Fabrizio Carta

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 75

Top Topics

Rheumatoid Arthritis

Pulmonary Fibrosis

Crystal Structure

Top Venues

Journal of medicinal chemistry

Molecules (Basel, Switzerland)

International journal of molecular sciences

Antioxidants (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Alejandro I Recio-Balsells, Renzo Carlucci, Simone Giovannuzzi, Fabrizio Carta, Claudiu T Supuran, Babu L Tekwani, Héctor R Morbidoni, Guillermo R Labadie
Repurposing antiparasitic N,N'-aliphatic diamine derivatives as promising antimycobacterial agents. Archiv der Pharmazie (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry 67 (4) (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry 67 (4) (2024)
Jaydeo T Kilbile, Suryakant B Sapkal, Gioele Renzi, Ilaria D'Agostino, Luigi Cutarella, Mattia Mori, Barbara De Filippis, Imadul Islam, Maria Luisa Massardi, Elena Somenza, Roberto Ronca, Yasinalli Tamboli, Fabrizio Carta, Claudiu T Supuran
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (6) (2024)
Mourad A M Aboul-Soud, Yazeed A Al-Sheikh, Hazem K Ghneim, Claudiu T Supuran, Fabrizio Carta
Kinase inhibitors: 20 years of success and many new challenges and recent trends in their patents. Expert opinion on therapeutic patents 34 (7) (2024)
Mourad A M Aboul-Soud, Yazeed A Al-Sheikh, Hazem K Ghneim, Claudiu T Supuran, Fabrizio Carta
Kinase inhibitors: 20 years of success and many new challenges and recent trends in their patents. Expert opinion on therapeutic patents (2024)
Arzu Gumus, Ilaria D'Agostino, Valentina Puca, Valentina Crocetta, Simone Carradori, Luigi Cutarella, Mattia Mori, Fabrizio Carta, Andrea Ageli, Clemente Capasso, Claudiu T Supuran
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α-carbonic anhydrase inhibitors. Archiv der Pharmazie (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry (2024)
Hakan Aslan, Gioele Renzi, Andrea Ageli, Ilaria D'Agostino, Roberto Ronca, Maria Luisa Massardi, Camilla Tavani, Simone Carradori, Marta Ferraroni, Paolo Governa, Fabrizio Manetti, Fabrizio Carta, Claudiu T Supuran
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC medicinal chemistry 15 (6) (2024)
Jaydeo T Kilbile, Suryakant B Sapkal, Gioele Renzi, Ilaria D'Agostino, Luigi Cutarella, Mattia Mori, Barbara De Filippis, Imadul Islam, Maria Luisa Massardi, Elena Somenza, Roberto Ronca, Yasinalli Tamboli, Fabrizio Carta, Claudiu T Supuran
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (6) (2024)
Hakan Aslan, Gioele Renzi, Andrea Ageli, Ilaria D'Agostino, Roberto Ronca, Maria Luisa Massardi, Camilla Tavani, Simone Carradori, Marta Ferraroni, Paolo Governa, Fabrizio Manetti, Fabrizio Carta, Claudiu T Supuran
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC medicinal chemistry 15 (6) (2024)
Marialuigia Fantacuzzi, Ilaria D'Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Mariangela Agamennone, Andrea Ageli, Filomena Sannio, Jean Denis Docquier, Clemente Capasso, Claudiu T Supuran
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Gioele Renzi, Fabrizio Carta, Claudiu T Supuran
The Integrase: An Overview of a Key Player Enzyme in the Antiviral Scenario. International journal of molecular sciences 24 (15) (2023)
Susanna Haapanen, Harlan Barker, Fabrizio Carta, Claudiu T Supuran, Seppo Parkkila
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors. Journal of medicinal chemistry (2023)
Thor Eysteinsson, Andrea García-Llorca, Arnar Oessur Hardarson, Daniela Vullo, Fabrizio Carta, Claudiu T Supuran
