Nicolotti Orazio (Orazio Nicolotti)

Scopus Author ID ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2018-2023
Publications (10 Years): 39

Top Venues

Molecules (Basel, Switzerland)

Journal of chemical information and modeling

Journal of clinical medicine

Pharmaceuticals (Basel, Switzerland)

Università degli Studi di Bari "Aldo Moro"

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Università degli Studi di Bari "Aldo Moro"

Italy

Assistant Professor :: Dipartimento di Farmacia - Scienze del Farmaco

Publications

Ashutosh Kumar Singh, Seong-Min Kim, Jong Min Oh, Mohamed A Abdelgawad, Mohammed M Ghoneim, T M Rangarajan, Sunil Kumar, Sachithra Thazhathuveedu Sudevan, Daniela Trisciuzzi, Nicolotti Orazio, Hoon Kim, Bijo Mathew
Exploration of a new class of monoamine oxidase B inhibitors by assembling benzyloxy pharmacophore on halogenated chalcones. Chemical biology & drug design (2023)
Nicola Gambacorta, Fulvio Ciriaco, Nicola Amoroso, Cosimo Damiano Altomare, Jürgen Bajorath, Nicolotti Orazio
CIRCE: Web-Based Platform for the Prediction of Cannabinoid Receptor Ligands Using Explainable Machine Learning. Journal of chemical information and modeling (2023)
Marco Paolino, Modesto de Candia, Rosa Purgatorio, Marco Catto, Mario Saletti, Anna Rita Tondo, Nicolotti Orazio, Andrea Cappelli, Antonella Brizzi, Claudia Mugnaini, Federico Corelli, Cosimo Damiano Altomare
Investigation on Novel E/Z 2-Benzylideneindan-1-One-Based Photoswitches with AChE and MAO-B Dual Inhibitory Activity. Molecules (Basel, Switzerland) 28 (15) (2023)
Daniela Trisciuzzi, Lydia Siragusa, Massimo Baroni, Ida Autiero, Nicolotti Orazio, Gabriele Cruciani
Getting Insights into Structural and Energetic Properties of Reciprocal Peptide-Protein Interactions. Journal of chemical information and modeling 62 (4) (2022)
Daniela Valeria Miniero, Nicola Gambacorta, Anna Spagnoletta, Vincenzo Tragni, Stefano Loizzo, Nicolotti Orazio, Ciro Leonardo Pierri, Annalisa De Palma
New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction. Journal of clinical medicine 11 (24) (2022)
Daniela Valeria Miniero, Nicola Gambacorta, Anna Spagnoletta, Vincenzo Tragni, Stefano Loizzo, Nicolotti Orazio, Ciro Leonardo Pierri, Annalisa De Palma
New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction. Journal of clinical medicine 11 (24) (2022)
Maria Vittoria Togo, Fabrizio Mastrolorito, Fulvio Ciriaco, Daniela Trisciuzzi, Anna Rita Tondo, Nicola Gambacorta, Loredana Bellantuono, Alfonso Monaco, Francesco Leonetti, Roberto Bellotti, Cosimo Damiano Altomare, Nicola Amoroso, Nicolotti Orazio
TIRESIA: An eXplainable Artificial Intelligence Platform for Predicting Developmental Toxicity. Journal of chemical information and modeling 63 (1) (2022)
Fulvio Ciriaco, Nicola Gambacorta, Daniela Trisciuzzi, Nicolotti Orazio
PLATO: A Predictive Drug Discovery Web Platform for Efficient Target Fishing and Bioactivity Profiling of Small Molecules. International journal of molecular sciences 23 (9) (2022)
Nisha Abdul Rehuman, Jong Min Oh, Mohamed Abdelwahab Abdelgawad, Eman A M Beshr, Mohammad A S Abourehab, Nicola Gambacorta, Nicolotti Orazio, Rakesh Kumar Jat, Hoon Kim, Bijo Mathew
Development of Halogenated-Chalcones Bearing with Dimethoxy Phenyl Head as Monoamine Oxidase-B Inhibitors. Pharmaceuticals (Basel, Switzerland) 15 (9) (2022)
