Serge Van Calenbergh (Serge van Calenbergh)

ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2016-2023
Publications (10 Years): 41

Top Venues

Journal of medicinal chemistry

International journal of molecular sciences

ChemMedChem

ACS medicinal chemistry letters

Universiteit Gent

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Universiteit Gent Aug 01 2010

Belgium

Full professor :: Pharmaceutics

Publications

Marzuq A Ungogo, Mustafa M Aldfer, Manal J Natto, Hainan Zhuang, Robyn Chisholm, Katy Walsh, MarieClaire McGee, Kayhan Ilbeigi, Jamal Ibrahim Asseri, Richard J S Burchmore, Guy Caljon, Serge Van Calenbergh, Harry P de Koning
Cloning and Characterization of Trypanosoma congolense and T. vivax Nucleoside Transporters Reveal the Potential of P1-Type Carriers for the Discovery of Broad-Spectrum Nucleoside-Based Therapeutics against Animal African Trypanosomiasis. International journal of molecular sciences 24 (4) (2023)
Simon Krols, Federica Matteucci, Kristof Van Hecke, Guy Caljon, Kenneth A Jacobson, Serge Van Calenbergh
Dual N 6 /C7-Substituted 7-Deazapurine and Tricyclic Ribonucleosides with Affinity for G Protein-Coupled Receptors. ACS medicinal chemistry letters 15 (1) (2023)
Marzuq A Ungogo, Mustafa M Aldfer, Manal J Natto, Hainan Zhuang, Robyn Chisholm, Katy Walsh, MarieClaire McGee, Kayhan Ilbeigi, Jamal Ibrahim Asseri, Richard J S Burchmore, Guy Caljon, Serge Van Calenbergh, Harry P de Koning
Cloning and Characterization of Trypanosoma congolense and T. vivax Nucleoside Transporters Reveal the Potential of P1-Type Carriers for the Discovery of Broad-Spectrum Nucleoside-Based Therapeutics against Animal African Trypanosomiasis. International journal of molecular sciences 24 (4) (2023)
Marzuq A Ungogo, Mustafa M Aldfer, Manal J Natto, Hainan Zhuang, Robyn Chisholm, Katy Walsh, MarieClaire McGee, Kayhan Ilbeigi, Jamal Ibrahim Asseri, Richard J S Burchmore, Guy Caljon, Serge Van Calenbergh, Harry P de Koning
Cloning and Characterization of Trypanosoma congolense and T. vivax Nucleoside Transporters Reveal the Potential of P1-Type Carriers for the Discovery of Broad-Spectrum Nucleoside-Based Therapeutics against Animal African Trypanosomiasis. International journal of molecular sciences 24 (4) (2023)
Simon Krols, Federica Matteucci, Kristof Van Hecke, Guy Caljon, Kenneth A Jacobson, Serge Van Calenbergh
Dual N 6 /C7-Substituted 7-Deazapurine and Tricyclic Ribonucleosides with Affinity for G Protein-Coupled Receptors. ACS medicinal chemistry letters 15 (1) (2023)
Marzuq A Ungogo, Mustafa M Aldfer, Manal J Natto, Hainan Zhuang, Robyn Chisholm, Katy Walsh, MarieClaire McGee, Kayhan Ilbeigi, Jamal Ibrahim Asseri, Richard J S Burchmore, Guy Caljon, Serge Van Calenbergh, Harry P de Koning
Cloning and Characterization of Trypanosoma congolense and T. vivax Nucleoside Transporters Reveal the Potential of P1-Type Carriers for the Discovery of Broad-Spectrum Nucleoside-Based Therapeutics against Animal African Trypanosomiasis. International journal of molecular sciences 24 (4) (2023)
Simon Krols, Federica Matteucci, Kristof Van Hecke, Guy Caljon, Kenneth A Jacobson, Serge Van Calenbergh
Dual N 6 /C7-Substituted 7-Deazapurine and Tricyclic Ribonucleosides with Affinity for G Protein-Coupled Receptors. ACS medicinal chemistry letters 15 (1) (2023)
Mustafa M Aldfer, Ibrahim A Alfayez, Hamza A A Elati, Nilanjana Gayen, Ehab Kotb Elmahallawy, Ana Milena Murillo, Sabrina Marsiccobetre, Serge Van Calenbergh, Ariel M Silber, Harry P de Koning
