Jacek Plewka

ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 21

Top Venues

ACS medicinal chemistry letters

Journal of medicinal chemistry

Nucleic acids research

RSC medicinal chemistry

Uniwersytet Jagielloński w Krakowie

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Uniwersytet Jagielloński w Krakowie Sep 01 2018

Poland

Post-doc :: Department of Chemistry

Publications

Aleksandra Hec-Gałązka, Urszula Tyrcha, Jan Barczyński, Przemyslaw Bielski, Michał Mikitiuk, Ganna P Gudz, Radoslaw Kitel, Bogdan M Musielak, Jacek Plewka, Tomasz Sitar, Tad A Holak
Nonsymmetrically Substituted 1,1'-Biphenyl-Based Small Molecule Inhibitors of the PD-1/PD-L1 Interaction. ACS medicinal chemistry letters 15 (6) (2024)
Robin van der Straat, Rosalie Draijer, Ewa Surmiak, Roberto Butera, Lennart Land, Katarzyna Magiera-Mularz, Bogdan Musielak, Jacek Plewka, Tad A Holak, Alexander S S Dömling
1,5-Disubstituted tetrazoles as PD-1/PD-L1 antagonists. RSC medicinal chemistry 15 (4) (2024)
Robin van der Straat, Rosalie Draijer, Ewa Surmiak, Roberto Butera, Lennart Land, Katarzyna Magiera-Mularz, Bogdan Musielak, Jacek Plewka, Tad A Holak, Alexander S S Dömling
1,5-Disubstituted tetrazoles as PD-1/PD-L1 antagonists. RSC medicinal chemistry 15 (4) (2024)
Aleksandra Hec-Gałązka, Urszula Tyrcha, Jan Barczyński, Przemyslaw Bielski, Michał Mikitiuk, Ganna P Gudz, Radoslaw Kitel, Bogdan M Musielak, Jacek Plewka, Tomasz Sitar, Tad A Holak
Nonsymmetrically Substituted 1,1'-Biphenyl-Based Small Molecule Inhibitors of the PD-1/PD-L1 Interaction. ACS medicinal chemistry letters 15 (6) (2024)
Alex Matsuda, Jacek Plewka, Michał Rawski, André Mourão, Weronika Zajko, Till Siebenmorgen, Leanid Kresik, Kinga Lis, Alisha N Jones, Magdalena Pachota, Abdulkarim Karim, Kinga Hartman, Shivlee Nirwal, Ravi Sonani, Yuliya Chykunova, Igor Minia, Paweł Mak, Markus Landthaler, Marcin Nowotny, Grzegorz Dubin, Michael Sattler, Piotr Suder, Grzegorz M Popowicz, Krzysztof Pyrc, Anna Czarna
Despite the odds: formation of the SARS-CoV-2 methylation complex. Nucleic acids research (2024)
Alex Matsuda, Jacek Plewka, Michał Rawski, André Mourão, Weronika Zajko, Till Siebenmorgen, Leanid Kresik, Kinga Lis, Alisha N Jones, Magdalena Pachota, Abdulkarim Karim, Kinga Hartman, Shivlee Nirwal, Ravi Sonani, Yuliya Chykunova, Igor Minia, Paweł Mak, Markus Landthaler, Marcin Nowotny, Grzegorz Dubin, Michael Sattler, Piotr Suder, Grzegorz M Popowicz, Krzysztof Pyrc, Anna Czarna
Despite the odds: formation of the SARS-CoV-2 methylation complex. Nucleic acids research 52 (11) (2024)
Alex Matsuda, Jacek Plewka, Michał Rawski, André Mourão, Weronika Zajko, Till Siebenmorgen, Leanid Kresik, Kinga Lis, Alisha N Jones, Magdalena Pachota, Abdulkarim Karim, Kinga Hartman, Shivlee Nirwal, Ravi Sonani, Yuliya Chykunova, Igor Minia, Paweł Mak, Markus Landthaler, Marcin Nowotny, Grzegorz Dubin, Michael Sattler, Piotr Suder, Grzegorz M Popowicz, Krzysztof Pyrc, Anna Czarna
Despite the odds: formation of the SARS-CoV-2 methylation complex. Nucleic acids research 52 (11) (2024)
Ewa Surmiak, Julia Ząber, Jacek Plewka, Grzegorz Wojtanowicz, Justyna Kocik-Krol, Oskar Kruc, Damian Muszak, Ismael Rodriguez, Bogdan M Musielak, Monica Viviano, Sabrina Castellano, Łukasz Skalniak, Katarzyna Magiera-Mularz, Tad A Holak, Justyna Kalinowska-Tłuścik
Solubilizer Tag Effect on PD-L1/Inhibitor Binding Properties for m -Terphenyl Derivatives. ACS medicinal chemistry letters 15 (1) (2023)
Ewa Surmiak, Julia Ząber, Jacek Plewka, Grzegorz Wojtanowicz, Justyna Kocik-Krol, Oskar Kruc, Damian Muszak, Ismael Rodriguez, Bogdan M Musielak, Monica Viviano, Sabrina Castellano, Łukasz Skalniak, Katarzyna Magiera-Mularz, Tad A Holak, Justyna Kalinowska-Tłuścik
Solubilizer Tag Effect on PD-L1/Inhibitor Binding Properties for m -Terphenyl Derivatives. ACS medicinal chemistry letters 15 (1) (2023)