Maria Vittoria Togo, Fabrizio Mastrolorito, Fulvio Ciriaco, Daniela Trisciuzzi, Anna Rita Tondo, Nicola Gambacorta, Loredana Bellantuono, Alfonso Monaco, Francesco Leonetti, Roberto Bellotti, Cosimo Damiano Altomare, Nicola Amoroso, Nicolotti Orazio
TIRESIA: An eXplainable Artificial Intelligence Platform for Predicting Developmental Toxicity. Journal of chemical information and modeling 63 (1) (2022)
Nicola Gambacorta, Leonardo Caputo, Laura Quintieri, Linda Monaci, Fulvio Ciriaco, Nicolotti Orazio
Rational Discovery of Antiviral Whey Protein-Derived Small Peptides Targeting the SARS-CoV-2 Main Protease. Biomedicines 10 (5) (2022)
Daniela Valeria Miniero, Nicola Gambacorta, Anna Spagnoletta, Vincenzo Tragni, Stefano Loizzo, Nicolotti Orazio, Ciro Leonardo Pierri, Annalisa De Palma
New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction. Journal of clinical medicine 11 (24) (2022)
Maria Vittoria Togo, Fabrizio Mastrolorito, Fulvio Ciriaco, Daniela Trisciuzzi, Anna Rita Tondo, Nicola Gambacorta, Loredana Bellantuono, Alfonso Monaco, Francesco Leonetti, Roberto Bellotti, Cosimo Damiano Altomare, Nicola Amoroso, Nicolotti Orazio
TIRESIA: An eXplainable Artificial Intelligence Platform for Predicting Developmental Toxicity. Journal of chemical information and modeling 63 (1) (2022)
Daniela Valeria Miniero, Nicola Gambacorta, Anna Spagnoletta, Vincenzo Tragni, Stefano Loizzo, Nicolotti Orazio, Ciro Leonardo Pierri, Annalisa De Palma
New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction. Journal of clinical medicine 11 (24) (2022)
Mehmet Abdullah Alagöz, Jong Min Oh, Yaren Nur Zenni, Zeynep Özdemir, Mohamed Abdelwahab Abdelgawad, Ibrahim A Naguib, Mohammed M Ghoneim, Nicola Gambacorta, Nicolotti Orazio, Hoon Kim, Bijo Mathew
Development of a Novel Class of Pyridazinone Derivatives as Selective MAO-B Inhibitors. Molecules (Basel, Switzerland) 27 (12) (2022)
Maria Vittoria Togo, Fabrizio Mastrolorito, Fulvio Ciriaco, Daniela Trisciuzzi, Anna Rita Tondo, Nicola Gambacorta, Loredana Bellantuono, Alfonso Monaco, Francesco Leonetti, Roberto Bellotti, Cosimo Damiano Altomare, Nicola Amoroso, Nicolotti Orazio
TIRESIA: An eXplainable Artificial Intelligence Platform for Predicting Developmental Toxicity. Journal of chemical information and modeling (2022)
Rosa Purgatorio, Nicola Gambacorta, Francesco Samarelli, Gianfranco Lopopolo, Modesto de Candia, Marco Catto, Nicolotti Orazio, Cosimo Damiano Altomare
Assessing the Role of a Malonamide Linker in the Design of Potent Dual Inhibitors of Factor Xa and Cholinesterases. Molecules (Basel, Switzerland) 27 (13) (2022)
Daniela Trisciuzzi, Lydia Siragusa, Massimo Baroni, Gabriele Cruciani, Nicolotti Orazio
An Integrated Machine Learning Model To Spot Peptide Binding Pockets in 3D Protein Screening. Journal of chemical information and modeling (2022)
Emanuele M Gargano, Abdelrahman Mohamed, Ahmed S Abdelsamie, Giuseppe Felice Mangiatordi, Hanna Drzewiecka, Paweł P Jagodziński, Arcangela Mazzini, Chris J van Koppen, Matthias W Laschke, Nicolotti Orazio, Angelo Carotti, Sandrine Marchais-Oberwinkler, Rolf Wolfgang Hartmann, Martin Frotscher
17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer. ACS medicinal chemistry letters 12 (12) (2021)
Alisa A Nevskaya, Lada V Anikina, Rosa Purgatorio, Marco Catto, Nicolotti Orazio, Modesto de Candia, Leonardo Pisani, Tatiana N Borisova, Almira R Miftyakhova, Aleksey V Varlamov, Elena Yu Nevskaya, Roman S Borisov, Leonid G Voskressensky, Cosimo Damiano Altomare