The Trypanosoma cruzi TcrNT2 Nucleoside Transporter Is a Conduit for the Uptake of 5-F-2'-Deoxyuridine and Tubercidin Analogues. Molecules (Basel, Switzerland) 27 (22) (2022)
Erine Craey, Fabian Hulpia, Jeroen Spanoghe, Simona Manzella, Lars E Larsen, Mathieu Sprengers, Dimitri De Bundel, Ilse Smolders, Evelien Carrette, Jean Delbeke, Kristl Vonck, Paul Boon, Serge Van Calenbergh, Wytse J Wadman, Robrecht Raedt
Ex Vivo Feedback Control of Neurotransmission Using a Photocaged Adenosine A1 Receptor Agonist. International journal of molecular sciences 23 (16) (2022)
Gustavo Daniel Campagnaro, Hamza A A Elati, Sofia Balaska, Maria Esther Martin Abril, Manal J Natto, Fabian Hulpia, Kelly Lee, Lilach Sheiner, Serge Van Calenbergh, Harry P de Koning
A Toxoplasma gondii Oxopurine Transporter Binds Nucleobases and Nucleosides Using Different Binding Modes. International journal of molecular sciences 23 (2) (2022)
Ludmila F de A Fiuza, Denise G J Batista, Roberson D Girão, Fabian Hulpia, Paula Finamore-Araújo, Mustafa M Aldfer, Ehab Kotb Elmahallawy, Harry P de Koning, Otacílio Moreira, Serge Van Calenbergh, Maria de Nazaré C Soeiro
Phenotypic Evaluation of Nucleoside Analogues against Trypanosoma cruzi Infection: In Vitro and In Vivo Approaches. Molecules (Basel, Switzerland) 27 (22) (2022)
Jakob Bouton, Ludmila Ferreira de Almeida Fiuza, Camila Cardoso Santos, Maria Angela Mazzarella, Maria de Nazaré Correia Soeiro, Louis Maes, Izet Karalic, Guy Caljon, Serge Van Calenbergh
Revisiting Pyrazolo[3,4-d]pyrimidine Nucleosides as Anti-Trypanosoma cruzi and Antileishmanial Agents. Journal of medicinal chemistry 64 (7) (2021)
Cai Lin, Ludmila Ferreira de Almeida Fiuza, Camila Cardoso Santos, Daniela Ferreira Nunes, Otacílio da Cruz Moreira, Jakob Bouton, Izet Karalic, Louis Maes, Guy Caljon, Fabian Hulpia, Maria de Nazaré Correia Soeiro, Serge Van Calenbergh
6-Methyl-7-Aryl-7-Deazapurine Nucleosides as Anti-Trypanosoma cruzi Agents: Structure-Activity Relationship and in vivo Efficacy. ChemMedChem 16 (14) (2021)
Manal J Natto, Fabian Hulpia, Eric R Kalkman, Susan Baillie, Amani Alhejeli, Yukiko Miyamoto, Lars Eckmann, Serge Van Calenbergh, Harry P de Koning
Deazapurine Nucleoside Analogues for the Treatment of Trichomonas vaginalis. ACS infectious diseases 7 (6) (2021)
Dorien Mabille, Camila Cardoso Santos, Rik Hendrickx, Mathieu Claes, Peter Takac, Christine Clayton, Sarah Hendrickx, Fabian Hulpia, Louis Maes, Serge Van Calenbergh, Guy Caljon
4E Interacting Protein as a Potential Novel Drug Target for Nucleoside Analogues in Trypanosoma brucei. Microorganisms 9 (4) (2021)
Wenjin Li, Joren Guillaume, Younis Baqi, Isabell Wachsmann, Volkmar Gieselmann, Serge Van Calenbergh, Christa Elisabeth Müller
Synthesis and structure-activity relationships of cerebroside analogues as substrates of cerebroside sulphotransferase and discovery of a competitive inhibitor. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Jakob Bouton, Serge Van Calenbergh, Jan Hullaert
Sydnone Ribosides as a Platform for the Synthesis of Pyrazole C-Nucleosides: A Unified Synthesis of Formycin B and Pyrazofurin. Organic letters 22 (23) (2020)
Thijs Van de Vyver, Bram Bogaert, Lynn De Backer, Freya Joris, Roberta Guagliardo, Jelter Van Hoeck, Pieterjan Merckx, Serge Van Calenbergh, Srinivas Ramishetti, Dan Peer, Katrien Remaut, Stefaan De Smedt, Koen Raemdonck
Cationic Amphiphilic Drugs Boost the Lysosomal Escape of Small Nucleic Acid Therapeutics in a Nanocarrier-Dependent Manner. ACS nano 14 (4) (2020)
Ruben De Coen, Lutz Nuhn, Chamani Perera, Maria Arista-Romero, Martijn D P Risseeuw, Alec Freyn, Raffael Nachbagauer, Lorenzo Albertazzi, Serge Van Calenbergh, David Adam Spiegel, Blake R Peterson, Bruno G De Geest
