Peter Brust

Publication Activity (10 Years)

Years Active: 2016-2023
Publications (10 Years): 38

Top Topics

Toxoplasma Gondii

Subarachnoid Hemorrhage

Top Venues

International journal of molecular sciences

Molecules (Basel, Switzerland)

Pharmaceuticals (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Sean Harrington, Jacob Pyche, Andrew R Burns, Tina Spalholz, Kaetlyn T Ryan, Rachel J Baker, Justin Ching, Lucien Rufener, Mark Lautens, Daniel Kulke, Alexandre Vernudachi, Mostafa Zamanian, Winnie Deuther-Conrad, Peter Brust, Peter J Roy
Nemacol is a small molecule inhibitor of C. elegans vesicular acetylcholine transporter with anthelmintic potential. Nature communications 14 (1) (2023)
Barbara Wenzel, Maximilian Schmid, Rodrigo Teodoro, Rareş-Petru Moldovan, Thu Hang Lai, Franziska Mitrach, Klaus Kopka, Björn Fischer, Michaela Schulz-Siegmund, Peter Brust, Michael C Hacker
Radiofluorination of an Anionic, Azide-Functionalized Teroligomer by Copper-Catalyzed Azide-Alkyne Cycloaddition. Nanomaterials (Basel, Switzerland) 13 (14) (2023)
Sean Harrington, Jacob Pyche, Andrew R Burns, Tina Spalholz, Kaetlyn T Ryan, Rachel J Baker, Justin Ching, Lucien Rufener, Mark Lautens, Daniel Kulke, Alexandre Vernudachi, Mostafa Zamanian, Winnie Deuther-Conrad, Peter Brust, Peter J Roy
Nemacol is a small molecule inhibitor of C. elegans vesicular acetylcholine transporter with anthelmintic potential. Nature communications 14 (1) (2023)
Rodrigo Teodoro, Daniel Gündel, Winnie Deuther-Conrad, Aleksandr Kazimir, Magali Toussaint, Barbara Wenzel, Guy Bormans, Evamarie Hey-Hawkins, Klaus Kopka, Peter Brust, Rareş-Petru Moldovan
Synthesis, Structure-Activity Relationships, Radiofluorination, and Biological Evaluation of [ 18 F]RM365, a Novel Radioligand for Imaging the Human Cannabinoid Receptor Type 2 (CB2R) in the Brain with PET. Journal of medicinal chemistry (2023)
Lea Ueberham, Daniel Gündel, Martin Kellert, Winnie Deuther-Conrad, Friedrich-Alexander Ludwig, Peter Lönnecke, Aleksandr Kazimir, Klaus Kopka, Peter Brust, Rareş-Petru Moldovan, Evamarie Hey-Hawkins
Development of the High-Affinity Carborane-Based Cannabinoid Receptor Type 2 PET Ligand [ 18 F]LUZ5- d 8 . Journal of medicinal chemistry (2023)
Barbara Wenzel, Stefan R Fritzsche, Magali Toussaint, Detlef Briel, Klaus Kopka, Peter Brust, Matthias Scheunemann, Winnie Deuther-Conrad
Radiosynthesis and Preclinical Evaluation of an 18 F-Labeled Triazolopyridopyrazine-Based Inhibitor for Neuroimaging of the Phosphodiesterase 2A (PDE2A). Pharmaceuticals (Basel, Switzerland) 15 (10) (2022)
Jan H Voss, Haneen Al-Hroub, Robin Gedschold, Jennifer M Dietrich, Evelyn Gaffal, Marieta Toma, Stefan Kehraus, Gabriele M König, Peter Brust, Bernd K Fleischmann, Daniela Wenzel, Winnie Deuther-Conrad, Christa Elisabeth Müller
Imaging of Gα q Proteins in Mouse and Human Organs and Tissues. Pharmaceutics 15 (1) (2022)