Homobivalent Lamellarin-Like Schiff Bases: In Vitro Evaluation of Their Cancer Cell Cytotoxicity and Multitargeting Anti-Alzheimer's Disease Potential. Molecules (Basel, Switzerland) 26 (2) (2021)
Nisha Abdul Rehuman, Jong Min Oh, Lekshmi R Nath, Ahmed Khames, Mohamed A Abdelgawad, Nicola Gambacorta, Nicolotti Orazio, Rakesh Kumar Jat, Hoon Kim, Bijo Mathew
Halogenated Coumarin-Chalcones as Multifunctional Monoamine Oxidase-B and Butyrylcholinesterase Inhibitors. ACS omega 6 (42) (2021)
Marialuigia Fantacuzzi, Marialucia Gallorini, Nicola Gambacorta, Alessandra Ammazzalorso, Zeineb Aturki, Marwa Balaha, Simone Carradori, Letizia Giampietro, Cristina Maccallini, Amelia Cataldi, Nicolotti Orazio, Rosa Amoroso, Barbara De Filippis
Design, Synthesis and Biological Evaluation of Aromatase Inhibitors Based on Sulfonates and Sulfonamides of Resveratrol. Pharmaceuticals (Basel, Switzerland) 14 (10) (2021)
Rosa Purgatorio, Nicola Gambacorta, Modesto de Candia, Marco Catto, Mariagrazia Rullo, Leonardo Pisani, Nicolotti Orazio, Cosimo Damiano Altomare
First-in-Class Isonipecotamide-Based Thrombin and Cholinesterase Dual Inhibitors with Potential for Alzheimer Disease. Molecules (Basel, Switzerland) 26 (17) (2021)
Alexander A Titov, Maxim S Kobzev, Marco Catto, Modesto de Candia, Nicola Gambacorta, Nunzio Denora, Leonardo Pisani, Nicolotti Orazio, Tatiana N Borisova, Alexey V Varlamov, Leonid G Voskressensky, Cosimo D Altomare
Away from Flatness: Unprecedented Nitrogen-Bridged Cyclopenta[a]indene Derivatives as Novel Anti-Alzheimer Multitarget Agents. ACS chemical neuroscience 12 (2) (2021)
Daniela Valeria Miniero, Anna Spagnoletta, Nicola Gambacorta, Vito Scalera, Ciro Leonardo Pierri, Nicolotti Orazio, Annalisa De Palma
The Interaction of Hemin, a Porphyrin Derivative, with the Purified Rat Brain 2-Oxoglutarate Carrier. Biomolecules 11 (8) (2021)
Anusree Venkidath, Jong Min Oh, Sanal Dev, Elham Amin, Shebina P Rasheed, Ajeesh Vengamthodi, Nicola Gambacorta, Ahmed Khames, Mohamed Abdelwahab Abdelgawad, Ginson George, Nicolotti Orazio, Hoon Kim, Bijo Mathew
Selected Class of Enamides Bearing Nitro Functionality as Dual-Acting with Highly Selective Monoamine Oxidase-B and BACE1 Inhibitors. Molecules (Basel, Switzerland) 26 (19) (2021)
Payyalot Koyiparambath Vishal, Jong Min Oh, Ahmed Khames, Mohamed Abdelwahab Abdelgawad, Aathira Sujathan Nair, Lekshmi R Nath, Nicola Gambacorta, Fulvio Ciriaco, Nicolotti Orazio, Hoon Kim, Bijo Mathew
Trimethoxylated Halogenated Chalcones as Dual Inhibitors of MAO-B and BACE-1 for the Treatment of Neurodegenerative Disorders. Pharmaceutics 13 (6) (2021)
Fulvio Ciriaco, Nicola Gambacorta, Domenico Alberga, Nicolotti Orazio
Quantitative Polypharmacology Profiling Based on a Multifingerprint Similarity Predictive Approach. Journal of chemical information and modeling 61 (10) (2021)
Rosa Purgatorio, Nicola Gambacorta, Marco Catto, Modesto de Candia, Leonardo Pisani, Alba Espargaró, Raimon Sabaté, Saverio Cellamare, Nicolotti Orazio, Cosimo D Altomare
Pharmacophore Modeling and 3D-QSAR Study of Indole and Isatin Derivatives as Antiamyloidogenic Agents Targeting Alzheimer's Disease. Molecules (Basel, Switzerland) 25 (23) (2020)
