Stephen L Buchwald

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 81

Top Topics

Reduced Graphene Oxide

Electron Transfer

Capillary Electrophoresis

Top Venues

Journal of the American Chemical Society

Angewandte Chemie (International ed. in English)

Organic letters

Science (New York, N.Y.)

This page only lists publications with an associated author ORCID identifier.

Publications

Jason Tao, Heemal H Dhanjee, Michael W Gribble, Veronika Kottisch, Jacob Rodriguez, Joseph S Brown, Holly Schmidt, Juhi Juneja, Fabienne Denhez, Peter S Lee, Daša Lipovšek, Stanley Krystek, Yihong Zhang, Patrick Bousquet, Yong Zhang, Bradley L Pentelute, Stephen L Buchwald
Site-Specific Antibody Prodrugs via S -Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues. Journal of the American Chemical Society (2024)
Subhash Garhwal, Yuyang Dong, Binh Khanh Mai, Peng Liu, Stephen L Buchwald
CuH-Catalyzed Regio- and Enantioselective Formal Hydroformylation of Vinyl Arenes. Journal of the American Chemical Society (2024)
Han-Jun Ai, Seoung-Tae Kim, Cecilia Liu, Stephen L Buchwald
Copper-Catalyzed Amination of Aryl Chlorides under Mild Reaction Conditions. Journal of the American Chemical Society (2024)
Michael J Strauss, Megan E Greaves, Seoung-Tae Kim, Christiana N Teijaro, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides. Angewandte Chemie (International ed. in English) 63 (19) (2024)
Kaibo Feng, Elaine Reichert Raguram, James R Howard, Ellyn Peters, Cecilia Liu, Matthew S Sigman, Stephen L Buchwald
Development of a Deactivation-Resistant Dialkylbiarylphosphine Ligand for Pd-Catalyzed Arylation of Secondary Amines. Journal of the American Chemical Society (2024)
Michael J Strauss, Megan E Greaves, Seoung-Tae Kim, Christiana N Teijaro, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides. Angewandte Chemie (International ed. in English) (2024)
Michael J Strauss, Megan E Greaves, Seoung-Tae Kim, Christiana N Teijaro, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides. Angewandte Chemie (International ed. in English) 63 (19) (2024)
Michael J Strauss, Kaylee X Liu, Megan E Greaves, Jakob C Dahl, Seoung-Tae Kim, Yong-Jin Wu, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Cu-Catalyzed Amination of Base-Sensitive Aryl Bromides and the Chemoselective N- and O-Arylation of Amino Alcohols. Journal of the American Chemical Society 146 (27) (2024)
Michael J Strauss, Megan E Greaves, Seoung-Tae Kim, Christiana N Teijaro, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides. Angewandte Chemie (International ed. in English) 63 (19) (2024)
Jason Tao, Heemal H Dhanjee, Michael W Gribble, Veronika Kottisch, Jacob Rodriguez, Joseph S Brown, Holly Schmidt, Juhi Juneja, Fabienne Denhez, Peter S Lee, Daša Lipovšek, Stanley Krystek, Yihong Zhang, Patrick Bousquet, Yong Zhang, Bradley L Pentelute, Stephen L Buchwald
Site-Specific Antibody Prodrugs via S -Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues. Journal of the American Chemical Society 146 (29) (2024)
Michael J Strauss, Kaylee X Liu, Megan E Greaves, Jakob C Dahl, Seoung-Tae Kim, Yong-Jin Wu, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Cu-Catalyzed Amination of Base-Sensitive Aryl Bromides and the Chemoselective N- and O-Arylation of Amino Alcohols. Journal of the American Chemical Society (2024)
Subhash Garhwal, Yuyang Dong, Binh Khanh Mai, Peng Liu, Stephen L Buchwald
CuH-Catalyzed Regio- and Enantioselective Formal Hydroformylation of Vinyl Arenes. Journal of the American Chemical Society 146 (20) (2024)
Michael J Strauss, Megan E Greaves, Seoung-Tae Kim, Christiana N Teijaro, Michael A Schmidt, Paul M Scola, Stephen L Buchwald
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides. Angewandte Chemie (International ed. in English) 63 (19) (2024)
