Neil P Grimster

ORCID

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 12

Top Venues

Journal of medicinal chemistry

ACS medicinal chemistry letters

RSC medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Adelphe M Mfuh, Jeffrey A Boerth, Gayathri Bommakanti, Christina Chan, Alex J Chinn, Erin Code, Patrick J Fricke, Kathryn A Giblin, Andrea Gohlke, Catherine Hansel, Niresh Hariparsad, Samantha J Hughes, Meizhong Jin, Vasudev Kantae, Stefan L Kavanagh, Michelle L Lamb, Jordan Lane, Rachel Moore, Taranee Puri, Taylor R Quinn, Iswarya Reddy, Graeme R Robb, Kevin J Robbins, Miguel Gancedo Rodrigo, Marianne Schimpl, Baljinder Singh, Meha Singh, Haoran Tang, Clare Thomson, Jarrod J Walsh, Jamie Ware, Iain D G Watson, Min-Wei Ye, Gail L Wrigley, Andrew X Zhang, Yun Zhang, Neil P Grimster
Discovery, Optimization, and Biological Evaluation of Arylpyridones as Cbl-b Inhibitors. Journal of medicinal chemistry 67 (2) (2024)
Taylor R Quinn, Kathryn A Giblin, Clare Thomson, Jeffrey A Boerth, Gayathri Bommakanti, Erin Braybrooke, Christina Chan, Alex J Chinn, Erin Code, Caifeng Cui, Yukai Fan, Neil P Grimster, Keishi Kohara, Michelle L Lamb, Lina Ma, Adelphe M Mfuh, Graeme R Robb, Kevin J Robbins, Marianne Schimpl, Haoran Tang, Jamie Ware, Gail L Wrigley, Lin Xue, Yun Zhang, Huimin Zhu, Samantha J Hughes
Accelerated Discovery of Carbamate Cbl-b Inhibitors Using Generative AI Models and Structure-Based Drug Design. Journal of medicinal chemistry 67 (16) (2024)
Adelphe M Mfuh, Jeffrey A Boerth, Gayathri Bommakanti, Christina Chan, Alex J Chinn, Erin Code, Patrick J Fricke, Kathryn A Giblin, Andrea Gohlke, Catherine Hansel, Niresh Hariparsad, Samantha J Hughes, Meizhong Jin, Vasudev Kantae, Stefan L Kavanagh, Michelle L Lamb, Jordan Lane, Rachel Moore, Taranee Puri, Taylor R Quinn, Iswarya Reddy, Graeme R Robb, Kevin J Robbins, Miguel Gancedo Rodrigo, Marianne Schimpl, Baljinder Singh, Meha Singh, Haoran Tang, Clare Thomson, Jarrod J Walsh, Jamie Ware, Iain D G Watson, Min-Wei Ye, Gail L Wrigley, Andrew X Zhang, Yun Zhang, Neil P Grimster
Discovery, Optimization, and Biological Evaluation of Arylpyridones as Cbl-b Inhibitors. Journal of medicinal chemistry (2024)
Taylor R Quinn, Kathryn A Giblin, Clare Thomson, Jeffrey A Boerth, Gayathri Bommakanti, Erin Braybrooke, Christina Chan, Alex J Chinn, Erin Code, Caifeng Cui, Yukai Fan, Neil P Grimster, Keishi Kohara, Michelle L Lamb, Lina Ma, Adelphe M Mfuh, Graeme R Robb, Kevin J Robbins, Marianne Schimpl, Haoran Tang, Jamie Ware, Gail L Wrigley, Lin Xue, Yun Zhang, Huimin Zhu, Samantha J Hughes
Accelerated Discovery of Carbamate Cbl-b Inhibitors Using Generative AI Models and Structure-Based Drug Design. Journal of medicinal chemistry (2024)
Taylor R Quinn, Kathryn A Giblin, Clare Thomson, Jeffrey A Boerth, Gayathri Bommakanti, Erin Braybrooke, Christina Chan, Alex J Chinn, Erin Code, Caifeng Cui, Yukai Fan, Neil P Grimster, Keishi Kohara, Michelle L Lamb, Lina Ma, Adelphe M Mfuh, Graeme R Robb, Kevin J Robbins, Marianne Schimpl, Haoran Tang, Jamie Ware, Gail L Wrigley, Lin Xue, Yun Zhang, Huimin Zhu, Samantha J Hughes
Accelerated Discovery of Carbamate Cbl-b Inhibitors Using Generative AI Models and Structure-Based Drug Design. Journal of medicinal chemistry 67 (16) (2024)
