Roland J Pieters (Roland Pieters)

ResearcherID Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 44

Top Venues

ACS chemical biology

International journal of molecular sciences

Molecules (Basel, Switzerland)

Journal of medicinal chemistry

Utrecht University

Massachusetts Institute of Technology (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Utrecht University Oct 16 1998

Netherlands

professor :: Chemical Biology & Drug Discovery

Education History

Massachusetts Institute of Technology Sep 01 1990 - Jan 10 1995

United States

PHD :: Department of Organic Chemistry

University of Groningen Sep 01 1984 - Aug 01 1990

Netherlands

MSC :: Organic Chemistry

Publications

Janja Sluga, Tihomir Tomašič, Marko Anderluh, Martina Hrast Rambaher, Gregor Bajc, Alen Sevšek, Nathaniel I Martin, Roland J Pieters, Marjana Novič, Katja Venko
Targeting N -Acetylglucosaminidase in Staphylococcus aureus with Iminosugar Inhibitors. Antibiotics (Basel, Switzerland) 13 (8) (2024)
Janja Sluga, Tihomir Tomašič, Marko Anderluh, Martina Hrast Rambaher, Gregor Bajc, Alen Sevšek, Nathaniel I Martin, Roland J Pieters, Marjana Novič, Katja Venko
Targeting N -Acetylglucosaminidase in Staphylococcus aureus with Iminosugar Inhibitors. Antibiotics (Basel, Switzerland) 13 (8) (2024)
Pouya Zaree, Ilhan Tomris, Sander D de Vos, Roosmarijn van der Woude, Frits M Flesch, Robertus J M Klein Gebbink, Robert P de Vries, Roland J Pieters
Facile electrochemical affinity measurements of small and large molecules. RSC advances 13 (14) (2023)
Robert M F van der Put, Bernard Metz, Roland J Pieters
Carriers and Antigens: New Developments in Glycoconjugate Vaccines. Vaccines 11 (2) (2023)
Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M Bouwman, Lin Liu, Zeshi Li, Jelle A Fok, María Ríos Carrasco, Roosmarijn van der Woude, Anne L M Kimpel, Mirte W Linthorst, Sinan E Kilavuzoglu, Enrico C J M Verpalen, Tom G Caniels, Rogier W Sanders, Balthasar A Heesters, Roland J Pieters, Jiménez-Barbero Jesús, John S Klassen, Geert-Jan Boons, Robert P de Vries
SARS-CoV-2 Spike N-Terminal Domain Engages 9- O -Acetylated α2-8-Linked Sialic Acids. ACS chemical biology (2023)
Robert M F van der Put, Bernard Metz, Roland J Pieters
Carriers and Antigens: New Developments in Glycoconjugate Vaccines. Vaccines 11 (2) (2023)
Pouya Zaree, Ilhan Tomris, Sander D de Vos, Roosmarijn van der Woude, Frits M Flesch, Robertus J M Klein Gebbink, Robert P de Vries, Roland J Pieters
Facile electrochemical affinity measurements of small and large molecules. RSC advances 13 (14) (2023)
Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M Bouwman, Lin Liu, Zeshi Li, Jelle A Fok, María Ríos Carrasco, Roosmarijn van der Woude, Anne L M Kimpel, Mirte W Linthorst, Sinan E Kilavuzoglu, Enrico C J M Verpalen, Tom G Caniels, Rogier W Sanders, Balthasar A Heesters, Roland J Pieters, Jiménez-Barbero Jesús, John S Klassen, Geert-Jan Boons, Robert P de Vries
SARS-CoV-2 Spike N-Terminal Domain Engages 9- O -Acetylated α2-8-Linked Sialic Acids. ACS chemical biology (2023)
Cyril Balsollier, Tihomir Tomašič, Daniel Yasini, Simon Bijkerk, Marko Anderluh, Roland J Pieters
Design of OSMI-4 Analogs Using Scaffold Hopping: Investigating the Importance of the Uridine Mimic in the Binding of OGT Inhibitors. ChemMedChem (2023)
Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M Bouwman, Lin Liu, Zeshi Li, Jelle A Fok, María Ríos Carrasco, Roosmarijn van der Woude, Anne L M Kimpel, Mirte W Linthorst, Sinan E Kilavuzoglu, Enrico C J M Verpalen, Tom G Caniels, Rogier W Sanders, Balthasar A Heesters, Roland J Pieters, Jiménez-Barbero Jesús, John S Klassen, Geert-Jan Boons, Robert P de Vries