Seoung-Tae Kim, Michael J Strauss, Albert Cabré, Stephen L Buchwald
Room-Temperature Cu-Catalyzed Amination of Aryl Bromides Enabled by DFT-Guided Ligand Design. Journal of the American Chemical Society (2023)
Elaine Reichert Raguram, Kaibo Feng, Aaron C Sather, Stephen L Buchwald
Pd-Catalyzed Amination of Base-Sensitive Five-Membered Heteroaryl Halides with Aliphatic Amines. Journal of the American Chemical Society 145 (6) (2023)
Simon L Rössler, Nathalie M Grob, Stephen L Buchwald, Bradley L Pentelute
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis. Science (New York, N.Y.) 379 (6635) (2023)
Nathalie M Grob, Clint Remarcik, Simon L Rössler, Jeffrey Y K Wong, John C K Wang, Jason Tao, Corey L Smith, Andrei Loas, Stephen L Buchwald, Dan L Eaton, Magdalena Preciado López, Bradley L Pentelute
Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders. ACS chemical biology (2023)
Elaine Reichert Raguram, Kaibo Feng, Aaron C Sather, Stephen L Buchwald
Pd-Catalyzed Amination of Base-Sensitive Five-Membered Heteroaryl Halides with Aliphatic Amines. Journal of the American Chemical Society 145 (6) (2023)
Simon L Rössler, Nathalie M Grob, Stephen L Buchwald, Bradley L Pentelute
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis. Science (New York, N.Y.) 379 (6635) (2023)
Elaine Reichert Raguram, Kaibo Feng, Aaron C Sather, Stephen L Buchwald
Pd-Catalyzed Amination of Base-Sensitive Five-Membered Heteroaryl Halides with Aliphatic Amines. Journal of the American Chemical Society (2023)
Dennis A Kutateladze, Binh Khanh Mai, Yuyang Dong, Yu Zhang, Peng Liu, Stephen L Buchwald
Stereoselective Synthesis of Trisubstituted Alkenes via Copper Hydride-Catalyzed Alkyne Hydroalkylation. Journal of the American Chemical Society (2023)
Yuxuan Ye, Seoung-Tae Kim, Ryan P King, Mu-Hyun Baik, Stephen L Buchwald
Studying Regioisomer Formation in the Pd-Catalyzed Fluorination of Cyclic Vinyl Triflates: Evidence for in situ Ligand Modification. Angewandte Chemie (International ed. in English) (2023)
Simon L Rössler, Nathalie M Grob, Stephen L Buchwald, Bradley L Pentelute
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis. Science (New York, N.Y.) 379 (6635) (2023)
Yuyang Dong, Alexander W Schuppe, Binh Khanh Mai, Peng Liu, Stephen L Buchwald
Confronting the Challenging Asymmetric Carbonyl 1,2-Addition Using Vinyl Heteroarene Pronucleophiles: Ligand-Controlled Regiodivergent Processes through a Dearomatized Allyl-Cu Species. Journal of the American Chemical Society 144 (13) (2022)
Sheng Feng, Yuyang Dong, Stephen L Buchwald
Enantioselective Hydrocarbamoylation of Alkenes. Angewandte Chemie (International ed. in English) 61 (31) (2022)
Martin Gazvoda, Heemal H Dhanjee, Jacob Rodriguez, Joseph S Brown, Charlotte E Farquhar, Nicholas L Truex, Andrei Loas, Stephen L Buchwald, Bradley L Pentelute
Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins. Journal of the American Chemical Society 144 (17) (2022)
Yuyang Dong, Kwangmin Shin, Binh Khanh Mai, Peng Liu, Stephen L Buchwald
Copper Hydride-Catalyzed Enantioselective Olefin Hydromethylation. Journal of the American Chemical Society 144 (36) (2022)
Anthony J Rojas, Justin M Wolfe, Heemal H Dhanjee, Ivan Buslov, Nicholas L Truex, Richard Y Liu, Walter Massefski, Bradley L Pentelute, Stephen L Buchwald
Palladium-peptide oxidative addition complexes for bioconjugation. Chemical science 13 (40) (2022)
James Levi Knippel, Anton Z Ni, Alexander W Schuppe, Stephen L Buchwald
A General Strategy for the Asymmetric Preparation of α-Stereogenic Allyl Silanes, Germanes, and Boronate Esters via Dual Copper Hydride- and Palladium-Catalysis. Angewandte Chemie (International ed. in English) 61 (47) (2022)
Martin Gazvoda, Heemal H Dhanjee, Jacob Rodriguez, Joseph S Brown, Charlotte E Farquhar, Nicholas L Truex, Andrei Loas, Stephen L Buchwald, Bradley L Pentelute