Membrane Permeability Is Required for the Vasodilatory Effect of Carbonic Anhydrase Inhibitors in Porcine Retinal Arteries. International journal of molecular sciences 24 (9) (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 66 (3) (2023)
Emanuela Berrino, Simone Carradori, Fabrizio Carta, Francesco Melfi, Marialucia Gallorini, Giulio Poli, Tiziano Tuccinardi, José G Fernández-Bolaños, Óscar López, Jacobus P Petzer, Anél Petzer, Paolo Guglielmi, Daniela Secci, Claudiu T Supuran
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration. Antioxidants (Basel, Switzerland) 12 (12) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Susanna Haapanen, Harlan Barker, Fabrizio Carta, Claudiu T Supuran, Seppo Parkkila
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors. Journal of medicinal chemistry 67 (1) (2023)
Susanna Haapanen, Harlan Barker, Fabrizio Carta, Claudiu T Supuran, Seppo Parkkila
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors. Journal of medicinal chemistry 67 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Aiva Plotniece, Arkadij Sobolev, Claudiu T Supuran, Fabrizio Carta, Fredrik Björkling, Henrik Franzyk, Jari T Yli-Kauhaluoma, Koen Augustyns, Paul Cos, Linda De Vooght, Matthias Govaerts, Juliana Aizawa, Päivi Tammela, Raivis Žalubovskis
Selected strategies to fight pathogenic bacteria. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Susanna Haapanen, Harlan Barker, Fabrizio Carta, Claudiu T Supuran, Seppo Parkkila
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors. Journal of medicinal chemistry 67 (1) (2023)
Susanna Haapanen, Harlan Barker, Fabrizio Carta, Claudiu T Supuran, Seppo Parkkila
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors. Journal of medicinal chemistry 67 (1) (2023)
Francesco Fiorentino, Fabrizio Carta, Dante Rotili, Antonello Mai, Claudiu T Supuran
State of the art of carbonic anhydrase activators. Future medicinal chemistry (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 66 (3) (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 66 (3) (2023)
Germán Benito, Ilaria D'Agostino, Simone Carradori, Marialuigia Fantacuzzi, Mariangela Agamennone, Valentina Puca, Rossella Grande, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Erlotinib-containing benzenesulfonamides as anti- Helicobacter pylori agents through carbonic anhydrase inhibition. Future medicinal chemistry (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Thor Eysteinsson, Andrea García-Llorca, Arnar Oessur Hardarson, Daniela Vullo, Fabrizio Carta, Claudiu T Supuran
Membrane Permeability Is Required for the Vasodilatory Effect of Carbonic Anhydrase Inhibitors in Porcine Retinal Arteries. International journal of molecular sciences 24 (9) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Susanna Haapanen, Harlan Barker, Fabrizio Carta, Claudiu T Supuran, Seppo Parkkila
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors. Journal of medicinal chemistry 67 (1) (2023)
Andrea Ageli, Marta Ferraroni, Carlotta Granchi, Filippo Minutolo, Xiaozhuo Chen, Pratik Shriwas, Emilio Russo, Antonio Leo, Silvia Selleri, Fabrizio Carta, Claudiu T Supuran
First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome. Journal of medicinal chemistry (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry (2023)
Aiva Plotniece, Arkadij Sobolev, Claudiu T Supuran, Fabrizio Carta, Fredrik Björkling, Henrik Franzyk, Jari T Yli-Kauhaluoma, Koen Augustyns, Paul Cos, Linda De Vooght, Matthias Govaerts, Juliana Aizawa, Päivi Tammela, Raivis Žalubovskis
Selected strategies to fight pathogenic bacteria. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Gianmarco Gualtieri, Annalisa Maruca, Roberta Rocca, Fabrizio Carta, Emanuela Berrino, Alessandro Salatino, Carolina Brescia, Roberta Torcasio, Manuel Crispo, Francesco Trapasso, Stefano Alcaro, Claudiu T Supuran, Giosuè Costa
