Koen Augustyns

ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 24

Top Venues

Journal of medicinal chemistry

Cell death and differentiation

Scientific reports

Journal of enzyme inhibition and medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Muhammet Tanc, Nicolò Filippi, Yentl Van Rymenant, Sergei Grintsevich, Isabel Pintelon, Marlies Verschuuren, Joni De Loose, Emile Verhulst, Euy Sung Moon, Lorenzo Cianni, Sigrid Stroobants, Koen Augustyns, Frank Roesch, Ingrid De Meester, Filipe Elvas, Pieter Van Der Veken
Druglike, 18 F-labeled PET Tracers Targeting Fibroblast Activation Protein. Journal of medicinal chemistry 67 (9) (2024)
Cédric Peleman, Stig Hellemans, Geraldine Veeckmans, Wout Arras, Hao Zheng, Ine Koeken, Emily Van San, Behrouz Hassannia, Magali Walravens, Edissa Kayirangwa, Nateneal Tamerat Beyene, Mikhaïl Alfons Van Herck, Winnok Harald De Vos, Isabel Pintelon, Luc van Nassauw, Baptiste Oosterlinck, Annemieke Smet, Lieve Vits, Eveline Dirinck, An Verrijken, Joris De Man, Annelies van Eyck, Wilhelmus Josephus Kwanten, Luisa Vonghia, Ann Driessen, Koen Augustyns, Shinya Toyokuni, Benedicte Y De Winter, Christophe Van Steenkiste, Sven Francque, Tom Vanden Berghe
Ferroptosis is a targetable detrimental factor in metabolic dysfunction-associated steatotic liver disease. Cell death and differentiation 31 (9) (2024)
Muhammet Tanc, Nicolò Filippi, Yentl Van Rymenant, Sergei Grintsevich, Isabel Pintelon, Marlies Verschuuren, Joni De Loose, Emile Verhulst, Euy Sung Moon, Lorenzo Cianni, Sigrid Stroobants, Koen Augustyns, Frank Roesch, Ingrid De Meester, Filipe Elvas, Pieter Van Der Veken
Druglike, 18 F-labeled PET Tracers Targeting Fibroblast Activation Protein. Journal of medicinal chemistry (2024)
Cédric Peleman, Stig Hellemans, Geraldine Veeckmans, Wout Arras, Hao Zheng, Ine Koeken, Emily Van San, Behrouz Hassannia, Magali Walravens, Edissa Kayirangwa, Nateneal Tamerat Beyene, Mikhaïl Alfons Van Herck, Winnok Harald De Vos, Isabel Pintelon, Luc van Nassauw, Baptiste Oosterlinck, Annemieke Smet, Lieve Vits, Eveline Dirinck, An Verrijken, Joris De Man, Annelies van Eyck, Wilhelmus Josephus Kwanten, Luisa Vonghia, Ann Driessen, Koen Augustyns, Shinya Toyokuni, Benedicte Y De Winter, Christophe Van Steenkiste, Sven Francque, Tom Vanden Berghe
Ferroptosis is a targetable detrimental factor in metabolic dysfunction-associated steatotic liver disease. Cell death and differentiation (2024)
Karuna Adhikari, Jonatan Dewulf, Christel Vangestel, Pieter Van Der Veken, Sigrid Stroobants, Filipe Elvas, Koen Augustyns
Characterization of Structurally Diverse 18 F-Labeled d-TCO Derivatives as a PET Probe for Bioorthogonal Pretargeted Imaging. ACS omega 8 (41) (2023)
Yang Zheng, Susanne Schroeder, Georgi K Kanev, Sanaa S Botros, Samia William Abdel-Sayed, Abdel-Nasser A Sabra, Louis Maes, Guy Caljon, Carmen Gil, Ana Martinez, Irene G Salado, Koen Augustyns, Ewald Edink, Maarten Sijm, Erik de Heuvel, Iwan J P de Esch, Tiffany van der Meer, Marco Siderius, Geert Jan Sterk, David Brown, Rob Leurs
To Target or Not to Target Schistosoma mansoni Cyclic Nucleotide Phosphodiesterase 4A? International journal of molecular sciences 24 (7) (2023)
Aiva Plotniece, Arkadij Sobolev, Claudiu T Supuran, Fabrizio Carta, Fredrik Björkling, Henrik Franzyk, Jari T Yli-Kauhaluoma, Koen Augustyns, Paul Cos, Linda De Vooght, Matthias Govaerts, Juliana Aizawa, Päivi Tammela, Raivis Žalubovskis