Thu Hang Lai, Barbara Wenzel, Rareş-Petru Moldovan, Peter Brust, Klaus Kopka, Rodrigo Teodoro
Automated radiosynthesis of the adenosine A 2A receptor-targeting radiotracer [ 18 F]FLUDA. Journal of labelled compounds & radiopharmaceuticals 65 (6) (2022)
Daniel Gündel, Winnie Deuther-Conrad, Lea Ueberham, Sarandeep Kaur, Elina Otikova, Rodrigo Teodoro, Magali Toussaint, Thu Hang Lai, Oliver Clauß, Matthias Scheunemann, Guy Bormans, Michael Bachmann, Klaus Kopka, Peter Brust, Rareş-Petru Moldovan
Structure-Based Design, Optimization, and Development of [ 18 F]LU13: A Novel Radioligand for Cannabinoid Receptor Type 2 Imaging in the Brain with PET. Journal of medicinal chemistry 65 (13) (2022)
Jan H Voss, Haneen Al-Hroub, Robin Gedschold, Jennifer M Dietrich, Evelyn Gaffal, Marieta Toma, Stefan Kehraus, Gabriele M König, Peter Brust, Bernd K Fleischmann, Daniela Wenzel, Winnie Deuther-Conrad, Christa Elisabeth Müller
Imaging of Gα q Proteins in Mouse and Human Organs and Tissues. Pharmaceutics 15 (1) (2022)
Oliver Clauß, Linda Schäker-Hübner, Barbara Wenzel, Magali Toussaint, Winnie Deuther-Conrad, Daniel Gündel, Rodrigo Teodoro, Sladjana Dukić-Stefanović, Friedrich-Alexander Ludwig, Klaus Kopka, Peter Brust, Finn K Hansen, Matthias Scheunemann
Development and Biological Evaluation of the First Highly Potent and Specific Benzamide-Based Radiotracer [ 18 F]BA3 for Imaging of Histone Deacetylases 1 and 2 in Brain. Pharmaceuticals (Basel, Switzerland) 15 (3) (2022)
Daniel Gündel, Magali Toussaint, Thu Hang Lai, Winnie Deuther-Conrad, Paul Cumming, Susann Schröder, Rodrigo Teodoro, Rareş-Petru Moldovan, Francisco Pan-Montojo, Bernhard Sattler, Klaus Kopka, Osama Sabri, Peter Brust
Quantitation of the A 2A Adenosine Receptor Density in the Striatum of Mice and Pigs with [ 18 F]FLUDA by Positron Emission Tomography. Pharmaceuticals (Basel, Switzerland) 15 (5) (2022)
Franziska Mitrach, Maximilian Schmid, Magali Toussaint, Sladjana Dukic-Stefanovic, Winnie Deuther-Conrad, Heike Franke, Alexander Ewe, Achim Aigner, Christian Wölk, Peter Brust, Michael C Hacker, Michaela Schulz-Siegmund
Amphiphilic Anionic Oligomer-Stabilized Calcium Phosphate Nanoparticles with Prospects in siRNA Delivery via Convection-Enhanced Delivery. Pharmaceutics 14 (2) (2022)
Daniel Gündel, Thu Hang Lai, Sladjana Dukic-Stefanovic, Rodrigo Teodoro, Winnie Deuther-Conrad, Magali Toussaint, Klaus Kopka, Rareş-Petru Moldovan, Peter Boknik, Britt Hofmann, Ulrich Gergs, Joachim Neumann, Peter Brust
Non-Invasive Assessment of Locally Overexpressed Human Adenosine 2A Receptors in the Heart of Transgenic Mice. International journal of molecular sciences 23 (3) (2022)
Jan H Voss, Haneen Al-Hroub, Robin Gedschold, Jennifer M Dietrich, Evelyn Gaffal, Marieta Toma, Stefan Kehraus, Gabriele M König, Peter Brust, Bernd K Fleischmann, Daniela Wenzel, Winnie Deuther-Conrad, Christa Elisabeth Müller