Uncovering Novel Capsaicin Inhibitory Activity towards Human Carbonic Anhydrase Isoforms IX and XII by Combining In Silico and In Vitro Studies. Antioxidants (Basel, Switzerland) 12 (5) (2023)
Emanuela Berrino, Simone Carradori, Fabrizio Carta, Francesco Melfi, Marialucia Gallorini, Giulio Poli, Tiziano Tuccinardi, José G Fernández-Bolaños, Óscar López, Jacobus P Petzer, Anél Petzer, Paolo Guglielmi, Daniela Secci, Claudiu T Supuran
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration. Antioxidants (Basel, Switzerland) 12 (12) (2023)
Chiara Testa, Anna Maria Papini, Reinhard Zeidler, Daniela Vullo, Fabrizio Carta, Claudiu T Supuran, Paolo Rovero
First studies on tumor associated carbonic anhydrases IX and XII monoclonal antibodies conjugated to small molecule inhibitors. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Arzu Gumus, Murat Bozdag, Atilla Akdemir, Andrea Ageli, Silvia Selleri, Fabrizio Carta, Claudiu T Supuran
Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII. Molecules (Basel, Switzerland) 27 (14) (2022)
Andrea Ageli, Alice Velluzzi, Silvia Selleri, Clemente Capasso, Costanza Spadini, Mattia Iannarelli, Clotilde S Cabassi, Fabrizio Carta, Claudiu T Supuran
Seleno Containing Compounds as Potent and Selective Antifungal Agents. ACS infectious diseases 8 (9) (2022)
Gioele Vannozzi, Daniela Vullo, Andrea Ageli, Marta Ferraroni, Jacob Combs, Carrie Lomelino, Jacob T Andring, Robert Mckenna, Gianluca Bartolucci, Marco Pallecchi, Laura Lucarini, Silvia Sgambellone, Emanuela Masini, Fabrizio Carta, Claudiu T Supuran
One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. Journal of medicinal chemistry 65 (1) (2021)
Emanuela Berrino, Bastien Michelet, Agnès Martin-Mingot, Fabrizio Carta, Claudiu T Supuran, Sébastien Thibaudeau
Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution. Angewandte Chemie (International ed. in English) 60 (43) (2021)
Murat Bozdag, Claudiu T Supuran, Davide Esposito, Andrea Ageli, Fabrizio Carta, Simona Maria Monti, Giuseppina De Simone, Vincenzo Alterio
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site. Chemical communications (Cambridge, England) 56 (59) (2021)
Emanuela Berrino, Simone Carradori, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran, Paolo Guglielmi, Cecilia Coletti, Roberto Paciotti, Helmut Schweikl, Francesca Maestrelli, Elisabetta Cerbai, Marialucia Gallorini
Dual Carbonic Anhydrase IX/XII Inhibitors and Carbon Monoxide Releasing Molecules Modulate LPS-Mediated Inflammation in Mouse Macrophages. Antioxidants (Basel, Switzerland) 10 (1) (2021)
Andrea Ageli, Marta Ferraroni, Akram A Da'dara, Silvia Selleri, Mariana Pinteala, Fabrizio Carta, Patrick J Skelly, Claudiu T Supuran
Structural Insights into Schistosoma mansoni Carbonic Anhydrase (SmCA) Inhibition by Selenoureido-Substituted Benzenesulfonamides. Journal of medicinal chemistry 64 (14) (2021)
Andrea Ageli, Emanuela Berrino, Simone Carradori, Claudiu T Supuran, Marzia Cirri, Fabrizio Carta, Gabriele Costantino
Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators. Molecules (Basel, Switzerland) 26 (23) (2021)
Marialucia Gallorini, Anna C Berardi, Alessia Ricci, Cristina Antonetti Lamorgese Passeri, Susi Zara, Francesco Oliva, Amelia Cataldi, Fabrizio Carta, Simone Carradori
Dual Acting Carbon Monoxide Releasing Molecules and Carbonic Anhydrase Inhibitors Differentially Modulate Inflammation in Human Tenocytes. Biomedicines 9 (2) (2021)
