Bradley L Pentelute (B L Pentelute)

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 87

Top Topics

Mass Spectrometry

Duchenne Muscular Dystrophy

Top Venues

Journal of the American Chemical Society

ACS chemical biology

ACS central science

The journal of physical chemistry. B

This page only lists publications with an associated author ORCID identifier.

Publications

Peiyuan Zhang, Xiyun Ye, John C K Wang, Hannah T Baddock, Zena Jensvold, Ian T Foe, Andrei Loas, Dan L Eaton, Qi Hao, Aaron H Nile, Bradley L Pentelute
Reversibly Reactive Affinity Selection-Mass Spectrometry Enables Identification of Covalent Peptide Binders. Journal of the American Chemical Society 146 (22) (2024)
Jason Tao, Heemal H Dhanjee, Michael W Gribble, Veronika Kottisch, Jacob Rodriguez, Joseph S Brown, Holly Schmidt, Juhi Juneja, Fabienne Denhez, Peter S Lee, Daša Lipovšek, Stanley Krystek, Yihong Zhang, Patrick Bousquet, Yong Zhang, Bradley L Pentelute, Stephen L Buchwald
Site-Specific Antibody Prodrugs via S -Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues. Journal of the American Chemical Society (2024)
Kwo-Kwang Abraham Wang, Jupneet Singh, John S Albin, Bradley L Pentelute, Elizabeth M Nolan
Class IIb Microcin MccM Interferes with Oxidative Phosphorylation in Escherichia coli . ACS chemical biology (2024)
Peiyuan Zhang, Xiyun Ye, John C K Wang, Corey L Smith, Silvino Sousa, Andrei Loas, Dan L Eaton, Magdalena Preciado López, Bradley L Pentelute
Development of an α-Klotho Recognizing High-Affinity Peptide Probe from In-Solution Enrichment. JACS Au 4 (4) (2024)
Bin Liu, Jacob Rodriguez, Landon J Kilgallon, Wencong Wang, Yuyan Wang, Aiden Wang, Yutong Dai, Hung V-T Nguyen, Bradley L Pentelute, Jeremiah A Johnson
An organometallic swap strategy for bottlebrush polymer-protein conjugate synthesis. Chemical communications (Cambridge, England) 60 (31) (2024)
Ahmet Yesilcimen, Alex J Callahan, Tara L Travaline, Satish Gandhesiri, Olena S Tokareva, Andrei Loas, John H McGee, Bradley L Pentelute
Rapid Production of Native and Mirror-Image Tumor Necrosis Factor-α Enabled by Automated Flow Peptide Synthesis Technology. The Journal of organic chemistry (2024)
Peiyuan Zhang, Xiyun Ye, John C K Wang, Corey L Smith, Silvino Sousa, Andrei Loas, Dan L Eaton, Magdalena Preciado López, Bradley L Pentelute
Development of an α-Klotho Recognizing High-Affinity Peptide Probe from In-Solution Enrichment. JACS Au 4 (4) (2024)
Alex J Callahan, Satish Gandhesiri, Tara L Travaline, Rahi M Reja, Lia Lozano Salazar, Stephanie Hanna, Yen-Chun Lee, Kunhua Li, Olena S Tokareva, Jean-Marie Swiecicki, Andrei Loas, Gregory L Verdine, John H McGee, Bradley L Pentelute
Mirror-image ligand discovery enabled by single-shot fast-flow synthesis of D-proteins. Nature communications 15 (1) (2024)
Nicholas L Truex, Somesh Mohapatra, Mariane Melo, Jacob Rodriguez, Na Li, Wuhbet Abraham, Deborah Sementa, Faycal Touti, Derin B Keskin, Catherine J Wu, Darrell J Irvine, Rafael Gomez-Bombarelli, Bradley L Pentelute
Design of Cytotoxic T Cell Epitopes by Machine Learning of Human Degrons. ACS central science 10 (4) (2024)
Anna Charalampidou, Thomas Nehls, Christian Meyners, Satish Gandhesiri, Sebastian J Pomplun, Bradley L Pentelute, Frederik Lermyte, Felix Hausch
Automated Flow Peptide Synthesis Enables Engineering of Proteins with Stabilized Transient Binding Pockets. ACS central science 10 (3) (2024)
Nicholas L Truex, Somesh Mohapatra, Mariane Melo, Jacob Rodriguez, Na Li, Wuhbet Abraham, Deborah Sementa, Faycal Touti, Derin B Keskin, Catherine J Wu, Darrell J Irvine, Rafael Gomez-Bombarelli, Bradley L Pentelute
Design of Cytotoxic T Cell Epitopes by Machine Learning of Human Degrons. ACS central science 10 (4) (2024)