Synthetic Rhamnose Glycopolymer Cell-Surface Receptor for Endogenous Antibody Recruitment. Biomacromolecules 21 (2) (2020)
Fabian Hulpia, Gustavo Daniel Campagnaro, Khalid J Alzahrani, Ibrahim A Alfayez, Marzuq A Ungogo, Dorien Mabille, Louis Maes, Harry P de Koning, Guy Caljon, Serge Van Calenbergh
Structure-Activity Relationship Exploration of 3'-Deoxy-7-deazapurine Nucleoside Analogues as Anti-Trypanosoma brucei Agents. ACS infectious diseases 6 (8) (2020)
Yanlin Jian, He Eun Forbes, Fabian Hulpia, Martijn D P Risseeuw, Guy Caljon, Hélène Munier-Lehmann, Helena I M Boshoff, Serge Van Calenbergh
2-((3,5-Dinitrobenzyl)thio)quinazolinones: Potent Antimycobacterial Agents Activated by Deazaflavin (F420)-Dependent Nitroreductase (Ddn). Journal of medicinal chemistry 64 (1) (2020)
Yanlin Jian, Fabian Hulpia, Martijn D P Risseeuw, He Eun Forbes, Guy Caljon, Hélène Munier-Lehmann, Helena I M Boshoff, Serge Van Calenbergh
1-(1-Arylethylpiperidin-4-yl)thymine Analogs as Antimycobacterial TMPK Inhibitors. Molecules (Basel, Switzerland) 25 (12) (2020)
Peter Blanckaert, Annelies Cannaert, Katleen Van Uytfanghe, Fabian Hulpia, Eric Deconinck, Serge Van Calenbergh, Christophe Pol Stove
Report on a novel emerging class of highly potent benzimidazole NPS opioids: Chemical and in vitro functional characterization of isotonitazene. Drug testing and analysis 12 (4) (2020)
Aurélie Crabbé, Lisa Ostyn, Sorien Staelens, Charlotte Rigauts, Martijn Risseeuw, Maarten Dhaenens, Simon Daled, Heleen Van Acker, Dieter Deforce, Serge Van Calenbergh, Tom Coenye
Host metabolites stimulate the bacterial proton motive force to enhance the activity of aminoglycoside antibiotics. PLoS pathogens 15 (4) (2019)
Jeroen Verhoeven, Fabian Hulpia, Ken Kersemans, Julie Bolcaen, Stef De Lombaerde, Jan Goeman, Benedicte Descamps, Giorgio Hallaert, Caroline Van den Broecke, Karel Deblaere, Christian Vanhove, Johan Van der Eycken, Serge Van Calenbergh, Ingeborg Goethals, Filip De Vos
New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma. Scientific reports 9 (1) (2019)
Fabian Hulpia, Dorien Mabille, Gustavo D Campagnaro, Gabriela Schumann, Louis Maes, Isabel Roditi, Anders Hofer, Harry P de Koning, Guy Caljon, Serge Van Calenbergh
Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness. Nature communications 10 (1) (2019)
Koen Venken, Peggy Jacques, Céline Mortier, Mark E Labadia, Tine Decruy, Julie Coudenys, Kathleen Hoyt, Anita L Wayne, Robert Hughes, Michael Turner, Sofie Van Gassen, Liesbet Martens, Dustin Smith, Christian Harcken, Joseph Wahle, Chao-Ting Wang, Eveline Verheugen, Nadia Schryvers, Gaëlle Varkas, Heleen Cypers, Ruth Wittoek, Yves Piette, Lieve Gyselbrecht, Serge Van Calenbergh, Filip Van den Bosch, Yvan Saeys, Gerald Nabozny, Dirk Elewaut
RORγt inhibition selectively targets IL-17 producing iNKT and γδ-T cells enriched in Spondyloarthritis patients. Nature communications 10 (1) (2019)
Rein Verbeke, Ine Lentacker, Karine Breckpot, Jonas Janssens, Serge Van Calenbergh, Stefaan De Smedt, Heleen Dewitte
Broadening the Message: A Nanovaccine Co-loaded with Messenger RNA and α-GalCer Induces Antitumor Immunity through Conventional and Natural Killer T Cells. ACS nano 13 (2) (2019)
Cai Lin, Fabian Hulpia, Cristiane França da Silva, Denise da Gama Jaen Batista, Kristof Van Hecke, Louis Maes, Guy Caljon, Maria de Nazaré C Soeiro, Serge Van Calenbergh
Discovery of Pyrrolo[2,3-b]pyridine (1,7-Dideazapurine) Nucleoside Analogues as Anti-Trypanosoma cruzi Agents. Journal of medicinal chemistry 62 (19) (2019)