Shawn Christopher Chafe, Frederick S Vizeacoumar, Geetha Venkateswaran, Oksana Nemirovsky, Shannon J Awrey, Wells S Brown, Paul C McDonald, Fabrizio Carta, Andrew Metcalfe, Joanna M Karasinska, Ling Huang, Senthil K Muthuswamy, David F Schaeffer, Daniel J Renouf, Claudiu T Supuran, Franco J Vizeacoumar, Shoukat Dedhar
Genome-wide synthetic lethal screen unveils novel CAIX-NFS1/xCT axis as a targetable vulnerability in hypoxic solid tumors. Science advances 7 (35) (2021)
Anna A Plyasova, Emanuela Berrino, Irina I Khan, Alexander V Veselovsky, Vadim S Pokrovsky, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Marina V Pokrovskaya, Svetlana S Alexandrova, Yulia A Gladilina, Nikolay N Sokolov, Abdullah Hilal, Fabrizio Carta, Dmitry D Zhdanov
Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors. Journal of medicinal chemistry 64 (15) (2021)
Kalyan Kumar Sethi, K M Abha Mishra, Saurabh M Verma, Daniela Vullo, Fabrizio Carta, Claudiu T Supuran
Synthesis and Human Carbonic Anhydrase I, II, IX, and XII Inhibition Studies of Sulphonamides Incorporating Mono-, Bi- and Tricyclic Imide Moieties. Pharmaceuticals (Basel, Switzerland) 14 (7) (2021)
Viviana De Luca, Andrea Ageli, Valeria Mazzone, Claudia Adelfio, Fabrizio Carta, Silvia Selleri, Vincenzo Carginale, Andrea Scaloni, Claudiu T Supuran, Clemente Capasso
Inhibitory Effects of Sulfonamide Derivatives on the β-Carbonic Anhydrase (MpaCA) from Malassezia pachydermatis, a Commensal, Pathogenic Fungus Present in Domestic Animals. International journal of molecular sciences 22 (22) (2021)
Felipe Raposo Passos Mansoldo, Fabrizio Carta, Andrea Ageli, Verônica da Silva Cardoso, Claudiu T Supuran, Alane Beatriz Vermelho
Chagas Disease: Perspectives on the Past and Present and Challenges in Drug Discovery. Molecules (Basel, Switzerland) 25 (22) (2020)
Majid Ali, Murat Bozdag, Umar Farooq, Andrea Ageli, Fabrizio Carta, Paola Berto, Giuseppe Zanotti, Claudiu T Supuran
Benzylaminoethyureido-Tailed Benzenesulfonamides: Design, Synthesis, Kinetic and X-ray Investigations on Human Carbonic Anhydrases. International journal of molecular sciences 21 (7) (2020)
Andrea Ageli, Marta Ferraroni, Mariana Pinteală, Stelian S Maier, Bogdan C Simionescu, Fabrizio Carta, Sonia Del Prete, Clemente Capasso, Claudiu T Supuran
Crystal Structure of a Tetrameric Type II β-Carbonic Anhydrase from the Pathogenic Bacterium Burkholderia pseudomallei. Molecules (Basel, Switzerland) 25 (10) (2020)
Giosuè Costa, Annalisa Maruca, Roberta Rocca, Francesca Alessandra Ambrosio, Emanuela Berrino, Fabrizio Carta, Francesco Mesiti, Alessandro Salatino, Delia Lanzillotta, Francesco Trapasso, Anna Artese, Stefano Alcaro, Claudiu T Supuran
In Silico Identification and Biological Evaluation of Antioxidant Food Components Endowed with IX and XII hCA Inhibition. Antioxidants (Basel, Switzerland) 9 (9) (2020)
Emanuela Berrino, Andrea Ageli, Dmitry D Zhdanov, Anna P Kiryukhina, Andrea Milaneschi, Alessandro De Luca, Murat Bozdag, Simone Carradori, Silvia Selleri, Gianluca Bartolucci, Thomas S Peat, Marta Ferraroni, Claudiu T Supuran, Fabrizio Carta
Azidothymidine "Clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors. Journal of medicinal chemistry 63 (13) (2020)
Andrea Ageli, Bogdan-Florin Craciun, Stelian S Maier, Bogdan C Simionescu, Andrea Milaneschi, Ghulam Abbas, Mariana Pinteală, Clemente Capasso, Stelian Sergiu Maier, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Evaluation of Thio- and Seleno-Acetamides Bearing Benzenesulfonamide as Inhibitor of Carbonic Anhydrases from Different Pathogenic Bacteria. International journal of molecular sciences 21 (2) (2020)