Selected strategies to fight pathogenic bacteria. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Pauline Puylaert, Lynn Roth, Melissa Van Praet, Isabel Pintelon, Catalina Dumitrascu, Alexander L N van Nuijs, Greta Klejborowska, Pieter-Jan D F Guns, Tom Vanden Berghe, Koen Augustyns, Guido R Y De Meyer, Wim Martinet
Effect of erythrophagocytosis-induced ferroptosis during angiogenesis in atherosclerotic plaques. Angiogenesis (2023)
Aiva Plotniece, Arkadij Sobolev, Claudiu T Supuran, Fabrizio Carta, Fredrik Björkling, Henrik Franzyk, Jari T Yli-Kauhaluoma, Koen Augustyns, Paul Cos, Linda De Vooght, Matthias Govaerts, Juliana Aizawa, Päivi Tammela, Raivis Žalubovskis
Selected strategies to fight pathogenic bacteria. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Emily Van San, Angela C Debruyne, Geraldine Veeckmans, Yulia Y Tyurina, Vladimir A Tyurin, Hao Zheng, Sze Men Choi, Koen Augustyns, Geert van Loo, Bernhard Michalke, Vivek Venkataramani, Shinya Toyokuni, Hülya Bayır, Peter Vandenabeele, Behrouz Hassannia, Tom Vanden Berghe
Ferroptosis contributes to multiple sclerosis and its pharmacological targeting suppresses experimental disease progression. Cell death and differentiation (2023)
Siham Benramdane, Joni De Loose, Nicolò Filippi, Margarida Espadinha, Olivier Beyens, Yentl Van Rymenant, Laura Dirkx, Murat Bozdag, Pim-Bart Feijens, Koen Augustyns, Guy Caljon, Hans De Winter, Ingrid De Meester, Pieter Van Der Veken
Highly Selective Inhibitors of Dipeptidyl Peptidase 9 (DPP9) Derived from the Clinically Used DPP4-Inhibitor Vildagliptin. Journal of medicinal chemistry (2023)
Samya Van Coillie, Emily Van San, Ines Goetschalckx, Bartosz Wiernicki, Banibrata Mukhopadhyay, Wulf Tonnus, Sze Men Choi, Ria Roelandt, Catalina Dumitrascu, Ludwig Lamberts, Geert Dams, Wannes Weyts, Jelle Huysentruyt, Behrouz Hassannia, Irina Ingold, Suhas Lele, Evelyne Meyer, Maya Berg, Ruth Seurinck, Yvan Saeys, An Vermeulen, Alexander L N van Nuijs, Marcus Conrad, Andreas Linkermann, Mohan Rajapurkar, Peter Vandenabeele, Eric Hoste, Koen Augustyns, Tom Vanden Berghe
Targeting ferroptosis protects against experimental (multi)organ dysfunction and death. Nature communications 13 (1) (2022)
Nikita Hanning, Michelle De Bruyn, Hannah Ceuleers, Tim Boogaerts, Maya Berg, Annemieke Smet, Heiko U De Schepper, Jurgen Joossens, Alexander L N van Nuijs, Joris G De Man, Koen Augustyns, Ingrid De Meester, Benedicte Y De Winter
Local Colonic Administration of a Serine Protease Inhibitor Improves Post-Inflammatory Visceral Hypersensitivity in Rats. Pharmaceutics 13 (6) (2021)
Irene G Salado, Abhimanyu K Singh, Carlos Moreno-Cinos, Guna Sakaine, Marco Siderius, Pieter Van Der Veken, An Matheeussen, Tiffany van der Meer, Payman Sadek, Sheraz Gul, Louis Maes, Geert-Jan Sterk, Rob Leurs, David Brown, Koen Augustyns
Lead Optimization of Phthalazinone Phosphodiesterase Inhibitors as Novel Antitrypanosomal Compounds. Journal of medicinal chemistry 63 (7) (2020)
Olga Balabon, Eleni Pitta, Maciej K Rogacki, Eugenia Meiler, Ruth Casanueva, Laura Guijarro, Sophie Huss, Eva Maria Lopez-Roman, Ángel Santos-Villarejo, Koen Augustyns, Lluis Ballell, David Barros Aguirre, Robert H Bates, Fraser Cunningham, Mónica Cacho, Pieter Van Der Veken
