Iacovos N Michaelides (Iacovos Michaelides)

Publication Activity (10 Years)

Years Active: 2021-2024
Publications (10 Years): 16

Top Topics

Recombinant Human

Top Venues

Journal of medicinal chemistry

ACS medicinal chemistry letters

RSC medicinal chemistry

Communications biology

This page only lists publications with an associated author ORCID identifier.

Publications

Simon C C Lucas, Afshan Ahmed, S Neha Ashraf, Argyrides Argyrou, Matthias R Bauer, Gian Marco De Donatis, Sylvain Demanze, Frederik Eisele, Lucia Fusani, Andreas Hock, Ganesh Kadamur, Shuyou Li, Abigail Macmillan-Jones, Iacovos N Michaelides, Christopher Phillips, Marie Rehnström, Magdalena Richter, Monica C Rodrigo-Brenni, Fiona Shilliday, Peng Wang, R Ian Storer
Optimization of Potent Ligands for the E3 Ligase DCAF15 and Evaluation of Their Use in Heterobifunctional Degraders. Journal of medicinal chemistry (2024)
Simon C C Lucas, Afshan Ahmed, S Neha Ashraf, Argyrides Argyrou, Matthias R Bauer, Gian Marco De Donatis, Sylvain Demanze, Frederik Eisele, Lucia Fusani, Andreas Hock, Ganesh Kadamur, Shuyou Li, Abigail Macmillan-Jones, Iacovos N Michaelides, Christopher Phillips, Marie Rehnström, Magdalena Richter, Monica C Rodrigo-Brenni, Fiona Shilliday, Peng Wang, R Ian Storer
Optimization of Potent Ligands for the E3 Ligase DCAF15 and Evaluation of Their Use in Heterobifunctional Degraders. Journal of medicinal chemistry 67 (7) (2024)
Simon C C Lucas, Afshan Ahmed, S Neha Ashraf, Argyrides Argyrou, Matthias R Bauer, Gian Marco De Donatis, Sylvain Demanze, Frederik Eisele, Lucia Fusani, Andreas Hock, Ganesh Kadamur, Shuyou Li, Abigail Macmillan-Jones, Iacovos N Michaelides, Christopher Phillips, Marie Rehnström, Magdalena Richter, Monica C Rodrigo-Brenni, Fiona Shilliday, Peng Wang, R Ian Storer
Optimization of Potent Ligands for the E3 Ligase DCAF15 and Evaluation of Their Use in Heterobifunctional Degraders. Journal of medicinal chemistry 67 (7) (2024)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry (2023)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry 66 (5) (2023)
Mateusz P Plesniak, Emilia K Taylor, Frederik Eisele, Christopher M B K Kourra, Iacovos N Michaelides, Alice Oram, Johan Wernevik, Zulma Santisteban Valencia, Hannah Rowbottom, Nadia Mann, Linda Fredlund, Valentyna Pivnytska, Anna Novén, Mohammad Pirmoradian, Thomas Lundbäck, R Ian Storer, Mariell Pettersson, Gian M De Donatis, Marie Rehnström
Rapid PROTAC Discovery Platform: Nanomole-Scale Array Synthesis and Direct Screening of Reaction Mixtures. ACS medicinal chemistry letters 14 (12) (2023)
Iacovos N Michaelides, Gavin W Collie
Correction to "E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology". Journal of medicinal chemistry (2023)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry 66 (5) (2023)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry 66 (5) (2023)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry (2023)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry 66 (5) (2023)
Iacovos N Michaelides, Gavin W Collie
E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology. Journal of medicinal chemistry 66 (5) (2023)
Mateusz P Plesniak, Emilia K Taylor, Frederik Eisele, Christopher M B K Kourra, Iacovos N Michaelides, Alice Oram, Johan Wernevik, Zulma Santisteban Valencia, Hannah Rowbottom, Nadia Mann, Linda Fredlund, Valentyna Pivnytska, Anna Novén, Mohammad Pirmoradian, Thomas Lundbäck, R Ian Storer, Mariell Pettersson, Gian M De Donatis, Marie Rehnström
Rapid PROTAC Discovery Platform: Nanomole-Scale Array Synthesis and Direct Screening of Reaction Mixtures. ACS medicinal chemistry letters 14 (12) (2023)
Iacovos N Michaelides, Gavin W Collie, Ulf Börjesson, Christina Vasalou, Omar Alkhatib, Louise Barlind, Tony Cheung, Ian L Dale, Kevin J Embrey, Edward J Hennessy, Puneet Khurana, Cheryl M Koh, Michelle L Lamb, Jianming Liu, Thomas A Moss, Daniel J O'Neill, Christopher Phillips, Joseph Shaw, Arjan Snijder, R Ian Storer, Christopher J Stubbs, Fujin Han, Chengzhi Li, Jingchuan Qiao, Dong-Qing Sun, Jingwen Wang, Peng Wang, Wenzhen Yang
Discovery and Optimization of the First ATP Competitive Type-III c-MET Inhibitor. Journal of medicinal chemistry (2023)
Richard Wang, Camilla Ascanelli, Ahmed Abdelbaki, Alex Fung, Tim Rasmusson, Iacovos N Michaelides, Karen Roberts, Catherine Lindon
Selective targeting of non-centrosomal AURKA functions through use of a targeted protein degradation tool. Communications biology 4 (1) (2021)
Matthias R Bauer, Paolo Di Fruscia, Simon C C Lucas, Iacovos N Michaelides, Jennifer E Nelson, R Ian Storer, Benjamin C Whitehurst
Put a ring on it: application of small aliphatic rings in medicinal chemistry. RSC medicinal chemistry 12 (4) (2021)