SARS-CoV-2 Spike N-Terminal Domain Engages 9- O -Acetylated α2-8-Linked Sialic Acids. ACS chemical biology 18 (5) (2023)
Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M Bouwman, Lin Liu, Zeshi Li, Jelle A Fok, María Ríos Carrasco, Roosmarijn van der Woude, Anne L M Kimpel, Mirte W Linthorst, Sinan E Kilavuzoglu, Enrico C J M Verpalen, Tom G Caniels, Rogier W Sanders, Balthasar A Heesters, Roland J Pieters, Jiménez-Barbero Jesús, John S Klassen, Geert-Jan Boons, Robert P de Vries
SARS-CoV-2 Spike N-Terminal Domain Engages 9- O -Acetylated α2-8-Linked Sialic Acids. ACS chemical biology 18 (5) (2023)
Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M Bouwman, Lin Liu, Zeshi Li, Jelle A Fok, María Ríos Carrasco, Roosmarijn van der Woude, Anne L M Kimpel, Mirte W Linthorst, Sinan E Kilavuzoglu, Enrico C J M Verpalen, Tom G Caniels, Rogier W Sanders, Balthasar A Heesters, Roland J Pieters, Jiménez-Barbero Jesús, John S Klassen, Geert-Jan Boons, Robert P de Vries
SARS-CoV-2 Spike N-Terminal Domain Engages 9- O -Acetylated α2-8-Linked Sialic Acids. ACS chemical biology 18 (5) (2023)
Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M Bouwman, Lin Liu, Zeshi Li, Jelle A Fok, María Ríos Carrasco, Roosmarijn van der Woude, Anne L M Kimpel, Mirte W Linthorst, Sinan E Kilavuzoglu, Enrico C J M Verpalen, Tom G Caniels, Rogier W Sanders, Balthasar A Heesters, Roland J Pieters, Jiménez-Barbero Jesús, John S Klassen, Geert-Jan Boons, Robert P de Vries
SARS-CoV-2 Spike N-Terminal Domain Engages 9- O -Acetylated α2-8-Linked Sialic Acids. ACS chemical biology (2023)
Maria Eleni Mavrogeni, Mostafa Asadpoor, Jo H Judernatz, Ingrid van Ark, Marc M S M Wösten, Karin Strijbis, Roland J Pieters, Gert Folkerts, Saskia Braber
Protective Effects of Alginate and Chitosan Oligosaccharides against Clostridioides difficile Bacteria and Toxin. Toxins 15 (10) (2023)
Reshmi Mukherjee, Victor J Somovilla, Fabrizio Chiodo, Sven Bruijns, Roland J Pieters, Johan Garssen, Yvette van Kooyk, Aletta D Kraneveld, Jeroen van Bergenhenegouwen
Human Milk Oligosaccharide 2'-Fucosyllactose Inhibits Ligand Binding to C-Type Lectin DC-SIGN but Not to Langerin. International journal of molecular sciences 23 (23) (2022)
Reshmi Mukherjee, Victor J Somovilla, Fabrizio Chiodo, Sven Bruijns, Roland J Pieters, Johan Garssen, Yvette van Kooyk, Aletta D Kraneveld, Jeroen van Bergenhenegouwen
Human Milk Oligosaccharide 2'-Fucosyllactose Inhibits Ligand Binding to C-Type Lectin DC-SIGN but Not to Langerin. International journal of molecular sciences 23 (23) (2022)
Reshmi Mukherjee, Victor J Somovilla, Fabrizio Chiodo, Sven Bruijns, Roland J Pieters, Johan Garssen, Yvette van Kooyk, Aletta D Kraneveld, Jeroen van Bergenhenegouwen
Human Milk Oligosaccharide 2'-Fucosyllactose Inhibits Ligand Binding to C-Type Lectin DC-SIGN but Not to Langerin. International journal of molecular sciences 23 (23) (2022)
Margherita Duca, Diksha Haksar, Jacq van Neer, Dominique M E Thies-Weesie, Dania Martínez-Alarcón, Hans de Cock, Annabelle Varrot, Roland J Pieters
Multivalent Fucosides Targeting β-Propeller Lectins from Lung Pathogens with Promising Anti-Adhesive Properties. ACS chemical biology (2022)
Robert M F van der Put, Arnoud Spies, Bernard Metz, Daniel Some, Roger Scherrers, Roland J Pieters, Maarten Danial
Validation of an FFF-MALS Method to Characterize the Production and Functionalization of Outer-Membrane Vesicles for Conjugate Vaccines. Analytical chemistry 94 (35) (2022)
