Marcin Dra G (Marcin Drąg, Marcin Drag)

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 33

Top Topics

Respiratory Syndrome Coronavirus

Fluorescent Probe

Crystal Structure

Top Venues

Protein science : a publication of the Protein Society

Journal of medicinal chemistry

ACS chemical neuroscience

Chemical science

This page only lists publications with an associated author ORCID identifier.

Publications

Griffin J Davis, Anthony O Omole, Yejin Jung, Wioletta Rut, Ronald Holewinski, Kiall F Suazo, Hong-Rae Kim, Mo Yang, Thorkell Andresson, Marcin Dra G, Euna Yoo
Chemical tools to define and manipulate interferon-inducible Ubl protease USP18. bioRxiv : the preprint server for biology (2024)
Wioletta Rut, Katarzyna Groborz, Xinyuanyuan Sun, Rolf Hilgenfeld, Marcin Dra G
Profiling of coronaviral M pro and enteroviral 3C pro specificity provides a framework for the development of broad-spectrum antiviral compounds. Protein science : a publication of the Protein Society 33 (9) (2024)
Griffin J Davis, Anthony O Omole, Yejin Jung, Wioletta Rut, Ronald Holewinski, Kiall F Suazo, Hong-Rae Kim, Mo Yang, Thorkell Andresson, Marcin Dra G, Euna Yoo
Chemical tools to define and manipulate interferon-inducible Ubl protease USP18. bioRxiv : the preprint server for biology (2024)
Natalia Malek, Radoslaw Gladysz, Natalia Stelmach, Marcin Dra G
Targeting Microglial Immunoproteasome: A Novel Approach in Neuroinflammatory-Related Disorders. ACS chemical neuroscience (2024)
Natalia Malek, Radoslaw Gladysz, Natalia Stelmach, Marcin Dra G
Targeting Microglial Immunoproteasome: A Novel Approach in Neuroinflammatory-Related Disorders. ACS chemical neuroscience 15 (14) (2024)
Natalia Malek, Radoslaw Gladysz, Natalia Stelmach, Marcin Dra G
Targeting Microglial Immunoproteasome: A Novel Approach in Neuroinflammatory-Related Disorders. ACS chemical neuroscience 15 (14) (2024)
Matthew W Mahoney, Jonathan Helander, Anoopjit S Kooner, Mariah Norman, Vishnu C Damalanka, Paolo De Bona, Paulina Kasperkiewicz, Wioletta Rut, Marcin Poreba, Maithri M Kashipathy, Kevin P Battaile, Scott Lovell, Anthony J O'Donoghue, Charles S Craik, Marcin Dra G, James W Janetka
Use of protease substrate specificity screening in the rational design of selective protease inhibitors with unnatural amino acids: Application to HGFA, matriptase, and hepsin. Protein science : a publication of the Protein Society 33 (8) (2024)
Natalia Malek, Radoslaw Gladysz, Natalia Stelmach, Marcin Dra G
Targeting Microglial Immunoproteasome: A Novel Approach in Neuroinflammatory-Related Disorders. ACS chemical neuroscience 15 (14) (2024)
Matthew W Mahoney, Jonathan Helander, Anoopjit S Kooner, Mariah Norman, Vishnu C Damalanka, Paolo De Bona, Paulina Kasperkiewicz, Wioletta Rut, Marcin Poreba, Maithri M Kashipathy, Kevin P Battaile, Scott Lovell, Anthony J O'Donoghue, Charles S Craik, Marcin Dra G, James W Janetka
Use of protease substrate specificity screening in the rational design of selective protease inhibitors with unnatural amino acids: Application to HGFA, matriptase, and hepsin. Protein science : a publication of the Protein Society 33 (8) (2024)
Wioletta Rut, Katarzyna Groborz, Xinyuanyuan Sun, Rolf Hilgenfeld, Marcin Dra G
Profiling of coronaviral M pro and enteroviral 3C pro specificity provides a framework for the development of broad-spectrum antiviral compounds. Protein science : a publication of the Protein Society 33 (9) (2024)
Matthew W Mahoney, Jonathan Helander, Anoopjit S Kooner, Mariah Norman, Vishnu C Damalanka, Paolo De Bona, Paulina Kasperkiewicz, Wioletta Rut, Marcin Poreba, Maithri M Kashipathy, Kevin P Battaile, Scott Lovell, Anthony J O'Donoghue, Charles S Craik, Marcin Dra G, James W Janetka