Correction to "Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins". Journal of the American Chemical Society 144 (22) (2022)
Sheng Feng, Stephen L Buchwald
CuH-Catalyzed Regio- and Enantioselective Hydrocarboxylation of Allenes: Toward Carboxylic Acids with Acyclic Quaternary Centers. Journal of the American Chemical Society 143 (13) (2021)
Ryan P King, Shane W Krska, Stephen L Buchwald
A Neophyl Palladacycle as an Air- and Thermally Stable Precursor to Oxidative Addition Complexes. Organic letters 23 (20) (2021)
Ryan P King, Shane W Krska, Stephen L Buchwald
A Ligand Exchange Process for the Diversification of Palladium Oxidative Addition Complexes. Organic letters 23 (15) (2021)
Chuan-Jin Hou, Alexander W Schuppe, James Levi Knippel, Anton Z Ni, Stephen L Buchwald
A Dual CuH- and Pd-Catalyzed Stereoselective Synthesis of Highly Substituted 1,3-Dienes. Organic letters 23 (22) (2021)
Alexander W Schuppe, James Levi Knippel, Gustavo M Borrajo-Calleja, Stephen L Buchwald
Enantioselective Hydroalkenylation of Olefins with Enol Sulfonates Enabled by Dual Copper Hydride and Palladium Catalysis. Journal of the American Chemical Society 143 (14) (2021)
Aaron J Mallek, Bradley L Pentelute, Stephen L Buchwald
Selective N-Arylation of p-Aminophenylalanine in Unprotected Peptides with Organometallic Palladium Reagents. Angewandte Chemie (International ed. in English) 60 (31) (2021)
James Levi Knippel, Yuxuan Ye, Stephen L Buchwald
Enantioselective C2-Allylation of Benzimidazoles Using 1,3-Diene Pronucleophiles. Organic letters 23 (6) (2021)
Jacob Rodriguez, Heemal H Dhanjee, Stephen L Buchwald
Amphiphilic Biaryl Monophosphine Ligands by Regioselective Sulfonation. Organic letters 23 (3) (2021)
Muhammad Jbara, Sebastian Pomplun, Carly K Schissel, Susana Wilson Hawken, Ann Boija, Isaac Klein, Jacob Rodriguez, Stephen L Buchwald, Bradley L Pentelute
Engineering Bioactive Dimeric Transcription Factor Analogs via Palladium Rebound Reagents. Journal of the American Chemical Society 143 (30) (2021)
Yiming Mo, Zhaohong Lu, Girish Rughoobur, Prashant Patil, Neil Gershenfeld, Akintunde I Akinwande, Stephen L Buchwald, Klavs F Jensen
Microfluidic electrochemistry for single-electron transfer redox-neutral reactions. Science (New York, N.Y.) 368 (6497) (2020)
Yuxuan Ye, Ilia Kevlishvili, Sheng Feng, Peng Liu, Stephen L Buchwald
Highly Enantioselective Synthesis of Indazoles with a C3-Quaternary Chiral Center Using CuH Catalysis. Journal of the American Chemical Society 142 (23) (2020)
Heemal H Dhanjee, Azin Saebi, Ivan Buslov, Alexander R Loftis, Stephen L Buchwald, Bradley L Pentelute
Correction to "Protein-Protein Cross-Coupling via Palladium-Protein Oxidative Addition Complexes from Cysteine Residues". Journal of the American Chemical Society 142 (28) (2020)
Hong Zhang, Paula Ruiz-Castillo, Alexander W Schuppe, Stephen L Buchwald
Improved Process for the Palladium-Catalyzed C-O Cross-Coupling of Secondary Alcohols. Organic letters 22 (14) (2020)
Scott D McCann, Elaine Reichert Raguram, Pedro Luis Arrechea, Stephen L Buchwald
Development of an Aryl Amination Catalyst with Broad Scope Guided by Consideration of Catalyst Stability. Journal of the American Chemical Society 142 (35) (2020)
Richard Y Liu, Joseph M Dennis, Stephen L Buchwald
The Quest for the Ideal Base: Rational Design of a Nickel Precatalyst Enables Mild, Homogeneous C-N Cross-Coupling. Journal of the American Chemical Society 142 (9) (2020)
Zhaohong Lu, Stephen L Buchwald
Enantioselective Preparation of Arenes with β-Stereogenic Centers: Confronting the 1,1-Disubstituted Olefin Problem Using CuH/Pd Cooperative Catalysis. Angewandte Chemie (International ed. in English) 59 (37) (2020)