Imaging of Gα q Proteins in Mouse and Human Organs and Tissues. Pharmaceutics 15 (1) (2022)
Jan H Voss, Haneen Al-Hroub, Robin Gedschold, Jennifer M Dietrich, Evelyn Gaffal, Marieta Toma, Stefan Kehraus, Gabriele M König, Peter Brust, Bernd K Fleischmann, Daniela Wenzel, Winnie Deuther-Conrad, Christa Elisabeth Müller
Imaging of Gα q Proteins in Mouse and Human Organs and Tissues. Pharmaceutics 15 (1) (2022)
Jan H Voss, Haneen Al-Hroub, Robin Gedschold, Jennifer M Dietrich, Evelyn Gaffal, Marieta Toma, Stefan Kehraus, Gabriele M König, Peter Brust, Bernd K Fleischmann, Daniela Wenzel, Winnie Deuther-Conrad, Christa Elisabeth Müller
Imaging of Gα q Proteins in Mouse and Human Organs and Tissues. Pharmaceutics 15 (1) (2022)
Thu Hang Lai, Magali Toussaint, Rodrigo Teodoro, Sladjana Dukić-Stefanović, Daniel Gündel, Friedrich-Alexander Ludwig, Barbara Wenzel, Susann Schröder, Bernhard Sattler, Rareş-Petru Moldovan, Björn H Falkenburger, Osama Sabri, Winnie Deuther-Conrad, Peter Brust
Improved in vivo PET imaging of the adenosine A2A receptor in the brain using [18F]FLUDA, a deuterated radiotracer with high metabolic stability. European journal of nuclear medicine and molecular imaging 48 (9) (2021)
Marcel Lindemann, Sladjana Dukic-Stefanovic, Sonja Hinz, Winnie Deuther-Conrad, Rodrigo Teodoro, Cathleen Juhl, Jörg Steinbach, Peter Brust, Christa Elisabeth Müller, Barbara Wenzel
Synthesis of Novel Fluorinated Xanthine Derivatives with High Adenosine A2B Receptor Binding Affinity. Pharmaceuticals (Basel, Switzerland) 14 (5) (2021)
Susann Schröder, Matthias Scheunemann, Barbara Wenzel, Peter Brust
Challenges on Cyclic Nucleotide Phosphodiesterases Imaging with Positron Emission Tomography: Novel Radioligands and (Pre-)Clinical Insights since 2016. International journal of molecular sciences 22 (8) (2021)
Thu Hang Lai, Magali Toussaint, Rodrigo Teodoro, Sladjana Dukić-Stefanović, Mathias Kranz, Winnie Deuther-Conrad, Rareş-Petru Moldovan, Peter Brust
Synthesis and Biological Evaluation of a Novel 18F-Labeled Radiotracer for PET Imaging of the Adenosine A2A Receptor. International journal of molecular sciences 22 (3) (2021)
Xiao-Ning Chai, Friedrich-Alexander Ludwig, Anne Müglitz, Michael Schaefer, Hai-Yan Yin, Peter Brust, Ralf Regenthal, Ute Krügel
Validation of an LC-MS/MS Method to Quantify the New TRPC6 Inhibitor SH045 (Larixyl N-methylcarbamate) and Its Application in an Exploratory Pharmacokinetic Study in Mice. Pharmaceuticals (Basel, Switzerland) 14 (3) (2021)
Thu Hang Lai, Susann Schröder, Magali Toussaint, Sladjana Dukić-Stefanović, Mathias Kranz, Friedrich-Alexander Ludwig, Steffen Fischer, Jörg Steinbach, Winnie Deuther-Conrad, Peter Brust, Rareş-Petru Moldovan
