Claudiu T Supuran (Claudiu Supuran, Claudiu T Supran)

ORCID

Publication Activity (10 Years)

Years Active: 2016-2024
Publications (10 Years): 586

Top Venues

Journal of enzyme inhibition and medicinal chemistry

Journal of medicinal chemistry

International journal of molecular sciences

Molecules (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Silvia Bua, Alessio Nocentini, Alessandro Bonardi, Giuseppe Palma, Giulia Ciampi, Angela Giliberti, Federica Iannelli, Francesca Bruzzese, Claudiu T Supuran, Filomena de Nigris
Harnessing Nitric Oxide-Donating Benzofuroxans for Targeted Inhibition of Carbonic Anhydrase IX in Cancer. Journal of medicinal chemistry (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Ehab S Taher, Adel A Marzouk, Walaa Hamada Abd-Allah, Simone Giovannuzzi, Tarek S Ibrahim, Claudiu T Supuran, Mohamed A El Hamd, Mohammed Farrag El-Behairy
Tailored Tetrasubstituted Imidazole Carrying the Benzenesulfonamide Fragments as Selective Human Carbonic Anhydrase IX/XII Inhibitors. ChemMedChem (2024)
Amit Kumar, Priyanka Arya, Simone Giovannuzzi, Brij Mohan, Neera Raghav, Claudiu T Supuran, Pawan K Sharma
Novel 1,2,4-triazoles as selective carbonic anhydrase inhibitors showing ancillary anticathepsin B activity. Future medicinal chemistry (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Salma M Hefny, Tarek F El-Moselhy, Nabaweya El-Din, Simone Giovannuzzi, Thamer Bin Traiki, Mansoor-Ali Vaali-Mohammed, Ahmed M El-Dessouki, Koki Yamaguchi, Masaharu Sugiura, Moataz A Shaldam, Claudiu T Supuran, Maha-Hamadien Abdulla, Wagdy M Eldehna, Haytham O Tawfik
Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR-2 as Potential Agents for Solid Tumors: X-ray, In Vitro , In Vivo , and In Silico Investigations of Coumarin-Based Thiazoles. Journal of medicinal chemistry (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Fawzy A Elbarbry, Tamer M Ibrahim, Mohamed A Abdelrahman, Claudiu T Supuran, Wagdy M Eldehna
Inhibitory Effect of Two Carbonic Anhydrases Inhibitors on the Activity of Major Cytochrome P450 Enzymes. European journal of drug metabolism and pharmacokinetics 49 (5) (2024)
Letizia Giampietro, Beatrice Marinacci, Alice Della Valle, Ilaria D'Agostino, Aldo Lauro, Mattia Mori, Simone Carradori, Alessandra Ammazzalorso, Barbara De Filippis, Cristina Maccallini, Andrea Ageli, Clemente Capasso, Santolo Francati, Adriano Mollica, Rossella Grande, Claudiu T Supuran
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies. Pharmaceuticals (Basel, Switzerland) 17 (8) (2024)
Ismail Koyuncu, Ebru Temiz, Behice Hande Sisman, Mustafa Durgun, Ozgür Yüksekdag, Simone Giovannuzzi, Claudiu T Supuran
Effective Anticancer Potential of a New Sulfonamide as a Carbonic Anhydrase IX Inhibitor Against Aggressive Tumors. ChemMedChem (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry 67 (5) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Viviana De Luca, Simone Giovannuzzi, Claudiu T Supuran, Clemente Capasso
A comprehensive investigation of the anion inhibition profile of a β-carbonic anhydrase from Acinetobacter baumannii for crafting innovative antimicrobial treatments. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry 67 (11) (2024)
Amit Kumar, Priyanka Arya, Simone Giovannuzzi, Brij Mohan, Neera Raghav, Claudiu T Supuran, Pawan K Sharma
Novel 1,2,4-triazoles as selective carbonic anhydrase inhibitors showing ancillary anticathepsin B activity. Future medicinal chemistry 16 (8) (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Ehab S Taher, Adel A Marzouk, Walaa Hamada Abd-Allah, Simone Giovannuzzi, Tarek S Ibrahim, Claudiu T Supuran, Mohamed A El Hamd, Mohammed Farrag El-Behairy