Use of protease substrate specificity screening in the rational design of selective protease inhibitors with unnatural amino acids: Application to HGFA, matriptase, and hepsin. Protein science : a publication of the Protein Society 33 (8) (2024)
Patrick Y A Reinke, Edmarcia Elisa de Souza, Sebastian Günther, Sven Falke, Julia Lieske, Wiebke Ewert, Jure Loboda, Alexander Herrmann, Aida Rahmani Mashhour, Katarina Karničar, Aleksandra Usenik, Nataša Lindič, Andreja Sekirnik, Viviane Fongaro Botosso, Gláucia Maria Machado Santelli, Josana Kapronezai, Marcelo Valdemir de Araújo, Taiana Tainá Silva-Pereira, Antônio Francisco de Souza Filho, Mariana Silva Tavares, Lizdany Flórez-Álvarez, Danielle Bruna Leal de Oliveira, Edison Luiz Durigon, Paula Roberta Giaretta, Marcos Bryan Heinemann, Maurice Hauser, Brandon Seychell, Hendrik Böhler, Wioletta Rut, Marcin Dra G, Tobias Beck, Russell J Cox, Henry N Chapman, Christian Betzel, Wolfgang Brehm, Winfried Hinrichs, Gregor Ebert, Sharissa L Latham, Ana Marcia de Sá Guimarães, Dusan Turk, Carsten Wrenger, Alke Meents
Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections. Communications biology 6 (1) (2023)
Yong Zou, Igor Sabljić, Natalia Horbach, Adrian N Dauphinee, Anna Åsman, Lucia Sancho Temino, Alyona E Minina, Marcin Dra G, Simon Stael, Marcin Poręba, Jerry Ståhlberg, Peter V Bozhkov
Thermoprotection by a cell membrane-localized metacaspase in a green alga. The Plant cell (2023)
Sylwia Modrzycka, Sonia Kołt, Ty E Adams, Stanisław Potoczek, James A Huntington, Paulina Kasperkiewicz-Wasilewska, Marcin Dra G
Fluorescent Activity-Based Probe To Image and Inhibit Factor XIa Activity in Human Plasma. Journal of medicinal chemistry 66 (6) (2023)
Sylwia Modrzycka, Sonia Kołt, Ty E Adams, Stanisław Potoczek, James A Huntington, Paulina Kasperkiewicz-Wasilewska, Marcin Dra G
Fluorescent Activity-Based Probe To Image and Inhibit Factor XIa Activity in Human Plasma. Journal of medicinal chemistry (2023)
Sizhu Amelia Chen, Elena Arutyunova, Jimmy Lu, Muhammad Bashir Khan, Wioletta Rut, Mikolaj Zmudzinski, Shima Shahbaz, Jegan Iyyathurai, Eman W Moussa, Zoe Turner, Bing Bai, Tess Lamer, James A Nieman, John C Vederas, Olivier Julien, Marcin Dra G, Shokrollah Elahi, Howard S Young, Mary Joanne Lemieux
SARS-CoV-2 M pro Protease Variants of Concern Display Altered Viral Substrate and Cell Host Target Galectin-8 Processing but Retain Sensitivity toward Antivirals. ACS central science 9 (4) (2023)
Sizhu Amelia Chen, Elena Arutyunova, Jimmy Lu, Muhammad Bashir Khan, Wioletta Rut, Mikolaj Zmudzinski, Shima Shahbaz, Jegan Iyyathurai, Eman W Moussa, Zoe Turner, Bing Bai, Tess Lamer, James A Nieman, John C Vederas, Olivier Julien, Marcin Dra G, Shokrollah Elahi, Howard S Young, Mary Joanne Lemieux
SARS-CoV-2 M pro Protease Variants of Concern Display Altered Viral Substrate and Cell Host Target Galectin-8 Processing but Retain Sensitivity toward Antivirals. ACS central science 9 (4) (2023)
Sylwia Modrzycka, Sonia Kołt, Ty E Adams, Stanisław Potoczek, James A Huntington, Paulina Kasperkiewicz-Wasilewska, Marcin Dra G
Fluorescent Activity-Based Probe To Image and Inhibit Factor XIa Activity in Human Plasma. Journal of medicinal chemistry 66 (6) (2023)
Radoslaw Gladysz, Natalia Malek, Wioletta Rut, Marcin Dra G
Investigation of the P1' and P2' sites of IQF substrates and their selectivity toward 20S proteasome subunits. Biological chemistry (2022)
Agata P Perlinska, Adam Stasiulewicz, Mai Lan Nguyen, Karolina W Swiderska, Mikolaj Zmudzinski, Alicja W Maksymiuk, Marcin Dra G, Joanna Ida Sulkowska
