Tihomir Tomašič (T Tomašič)

ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 61

Top Venues

Journal of medicinal chemistry

International journal of molecular sciences

RSC advances

Journal of chemical information and modeling

University of Ljubljana, Faculty of Pharmacy

University of Ljubljana, Faculty of Pharmacy (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

University of Ljubljana, Faculty of Pharmacy Jun 01 2011

Slovenia

Associate Professor :: Chair of Pharmaceutical Chemistry

Education History

University of Ljubljana, Faculty of Pharmacy Nov 01 2006 - Apr 20 2011

Slovenia

PHD

University of Ljubljana, Faculty of Pharmacy Sep 01 2000 - Apr 22 2006

Slovenia

MSC

Publications

Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Andrej Emanuel Cotman, Federica Fulgheri, Martina Piga, Peter Peršolja, Davide Benedetto Tiz, Žiga Skok, Martina Durcik, Maša Sterle, Jaka Dernovšek, Cristina D Cruz, Päivi Tammela, Petra Éva Szili, Lejla Daruka, Csaba Pál, Anamarija Zega, Lucija Peterlin Mašič, Janez Ilaš, Tihomir Tomašič, Danijel Kikelj, Nace Zidar
New N -phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity. RSC advances 14 (39) (2024)
Martina Durcik, Cristina D Cruz, Mariano Andrea Scorciapino, Janez Ilaš, Päivi Tammela, Matteo Ceccarelli, Lucija Peterlin Mašič, Tihomir Tomašič
Benzothiazole DNA gyrase inhibitors and their conjugates with siderophore mimics: design, synthesis and evaluation. RSC advances 14 (5) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Živa Zajec, Jaka Dernovšek, Jernej Cingl, Iza Ogris, Marius Gedgaudas, Asta Zubrienė, Ana Mitrović, Simona Golič Grdadolnik, Martina Gobec, Tihomir Tomašič
New Class of Hsp90 C-Terminal Domain Inhibitors with Anti-tumor Properties against Triple-Negative Breast Cancer. Journal of medicinal chemistry 67 (15) (2024)
Živa Zajec, Jaka Dernovšek, Jernej Cingl, Iza Ogris, Marius Gedgaudas, Asta Zubrienė, Ana Mitrović, Simona Golič Grdadolnik, Martina Gobec, Tihomir Tomašič
New Class of Hsp90 C-Terminal Domain Inhibitors with Anti-tumor Properties against Triple-Negative Breast Cancer. Journal of medicinal chemistry 67 (15) (2024)
Živa Zajec, Jaka Dernovšek, Jernej Cingl, Iza Ogris, Marius Gedgaudas, Asta Zubrienė, Ana Mitrović, Simona Golič Grdadolnik, Martina Gobec, Tihomir Tomašič
New Class of Hsp90 C-Terminal Domain Inhibitors with Anti-tumor Properties against Triple-Negative Breast Cancer. Journal of medicinal chemistry 67 (15) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Janja Sluga, Tihomir Tomašič, Marko Anderluh, Martina Hrast Rambaher, Gregor Bajc, Alen Sevšek, Nathaniel I Martin, Roland J Pieters, Marjana Novič, Katja Venko
Targeting N -Acetylglucosaminidase in Staphylococcus aureus with Iminosugar Inhibitors. Antibiotics (Basel, Switzerland) 13 (8) (2024)
Živa Zajec, Jaka Dernovšek, Jernej Cingl, Iza Ogris, Marius Gedgaudas, Asta Zubrienė, Ana Mitrović, Simona Golič Grdadolnik, Martina Gobec, Tihomir Tomašič
New Class of Hsp90 C-Terminal Domain Inhibitors with Anti-tumor Properties against Triple-Negative Breast Cancer. Journal of medicinal chemistry (2024)
Živa Zajec, Jaka Dernovšek, Jernej Cingl, Iza Ogris, Marius Gedgaudas, Asta Zubrienė, Ana Mitrović, Simona Golič Grdadolnik, Martina Gobec, Tihomir Tomašič
New Class of Hsp90 C-Terminal Domain Inhibitors with Anti-tumor Properties against Triple-Negative Breast Cancer. Journal of medicinal chemistry 67 (15) (2024)