Tailored Tetrasubstituted Imidazole Carrying the Benzenesulfonamide Fragments as Selective Human Carbonic Anhydrase IX/XII Inhibitors. ChemMedChem 19 (10) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Martina Palomba, Andrea Angeli, Riccardo Galdini, Alexandra Joana Hughineata, Gelson Perin, Eder Joao Lenardao, Francesca Marini, Claudio Santi, Claudiu T Supuran, Luana Bagnoli
Iodine/Oxone® oxidative system for the synthesis of selenylindoles bearing a benzenesulfonamide moiety as carbonic anhydrase I, II, IX, and XII inhibitors. Organic & biomolecular chemistry (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry 67 (4) (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry 67 (5) (2024)
Molly S Youse, Nader S Abutaleb, Alessio Nocentini, Abdallah S Abdelsattar, Farman Ali, Claudiu T Supuran, Mohamed N Seleem, Daniel P Flaherty
Optimization of Ethoxzolamide Analogs with Improved Pharmacokinetic Properties for In Vivo Efficacy against Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry 67 (4) (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry (2024)
Mehmet Onyilmaz, Murat Koca, Andrea Ammara, Mustafa Degirmenci, Claudiu T Supuran
Isocoumarins incorporating chalcone moieties act as isoform selective tumor-associated carbonic anhydrase inhibitors. Future medicinal chemistry 16 (13) (2024)
Haytham O Tawfik, Mohamed M Saleh, Andrea Ammara, Eman F Khaleel, Rehab Badi, Yomna T T Khater, Rabab Ahmed Rasheed, Ahmed A Attia, Salma M Hefny, Eslam B Elkaeed, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna, Moataz A Shaldam
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma. Journal of medicinal chemistry 67 (2) (2024)
Muhammed Trawally, Kübra Demir-Yazıcı, Andrea Ageli, Kerem Kaya, Atilla Akdemir, Claudiu T Supuran, Özlen Güzel-Akdemir
Thiosemicarbazone-benzenesulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies. Anti-cancer agents in medicinal chemistry 24 (9) (2024)
Jaydeo T Kilbile, Suryakant B Sapkal, Gioele Renzi, Ilaria D'Agostino, Luigi Cutarella, Mattia Mori, Barbara De Filippis, Imadul Islam, Maria Luisa Massardi, Elena Somenza, Roberto Ronca, Yasinalli Tamboli, Fabrizio Carta, Claudiu T Supuran
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (6) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Fawzy A Elbarbry, Tamer M Ibrahim, Mohamed A Abdelrahman, Claudiu T Supuran, Wagdy M Eldehna
Inhibitory Effect of Two Carbonic Anhydrases Inhibitors on the Activity of Major Cytochrome P450 Enzymes. European journal of drug metabolism and pharmacokinetics 49 (5) (2024)
Mourad A M Aboul-Soud, Yazeed A Al-Sheikh, Hazem K Ghneim, Claudiu T Supuran, Fabrizio Carta
Kinase inhibitors: 20 years of success and many new challenges and recent trends in their patents. Expert opinion on therapeutic patents 34 (7) (2024)
Mehmet Onyilmaz, Murat Koca, Andrea Ammara, Mustafa Degirmenci, Claudiu T Supuran
Isocoumarins incorporating chalcone moieties act as isoform selective tumor-associated carbonic anhydrase inhibitors. Future medicinal chemistry 16 (13) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Mourad A M Aboul-Soud, Yazeed A Al-Sheikh, Hazem K Ghneim, Claudiu T Supuran, Fabrizio Carta
Kinase inhibitors: 20 years of success and many new challenges and recent trends in their patents. Expert opinion on therapeutic patents (2024)
Giuseppina De Simone, Claudiu T Supuran
Anticancer drugs: where are we now? Expert opinion on therapeutic patents 34 (7) (2024)
Ismail Koyuncu, Ebru Temiz, Behice Hande Sisman, Mustafa Durgun, Ozgür Yüksekdag, Simone Giovannuzzi, Claudiu T Supuran
Effective Anticancer Potential of a New Sulfonamide as a Carbonic Anhydrase IX Inhibitor Against Aggressive Tumors. ChemMedChem 19 (9) (2024)
Arzu Gumus, Ilaria D'Agostino, Valentina Puca, Valentina Crocetta, Simone Carradori, Luigi Cutarella, Mattia Mori, Fabrizio Carta, Andrea Ageli, Clemente Capasso, Claudiu T Supuran
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α-carbonic anhydrase inhibitors. Archiv der Pharmazie (2024)
