Claudiu T Supuran (Claudiu Supuran, Claudiu T Supran)

ORCID

Publication Activity (10 Years)

Years Active: 2016-2023
Publications (10 Years): 487

Top Venues

Journal of enzyme inhibition and medicinal chemistry

International journal of molecular sciences

Journal of medicinal chemistry

Molecules (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Claudiu T Supuran, Raivis Žalubovskis
2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Marialuigia Fantacuzzi, Ilaria D'Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Mariangela Agamennone, Andrea Ageli, Filomena Sannio, Jean Denis Docquier, Clemente Capasso, Claudiu T Supuran
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Gioele Renzi, Fabrizio Carta, Claudiu T Supuran
The Integrase: An Overview of a Key Player Enzyme in the Antiviral Scenario. International journal of molecular sciences 24 (15) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris V Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Farhat Ramzan, Syed Ayaz Nabi, Mehak Saba Lone, Alessandro Bonardi, Aabid Hamid, Sameena Bano, Kalicharan Sharma, Syed Shafi, Mohammed Samim, Kalim Javed, Claudiu T Supuran
Synthesis, biological evaluation and theoretical studies of ( E )-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Viviana De Luca, Clemente Capasso, Claudiu T Supuran, Raivis Žalubovskis
Novel thiazolone-benzenesulphonamide inhibitors of human and bacterial carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Niccolò Paoletti, Claudiu T Supuran
Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (7) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Mai H ElNaggar, Abdullah A Elgazar, Ghada Gamal, Shimaa M Hamed, Zainab M Elsayed, Mohamed K El-Ashrey, Amira Abood, Mahmoud A El Hassab, Ahmed M Soliman, Ramadan A El-Domany, Farid A Badria, Claudiu T Supuran, Wagdy M Eldehna
Identification of sulphonamide-tethered N -((triazol-4-yl)methyl)isatin derivatives as inhibitors of SARS-CoV-2 main protease. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Doretta Cuffaro, Riccardo Di Leo, Lidia Ciccone, Alessio Nocentini, Claudiu T Supuran, Elisa Nuti, Armando Rossello
New isoxazolidinyl-based N -alkylethanolamines as new activators of human brain carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Thor Eysteinsson, Andrea García-Llorca, Arnar Oessur Hardarson, Daniela Vullo, Fabrizio Carta, Claudiu T Supuran
Membrane Permeability Is Required for the Vasodilatory Effect of Carbonic Anhydrase Inhibitors in Porcine Retinal Arteries. International journal of molecular sciences 24 (9) (2023)
Moataz A Shaldam, Hadia Almahli, Andrea Ageli, Rehab Mustafa Badi, Eman F Khaleel, Abdelrahman I Zain-Alabdeen, Zainab M Elsayed, Eslam B Elkaeed, Rofaida Salem, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Claudiu T Supuran
Latest advances in specific inhibition of tumor-associated carbonic anhydrases. Future medicinal chemistry 15 (1) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Viviana De Luca, Clemente Capasso, Claudiu T Supuran
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Ashok Aspatwar, Alessandro Bonardi, Heidi Aisala, Ksenia Zueva, Craig Robert Primmer, Jaakko Lumme, Seppo Parkkila, Claudiu T Supuran
Sulphonamide inhibition studies of the β-carbonic anhydrase GsaCAβ present in the salmon platyhelminth parasite Gyrodactylus salaris . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris V Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Lisa Sequeira, Simona Distinto, Rita Meleddu, Marco Gaspari, Andrea Ageli, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Fernanda Borges, Eugenio Uriarte, Stefano Alcaro, Claudiu T Supuran, Elias Maccioni
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Moataz A Shaldam, Ahmed F Khalil, Hadia Almahli, Maiy Y Jaballah, Andrea Angeli, Eman F Khaleel, Rehab Mustafa Badi, Eslam B Elkaeed, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Identification of 3-(5-cyano-6-oxo-pyridin-2-yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity. Archiv der Pharmazie (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 66 (3) (2023)