Reshmi Mukherjee, Victor J Somovilla, Fabrizio Chiodo, Sven Bruijns, Roland J Pieters, Johan Garssen, Yvette van Kooyk, Aletta D Kraneveld, Jeroen van Bergenhenegouwen
Human Milk Oligosaccharide 2'-Fucosyllactose Inhibits Ligand Binding to C-Type Lectin DC-SIGN but Not to Langerin. International journal of molecular sciences 23 (23) (2022)
Reshmi Mukherjee, Victor J Somovilla, Fabrizio Chiodo, Sven Bruijns, Roland J Pieters, Johan Garssen, Yvette van Kooyk, Aletta D Kraneveld, Jeroen van Bergenhenegouwen
Human Milk Oligosaccharide 2'-Fucosyllactose Inhibits Ligand Binding to C-Type Lectin DC-SIGN but Not to Langerin. International journal of molecular sciences 23 (23) (2022)
Veronica Ayechu-Muruzabal, Melanie van de Kaa, Reshmi Mukherjee, Johan Garssen, Bernd Stahl, Roland J Pieters, Belinda Van't Land, Aletta D Kraneveld, Linette E M Willemsen
Modulation of the Epithelial-Immune Cell Crosstalk and Related Galectin Secretion by DP3-5 Galacto-Oligosaccharides and β-3'Galactosyllactose. Biomolecules 12 (3) (2022)
Xuan Wei, Wenjuan Du, Margherita Duca, Guangyun Yu, Erik de Vries, Cornelis A M de Haan, Roland J Pieters
Preventing Influenza A Virus Infection by Mixed Inhibition of Neuraminidase and Hemagglutinin by Divalent Inhibitors. Journal of medicinal chemistry 65 (10) (2022)
Elena M Loi, Tihomir Tomašič, Cyril Balsollier, Kevin van Eekelen, Matjaž Weiss, Martina Gobec, Matthew G Alteen, David J Vocadlo, Roland J Pieters, Marko Anderluh
Discovery of a New Drug-like Series of OGT Inhibitors by Virtual Screening. Molecules (Basel, Switzerland) 27 (6) (2022)
Zhongkai Lu, Zhicheng Liu, Xia Li, Xinfang Qin, Haofei Hong, Zhifang Zhou, Roland J Pieters, Jie Shi, Zhimeng Wu
Nanobody-Based Bispecific Neutralizer for Shiga Toxin-Producing E. coli . ACS infectious diseases 8 (2) (2022)
Gerlof P Bosman, Sergio Oliveira, Peter J Simons, Javier Sastre Torano, Govert W Somsen, Leon M J Knippels, Rob Haselberg, Roland J Pieters, Johan Garssen, Karen Knipping
Limited Lactosylation of Beta-Lactoglobulin from Cow's Milk Exerts Strong Influence on Antigenicity and Degranulation of Mast Cells. Nutrients 13 (6) (2021)
Nishant V Sewgobind, Sanne Albers, Roland J Pieters
Functions and Inhibition of Galectin-7, an Emerging Target in Cellular Pathophysiology. Biomolecules 11 (11) (2021)
Mostafa Asadpoor, Georgia-Nefeli Ithakisiou, Paul A J Henricks, Roland J Pieters, Gert Folkerts, Saskia Braber
Non-Digestible Oligosaccharides and Short Chain Fatty Acids as Therapeutic Targets against Enterotoxin-Producing Bacteria and Their Toxins. Toxins 13 (3) (2021)
Xiangjie Su, Mercedes Ramírez-Escudero, Feilong Sun, Joep B van den Dikkenberg, Mies J van Steenbergen, Roland J Pieters, Bert J C Janssen, Peter M van Hasselt, Wim E Hennink, Cornelus F van Nostrum
Internalization and Transport of PEGylated Lipid-Based Mixed Micelles across Caco-2 Cells Mediated by Scavenger Receptor B1. Pharmaceutics 13 (12) (2021)
Cyril Balsollier, Roland J Pieters, Marko Anderluh
Overview of the Assays to Probe O-Linked β-N-Acetylglucosamine Transferase Binding and Activity. Molecules (Basel, Switzerland) 26 (4) (2021)
Diksha Haksar, Mostafa Asadpoor, Torben Heise, Jie Shi, Saskia Braber, Gert Folkerts, Lluis Ballell, Janneth Rodrigues, Roland J Pieters
Fighting Shigella by Blocking Its Disease-Causing Toxin. Journal of medicinal chemistry 64 (9) (2021)
Jie Shi, Suhela Sharif, Cyril Balsollier, Rob Ruijtenbeek, Roland J Pieters, Seino A K Jongkees