Elena Lucarini, Vanessa D'Antogiovanni, Luca Antonioli, Carla Ghelardini, Lorenzo Di Cesare Mannelli, Marta Ferraroni, Maria Locuoco, Antonella Capperucci, Damiano Tanini, Andrea Ageli, Claudiu T Supuran
Study of Chalcogen Aspirin Derivatives with Carbonic Anhydrase Inhibitory Properties for Treating Inflammatory Pain. ACS medicinal chemistry letters 15 (9) (2024)
Ehab S Taher, Adel A Marzouk, Walaa Hamada Abd-Allah, Simone Giovannuzzi, Tarek S Ibrahim, Claudiu T Supuran, Mohamed A El Hamd, Mohammed Farrag El-Behairy
Tailored Tetrasubstituted Imidazole Carrying the Benzenesulfonamide Fragments as Selective Human Carbonic Anhydrase IX/XII Inhibitors. ChemMedChem 19 (10) (2024)
Galina I Buravchenko, Alexander M Scherbakov, Stepan K Krymov, Diana I Salnikova, George V Zatonsky, Dominique Schols, Daniela Vullo, Claudiu T Supuran, Galina I Buravchenko
Synthesis and evaluation of sulfonamide derivatives of quinoxaline 1,4-dioxides as carbonic anhydrase inhibitors. RSC advances 14 (32) (2024)
Viviana De Luca, Simone Giovannuzzi, Claudiu T Supuran, Clemente Capasso
A comprehensive investigation of the anion inhibition profile of a β-carbonic anhydrase from Acinetobacter baumannii for crafting innovative antimicrobial treatments. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Fawzy A Elbarbry, Tamer M Ibrahim, Mohamed A Abdelrahman, Claudiu T Supuran, Wagdy M Eldehna
Inhibitory Effect of Two Carbonic Anhydrases Inhibitors on the Activity of Major Cytochrome P450 Enzymes. European journal of drug metabolism and pharmacokinetics 49 (5) (2024)
Ismail Koyuncu, Ebru Temiz, Behice Hande Sisman, Mustafa Durgun, Ozgür Yüksekdag, Simone Giovannuzzi, Claudiu T Supuran
Effective Anticancer Potential of a New Sulfonamide as a Carbonic Anhydrase IX Inhibitor Against Aggressive Tumors. ChemMedChem 19 (9) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Amit Kumar, Priyanka Arya, Simone Giovannuzzi, Brij Mohan, Neera Raghav, Claudiu T Supuran, Pawan K Sharma
Novel 1,2,4-triazoles as selective carbonic anhydrase inhibitors showing ancillary anticathepsin B activity. Future medicinal chemistry (2024)
Davide Moi, Serena Vittorio, Andrea Ageli, Claudiu T Supuran, Valentina Onnis
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (4) (2024)
Haytham O Tawfik, Mohamed M Saleh, Andrea Ammara, Eman F Khaleel, Rehab Badi, Yomna T T Khater, Rabab Ahmed Rasheed, Ahmed A Attia, Salma M Hefny, Eslam B Elkaeed, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna, Moataz A Shaldam
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma. Journal of medicinal chemistry (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Amit Kumar, Priyanka Arya, Simone Giovannuzzi, Brij Mohan, Neera Raghav, Claudiu T Supuran, Pawan K Sharma
Novel 1,2,4-triazoles as selective carbonic anhydrase inhibitors showing ancillary anticathepsin B activity. Future medicinal chemistry 16 (8) (2024)
Martina Palomba, Andrea Angeli, Riccardo Galdini, Alexandra Joana Hughineata, Gelson Perin, Eder Joao Lenardao, Francesca Marini, Claudio Santi, Claudiu T Supuran, Luana Bagnoli
Iodine/Oxone® oxidative system for the synthesis of selenylindoles bearing a benzenesulfonamide moiety as carbonic anhydrase I, II, IX, and XII inhibitors. Organic & biomolecular chemistry 22 (32) (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Claudiu T Supuran
Fighting antibacterial drug resistance. Expert opinion on therapeutic patents 34 (6) (2024)
Giuseppina De Simone, Claudiu T Supuran
Anticancer drugs: where are we now? Expert opinion on therapeutic patents (2024)
Amit Kumar, Priyanka Arya, Simone Giovannuzzi, Brij Mohan, Neera Raghav, Claudiu T Supuran, Pawan K Sharma
Novel 1,2,4-triazoles as selective carbonic anhydrase inhibitors showing ancillary anticathepsin B activity. Future medicinal chemistry (2024)