Janja Sluga, Tihomir Tomašič, Marko Anderluh, Martina Hrast Rambaher, Gregor Bajc, Alen Sevšek, Nathaniel I Martin, Roland J Pieters, Marjana Novič, Katja Venko
Targeting N -Acetylglucosaminidase in Staphylococcus aureus with Iminosugar Inhibitors. Antibiotics (Basel, Switzerland) 13 (8) (2024)
Jaka Dernovšek, Nina Gradišek, Živa Zajec, Dunja Urbančič, Jernej Cingl, Tjaša Goričan, Simona Golič Grdadolnik, Tihomir Tomašič
Discovery of new Hsp90-Cdc37 protein-protein interaction inhibitors: in silico screening and optimization of anticancer activity. RSC advances 14 (39) (2024)
Sjors van Klaveren, Mujtaba Hassan, Maria Håkansson, Richard E Johnsson, Jessica Larsson, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Tihomir Tomašič, Ulf J Nilsson
Galectin-8N-Selective 4-Halophenylphthalazinone-Galactals Double π-Stack in a Unique Pocket. ACS medicinal chemistry letters 15 (8) (2024)
Sjors van Klaveren, Mujtaba Hassan, Maria Håkansson, Richard E Johnsson, Jessica Larsson, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Tihomir Tomašič, Ulf J Nilsson
Galectin-8N-Selective 4-Halophenylphthalazinone-Galactals Double π-Stack in a Unique Pocket. ACS medicinal chemistry letters 15 (8) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Martina Durcik, Cristina D Cruz, Mariano Andrea Scorciapino, Janez Ilaš, Päivi Tammela, Matteo Ceccarelli, Lucija Peterlin Mašič, Tihomir Tomašič
Benzothiazole DNA gyrase inhibitors and their conjugates with siderophore mimics: design, synthesis and evaluation. RSC advances 14 (5) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling (2024)
Anne-Sophie Depuydt, Piyush A Patel, Žan Toplak, Chinmaya Bhat, Manuela Voráčová, Irene Eteläinen, Fiammetta Vitulano, Tanja Bruun, Antti Lempinen, Nives Hribernik, Eero Mäki-Lohiluoma, Louise Hendrickx, Ernesto Lopes Pinheiro-Junior, Tihomir Tomašič, Lucija Peterlin Mašič, Jari T Yli-Kauhaluoma, Paula S Kiuru, Jan Tytgat, Steve Peigneur
Structure-Function Studies of Sponge-Derived Compounds on the Cardiac Ca V 3.1 Channel. International journal of molecular sciences 24 (4) (2023)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A Pardo, Diarmaid Hughes, Douglas L Huseby, Talía Berruga Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus . Journal of medicinal chemistry 66 (6) (2023)
C Sturtzel, S Grissenberger, P Bozatzi, E Scheuringer, A Wenninger-Weinzierl, Z Zajec, J Dernovšek, Susana Pascoal, V Gehl, A Kutsch, A Granig, Firkret Rifatbegovic, Manon Carré, A Lang, I Valtingojer, J Moll, D Lötsch, F Erhart, Georg Widhalm, D Surdez, O Delattre, N André, J Stampfl, Tihomir Tomašič, Sabine Taschner-Mandl, Martin Distel
Refined high-content imaging-based phenotypic drug screening in zebrafish xenografts. NPJ precision oncology 7 (1) (2023)
Anne-Sophie Depuydt, Piyush A Patel, Žan Toplak, Chinmaya Bhat, Manuela Voráčová, Irene Eteläinen, Fiammetta Vitulano, Tanja Bruun, Antti Lempinen, Nives Hribernik, Eero Mäki-Lohiluoma, Louise Hendrickx, Ernesto Lopes Pinheiro-Junior, Tihomir Tomašič, Lucija Peterlin Mašič, Jari T Yli-Kauhaluoma, Paula S Kiuru, Jan Tytgat, Steve Peigneur
Structure-Function Studies of Sponge-Derived Compounds on the Cardiac Ca V 3.1 Channel. International journal of molecular sciences 24 (4) (2023)
Anne-Sophie Depuydt, Piyush A Patel, Žan Toplak, Chinmaya Bhat, Manuela Voráčová, Irene Eteläinen, Fiammetta Vitulano, Tanja Bruun, Antti Lempinen, Nives Hribernik, Eero Mäki-Lohiluoma, Louise Hendrickx, Ernesto Lopes Pinheiro-Junior, Tihomir Tomašič, Lucija Peterlin Mašič, Jari T Yli-Kauhaluoma, Paula S Kiuru, Jan Tytgat, Steve Peigneur