Jakob Bouton, Kristof Van Hecke, Reuven Rasooly, Serge Van Calenbergh
Synthesis of pyrrolidine-based hamamelitannin analogues as quorum sensing inhibitors in Staphylococcus aureus. Beilstein journal of organic chemistry 14 (2018)
Mingcheng Qian, Lakshmi Vasudevan, Jelle Huysentruyt, Martijn D P Risseeuw, Christophe Stove, Patrick M L Vanderheyden, Kathleen Van Craenenbroeck, Serge Van Calenbergh
Design, Synthesis, and Biological Evaluation of Bivalent Ligands Targeting Dopamine D2 -Like Receptors and the μ-Opioid Receptor. ChemMedChem 13 (9) (2018)
Mingcheng Qian, Elise Wouters, James A R Dalton, Martijn D P Risseeuw, René A J Crans, Christophe Pol Stove, Jesus Giraldo, Kathleen Van Craenenbroeck, Serge Van Calenbergh
Synthesis toward Bivalent Ligands for the Dopamine D2 and Metabotropic Glutamate 5 Receptors. Journal of medicinal chemistry 61 (18) (2018)
Jonas Janssens, Aruna Bitra, Jing Wang, Tine Decruy, Koen Venken, Johan van der Eycken, Dirk Elewaut, Dirk M Zajonc, Serge Van Calenbergh
4"-O-Alkylated α-Galactosylceramide Analogues as iNKT-Cell Antigens: Synthetic, Biological, and Structural Studies. ChemMedChem 14 (1) (2018)
Lijun Song, Romain Merceron, Begoña Gracia, Ainhoa Lucía Quintana, Martijn D P Risseeuw, Fabian Hulpia, Paul Cos, José A Aínsa, Hélène Munier-Lehmann, Savvas N Savvides, Serge Van Calenbergh
Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors. Journal of medicinal chemistry 61 (7) (2018)
Joren Guillaume, Toshiyuki Seki, Tine Decruy, Koen Venken, Dirk Elewaut, Moriya Tsuji, Serge Van Calenbergh
Synthesis of C6''-modified α-C-GalCer analogues as mouse and human iNKT cell agonists. Organic & biomolecular chemistry 15 (10) (2018)
Fabian Hulpia, Kristof Van Hecke, Cristiane França da Silva, Denise da Gama Jaen Batista, Louis Maes, Guy Caljon, Maria de Nazaré C Soeiro, Serge Van Calenbergh
Discovery of Novel 7-Aryl 7-Deazapurine 3'-Deoxy-ribofuranosyl Nucleosides with Potent Activity against Trypanosoma cruzi. Journal of medicinal chemistry 61 (20) (2018)
Arno Vermote, Serge Van Calenbergh
Small-Molecule Potentiators for Conventional Antibiotics against Staphylococcus aureus. ACS infectious diseases 3 (11) (2017)
Benoit Louage, Mies J van Steenbergen, Lutz Nuhn, Martijn D P Risseeuw, Izet Karalic, Johan Winne, Serge Van Calenbergh, Wim E Hennink, Bruno G De Geest
Micellar Paclitaxel-Initiated RAFT Polymer Conjugates with Acid-Sensitive Behavior. ACS macro letters 6 (3) (2017)
Annelein M Stax, Jessica Tuengel, Enrico Girardi, Naoki Kitano, Lenka L Allan, Victor Liu, Dongjun Zheng, William J Panenka, Joren Guillaume, Chi-Huey Wong, Serge Van Calenbergh, Dirk M Zajonc, Peter van den Elzen
Autoreactivity to Sulfatide by Human Invariant NKT Cells. Journal of immunology (Baltimore, Md. : 1950) 199 (1) (2017)
Joren Guillaume, Jing Wang, Jonas Janssens, Soumya G Remesh, Martijn D P Risseeuw, Tine Decruy, Mathy Froeyen, Dirk Elewaut, Dirk M Zajonc, Serge Van Calenbergh
Galactosylsphingamides: new α-GalCer analogues to probe the F'-pocket of CD1d. Scientific reports 7 (1) (2017)
Sanjeewani Sooriyaarachchi, René Chofor, Martijn D P Risseeuw, Terese Bergfors, Jenny Pouyez, Cynthia S Dowd, Louis Maes, Johan Wouters, T Alwyn Jones, Serge Van Calenbergh, Sherry L Mowbray
Targeting an Aromatic Hotspot in Plasmodium falciparum 1-Deoxy-d-xylulose-5-phosphate Reductoisomerase with β-Arylpropyl Analogues of Fosmidomycin. ChemMedChem 11 (18) (2016)

Serge Van Calenbergh.css-eqlu8i{font-size:small;padding-left:4px;} (Serge van Calenbergh)

Publication Activity (10 Years)

Top Topics

Top Venues

Serge Van Calenbergh (Serge van Calenbergh)