Andrea Ageli, Mikel Etxebeste-Mitxeltorena, Carmen Sanmartin, Socorro Espuelas, Esther Moreno, Amaya Azqueta, Seppo Parkkila, Fabrizio Carta, Claudiu T Supuran
Tellurides Bearing Sulfonamides as Novel Inhibitors of Leishmanial Carbonic Anhydrase with Potent Antileishmanial Activity. Journal of medicinal chemistry 63 (8) (2020)
Andrea Ageli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A Donald, Shoukat Dedhar, Claudiu T Supuran
Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 10 (10) (2020)
Laura Lucarini, Mariaconcetta Durante, Silvia Sgambellone, Cecilia Lanzi, Elisabetta Bigagli, Ozlem Akgul, Emanuela Masini, Claudiu T Supuran, Fabrizio Carta
Effects of New NSAID-CAI Hybrid Compounds in Inflammation and Lung Fibrosis. Biomolecules 10 (9) (2020)
Emanuela Berrino, Lisa Milazzo, Laura Micheli, Daniela Vullo, Andrea Angeli, Murat Bozdag, Alessio Nocentini, Marta Menicatti, Gianluca Bartolucci, Lorenzo di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran, Fabrizio Carta
Synthesis and Evaluation of Carbonic Anhydrase Inhibitors with Carbon Monoxide Releasing Properties for the Management of Rheumatoid Arthritis. Journal of medicinal chemistry 62 (15) (2019)
Fabrizio Carta, Pascal Dumy, Claudiu T Supuran, Jean-Yves Winum
Multivalent Carbonic Anhydrases Inhibitors. International journal of molecular sciences 20 (21) (2019)
Silvia Bua, Laura Lucarini, Laura Micheli, Marta Menicatti, Gianluca Bartolucci, Silvia Selleri, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Emanuela Masini, Fabrizio Carta, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Bioisosteric Development of Multitarget Nonsteroidal Anti-Inflammatory Drug-Carbonic Anhydrases Inhibitor Hybrids for the Management of Rheumatoid Arthritis. Journal of medicinal chemistry 63 (5) (2019)
Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, Claudiu T Supuran, Fiorella Casamenti, M Beatrice Passani, Silvia Fossati
A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease. International journal of molecular sciences 20 (19) (2019)
Ashok Aspatwar, Jean-Yves Winum, Fabrizio Carta, Claudiu T Supuran, Milka Marjut Hammarén, Mataleena Parikka, Seppo Parkkila
Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on In Vitro and In Vivo Studies. Molecules (Basel, Switzerland) 23 (11) (2018)
Alessio Nocentini, Mariangela Ceruso, Silvia Bua, Carrie L Lomelino, Jacob T Andring, Robert McKenna, Cecilia Lanzi, Silvia Sgambellone, Riccardo Pecori, Rosanna Matucci, Luca Filippi, Paola Gratteri, Fabrizio Carta, Emanuela Masini, Silvia Selleri, Claudiu T Supuran
Discovery of β-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy. Journal of medicinal chemistry 61 (12) (2018)
Ozlem Akgul, Lorenzo Di Cesare Mannelli, Daniela Vullo, Andrea Angeli, Carla Ghelardini, Gianluca Bartolucci, Abdulmalik Saleh Alfawaz Altamimi, Andrea Scozzafava, Claudiu T Supuran, Fabrizio Carta
Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis. Journal of medicinal chemistry 61 (11) (2018)
Murat Bozdag, Fabrizio Carta, Mariangela Ceruso, Marta Ferraroni, Paul C McDonald, Shoukat Dedhar, Claudiu T Supuran
Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX. Journal of medicinal chemistry 61 (14) (2018)
Silvia Bua, Lorenzo Di Cesare Mannelli, Daniela Vullo, Carla Ghelardini, Gianluca Bartolucci, Andrea Scozzafava, Claudiu T Supuran, Fabrizio Carta
Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 60 (3) (2017)
Fabrizio Carta, Alexander Birkmann, Tamara Pfaff, Helmut Buschmann, Wilfried Schwab, Holger Zimmermann, Alfonso Maresca, Claudiu T Supuran
Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action. Journal of medicinal chemistry 60 (7) (2017)