Structure-Function Studies of Sponge-Derived Compounds on the Cardiac Ca V 3.1 Channel. International journal of molecular sciences 24 (4) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A Pardo, Diarmaid Hughes, Douglas L Huseby, Talía Berruga Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus . Journal of medicinal chemistry 66 (6) (2023)
Maša Sterle, Martina Durcik, Clare E M Stevenson, Sara R Henderson, Petra Eva Szili, Marton Czikkely, David M Lawson, Anthony Maxwell, Dominique Cahard, Danijel Kikelj, Nace Zidar, Csaba Pal, Lucija Peterlin Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega
Exploring the 5-Substituted 2-Aminobenzothiazole-Based DNA Gyrase B Inhibitors Active against ESKAPE Pathogens. ACS omega 8 (27) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
C Sturtzel, S Grissenberger, P Bozatzi, E Scheuringer, A Wenninger-Weinzierl, Z Zajec, J Dernovšek, Susana Pascoal, V Gehl, A Kutsch, A Granig, Firkret Rifatbegovic, Manon Carré, A Lang, I Valtingojer, J Moll, D Lötsch, F Erhart, Georg Widhalm, D Surdez, O Delattre, N André, J Stampfl, Tihomir Tomašič, Sabine Taschner-Mandl, Martin Distel
Refined high-content imaging-based phenotypic drug screening in zebrafish xenografts. NPJ precision oncology 7 (1) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry (2023)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A Pardo, Diarmaid Hughes, Douglas L Huseby, Talía Berruga Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus . Journal of medicinal chemistry (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Anne-Sophie Depuydt, Piyush A Patel, Žan Toplak, Chinmaya Bhat, Manuela Voráčová, Irene Eteläinen, Fiammetta Vitulano, Tanja Bruun, Antti Lempinen, Nives Hribernik, Eero Mäki-Lohiluoma, Louise Hendrickx, Ernesto Lopes Pinheiro-Junior, Tihomir Tomašič, Lucija Peterlin Mašič, Jari T Yli-Kauhaluoma, Paula S Kiuru, Jan Tytgat, Steve Peigneur
Structure-Function Studies of Sponge-Derived Compounds on the Cardiac Ca V 3.1 Channel. International journal of molecular sciences 24 (4) (2023)
C Sturtzel, S Grissenberger, P Bozatzi, E Scheuringer, A Wenninger-Weinzierl, Z Zajec, J Dernovšek, Susana Pascoal, V Gehl, A Kutsch, A Granig, Firkret Rifatbegovic, Manon Carré, A Lang, I Valtingojer, J Moll, D Lötsch, F Erhart, Georg Widhalm, D Surdez, O Delattre, N André, J Stampfl, Tihomir Tomašič, Sabine Taschner-Mandl, Martin Distel
Refined high-content imaging-based phenotypic drug screening in zebrafish xenografts. NPJ precision oncology 7 (1) (2023)
Anne-Sophie Depuydt, Piyush A Patel, Žan Toplak, Chinmaya Bhat, Manuela Voráčová, Irene Eteläinen, Fiammetta Vitulano, Tanja Bruun, Antti Lempinen, Nives Hribernik, Eero Mäki-Lohiluoma, Louise Hendrickx, Ernesto Lopes Pinheiro-Junior, Tihomir Tomašič, Lucija Peterlin Mašič, Jari T Yli-Kauhaluoma, Paula S Kiuru, Jan Tytgat, Steve Peigneur
Structure-Function Studies of Sponge-Derived Compounds on the Cardiac Ca V 3.1 Channel. International journal of molecular sciences 24 (4) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
C Sturtzel, S Grissenberger, P Bozatzi, E Scheuringer, A Wenninger-Weinzierl, Z Zajec, J Dernovšek, Susana Pascoal, V Gehl, A Kutsch, A Granig, Firkret Rifatbegovic, Manon Carré, A Lang, I Valtingojer, J Moll, D Lötsch, F Erhart, Georg Widhalm, D Surdez, O Delattre, N André, J Stampfl, Tihomir Tomašič, Sabine Taschner-Mandl, Martin Distel