Development of 18F-Labeled Radiotracers for PET Imaging of the Adenosine A2A Receptor: Synthesis, Radiolabeling and Preliminary Biological Evaluation. International journal of molecular sciences 22 (5) (2021)
Rodrigo Teodoro, Daniel Gündel, Winnie Deuther-Conrad, Lea Ueberham, Magali Toussaint, Guy Bormans, Peter Brust, Rareş-Petru Moldovan
Development of [18F]LU14 for PET Imaging of Cannabinoid Receptor Type 2 in the Brain. International journal of molecular sciences 22 (15) (2021)
Daniel Gündel, Masoud Sadeghzadeh, Winnie Deuther-Conrad, Barbara Wenzel, Paul Cumming, Magali Toussaint, Friedrich-Alexander Ludwig, Rareş-Petru Moldovan, Mathias Kranz, Rodrigo Teodoro, Bernhard Sattler, Osama Sabri, Peter Brust
Preclinical Evaluation of [18F]FACH in Healthy Mice and Piglets: An 18F-Labeled Ligand for Imaging of Monocarboxylate Transporters with PET. International journal of molecular sciences 22 (4) (2021)
Rareş-Petru Moldovan, Daniel Gündel, Rodrigo Teodoro, Friedrich-Alexander Ludwig, Steffen Fischer, Magali Toussaint, Dirk Schepmann, Bernhard Wünsch, Peter Brust, Winnie Deuther-Conrad
Design, Radiosynthesis and Preliminary Biological Evaluation in Mice of a Brain-Penetrant 18F-Labelled σ2 Receptor Ligand. International journal of molecular sciences 22 (11) (2021)
Masoud Sadeghzadeh, Barbara Wenzel, Daniel Gündel, Winnie Deuther-Conrad, Magali Toussaint, Rareş-Petru Moldovan, Steffen Fischer, Friedrich-Alexander Ludwig, Rodrigo Teodoro, Shirisha Jonnalagadda, Sravan K Jonnalagadda, Gerrit Schüürmann, Venkatram R Mereddy, Lester R Drewes, Peter Brust
Development of Novel Analogs of the Monocarboxylate Transporter Ligand FACH and Biological Validation of One Potential Radiotracer for Positron Emission Tomography (PET) Imaging. Molecules (Basel, Switzerland) 25 (10) (2020)
Ivana I Jevtić, Thu Hang Lai, Jelena Z Penjišević, Sladjana Dukić-Stefanović, Deana B Andrić, Peter Brust, Sladjana V Kostić-Rajačić, Rodrigo Teodoro
Newly Synthesized Fluorinated Cinnamylpiperazines Possessing Low In Vitro MAO-B Binding. Molecules (Basel, Switzerland) 25 (21) (2020)
Bernhard Sattler, Mathias Kranz, Barbara Wenzel, Nalin T Jain, Rareş-Petru Moldovan, Magali Toussaint, Winnie Deuther-Conrad, Friedrich-Alexander Ludwig, Rodrigo Teodoro, Tatjana Sattler, Masoud Sadeghzadeh, Osama Sabri, Peter Brust
Preclinical Incorporation Dosimetry of [18F]FACH-A Novel 18F-Labeled MCT1/MCT4 Lactate Transporter Inhibitor for Imaging Cancer Metabolism with PET. Molecules (Basel, Switzerland) 25 (9) (2020)
Kuntarat Arunrungvichian, Sumet Chongruchiroj, Jiradanai Sarasamkan, Gerrit Schüürmann, Peter Brust, Opa Vajragupta
In Silico Finding of Key Interaction Mediated α3β4 and α7 Nicotinic Acetylcholine Receptor Ligand Selectivity of Quinuclidine-Triazole Chemotype. International journal of molecular sciences 21 (17) (2020)
Magali Toussaint, Winnie Deuther-Conrad, Mathias Kranz, Steffen Fischer, Friedrich-Alexander Ludwig, Tareq A Juratli, Marianne Patt, Bernhard Wünsch, Gabriele Schackert, Osama Sabri, Peter Brust