Salma M Hefny, Tarek F El-Moselhy, Nabaweya El-Din, Simone Giovannuzzi, Thamer Bin Traiki, Mansoor-Ali Vaali-Mohammed, Ahmed M El-Dessouki, Koki Yamaguchi, Masaharu Sugiura, Moataz A Shaldam, Claudiu T Supuran, Maha-Hamadien Abdulla, Wagdy M Eldehna, Haytham O Tawfik
Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR-2 as Potential Agents for Solid Tumors: X-ray, In Vitro , In Vivo , and In Silico Investigations of Coumarin-Based Thiazoles. Journal of medicinal chemistry 67 (9) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Davide Moi, Serena Vittorio, Andrea Ageli, Claudiu T Supuran, Valentina Onnis
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (4) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Fawzy A Elbarbry, Tamer M Ibrahim, Mohamed A Abdelrahman, Claudiu T Supuran, Wagdy M Eldehna
Inhibitory Effect of Two Carbonic Anhydrases Inhibitors on the Activity of Major Cytochrome P450 Enzymes. European journal of drug metabolism and pharmacokinetics (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry (2024)
Mehmet Onyilmaz, Murat Koca, Andrea Ammara, Mustafa Degirmenci, Claudiu T Supuran
Isocoumarins incorporating chalcone moieties act as isoform selective tumor-associated carbonic anhydrase inhibitors. Future medicinal chemistry 16 (13) (2024)
Viviana De Luca, Simone Giovannuzzi, Clemente Capasso, Claudiu T Supuran
Cloning, expression, and purification of an α-carbonic anhydrase from Toxoplasma gondii to unveil its kinetic parameters and anion inhibition profile. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Claudiu T Supuran
Fighting antibacterial drug resistance. Expert opinion on therapeutic patents (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry (2024)
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Letizia Giampietro, Beatrice Marinacci, Alice Della Valle, Ilaria D'Agostino, Aldo Lauro, Mattia Mori, Simone Carradori, Alessandra Ammazzalorso, Barbara De Filippis, Cristina Maccallini, Andrea Ageli, Clemente Capasso, Santolo Francati, Adriano Mollica, Rossella Grande, Claudiu T Supuran
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies. Pharmaceuticals (Basel, Switzerland) 17 (8) (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Morteza Abdoli, Alessandro Bonardi, Claudiu T Supuran, Raivis Žalubovskis
Synthesis and Carbonic Anhydrase I, II, IX, and XII Inhibition Studies with a Series of Cyclic Sulfonyl Guanidines. ChemMedChem (2024)
Galina I Buravchenko, Alexander M Scherbakov, Stepan K Krymov, Diana I Salnikova, George V Zatonsky, Dominique Schols, Daniela Vullo, Claudiu T Supuran, Galina I Buravchenko
Synthesis and evaluation of sulfonamide derivatives of quinoxaline 1,4-dioxides as carbonic anhydrase inhibitors. RSC advances 14 (32) (2024)
Hakan Aslan, Gioele Renzi, Andrea Ageli, Ilaria D'Agostino, Roberto Ronca, Maria Luisa Massardi, Camilla Tavani, Simone Carradori, Marta Ferraroni, Paolo Governa, Fabrizio Manetti, Fabrizio Carta, Claudiu T Supuran
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC medicinal chemistry 15 (6) (2024)
Viviana De Luca, Simone Giovannuzzi, Clemente Capasso, Claudiu T Supuran
Cloning, expression, and purification of an α-carbonic anhydrase from Toxoplasma gondii to unveil its kinetic parameters and anion inhibition profile. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessio Nocentini, Alessia Costa, Alessandro Bonardi, Andrea Ammara, Simone Giovannuzzi, Andrea Petreni, Gianluca Bartolucci, Barbara Rani, Manuela Leri, Monica Bucciantini, José G Fernández-Bolaños, Óscar López, Maria Beatrice Passani, Gustavo Provensi, Paola Gratteri, Claudiu T Supuran
Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases. Journal of medicinal chemistry (2024)