Refined high-content imaging-based phenotypic drug screening in zebrafish xenografts. NPJ precision oncology 7 (1) (2023)
Špela Gubič, Louise Antonia Hendrickx, Xiaoyi Shi, Žan Toplak, Štefan Možina, Kenny M Van Theemsche, Ernesto Lopes Pinheiro-Junior, Steve Peigneur, Alain J Labro, Luis A Pardo, Jan Tytgat, Tihomir Tomašič, Lucija Peterlin Mašič
Correction: Gubič et al. Design of New Potent and Selective Thiophene-Based K V 1.3 Inhibitors and Their Potential for Anticancer Activity. Cancers 2022, 14 , 2595. Cancers 15 (11) (2023)
Sjors van Klaveren, Jaka Dernovšek, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Ulf J Nilsson, Tihomir Tomašič
Design and synthesis of novel 3-triazolyl-1-thiogalactosides as galectin-1, -3 and -8 inhibitors. RSC advances 12 (29) (2022)
Andrej Emanuel Cotman, Pavel A Dub, Maša Sterle, Matic Lozinšek, Jaka Dernovšek, Živa Zajec, Anamarija Zega, Tihomir Tomašič, Dominique Cahard
Catalytic Stereoconvergent Synthesis of Homochiral β-CF 3 , β-SCF 3 , and β-OCF 3 Benzylic Alcohols. ACS organic & inorganic Au 2 (5) (2022)
Živa Zajec, Jaka Dernovšek, Martina Gobec, Tihomir Tomašič
In Silico Discovery and Optimisation of a Novel Structural Class of Hsp90 C-Terminal Domain Inhibitors. Biomolecules 12 (7) (2022)
Samo Guzelj, Tihomir Tomašič, Žiga Jakopin
Novel Scaffolds for Modulation of NOD2 Identified by Pharmacophore-Based Virtual Screening. Biomolecules 12 (8) (2022)
Špela Gubič, Žan Toplak, Xiaoyi Shi, Jaka Dernovšek, Louise Antonia Hendrickx, Ernesto Lopes Pinheiro-Junior, Steve Peigneur, Jan Tytgat, Luis A Pardo, Lucija Peterlin Mašič, Tihomir Tomašič
New Diarylamine K V 10.1 Inhibitors and Their Anticancer Potential. Pharmaceutics 14 (9) (2022)
Elena M Loi, Tihomir Tomašič, Cyril Balsollier, Kevin van Eekelen, Matjaž Weiss, Martina Gobec, Matthew G Alteen, David J Vocadlo, Roland J Pieters, Marko Anderluh
Discovery of a New Drug-like Series of OGT Inhibitors by Virtual Screening. Molecules (Basel, Switzerland) 27 (6) (2022)
Žan Toplak, Franci Merzel, Luis A Pardo, Lucija Peterlin Mašič, Tihomir Tomašič
Molecular Dynamics-Derived Pharmacophore Model Explaining the Nonselective Aspect of KV10.1 Pore Blockers. International journal of molecular sciences 22 (16) (2021)
Benedetta Girardi, Martina Manna, Sjors Van Klaveren, Tihomir Tomašič, Žiga Jakopin, Hakon Leffler, Ulf J Nilsson, Daniel Ricklin, Janez Mravljak, Oliver Schwardt, Marko Anderluh
Selective Monovalent Galectin-8 Ligands Based on 3-Lactoylgalactoside. ChemMedChem (2021)
Žan Toplak, Louise Antonia Hendrickx, Špela Gubič, Štefan Možina, Bojana Žegura, Alja Štern, Matjaž Novak, Xiaoyi Shi, Steve Peigneur, Jan Tytgat, Tihomir Tomašič, Luis A Pardo, Lucija Peterlin Mašič
3D Pharmacophore-Based Discovery of Novel KV10.1 Inhibitors with Antiproliferative Activity. Cancers 13 (6) (2021)
Sjors van Klaveren, Anders P Sundin, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Ulf J Nilsson, Tihomir Tomašič
Selective Galectin-8N Ligands: The Design and Synthesis of Phthalazinone-d-Galactals. ChemMedChem 17 (6) (2021)
Žan Toplak, Louise A Hendrickx, Reham Abdelaziz, Xiaoyi Shi, Steve Peigneur, Tihomir Tomašič, Jan Tytgat, Lucija Peterlin-Mašič, Luis A Pardo
Overcoming challenges of HERG potassium channel liability through rational design: Eag1 inhibitors for cancer treatment. Medicinal research reviews 42 (1) (2021)
Jaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič
