavětínská, Evzen Boura, Radim Nencka
Novel analogues of a nonnucleoside SARS-CoV-2 RdRp inhibitor as potential antivirotics. Beilstein journal of organic chemistry 20 (2024)
Hugo Kocek, Dominika Chalupská, Milan Dejmek, Alexandra Dvořáková, Michala Zgarbová, Michal Šála, Karel Chalupský, Petra Krafčíková, Tomáš Otava, Matúš Drexler, Eliška Procházková, Blanka Klepetářová, Milan Štefek, Ján Kozic, Helena Mertlíková-Kaiserová, Evzen Boura, Jan Weber, Radim Nencka
Discovery of highly potent SARS-CoV-2 nsp14 methyltransferase inhibitors based on adenosine 5'-carboxamides. RSC medicinal chemistry (2024)
Hugo Kocek, Dominika Chalupská, Milan Dejmek, Alexandra Dvořáková, Michala Zgarbová, Michal Šála, Karel Chalupský, Petra Krafčíková, Tomáš Otava, Matúš Drexler, Eliška Procházková, Blanka Klepetářová, Milan Štefek, Ján Kozic, Helena Mertlíková-Kaiserová, Evzen Boura, Jan Weber, Radim Nencka
Discovery of highly potent SARS-CoV-2 nsp14 methyltransferase inhibitors based on adenosine 5'-carboxamides. RSC medicinal chemistry (2024)
Luca Julianna Tóth, Kateřina Krejčová, Milan Dejmek, Eva Žilecká, Blanka Klepetářová, Lenka Poštová Slavětínská, Evzen Boura, Radim Nencka
Novel analogues of a nonnucleoside SARS-CoV-2 RdRp inhibitor as potential antivirotics. Beilstein journal of organic chemistry 20 (2024)
Milan Štefek, Dominika Chalupská, Karel Chalupský, Michala Zgarbová, Alexandra Dvořáková, Petra Krafčíková, Alice Shi Ming Li, Michal Šála, Milan Dejmek, Tomáš Otava, Ema Chaloupecká, Jaroslav Kozák, Ján Kozic, Masoud Vedadi, Jan Weber, Helena Mertlíková-Kaiserová, Radim Nencka
Rational Design of Highly Potent SARS-CoV-2 nsp14 Methyltransferase Inhibitors. ACS omega 8 (30) (2023)
Courtney Chambers, Katerina Cermakova, Yuen San Chan, Kristen J Kurtz, Katharina Wohlan, Andrew Henry Lewis, Christiana Wang, Anh Pham, Milan Dejmek, Michal Šála, Mario Loeza Cabrera, Rogelio Aguilar, Radim Nencka, H Daniel Lacorazza, Rachel E Rau, H Courtney Hodges
SWI/SNF blockade disrupts PU.1-directed enhancer programs in normal hematopoietic cells and acute myeloid leukemia. Cancer research (2023)
Courtney Chambers, Katerina Cermakova, Yuen San Chan, Kristen J Kurtz, Katharina Wohlan, Andrew Henry Lewis, Christiana Wang, Anh Pham, Milan Dejmek, Michal Šála, Mario Loeza Cabrera, Rogelio Aguilar, Radim Nencka, H Daniel Lacorazza, Rachel E Rau, H Courtney Hodges
SWI/SNF blockade disrupts PU.1-directed enhancer programs in normal hematopoietic cells and acute myeloid leukemia. Cancer research (2023)
Petra Břehová, Eva Řezníčková, Kryštof Škach, Radek Jorda, Milan Dejmek, Veronika Vojáčková, Michal Šála, Markéta Kovalová, Martin Dračínský, Alexandra Dolníková, Timotej Strmeň, Monika Kinnertová, Karel Chalupský, Alexandra Dvořáková, Tomáš Gucký, Helena Mertlíková Kaiserová, Pavel Klener, Radim Nencka, Vladimir Kryštof
Inhibition of FLT3-ITD Kinase in Acute Myeloid Leukemia by New Imidazo[1,2- b ]pyridazine Derivatives Identified by Scaffold Hopping. Journal of medicinal chemistry (2023)
Zdeněk Vavřina, Pavla Perlíková, Nemanja Milisavljević, Florian Chevrier, Miroslav Smola, Joshua Smith, Milan Dejmek, Vojtěch Havlíček, Miloš Buděšínský, Radek Liboska, Lenka Vanekova, Jiří Brynda, Evzen Boura, Pavlína Řezáčová, Michal Hocek, Gabriel Birkuš
Design, Synthesis, and Biochemical and Biological Evaluation of Novel 7-Deazapurine Cyclic Dinucleotide Analogues as STING Receptor Agonists. Journal of medicinal chemistry 65 (20) (2022)
Marketa Pimkova Polidarova, Lenka Vanekova, Petra Břehová, Milan Dejmek, Zdeněk Vavřina, Gabriel Birkuš, Andrea Brazdova
Synthetic Stimulator of Interferon Genes (STING) Agonists Induce a Cytokine-Mediated Anti-Hepatitis B Virus Response in Nonparenchymal Liver Cells. ACS infectious diseases (2022)
Miroslav Smola, Ondrej Gutten, Milan Dejmek, Milan Kožíšek, Thomas Evangelidis, Zahra Aliakbar Tehrani, Barbora Novotná, Radim Nencka, Gabriel Birkuš, Lubomír Rulíšek, Evzen Boura
Ligand Strain and Its Conformational Complexity Is a Major Factor in the Binding of Cyclic Dinucleotides to STING Protein. Angewandte Chemie (International ed. in English) 60 (18) (2021)