Claudiu T Supuran
Latest advances in specific inhibition of tumor-associated carbonic anhydrases. Future medicinal chemistry (2023)
Annachiara Sarnella, Ylenia Ferrara, Sandra Albanese, Daniela Omodei, Gennaro Chiappetta, Giuseppina De Simone, Claudiu T Supuran, Antonella Zannetti
Inhibition of Bone Marrow-Mesenchymal Stem Cell-Induced Carbonic Anhydrase IX Potentiates Chemotherapy Efficacy in Triple-Negative Breast Cancer Cells. Cells 12 (2) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Morteza Abdoli, Alessandro Bonardi, Claudiu T Supuran, Raivis Žalubovskis
Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Shaimaa M Aboukhatwa, Peter A Sidhom, Andrea Ageli, Claudiu T Supuran, Haytham O Tawfik
Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids. ACS omega 8 (8) (2023)
Simone Giovannuzzi, Anil Kumar Marapaka, Nader S Abutaleb, Fabrizio Carta, Hsin-Wen Liang, Alessio Nocentini, Luigi Pisano, Mohamed N Seleem, Daniel P Flaherty, Claudiu T Supuran
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Md Abu Sufian, Sabina Zamanova, Ahmed M Shabana, Brianna Kemp, Utpal K Mondal, Claudiu T Supuran, Marc A Ilies
Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors. International journal of molecular sciences 24 (5) (2023)
Morteza Abdoli, Alessandro Bonardi, Niccolò Paoletti, Ashok Aspatwar, Seppo Parkkila, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N -((4-Sulfamoylphenyl)carbamothioyl) Amides. Molecules (Basel, Switzerland) 28 (10) (2023)
Doretta Cuffaro, Riccardo Di Leo, Lidia Ciccone, Alessio Nocentini, Claudiu T Supuran, Elisa Nuti, Armando Rossello
New isoxazolidinyl-based N -alkylethanolamines as new activators of human brain carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Alessandro Bonardi, Claudiu T Supuran, Raivis Žalubovskis
Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Claudiu T Supuran
Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Carbonic Anhydrase Inhibitors as Novel Antibacterials in the Era of Antibiotic Resistance: Where Are We Now? Antibiotics (Basel, Switzerland) 12 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Bader I Huwaimel, Sravan K Jonnalagadda, Shirisha Jonnalagadda, Shikha Kumari, Alessio Nocentini, Claudiu T Supuran, Paul C Trippier
Selective carbonic anhydrase IX and XII inhibitors based around a functionalized coumarin scaffold. Drug development research (2023)
Heba Abdelrasheed Allam, Mohamed E Albakry, Walaa R Mahmoud, Alessandro Bonardi, Shaimaa A Moussa, Samy Mohamady, Hatem A Abdel-Aziz, Claudiu T Supuran, Hany S Ibrahim
Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Moataz A Shaldam, Hadia Almahli, Andrea Ageli, Rehab Mustafa Badi, Eman F Khaleel, Abdelrahman I Zain-Alabdeen, Zainab M Elsayed, Eslam B Elkaeed, Rofaida Salem, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Aiva Plotniece, Arkadij Sobolev, Claudiu T Supuran, Fabrizio Carta, Fredrik Björkling, Henrik Franzyk, Jari T Yli-Kauhaluoma, Koen Augustyns, Paul Cos, Linda De Vooght, Matthias Govaerts, Juliana Aizawa, Päivi Tammela, Raivis Žalubovskis
Selected strategies to fight pathogenic bacteria. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Viviana De Luca, Clemente Capasso, Claudiu T Supuran, Raivis Žalubovskis
Investigation of carbonic anhydrase inhibitory potency of ( Z/E )-alkyl N '-benzyl- N -(arylsulfonyl)-carbamimidothioates. Future medicinal chemistry 15 (7) (2023)
Heba Abdelrasheed Allam, Mohamed E Albakry, Walaa R Mahmoud, Alessandro Bonardi, Shaimaa A Moussa, Samy Mohamady, Hatem A Abdel-Aziz, Claudiu T Supuran, Hany S Ibrahim
Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Viviana De Luca, Clemente Capasso, Claudiu T Supuran, Raivis Žalubovskis
Investigation of carbonic anhydrase inhibitory potency of ( Z/E )-alkyl N '-benzyl- N -(arylsulfonyl)-carbamimidothioates. Future medicinal chemistry (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T Supuran, Raivis Žalubovskis
Aryl derivatives of 3 H -1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Xiaojing Huang, Daniel Winter, Dominic J Glover, Claudiu T Supuran, W Alexander Donald