Structure-Activity Relationships of Benzothiazole-Based Hsp90 C-Terminal-Domain Inhibitors. Pharmaceutics 13 (8) (2021)
Tihomir Tomašič, Asta Zubrienė, Žiga Skok, Riccardo Martini, Stane Pajk, Gobec Izidor Sosič, Janez Ilaš, Daumantas Matulis, Sharon D Bryant
Selective DNA Gyrase Inhibitors: Multi-Target in Silico Profiling with 3D-Pharmacophores. Pharmaceuticals (Basel, Switzerland) 14 (8) (2021)
Špela Gubič, Louise A Hendrickx, Žan Toplak, Maša Sterle, Steve Peigneur, Tihomir Tomašič, Luis A Pardo, Jan Tytgat, Anamarija Zega, Lucija Peterlin Mašič
Discovery of KV 1.3 ion channel inhibitors: Medicinal chemistry approaches and challenges. Medicinal research reviews 41 (4) (2021)
Mujtaba Hassan, Floriane Baussière, Samo Guzelj, Anders P Sundin, Maria Håkansson, Rebeka Kovačič, Hakon Leffler, Tihomir Tomašič, Marko Anderluh, Žiga Jakopin, Ulf J Nilsson
Structure-Guided Design of d-Galactal Derivatives with High Affinity and Selectivity for the Galectin-8 N-Terminal Domain. ACS medicinal chemistry letters 12 (11) (2021)
Martina Durcik, Žiga Skok, Janez Ilaš, Nace Zidar, Anamarija Zega, Petra Éva Szili, Gábor Draskovits, Tamás Révész, Danijel Kikelj, Akos Nyerges, Csaba Pál, Lucija Peterlin Mašič, Tihomir Tomašič
Hybrid Inhibitors of DNA Gyrase A and B: Design, Synthesis and Evaluation. Pharmaceutics 13 (1) (2020)
Elena Maria Loi, Matjaž Weiss, Stane Pajk, Martina Gobec, Tihomir Tomašič, Roland J Pieters, Marko Anderluh
Intracellular Hydrolysis of Small-Molecule O-Linked N-Acetylglucosamine Transferase Inhibitors Differs among Cells and Is Not Required for Its Inhibition. Molecules (Basel, Switzerland) 25 (15) (2020)
Akos Nyerges, Tihomir Tomašič, Martina Durcik, Tamas Revesz, Petra Szili, Gabor Draskovits, Ferenc Bogar, Žiga Skok, Nace Zidar, Janez Ilaš, Anamarija Zega, Danijel Kikelj, Lejla Daruka, Balint Kintses, Balint Vasarhelyi, Imre Foldesi, Diána Kata, Martin Welin, Yengo Raymond Kimbung, Dorota Focht, Lucija Peterlin Mašič, Csaba Pál
Rational design of balanced dual-targeting antibiotics with limited resistance. PLoS biology 18 (10) (2020)
Tihomir Tomašič, Martina Durcik, Bradley M Keegan, Darja Gramec Skledar, Živa Zajec, Brian S J Blagg, Sharon D Bryant
Discovery of Novel Hsp90 C-Terminal Inhibitors Using 3D-Pharmacophores Derived from Molecular Dynamics Simulations. International journal of molecular sciences 21 (18) (2020)
Katja-Emilia Lillsunde, Tihomir Tomašič, Philipp Schult, Volker Lohmann, Danijel Kikelj, Päivi Tammela
Inhibition of Hepatitis C Replication by Targeting the Molecular Chaperone Hsp90: Synthesis and Biological Evaluation of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazole Derivatives. ChemMedChem 14 (3) (2019)
Nace Zidar, Helena Macut, Tihomir Tomašič, Lucija Peterlin Mašič, Janez Ilaš, Anamarija Zega, Päivi Tammela, Danijel Kikelj
New N-phenyl-4,5-dibromopyrrolamides as DNA gyrase B inhibitors. MedChemComm 10 (6) (2019)
Hao Zhang, Tihomir Tomašič, Jie Shi, Matjaž Weiss, Rob Ruijtenbeek, Marko Anderluh, Roland J Pieters
Inhibition of O-GlcNAc transferase (OGT) by peptidic hybrids. MedChemComm 9 (5) (2018)
Tihomir Tomašič, Michaela Barančoková, Nace Zidar, Janez Ilaš, Päivi Tammela, Danijel Kikelj
Design, synthesis, and biological evaluation of 1-ethyl-3-(thiazol-2-yl)urea derivatives as Escherichia coli DNA gyrase inhibitors. Archiv der Pharmazie 351 (1) (2017)

Tihomir Tomašič.css-eqlu8i{font-size:small;padding-left:4px;} (T Tomašič)

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Tihomir Tomašič (T Tomašič)