Optimization of Hydantoins as Potent Antimycobacterial Decaprenylphosphoryl-β-d-Ribose Oxidase (DprE1) Inhibitors. Journal of medicinal chemistry 63 (10) (2020)
Nathalia M de Vasconcelos, Gwendolyn Vliegen, Amanda Gonçalves, Emilie De Hert, Rosa Martín-Pérez, Nina Van Opdenbosch, Anvesh Jallapally, Ruth Geiss-Friedlander, Anne-Marie Lambeir, Koen Augustyns, Pieter Van Der Veken, Ingrid De Meester, Mohamed Lamkanfi
DPP8/DPP9 inhibition elicits canonical Nlrp1b inflammasome hallmarks in murine macrophages. Life science alliance 2 (1) (2019)
Carlos Moreno-Cinos, Elisa Sassetti, Irene G Salado, Gesa Witt, Siham Benramdane, Laura Reinhardt, Cristina D Cruz, Jurgen Joossens, Pieter Van Der Veken, Heike Brötz-Oesterhelt, Päivi Tammela, Mathias Winterhalter, Philip Gribbon, Björn Windshügel, Koen Augustyns
α-Amino Diphenyl Phosphonates as Novel Inhibitors of Escherichia coli ClpP Protease. Journal of medicinal chemistry 62 (2) (2019)
Sofie Martens, Vera Goossens, Lars Devisscher, Sam Hofmans, Polien Claeys, Marnik Vuylsteke, Nozomi Takahashi, Koen Augustyns, Peter Vandenabeele
RIPK1-dependent cell death: a novel target of the Aurora kinase inhibitor Tozasertib (VX-680). Cell death & disease 9 (2) (2018)
Dries Van Rompaey, Kenneth Verstraete, Frank Peelman, Savvas N Savvides, Koen Augustyns, Pieter Van Der Veken, Hans De Winter
Author Correction: Virtual screening for inhibitors of the human TSLP:TSLPR interaction. Scientific reports 8 (1) (2018)
Lars Devisscher, Samya Van Coillie, Sam Hofmans, Dries Van Rompaey, Kenneth Goossens, Eline Meul, Louis Maes, Hans De Winter, Pieter Van Der Veken, Peter Vandenabeele, Tom Vanden Berghe, Koen Augustyns
Discovery of Novel, Drug-Like Ferroptosis Inhibitors with in Vivo Efficacy. Journal of medicinal chemistry 61 (22) (2018)
Sam Hofmans, Lars Devisscher, Sofie Martens, Dries Van Rompaey, Kenneth Goossens, Tatyana Divert, Wim Nerinckx, Nozomi Takahashi, Hans De Winter, Pieter Van Der Veken, Vera Goossens, Peter Vandenabeele, Koen Augustyns
Tozasertib Analogues as Inhibitors of Necroptotic Cell Death. Journal of medicinal chemistry 61 (5) (2018)
Maciej K Rogacki, Eleni Pitta, Olga Balabon, Sophie Huss, Eva Maria Lopez-Roman, Argyrides Argyrou, Delia Blanco-Ruano, Monica Cacho, Christophe M L Vande Velde, Koen Augustyns, Lluis Ballell, David Barros Aguirre, Robert H Bates, Fraser Cunningham, Pieter Van Der Veken
Identification and Profiling of Hydantoins-A Novel Class of Potent Antimycobacterial DprE1 Inhibitors. Journal of medicinal chemistry 61 (24) (2018)
Dries Van Rompaey, Kenneth Verstraete, Frank Peelman, Savvas N Savvides, Koen Augustyns, Pieter Van Der Veken, Hans De Winter
Virtual screening for inhibitors of the human TSLP:TSLPR interaction. Scientific reports 7 (1) (2017)
Sofie Martens, Manhyung Jeong, Wulf Tonnus, Friederike Feldmann, Sam Hofmans, Vera Goossens, Nozomi Takahashi, Jan Hinrich Bräsen, Eun Woo Lee, Pieter Van der Veken, Jurgen Joossens, Koen Augustyns, Simone Fulda, Andreas Linkermann, Jaekyoung Son, Peter Vandenabeele
Sorafenib tosylate inhibits directly necrosome complex formation and protects in mouse models of inflammation and tissue injury. Cell death & disease 8 (6) (2017)

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Publication Activity (10 Years)

Top Topics

Top Venues

Koen Augustyns