Boyoung Y Park, Michael T Pirnot, Stephen L Buchwald
Visible Light-Mediated (Hetero)aryl Amination Using Ni(II) Salts and Photoredox Catalysis in Flow: A Synthesis of Tetracaine. The Journal of organic chemistry 85 (5) (2020)
Richard Y Liu, Stephen L Buchwald
CuH-Catalyzed Olefin Functionalization: From Hydroamination to Carbonyl Addition. Accounts of chemical research 53 (6) (2020)
Heemal H Dhanjee, Azin Saebi, Ivan Buslov, Alexander R Loftis, Stephen L Buchwald, Bradley L Pentelute
Protein-Protein Cross-Coupling via Palladium-Protein Oxidative Addition Complexes from Cysteine Residues. Journal of the American Chemical Society 142 (20) (2020)
Sheng Guo, Jiaqi Zhu, Stephen L Buchwald
Enantioselective Synthesis of β-Amino Acid Derivatives Enabled by Ligand-Controlled Reversal of Hydrocupration Regiochemistry. Angewandte Chemie (International ed. in English) 59 (47) (2020)
Heemal H Dhanjee, Ivan Buslov, Ian W Windsor, Ronald T Raines, Bradley L Pentelute, Stephen L Buchwald
Palladium-Protein Oxidative Addition Complexes by Amine-Selective Acylation. Journal of the American Chemical Society 142 (51) (2020)
Michael W Gribble, Richard Y Liu, Stephen L Buchwald
Evidence for Simultaneous Dearomatization of Two Aromatic Rings under Mild Conditions in Cu(I)-Catalyzed Direct Asymmetric Dearomatization of Pyridine. Journal of the American Chemical Society 142 (25) (2020)
Yujing Zhou, Lin Zhou, Luke T Jesikiewicz, Peng Liu, Stephen L Buchwald
Synthesis of Pyrroles through the CuH-Catalyzed Coupling of Enynes and Nitriles. Journal of the American Chemical Society 142 (22) (2020)
Achim Link, Yujing Zhou, Stephen L Buchwald
CuH-Catalyzed Asymmetric Reductive Amidation of α,β-Unsaturated Carboxylic Acids. Organic letters 22 (14) (2020)
Mycah R Uehling, Ryan P King, Shane W Krska, Tim Cernak, Stephen L Buchwald
Pharmaceutical diversification via palladium oxidative addition complexes. Science (New York, N.Y.) 363 (6425) (2019)
Corin C Wagen, Bryan T Ingoglia, Stephen L Buchwald
Unexpected Formation of Hexasubstituted Arenes through a 2-fold Palladium-Mediated Ligand Arylation. The Journal of organic chemistry 84 (19) (2019)
Chengxi Li, Richard Y Liu, Luke T Jesikiewicz, Yang Yang, Peng Liu, Stephen L Buchwald
CuH-Catalyzed Enantioselective Ketone Allylation with 1,3-Dienes: Scope, Mechanism, and Applications. Journal of the American Chemical Society 141 (12) (2019)
Saki Ichikawa, Stephen L Buchwald
Asymmetric Synthesis of γ-Amino Alcohols by Copper-Catalyzed Hydroamination. Organic letters 21 (21) (2019)
Liela Bayeh-Romero, Stephen L Buchwald
Copper Hydride Catalyzed Enantioselective Synthesis of Axially Chiral 1,3-Disubstituted Allenes. Journal of the American Chemical Society 141 (35) (2019)
Yuxuan Ye, Seoung-Tae Kim, Jinhoon Jeong, Mu-Hyun Baik, Stephen L Buchwald
CuH-Catalyzed Enantioselective Alkylation of Indole Derivatives with Ligand-Controlled Regiodivergence. Journal of the American Chemical Society 141 (9) (2019)
Richard Y Liu, Yujing Zhou, Yang Yang, Stephen L Buchwald
Enantioselective Allylation Using Allene, a Petroleum Cracking Byproduct. Journal of the American Chemical Society 141 (6) (2019)
Alexander W Schuppe, Gustavo M Borrajo-Calleja, Stephen L Buchwald
Enantioselective Olefin Hydrocyanation without Cyanide. Journal of the American Chemical Society 141 (47) (2019)
Chengxi Li, Kwangmin Shin, Richard Y Liu, Stephen L Buchwald
Engaging Aldehydes in CuH-Catalyzed Reductive Coupling Reactions: Stereoselective Allylation with Unactivated 1,3-Diene Pronucleophiles. Angewandte Chemie (International ed. in English) 58 (47) (2019)
Saki Ichikawa, Xi-Jie Dai, Stephen L Buchwald
Regio- and Enantioselective Synthesis of 1,2-Diamine Derivatives by Copper-Catalyzed Hydroamination. Organic letters 21 (11) (2019)