Francesca Carofiglio, Antonio Lopalco, Angela Lopedota, Annalisa Cutrignelli, Nicolotti Orazio, Nunzio Denora, Angela Stefanachi, Francesco Leonetti
Bcr-Abl Tyrosine Kinase Inhibitors in the Treatment of Pediatric CML. International journal of molecular sciences 21 (12) (2020)
Francesca Carofiglio, Daniela Trisciuzzi, Nicola Gambacorta, Francesco Leonetti, Angela Stefanachi, Nicolotti Orazio
Bcr-Abl Allosteric Inhibitors: Where We Are and Where We Are Going to. Molecules (Basel, Switzerland) 25 (18) (2020)
Anna Rita Tondo, Leonardo Caputo, Giuseppe Felice Mangiatordi, Linda Monaci, Giovanni Lentini, Antonio Francesco Logrieco, Michele Montaruli, Nicolotti Orazio, Laura Quintieri
Structure-Based Identification and Design of Angiotensin Converting Enzyme-Inhibitory Peptides from Whey Proteins. Journal of agricultural and food chemistry 68 (2) (2020)
Muhammed Çeçen, Jong Min Oh, Zeynep Özdemir, Saliha Ebru Büyüktuncel, Mehtap Uysal, Mohamed A Abdelgawad, Arafa Musa, Nicola Gambacorta, Nicolotti Orazio, Bijo Mathew, Hoon Kim
Design, Synthesis, and Biological Evaluation of Pyridazinones Containing the (2-Fluorophenyl) Piperazine Moiety as Selective MAO-B Inhibitors. Molecules (Basel, Switzerland) 25 (22) (2020)
Ashique Palakkathondi, Jong Min Oh, Sanal Dev, T M Rangarajan, Swafvan Kaipakasseri, Fathima Sahla Kavully, Nicola Gambacorta, Nicolotti Orazio, Hoon Kim, Bijo Mathew
(Hetero-)(arylidene)arylhydrazides as Multitarget-Directed Monoamine Oxidase Inhibitors. ACS combinatorial science 22 (11) (2020)
Ilaria Cicalini, Barbara De Filippis, Nicola Gambacorta, Antonio Di Michele, Silvia Valentinuzzi, Alessandra Ammazzalorso, Alice Della Valle, Rosa Amoroso, Nicolotti Orazio, Piero Del Boccio, Letizia Giampietro
Development of a Rapid Mass Spectrometric Determination of AMP and Cyclic AMP for PDE3 Activity Study: Application and Computational Analysis for Evaluating the Effect of a Novel 2-oxo-1,2-dihydropyridine-3-carbonitrile Derivative as PDE-3 Inhibitor. Molecules (Basel, Switzerland) 25 (8) (2020)
Domenico Alberga, Gambacorta Nicola, Trisciuzzi Daniela, Ciriaco Fulvio, Amoroso Nicola, Nicolotti Orazio
De Novo Drug Design of Targeted Chemical Libraries Based on Artificial Intelligence and Pair-Based Multiobjective Optimization. Journal of chemical information and modeling 60 (10) (2020)
Giuseppe Felice Mangiatordi, Tatiana Guzzo, Eugenio Claudio Rossano, Daniela Trisciuzzi, Domenico Alberga, Giovanni Fasciglione, Massimiliano Coletta, Alessandra Topai, Nicolotti Orazio
Design, Synthesis, and Biological Evaluation of Tetrahydro-β-carboline Derivatives as Selective Sub-Nanomolar Gelatinase Inhibitors. ChemMedChem 13 (13) (2018)
Domenico Alberga, Daniela Trisciuzzi, Michele Montaruli, Francesco Leonetti, Giuseppe Felice Mangiatordi, Nicolotti Orazio
A New Approach for Drug Target and Bioactivity Prediction: The Multifingerprint Similarity Search Algorithm (MuSSeL). Journal of chemical information and modeling 59 (1) (2018)
Giuseppe Felice Mangiatordi, Daniela Trisciuzzi, Rosamaria Iacobazzi, Nunzio Denora, Leonardo Pisani, Marco Catto, Francesco Leonetti, Domenico Alberga, Nicolotti Orazio
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitors. Chemical biology & drug design 92 (1) (2018)

Nicolotti Orazio.css-eqlu8i{font-size:small;padding-left:4px;} (Orazio Nicolotti)

Publication Activity (10 Years)

Top Topics

Top Venues

Nicolotti Orazio (Orazio Nicolotti)