Effects of Phosphorylation on the Activity, Inhibition and Stability of Carbonic Anhydrases. International journal of molecular sciences 24 (11) (2023)
Claudiu T Supuran
Progress of Section "Biochemistry" in 2022. International journal of molecular sciences 24 (6) (2023)
Annachiara Sarnella, Ylenia Ferrara, Sandra Albanese, Daniela Omodei, Gennaro Chiappetta, Giuseppina De Simone, Claudiu T Supuran, Antonella Zannetti
Inhibition of Bone Marrow-Mesenchymal Stem Cell-Induced Carbonic Anhydrase IX Potentiates Chemotherapy Efficacy in Triple-Negative Breast Cancer Cells. Cells 12 (2) (2023)
Heba Abdelrasheed Allam, Mohamed E Albakry, Walaa R Mahmoud, Alessandro Bonardi, Shaimaa A Moussa, Samy Mohamady, Hatem A Abdel-Aziz, Claudiu T Supuran, Hany S Ibrahim
Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Tuba Tekeli, Suleyman Akocak, Andrea Petreni, Nebih Lolak, Servet Çete, Claudiu T Supuran
Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Valentina Puca, Gabriele Turacchio, Beatrice Marinacci, Claudiu T Supuran, Clemente Capasso, Pamela Di Giovanni, Ilaria D'Agostino, Simone Carradori, Rossella Grande
Antimicrobial and Antibiofilm Activities of Carvacrol, Amoxicillin and Salicylhydroxamic Acid Alone and in Combination vs. Helicobacter pylori: Towards a New Multi-Targeted Therapy. International journal of molecular sciences 24 (5) (2023)
Francesco Fiorentino, Fabrizio Carta, Dante Rotili, Antonello Mai, Claudiu T Supuran
State of the art of carbonic anhydrase activators. Future medicinal chemistry (2023)
Md Abu Sufian, Sabina Zamanova, Ahmed M Shabana, Brianna Kemp, Utpal K Mondal, Claudiu T Supuran, Marc A Ilies
Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors. International journal of molecular sciences 24 (5) (2023)
Bader I Huwaimel, Sravan K Jonnalagadda, Shirisha Jonnalagadda, Shikha Kumari, Alessio Nocentini, Claudiu T Supuran, Paul C Trippier
Selective carbonic anhydrase IX and XII inhibitors based around a functionalized coumarin scaffold. Drug development research (2023)
Morteza Abdoli, Claudiu T Supuran, Raivis Žalubovskis
2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Ashok Aspatwar, Alessandro Bonardi, Heidi Aisala, Ksenia Zueva, Craig Robert Primmer, Jaakko Lumme, Seppo Parkkila, Claudiu T Supuran
Sulphonamide inhibition studies of the β-carbonic anhydrase GsaCAβ present in the salmon platyhelminth parasite Gyrodactylus salaris . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Annachiara Sarnella, Ylenia Ferrara, Sandra Albanese, Daniela Omodei, Gennaro Chiappetta, Giuseppina De Simone, Claudiu T Supuran, Antonella Zannetti
Inhibition of Bone Marrow-Mesenchymal Stem Cell-Induced Carbonic Anhydrase IX Potentiates Chemotherapy Efficacy in Triple-Negative Breast Cancer Cells. Cells 12 (2) (2023)
Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 66 (3) (2023)
Ashraf K El-Damasy, Hyun Ji Kim, Alessio Nocentini, Seon Hee Seo, Wagdy M Eldehna, Eun-Kyoung Bang, Claudiu T Supuran, Gyochang Keum
Discovery of new 6-ureido/amidocoumarins as highly potent and selective inhibitors for the tumour-relevant carbonic anhydrases IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Heba Abdelrasheed Allam, Mohamed E Albakry, Walaa R Mahmoud, Alessandro Bonardi, Shaimaa A Moussa, Samy Mohamady, Hatem A Abdel-Aziz, Claudiu T Supuran, Hany S Ibrahim
Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci, Claudiu T Supuran
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of medicinal chemistry 66 (3) (2023)
Mónica Martínez-Montiel, Laura L Romero-Hernández, Simone Giovannuzzi, Paloma Begines, Adrián Puerta, Ana I Ahuja-Casarín, Miguel X Fernandes, Penélope Merino-Montiel, Sara Montiel-Smith, Alessio Nocentini, José Manuel Padrón, Claudiu T Supuran, José G Fernández-Bolaños, Óscar López
Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (11) (2023)
Claudiu T Supuran
Progress of Section "Biochemistry" in 2022. International journal of molecular sciences 24 (6) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Md Abu Sufian, Sabina Zamanova, Ahmed M Shabana, Brianna Kemp, Utpal K Mondal, Claudiu T Supuran, Marc A Ilies
Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors. International journal of molecular sciences 24 (5) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Belma Zengin Kurt, Gulsen Celebi, Dilek Ozturk Civelek, Andrea Ageli, Atilla Akdemir, Fatih Sonmez, Claudiu T Supuran
Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS omega 8 (6) (2023)
Germán Benito, Ilaria D'Agostino, Simone Carradori, Marialuigia Fantacuzzi, Mariangela Agamennone, Valentina Puca, Rossella Grande, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Erlotinib-containing benzenesulfonamides as anti- Helicobacter pylori agents through carbonic anhydrase inhibition. Future medicinal chemistry (2023)
Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Mudasir Nabi Peerzada, Daniela Vullo, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Amir Azam
Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors. ACS medicinal chemistry letters 14 (6) (2023)
Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T Supuran
Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Marjan Sobati, Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Inhibition Profiles of Some Novel Sulfonamide-Incorporated α-Aminophosphonates on Human Carbonic Anhydrases. ACS medicinal chemistry letters 14 (8) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Simone Giovannuzzi, Viviana De Luca, Clemente Capasso, Claudiu T Supuran
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Claudiu T Supuran
Progress of Section "Biochemistry" in 2022. International journal of molecular sciences 24 (6) (2023)
Lalit Vats, Priyanka Arya, Rajiv Kumar, Simone Giovannuzzi, Neera Raghav, Claudiu T Supuran, Pawan K Sharma
Keto-bridged dual triazole-linked benzenesulfonamides as potent carbonic anhydrase and cathepsin B inhibitors. Future medicinal chemistry (2023)
Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T Supuran
Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Thor Eysteinsson, Andrea García-Llorca, Arnar Oessur Hardarson, Daniela Vullo, Fabrizio Carta, Claudiu T Supuran
Membrane Permeability Is Required for the Vasodilatory Effect of Carbonic Anhydrase Inhibitors in Porcine Retinal Arteries. International journal of molecular sciences 24 (9) (2023)
Davide Ialongo, Antonella Messore, Valentina Noemi Madia, Valeria Tudino, Alessio Nocentini, Paola Gratteri, Simone Giovannuzzi, Claudiu T Supuran, Alice Nicolai, Susanna Scarpa, Samanta Taurone, Michele Camarda, Marco Artico, Veronica Papa, Francesco Saccoliti, Luigi Scipione, Roberto Di Santo, Roberta Costi
Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII. Pharmaceuticals (Basel, Switzerland) 16 (2) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Simone Carradori, Andrea Ageli, Patrick Severin Sfragano, Xheila Yzeiri, Massimo Calamante, Damiano Tanini, Antonella Capperucci, Hannah Kunstek, Mihayl Varbanov, Clemente Capasso, Claudiu T Supuran
Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents. International journal of molecular sciences 24 (11) (2023)
Jekateri Na Ivanova, Alessio Nocentini, Kaspars Tars, Ja Nis Leita Ns, Elviss Dvinskis, Andris Kazaks, Ilona Domračeva, Claudiu T Supuran, Raivis Žalubovskis
Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect. Journal of medicinal chemistry (2023)
Claudiu T Supuran
Latest advances in specific inhibition of tumor-associated carbonic anhydrases. Future medicinal chemistry 15 (1) (2023)
Morteza Abdoli, Claudiu T Supuran, Raivis Žalubovskis
2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Viviana De Luca, Clemente Capasso, Claudiu T Supuran, Raivis Žalubovskis
Investigation of carbonic anhydrase inhibitory potency of ( Z/E )-alkyl N '-benzyl- N -(arylsulfonyl)-carbamimidothioates. Future medicinal chemistry 15 (7) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)

Claudiu T Supuran.css-eqlu8i{font-size:small;padding-left:4px;} (Claudiu Supuran, Claudiu T Supran)

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Claudiu T Supuran (Claudiu Supuran, Claudiu T Supran)