Sigma-1 Receptor Positron Emission Tomography: A New Molecular Imaging Approach Using (S)-(-)-[18F]Fluspidine in Glioblastoma. Molecules (Basel, Switzerland) 25 (9) (2020)
Susann Schröder, Thu Hang Lai, Magali Toussaint, Mathias Kranz, Alexandra Chovsepian, Qi Shang, Sladjana Dukić-Stefanović, Winnie Deuther-Conrad, Rodrigo Teodoro, Barbara Wenzel, Rareş-Petru Moldovan, Francisco Pan-Montojo, Peter Brust
PET Imaging of the Adenosine A2A Receptor in the Rotenone-Based Mouse Model of Parkinson's Disease with [18F]FESCH Synthesized by a Simplified Two-Step One-Pot Radiolabeling Strategy. Molecules (Basel, Switzerland) 25 (7) (2020)
Masoud Sadeghzadeh, Rareş-Petru Moldovan, Rodrigo Teodoro, Peter Brust, Barbara Wenzel
One-step radiosynthesis of the MCTs imaging agent [18F]FACH by aliphatic 18F-labelling of a methylsulfonate precursor containing an unprotected carboxylic acid group. Scientific reports 9 (1) (2019)
Friedrich-Alexander Ludwig, Steffen Fischer, René Smits, Winnie Deuther-Conrad, Alexander Hoepping, Solveig Tiepolt, Marianne Patt, Osama Sabri, Peter Brust
Exploring the Metabolism of (+)-[18F]Flubatine in Vitro and in Vivo: LC-MS/MS Aided Identification of Radiometabolites in a Clinical PET Study. Molecules (Basel, Switzerland) 23 (2) (2018)
Mathias Kranz, Ralf Bergmann, Torsten Kniess, Birgit Belter, Christin Neuber, Zhengxin Cai, Gang Deng, Steffen Fischer, Jiangbing Zhou, Yiyun Huang, Peter Brust, Winnie Deuther-Conrad, Jens Pietzsch
Bridging from Brain to Tumor Imaging: (S)-(-)- and (R)-(+)-[18F]Fluspidine for Investigation of Sigma-1 Receptors in Tumor-Bearing Mice. Molecules (Basel, Switzerland) 23 (3) (2018)
Melanie Bergkemper, Elisabeth Kronenberg, Simone Thum, Frederik Börgel, Constantin Daniliuc, Dirk Schepmann, Francisco Rafael Nieto, Peter Brust, Raquel F Reinoso, Inés Alvarez, Bernhard Wünsch
Synthesis, Receptor Affinity, and Antiallodynic Activity of Spirocyclic σ Receptor Ligands with Exocyclic Amino Moiety. Journal of medicinal chemistry 61 (21) (2018)
Susann Schröder, Barbara Wenzel, Winnie Deuther-Conrad, Rodrigo Teodoro, Mathias Kranz, Matthias Scheunemann, Ute Egerland, Norbert Höfgen, Detlef Briel, Jörg Steinbach, Peter Brust
Investigation of an 18F-labelled Imidazopyridotriazine for Molecular Imaging of Cyclic Nucleotide Phosphodiesterase 2A. Molecules (Basel, Switzerland) 23 (3) (2018)
Mathias Kranz, Bernhard Sattler, Solveig Tiepolt, Stephan Wilke, Winnie Deuther-Conrad, Cornelius K Donat, Steffen Fischer, Marianne Patt, Andreas Schildan, Jörg Patt, René Smits, Alexander Hoepping, Jörg Steinbach, Osama Sabri, Peter Brust
Radiation dosimetry of the α4β2 nicotinic receptor ligand (+)-[18F]flubatine, comparing preclinical PET/MRI and PET/CT to first-in-human PET/CT results. EJNMMI physics 3 (1) (2016)