C-Terminal Tag Location Hampers in Vitro Profiling of OGT Peptide Substrates by mRNA Display. Chembiochem : a European journal of chemical biology 22 (4) (2020)
Elena Maria Loi, Matjaž Weiss, Stane Pajk, Martina Gobec, Tihomir Tomašič, Roland J Pieters, Marko Anderluh
Intracellular Hydrolysis of Small-Molecule O-Linked N-Acetylglucosamine Transferase Inhibitors Differs among Cells and Is Not Required for Its Inhibition. Molecules (Basel, Switzerland) 25 (15) (2020)
Hao Zhang, Hans Ippel, Michelle C Miller, Tse J Wong, Arjan W Griffioen, Kevin H Mayo, Roland J Pieters
Hybrid ligands with calixarene and thiodigalactoside groups: galectin binding and cytotoxicity. Organic chemistry frontiers : an international journal of organic chemistry 6 (16) (2019)
Diksha Haksar, Eyleen de Poel, Linda Quarles van Ufford, Sumati Bhatia, Rainer Haag, Jeffrey Beekman, Roland J Pieters
Strong Inhibition of Cholera Toxin B Subunit by Affordable, Polymer-Based Multivalent Inhibitors. Bioconjugate chemistry 30 (3) (2019)
Suhela Sharif, Jie Shi, Rob Ruijtenbeek, Roland J Pieters
Study of cross talk between phosphatases and OGA on a ZO-3-derived peptide. Amino acids 51 (4) (2019)
Wenjing Lu, Wenjuan Du, Víctor J Somovilla, Guangyun Yu, Diksha Haksar, Erik de Vries, Geert-Jan Boons, Robert P de Vries, Cornelis A M de Haan, Roland J Pieters
Enhanced Inhibition of Influenza A Virus Adhesion by Di- and Trivalent Hemagglutinin Inhibitors. Journal of medicinal chemistry 62 (13) (2019)
Sauli Haataja, Priya Verma, Ou Fu, Anastassios C Papageorgiou, Sakari Pöysti, Roland J Pieters, Ulf J Nilsson, Jukka Finne
Rationally Designed Chemically Modified Glycodendrimer Inhibits Streptococcus suis Adhesin SadP at Picomolar Concentrations. Chemistry (Weinheim an der Bergstrasse, Germany) 24 (8) (2018)
Hao Zhang, Dominic Laaf, Lothar Elling, Roland J Pieters
Thiodigalactoside-Bovine Serum Albumin Conjugates as High-Potency Inhibitors of Galectin-3: An Outstanding Example of Multivalent Presentation of Small Molecule Inhibitors. Bioconjugate chemistry 29 (4) (2018)
Hao Zhang, Tihomir Tomašič, Jie Shi, Matjaž Weiss, Rob Ruijtenbeek, Marko Anderluh, Roland J Pieters
Inhibition of O-GlcNAc transferase (OGT) by peptidic hybrids. MedChemComm 9 (5) (2018)
Teresa Mena-Barragán, M Isabel García-Moreno, Alen Sevšek, Tetsuya Okazaki, Eiji Nanba, Katsumi Higaki, Nathaniel I Martin, Roland J Pieters, José Manuel García Fernández, Carmen Ortiz Mellet
Probing the Inhibitor versus Chaperone Properties of sp²-Iminosugars towards Human β-Glucocerebrosidase: A Picomolar Chaperone for Gaucher Disease. Molecules (Basel, Switzerland) 23 (4) (2018)
Alen Sevšek, Luka Šrot, Jakob Rihter, Maša Čelan, Linda Quarles van Ufford, Ed E Moret, Nathaniel I Martin, Roland J Pieters
N-Guanidino Derivatives of 1,5-Dideoxy-1,5-imino-d-xylitol are Potent, Selective, and Stable Inhibitors of β-Glucocerebrosidase. ChemMedChem 12 (7) (2017)
Alen Sevšek, Javier Sastre Toraño, Linda Quarles van Ufford, Ed E Moret, Roland J Pieters, Nathaniel I Martin
Orthoester functionalized N-guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol as pH-responsive inhibitors of β-glucocerebrosidase. MedChemComm 8 (11) (2017)
Jie Shi, Tihomir Tomašič, Suhela Sharif, Arwin J Brouwer, Marko Anderluh, Rob Ruijtenbeek, Roland J Pieters
Peptide microarray analysis of the cross-talk between O-GlcNAcylation and tyrosine phosphorylation. FEBS letters 591 (13) (2017)

Roland J Pieters.css-eqlu8i{font-size:small;padding-left:4px;} (Roland Pieters)

Publication Activity (10 Years)

Top Topics

Top Venues

Roland J Pieters (Roland Pieters)