Adelphe M Mfuh, Jeffrey A Boerth, Gayathri Bommakanti, Christina Chan, Alex J Chinn, Erin Code, Patrick J Fricke, Kathryn A Giblin, Andrea Gohlke, Catherine Hansel, Niresh Hariparsad, Samantha J Hughes, Meizhong Jin, Vasudev Kantae, Stefan L Kavanagh, Michelle L Lamb, Jordan Lane, Rachel Moore, Taranee Puri, Taylor R Quinn, Iswarya Reddy, Graeme R Robb, Kevin J Robbins, Miguel Gancedo Rodrigo, Marianne Schimpl, Baljinder Singh, Meha Singh, Haoran Tang, Clare Thomson, Jarrod J Walsh, Jamie Ware, Iain D G Watson, Min-Wei Ye, Gail L Wrigley, Andrew X Zhang, Yun Zhang, Neil P Grimster
Discovery, Optimization, and Biological Evaluation of Arylpyridones as Cbl-b Inhibitors. Journal of medicinal chemistry 67 (2) (2024)
Magnus Nilsson, Kristina Berggren, Susanne Berglund, Silvia Cerboni, Mia Collins, Göran Dahl, David Elmqvist, Neil P Grimster, Ramon Hendrickx, Johan R Johansson, Jason G Kettle, Matti Lepistö, Magdalena Rhedin, Amir Smailagic, Qibin Su, Tiiu Wennberg, Allan Wu, Torben Österlund, Thomas Naessens, Suman Mitra
Discovery of the Potent and Selective Inhaled Janus Kinase 1 Inhibitor AZD4604 and Its Preclinical Characterization. Journal of medicinal chemistry (2023)
Jeffrey A Boerth, Alex J Chinn, Marianne Schimpl, Gayathri Bommakanti, Christina Chan, Erin L Code, Kathryn A Giblin, Andrea Gohlke, Catherine S Hansel, Meizhong Jin, Stefan L Kavanagh, Michelle L Lamb, Jordan S Lane, Carrie J B Larner, Adelphe M Mfuh, Rachel K Moore, Taranee Puri, Taylor R Quinn, Minwei Ye, Kevin J Robbins, Miguel Gancedo Rodrigo, Haoran Tang, Jarrod Walsh, Jamie Ware, Gail L Wrigley, Iswarya Karapa Reddy, Yun Zhang, Neil P Grimster
Discovery of a Novel Benzodiazepine Series of Cbl-b Inhibitors for the Enhancement of Antitumor Immunity. ACS medicinal chemistry letters 14 (12) (2023)
Jeffrey A Boerth, Alex J Chinn, Marianne Schimpl, Gayathri Bommakanti, Christina Chan, Erin L Code, Kathryn A Giblin, Andrea Gohlke, Catherine S Hansel, Meizhong Jin, Stefan L Kavanagh, Michelle L Lamb, Jordan S Lane, Carrie J B Larner, Adelphe M Mfuh, Rachel K Moore, Taranee Puri, Taylor R Quinn, Minwei Ye, Kevin J Robbins, Miguel Gancedo Rodrigo, Haoran Tang, Jarrod Walsh, Jamie Ware, Gail L Wrigley, Iswarya Karapa Reddy, Yun Zhang, Neil P Grimster
Discovery of a Novel Benzodiazepine Series of Cbl-b Inhibitors for the Enhancement of Antitumor Immunity. ACS medicinal chemistry letters 14 (12) (2023)
Neil P Grimster
Covalent PROTACs: the best of both worlds? RSC medicinal chemistry 12 (9) (2021)
Qibin Su, Erica Banks, Geraldine Bebernitz, Kirsten Bell, Cassandra F Borenstein, Huawei Chen, Claudio E Chuaqui, Nanhua Deng, Andrew D Ferguson, Sameer Kawatkar, Neil P Grimster, Linette Ruston, Paul D Lyne, Jon A Read, Xianyou Peng, Xiaohui Pei, Stephen Fawell, Zhanlei Tang, Scott Throner, Melissa M Vasbinder, Haoyu Wang, Jon Winter-Holt, Richard Woessner, Allan Wu, Wenzhan Yang, Michael Zinda, Jason G Kettle
Discovery of (2R)-N-[3-[2-[(3-Methoxy-1-methyl-pyrazol-4-yl)amino]pyrimidin-4-yl]-1H-indol-7-yl]-2-(4-methylpiperazin-1-yl)propenamide (AZD4205) as a Potent and Selective Janus Kinase 1 Inhibitor. Journal of medicinal chemistry 63 (9) (2020)
Neil P Grimster, Erica Anderson, Marat Alimzhanov, Geraldine Bebernitz, Kirsten Bell, Claudio Chuaqui, Tracy Deegan, Andrew D Ferguson, Thomas Gero, Andreas Harsch, Dennis Huszar, Aarti Kawatkar, Jason G Kettle, Paul Lyne, Jon A Read, Caroline Rivard Costa, Linette Ruston, Patricia Schroeder, Jie Shi, Qibin Su, Scott Throner, Dorin Toader, Melissa Vasbinder, Richard Woessner, Haixia Wang, Allan Wu, Minwei Ye, Weijia Zheng, Michael Zinda
Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors. Journal of medicinal chemistry 61 (12) (2018)

Neil P Grimster.css-eqlu8i{font-size:small;padding-left:4px;}

Publication Activity (10 Years)

Top Topics

Top Venues

Neil P Grimster