Amino acid variants of SARS-CoV-2 papain-like protease have impact on drug binding. PLoS computational biology 18 (11) (2022)
Sylwia Modrzycka, Sonia Kołt, Stéphanie G I Polderdijk, Ty E Adams, Stanisław Potoczek, James A Huntington, Paulina Kasperkiewicz-Wasilewska, Marcin Dra G
Parallel imaging of coagulation pathway proteases activated protein C, thrombin, and factor Xa in human plasma. Chemical science 13 (23) (2022)
Izabela Nawrot-Hadzik, Mikolaj Zmudzinski, Adam Matkowski, Robert Preissner, Małgorzata Kęsik-Brodacka, Jakub Hadzik, Marcin Dra G, Renata Abel
Reynoutria Rhizomes as a Natural Source of SARS-CoV-2 Mpro Inhibitors-Molecular Docking and In Vitro Study. Pharmaceuticals (Basel, Switzerland) 14 (8) (2021)
Izabela Maluch, Justyna Grzymska, Scott J Snipas, Guy S Salvesen, Marcin Dra G
Evaluation of the effects of phosphorylation of synthetic peptide substrates on their cleavage by caspase-3 and -7. The Biochemical journal 478 (12) (2021)
Marcin Poręba, Katarzyna M Groborz, Wioletta Rut, Milind Pore, Scott J Snipas, Matej Vizovisek, Boris Turk, Peter Kuhn, Marcin Dra G, Guy S Salvesen
Multiplexed Probing of Proteolytic Enzymes Using Mass Cytometry-Compatible Activity-Based Probes. Journal of the American Chemical Society 142 (39) (2020)
Wioletta Rut, Mikolaj Zmudzinski, Scott J Snipas, Miklos Bekes, Tony T Huang, Marcin Dra G
Engineered unnatural ubiquitin for optimal detection of deubiquitinating enzymes. Chemical science 11 (23) (2020)
Wioletta Rut, Zongyang Lv, Mikolaj Zmudzinski, Stephanie Patchett, Digant Nayak, Scott J Snipas, Farid El Oualid, Tony T Huang, Miklós Békés, Marcin Dra G, Shaun K Olsen
Activity profiling and crystal structures of inhibitor-bound SARS-CoV-2 papain-like protease: A framework for anti-COVID-19 drug design. Science advances 6 (42) (2020)
Sonia Kolt, Tomasz Janiszewski, Dion Kaiserman, Sylwia Modrzycka, Scott J Snipas, Guy Salvesen, Marcin Dra G, Phillip I Bird, Paulina Kasperkiewicz-Wasilewska
Detection of Active Granzyme A in NK92 Cells with Fluorescent Activity-Based Probe. Journal of medicinal chemistry 63 (6) (2020)
Wioletta Rut, Katarzyna Groborz, Linlin Zhang, Xinyuanyuan Sun, Mikolaj Zmudzinski, Bartłomiej Pawlik, Xinyu Wang, Dirk Jochmans, Johan Neyts, Wojciech Mlynarski, Rolf Hilgenfeld, Marcin Dra G
SARS-CoV-2 Mpro inhibitors and activity-based probes for patient-sample imaging. Nature chemical biology 17 (2) (2020)
Marcin Poręba, Katarzyna Groborz, Matej Vizovisek, Marco Maruggi, Dusan Turk, Boris Turk, Garth Powis, Marcin Dra G, Guy S Salvesen
Fluorescent probes towards selective cathepsin B detection and visualization in cancer cells and patient samples. Chemical science 10 (36) (2019)
Izabela Maluch, Justyna Czarna, Marcin Dra G
Applications of Unnatural Amino Acids in Protease Probes. Chemistry, an Asian journal 14 (23) (2019)
Wioletta Rut, Marcin Poręba, Paulina Kasperkiewicz, Scott J Snipas, Marcin Dra G
Selective Substrates and Activity-Based Probes for Imaging of the Human Constitutive 20S Proteasome in Cells and Blood Samples. Journal of medicinal chemistry 61 (12) (2018)
Marcin Poreba, Wioletta Rut, Matej Vizovisek, Katarzyna Groborz, Paulina Kasperkiewicz, Darren Finlay, Kristiina Vuori, Dusan Turk, Boris Turk, Guy S Salvesen, Marcin Dra G
Selective imaging of cathepsin L in breast cancer by fluorescent activity-based probes. Chemical science 9 (8) (2018)
Paulina Kasperkiewicz, Yoav Altman, Maximiliano D'Angelo, Guy S Salvesen, Marcin Dra G
Toolbox of Fluorescent Probes for Parallel Imaging Reveals Uneven Location of Serine Proteases in Neutrophils. Journal of the American Chemical Society 139 (29) (2017)