Muhammed Trawally, Kübra Demir-Yazıcı, Andrea Ageli, Kerem Kaya, Atilla Akdemir, Claudiu T Supuran, Özlen Güzel-Akdemir
Thiosemicarbazone-benzene Sulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies. Anti-cancer agents in medicinal chemistry (2024)
Haytham O Tawfik, Mohamed M Saleh, Andrea Ammara, Eman F Khaleel, Rehab Badi, Yomna T T Khater, Rabab Ahmed Rasheed, Ahmed A Attia, Salma M Hefny, Eslam B Elkaeed, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna, Moataz A Shaldam
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma. Journal of medicinal chemistry 67 (2) (2024)
Viviana De Luca, Simone Giovannuzzi, Clemente Capasso, Claudiu T Supuran
Cloning, expression, and purification of an α-carbonic anhydrase from Toxoplasma gondii to unveil its kinetic parameters and anion inhibition profile. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Jaydeo T Kilbile, Suryakant B Sapkal, Gioele Renzi, Ilaria D'Agostino, Luigi Cutarella, Mattia Mori, Barbara De Filippis, Imadul Islam, Maria Luisa Massardi, Elena Somenza, Roberto Ronca, Yasinalli Tamboli, Fabrizio Carta, Claudiu T Supuran
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (6) (2024)
Viviana De Luca, Simone Giovannuzzi, Claudiu T Supuran, Clemente Capasso
A comprehensive investigation of the anion inhibition profile of a β-carbonic anhydrase from Acinetobacter baumannii for crafting innovative antimicrobial treatments. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Davide Moi, Serena Vittorio, Andrea Ageli, Claudiu T Supuran, Valentina Onnis
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (4) (2024)
Hakan Aslan, Gioele Renzi, Andrea Ageli, Ilaria D'Agostino, Roberto Ronca, Maria Luisa Massardi, Camilla Tavani, Simone Carradori, Marta Ferraroni, Paolo Governa, Fabrizio Manetti, Fabrizio Carta, Claudiu T Supuran
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC medicinal chemistry 15 (6) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Claudiu T Supuran, Raivis Žalubovskis
2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Marialuigia Fantacuzzi, Ilaria D'Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Mariangela Agamennone, Andrea Ageli, Filomena Sannio, Jean Denis Docquier, Clemente Capasso, Claudiu T Supuran
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Gioele Renzi, Fabrizio Carta, Claudiu T Supuran
The Integrase: An Overview of a Key Player Enzyme in the Antiviral Scenario. International journal of molecular sciences 24 (15) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris Valerievich Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Farhat Ramzan, Syed Ayaz Nabi, Mehak Saba Lone, Alessandro Bonardi, Aabid Hamid, Sameena Bano, Kalicharan Sharma, Syed Shafi, Mohammed Samim, Kalim Javed, Claudiu T Supuran
Synthesis, biological evaluation and theoretical studies of ( E )-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Viviana De Luca, Clemente Capasso, Claudiu T Supuran, Raivis Žalubovskis
Novel thiazolone-benzenesulphonamide inhibitors of human and bacterial carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Niccolò Paoletti, Claudiu T Supuran
Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (7) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Mai H ElNaggar, Abdullah A Elgazar, Ghada Gamal, Shimaa M Hamed, Zainab M Elsayed, Mohamed K El-Ashrey, Amira Abood, Mahmoud A El Hassab, Ahmed M Soliman, Ramadan A El-Domany, Farid A Badria, Claudiu T Supuran, Wagdy M Eldehna
Identification of sulphonamide-tethered N -((triazol-4-yl)methyl)isatin derivatives as inhibitors of SARS-CoV-2 main protease. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)

Claudiu T Supuran.css-eqlu8i{font-size:small;padding-left:4px;} (Claudiu Supuran, Claudiu T Supran)

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Claudiu T Supuran (Claudiu Supuran, Claudiu T Supran)