Michael Gajhede

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 14

Top Venues

Research square

Journal of medicinal chemistry

The FEBS journal

Chembiochem : a European journal of chemical biology

Københavns Universitet

Københavns Universitet (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Københavns Universitet Sep 01 2002

Denmark

Professor :: Drug Design and Pharmacology

Education History

Københavns Universitet Jul 15 1984 - Jul 15 1988

Denmark

PHD :: Chemistry

Publications

David E Gloriam, Thor Thorsen, Yashraj Kulkarni, David A Sykes, Andreas Bøggild, Taner Drace, Pattarin Hompluem, Christos Iliopoulos-Tsoutsouvas, Spyros P Nikas, Henrik Daver, Alexandros Makriyannis, Poul Nissen, Michael Gajhede, Dmitry B Veprintsev, Thomas Boesen, Jette Kastrup
Structural basis of Δ9-THC analog activity at the Cannabinoid 1 receptor. Research square (2024)
David E Gloriam, Thor Thorsen, Yashraj Kulkarni, David A Sykes, Andreas Bøggild, Taner Drace, Pattarin Hompluem, Christos Iliopoulos-Tsoutsouvas, Spyros P Nikas, Henrik Daver, Alexandros Makriyannis, Poul Nissen, Michael Gajhede, Dmitry B Veprintsev, Thomas Boesen, Jette Kastrup
Structural basis of Δ 9 -THC analog activity at the Cannabinoid 1 receptor. Research square (2024)
Yasmin Bay, Raminta Venskutonytė, Stine M Frantsen, Thor S Thorsen, Maria Musgaard, Karla A Frydenvang, Pierre Francotte, Bernard Pirotte, Philip Charles Biggin, Anders S Kristensen, Thomas Boesen, Darryl S Pickering, Michael Gajhede, Jette Sandholm Kastrup
Small-molecule positive allosteric modulation of homomeric kainate receptors GluK1-3: development of screening assays and insight into GluK3 structure. The FEBS journal 291 (7) (2024)
David E Gloriam, Thor Thorsen, Yashraj Kulkarni, David A Sykes, Andreas Bøggild, Taner Drace, Pattarin Hompluem, Christos Iliopoulos-Tsoutsouvas, Spyros P Nikas, Henrik Daver, Alexandros Makriyannis, Poul Nissen, Michael Gajhede, Dmitry B Veprintsev, Thomas Boesen, Jette Kastrup
Structural basis of Δ9-THC analog activity at the Cannabinoid 1 receptor. Research square (2024)
Yasmin Bay, Raminta Venskutonytė, Stine M Frantsen, Thor S Thorsen, Maria Musgaard, Karla A Frydenvang, Pierre Francotte, Bernard Pirotte, Philip Charles Biggin, Anders S Kristensen, Thomas Boesen, Darryl S Pickering, Michael Gajhede, Jette Sandholm Kastrup
Small-molecule positive allosteric modulation of homomeric kainate receptors GluK1-3: development of screening assays and insight into GluK3 structure. The FEBS journal 291 (7) (2024)
Yasmin Bay, Raminta Venskutonytė, Stine M Frantsen, Thor S Thorsen, Maria Musgaard, Karla A Frydenvang, Pierre Francotte, Bernard Pirotte, Philip Charles Biggin, Anders S Kristensen, Thomas Boesen, Darryl S Pickering, Michael Gajhede, Jette Sandholm Kastrup
Small-molecule positive allosteric modulation of homomeric kainate receptors GluK1-3: development of screening assays and insight into GluK3 structure. The FEBS journal (2023)
Jie Zang, Felix Peters, Yves Cambet, Eugenia Cifuentes-Pagano, Munira Mohamed Shishay Hissabu, Christopher M Dustin, Lars Henrik Svensson, Martin Mariboe Olesen, Mathias Feldt Lomholt Poulsen, Stig Jacobsen, Pernille Sønderby Tuelung, Dilip Narayanan, Annette Eva Langkilde, Michael Gajhede, Patrick J Pagano, Vincent Jaquet, Frederik Vilhardt, Anders Bach
Targeting NOX2 with Bivalent Small-Molecule p47phox-p22phox Inhibitors. Journal of medicinal chemistry (2023)
Sara Dam Kobberø, Michael Gajhede, Osman Asghar Mirza, Søren Kløverpris, Troels Rønn Kjær, Jakob Hauge Mikkelsen, Thomas Boesen, Claus Oxvig
Structure of the proteolytic enzyme PAPP-A with the endogenous inhibitor stanniocalcin-2 reveals its inhibitory mechanism. Nature communications 13 (1) (2022)
Dilip Narayanan, Kim T Tran, Jakob S Pallesen, Sara M Ø Solbak, Yuting Qin, Elina Mukminova, Martina Luchini, Kristina O Vasilyeva, Dorleta González Chichón, Georgia Goutsiou, Cecilie Poulsen, Nanna Haapanen, Grzegorz M Popowicz, Michael Sattler, David Olagnier, Michael Gajhede, Anders Bach
Development of Noncovalent Small-Molecule Keap1-Nrf2 Inhibitors by Fragment-Based Drug Discovery. Journal of medicinal chemistry 65 (21) (2022)
Jakob S Pallesen, Dilip Narayanan, Kim T Tran, Sara M Ø Solbak, Giuseppe Marseglia, Louis M E Sørensen, Lars J Høj, Federico Munafò, Rosa M C Carmona, Anthony D Garcia, Haritha L Desu, Roberta Brambilla, Tommy N Johansen, Grzegorz M Popowicz, Michael Sattler, Michael Gajhede, Anders Bach
Deconstructing Noncovalent Kelch-like ECH-Associated Protein 1 (Keap1) Inhibitors into Fragments to Reconstruct New Potent Compounds. Journal of medicinal chemistry 64 (8) (2021)
Malene J Petersen, Xamuel L Lund, Susan J Semple, Bevan J Buirchell, Henrik Franzyk, Michael Gajhede, Kenneth Thermann Kongstad, Jan Stenvang, Dan Staerk
Reversal of ABCG2/BCRP-Mediated Multidrug Resistance by 5,3',5'-Trihydroxy-3,6,7,4'-Tetramethoxyflavone Isolated from the Australian Desert Plant Eremophila galeata Chinnock. Biomolecules 11 (10) (2021)
Sarah E Jones, Lars Olsen, Jerzy Dorosz, Signe T Seger, Jan L Andersson, Line H Kristensen, Michael Gajhede
Peptides Derived from Histone 3 and Modified at Position 18 Inhibit Histone Demethylase KDM6 Enzymes. Chembiochem : a European journal of chemical biology 19 (17) (2018)
Jerzy Dorosz, Lars Olsen, Signe Teuber Seger, Cornelia Steinhauer, Giorgos Bouras, Charlotte Helgstrand, Anders Wiuf, Michael Gajhede
Structure-Based Design of a New Scaffold for Cell-Penetrating Peptidic Inhibitors of the Histone Demethylase PHF8. Chembiochem : a European journal of chemical biology 18 (14) (2017)
Sarah E Jones, Lars Olsen, Michael Gajhede
Structural Basis of Histone Demethylase KDM6B Histone 3 Lysine 27 Specificity. Biochemistry 57 (5) (2017)

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Publication Activity (10 Years)

Top Topics

Top Venues

Michael Gajhede