Marta A Ważyńska, Roberto Butera, Marta Requesens, Annechien Plat, Tryfon Zarganes-Tzitzikas, Constantinos G Neochoritis, Jacek Plewka, Lukasz Skalniak, Justyna Kocik-Krol, Bogdan Musielak, Katarzyna Magiera-Mularz, Ismael Rodriguez, Simon N Blok, Marco de Bruyn, Hans W Nijman, Philip H Elsinga, Tad A Holak, Alexander S S Dömling
Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors. Journal of medicinal chemistry (2023)
Hua Zhang, Shijia Zhou, Jacek Plewka, Caiyun Wu, Mengyu Zhu, Qimeng Yu, Bogdan M Musielak, Xiao Wang, Annoor Awadasseid, Katarzyna Magiera-Mularz, Yanling Wu, Wen Zhang
Design, Synthesis, and Antitumor Activity Evaluation of 2-Arylmethoxy-4-(2,2'-dihalogen-substituted biphenyl-3-ylmethoxy) Benzylamine Derivatives as Potent PD-1/PD-L1 Inhibitors. Journal of medicinal chemistry (2023)
Marta Cegłowska, Karolina Szubert, Beata Grygier, Marzena Lenart, Jacek Plewka, Aleksandra Milewska, Kinga Lis, Artur Szczepański, Yuliya Chykunova, Emilia Barreto Duran, Krzysztof Pyrc, Alicja Kosakowska, Hanna Mazur-Marzec
Pseudanabaena galeata CCNP1313-Biological Activity and Peptides Production. Toxins 14 (5) (2022)
Damian Muszak, Ewa Surmiak, Jacek Plewka, Katarzyna Magiera-Mularz, Justyna Kocik-Krol, Bogdan M Musielak, Dominik Sala, Radoslaw Kitel, Malgorzata Stec, Kazimierz Weglarczyk, Maciej Siedlar, Alexander S S Dömling, Łukasz Skalniak, Tad A Holak
Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction. Journal of medicinal chemistry 64 (15) (2021)
Roberto Butera, Marta Ważyńska, Katarzyna Magiera-Mularz, Jacek Plewka, Bogdan M Musielak, Ewa Surmiak, Dominik Sala, Radoslaw Kitel, Marco de Bruyn, Hans W Nijman, Philip H Elsinga, Tad A Holak, Alexander S S Dömling
Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists. ACS medicinal chemistry letters 12 (5) (2021)
Ewa Surmiak, Katarzyna Magiera-Mularz, Bogdan M Musielak, Damian Muszak, Justyna Kocik-Krol, Radoslaw Kitel, Jacek Plewka, Tad A Holak, Łukasz Skalniak
PD-L1 Inhibitors: Different Classes, Activities, and Mechanisms of Action. International journal of molecular sciences 22 (21) (2021)
Magdalena Konieczny, Bogdan M Musielak, Justyna Kocik-Krol, Łukasz Skalniak, Dominik Sala, Miroslawa Czub, Katarzyna Magiera-Mularz, Ismael Rodriguez, Maja Myrcha, Malgorzata Stec, Maciej Siedlar, Tad A Holak, Jacek Plewka
Di-bromo-Based Small-Molecule Inhibitors of the PD-1/PD-L1 Immune Checkpoint. Journal of medicinal chemistry 63 (19) (2020)
Bogdan M Musielak, Weronika Janczyk, Ismael Rodriguez, Jacek Plewka, Dominik Sala, Katarzyna Magiera-Mularz, Tad A Holak
Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions. Molecules (Basel, Switzerland) 25 (13) (2020)
Bogdan M Musielak, Justyna Kocik-Krol, Łukasz Skalniak, Katarzyna Magiera-Mularz, Dominik Sala, Miroslawa Czub, Malgorzata Stec, Maciej Siedlar, Tad A Holak, Jacek Plewka
CA-170 - A Potent Small-Molecule PD-L1 Inhibitor or Not? Molecules (Basel, Switzerland) 24 (15) (2019)
Gonçalo F L da Silva, Jacek Plewka, Helga C Lichtenegger, Ana Cristina Dias-Cabral, Alois Jungbauer, Rupert Tscheließnig
The pearl necklace model in protein A chromatography: Molecular mechanisms at the resin interface. Biotechnology and bioengineering 116 (1) (2018)
Jacek Plewka, Gonçalo L Silva, Rupert Tscheließnig, Harald Rennhofer, Ana Cristina Dias-Cabral, Alois Jungbauer, Helga C Lichtenegger
Antibody adsorption in protein-A affinity chromatography - in situ measurement of nanoscale structure by small-angle X-ray scattering. Journal of separation science 41 (22) (2018)
Marcin D Roganowicz, Sevnur Komurlu, Santanu Mukherjee, Jacek Plewka, Steven L Alam, Katarzyna A Skorupka, Yueping Wan, Damian Dawidowski, David S Cafiso, Barbie K Ganser-Pornillos, Edward M Campbell, Owen Pornillos
TRIM5α SPRY/coiled-coil interactions optimize avid retroviral capsid recognition. PLoS pathogens 13 (10) (2017)

Jacek Plewka.css-eqlu8i{font-size:small;padding-left:4px;}

Publication Activity (10 Years)

Top Topics

Top Venues

Jacek Plewka