Xi-Jie Dai, Oliver D Engl, Thierry León, Stephen L Buchwald
Catalytic Asymmetric Synthesis of α-Arylpyrrolidines and Benzo-fused Nitrogen Heterocycles. Angewandte Chemie (International ed. in English) 58 (11) (2019)
Joseph M Dennis, Nicholas A White, Richard Y Liu, Stephen L Buchwald
Breaking the Base Barrier: An Electron-Deficient Palladium Catalyst Enables the Use of a Common Soluble Base in C-N Coupling. Journal of the American Chemical Society 140 (13) (2018)
Richard Y Liu, Minwoo Bae, Stephen L Buchwald
Mechanistic Insight Facilitates Discovery of a Mild and Efficient Copper-Catalyzed Dehydration of Primary Amides to Nitriles Using Hydrosilanes. Journal of the American Chemical Society 140 (5) (2018)
Yujing Zhou, Jeffrey S Bandar, Richard Y Liu, Stephen L Buchwald
CuH-Catalyzed Asymmetric Reduction of α,β-Unsaturated Carboxylic Acids to β-Chiral Aldehydes. Journal of the American Chemical Society 140 (2) (2018)
Andy A Thomas, Klaus Speck, Ilia Kevlishvili, Zhaohong Lu, Peng Liu, Stephen L Buchwald
Mechanistically Guided Design of Ligands That Significantly Improve the Efficiency of CuH-Catalyzed Hydroamination Reactions. Journal of the American Chemical Society 140 (42) (2018)
Saki Ichikawa, Shaolin Zhu, Stephen L Buchwald
A Modified System for the Synthesis of Enantioenriched N-Arylamines through Copper-Catalyzed Hydroamination. Angewandte Chemie (International ed. in English) 57 (28) (2018)
Hong Zhang, Paula Ruiz-Castillo, Stephen L Buchwald
Palladium-Catalyzed C-O Cross-Coupling of Primary Alcohols. Organic letters 20 (6) (2018)
Erica Y Tsai, Richard Y Liu, Yang Yang, Stephen L Buchwald
A Regio- and Enantioselective CuH-Catalyzed Ketone Allylation with Terminal Allenes. Journal of the American Chemical Society 140 (6) (2018)
Erica Y Tsai, Richard Y Liu, Yang Yang, Stephen L Buchwald
Correction to "A Regio- and Enantioselective CuH-Catalyzed Ketone Allylation with Terminal Allenes". Journal of the American Chemical Society 140 (19) (2018)
Yujing Zhou, Oliver D Engl, Jeffrey S Bandar, Emma D Chant, Stephen L Buchwald
CuH-Catalyzed Asymmetric Hydroamidation of Vinylarenes. Angewandte Chemie (International ed. in English) 57 (22) (2018)
R Kashif M Khan, Yang Zhao, Tal D Scully, Stephen L Buchwald
Catalytic Arylhydroxylation of Dehydroalanine in Continuous Flow for Simple Access to Unnatural Amino Acids. Chemistry (Weinheim an der Bergstrasse, Germany) 24 (57) (2018)
Michael W Gribble, Sheng Guo, Stephen L Buchwald
Asymmetric Cu-Catalyzed 1,4-Dearomatization of Pyridines and Pyridazines without Preactivation of the Heterocycle or Nucleophile. Journal of the American Chemical Society 140 (15) (2018)
Sheng Guo, Jeffrey C Yang, Stephen L Buchwald
A Practical Electrophilic Nitrogen Source for the Synthesis of Chiral Primary Amines by Copper-Catalyzed Hydroamination. Journal of the American Chemical Society 140 (46) (2018)
Koji Kubota, Peng Dai, Bradley L Pentelute, Stephen L Buchwald
Palladium Oxidative Addition Complexes for Peptide and Protein Cross-linking. Journal of the American Chemical Society 140 (8) (2018)
Anthony J Rojas, Chi Zhang, Ekaterina V Vinogradova, Nathan H Buchwald, John Reilly, Bradley L Pentelute, Stephen L Buchwald
Divergent unprotected peptide macrocyclisation by palladium-mediated cysteine arylation. Chemical science 8 (6) (2017)
Gang Lu, Richard Y Liu, Yang Yang, Cheng Fang, Daniel S Lambrecht, Stephen L Buchwald, Peng Liu
Ligand-Substrate Dispersion Facilitates the Copper-Catalyzed Hydroamination of Unactivated Olefins. Journal of the American Chemical Society 139 (46) (2017)
Stig D Friis, Michael T Pirnot, Lauren N Dupuis, Stephen L Buchwald
A Dual Palladium and Copper Hydride Catalyzed Approach for Alkyl-Aryl Cross-Coupling of Aryl Halides and Olefins. Angewandte Chemie (International ed. in English) 56 (25) (2017)