Alex J Callahan, Satish Gandhesiri, Tara L Travaline, Rahi M Reja, Lia Lozano Salazar, Stephanie Hanna, Yen-Chun Lee, Kunhua Li, Olena S Tokareva, Jean-Marie Swiecicki, Andrei Loas, Gregory L Verdine, John H McGee, Bradley L Pentelute
Mirror-image ligand discovery enabled by single-shot fast-flow synthesis of D-proteins. Nature communications 15 (1) (2024)
Jiayuan Miao, Arghya Pratim Ghosh, Minh Ngoc Ho, Chengxi Li, Xuejian Huang, Bradley L Pentelute, James D Baleja, Yu-Shan Lin
Assessing the Performance of Peptide Force Fields for Modeling the Solution Structural Ensembles of Cyclic Peptides. The journal of physical chemistry. B 128 (22) (2024)
Jiayuan Miao, Arghya Pratim Ghosh, Minh Ngoc Ho, Chengxi Li, Xuejian Huang, Bradley L Pentelute, James D Baleja, Yu-Shan Lin
Assessing the Performance of Peptide Force Fields for Modeling the Solution Structural Ensembles of Cyclic Peptides. The journal of physical chemistry. B 128 (22) (2024)
Nicholas L Truex, Somesh Mohapatra, Mariane Melo, Jacob Rodriguez, Na Li, Wuhbet Abraham, Deborah Sementa, Faycal Touti, Derin B Keskin, Catherine J Wu, Darrell J Irvine, Rafael Gomez-Bombarelli, Bradley L Pentelute
Design of Cytotoxic T Cell Epitopes by Machine Learning of Human Degrons. ACS central science 10 (4) (2024)
Xin Gu, Yu-An Zhang, Shuo Zhang, Leon Wang, Xiyun Ye, Gino Occhialini, Jonah Barbour, Bradley L Pentelute, Alison E Wendlandt
Synthesis of non-canonical amino acids through dehydrogenative tailoring. Nature (2024)
Peiyuan Zhang, Xiyun Ye, John C K Wang, Hannah T Baddock, Zena Jensvold, Ian T Foe, Andrei Loas, Dan L Eaton, Qi Hao, Aaron H Nile, Bradley L Pentelute
Reversibly Reactive Affinity Selection-Mass Spectrometry Enables Identification of Covalent Peptide Binders. Journal of the American Chemical Society (2024)
Jason Tao, Heemal H Dhanjee, Michael W Gribble, Veronika Kottisch, Jacob Rodriguez, Joseph S Brown, Holly Schmidt, Juhi Juneja, Fabienne Denhez, Peter S Lee, Daša Lipovšek, Stanley Krystek, Yihong Zhang, Patrick Bousquet, Yong Zhang, Bradley L Pentelute, Stephen L Buchwald
Site-Specific Antibody Prodrugs via S -Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues. Journal of the American Chemical Society 146 (29) (2024)
Alex J Callahan, Satish Gandhesiri, Tara L Travaline, Rahi M Reja, Lia Lozano Salazar, Stephanie Hanna, Yen-Chun Lee, Kunhua Li, Olena S Tokareva, Jean-Marie Swiecicki, Andrei Loas, Gregory L Verdine, John H McGee, Bradley L Pentelute
Mirror-image ligand discovery enabled by single-shot fast-flow synthesis of D-proteins. Nature communications 15 (1) (2024)
Bin Liu, Jacob Rodriguez, Landon J Kilgallon, Wencong Wang, Yuyan Wang, Aiden Wang, Yutong Dai, Hung V-T Nguyen, Bradley L Pentelute, Jeremiah A Johnson
An organometallic swap strategy for bottlebrush polymer-protein conjugate synthesis. Chemical communications (Cambridge, England) 60 (31) (2024)
Jiayuan Miao, Arghya Pratim Ghosh, Minh Ngoc Ho, Chengxi Li, Xuejian Huang, Bradley L Pentelute, James D Baleja, Yu-Shan Lin
Assessing the Performance of Peptide Force Fields for Modeling the Solution Structural Ensembles of Cyclic Peptides. The journal of physical chemistry. B 128 (22) (2024)
Nicholas L Truex, Somesh Mohapatra, Mariane Melo, Jacob Rodriguez, Na Li, Wuhbet Abraham, Deborah Sementa, Faycal Touti, Derin B Keskin, Catherine J Wu, Darrell J Irvine, Rafael Gomez-Bombarelli, Bradley L Pentelute
Design of Cytotoxic T Cell Epitopes by Machine Learning of Human Degrons. ACS central science 10 (4) (2024)
Bin Liu, Jacob Rodriguez, Landon J Kilgallon, Wencong Wang, Yuyan Wang, Aiden Wang, Yutong Dai, Hung V-T Nguyen, Bradley L Pentelute, Jeremiah A Johnson
An organometallic swap strategy for bottlebrush polymer-protein conjugate synthesis. Chemical communications (Cambridge, England) (2024)
Anna Charalampidou, Thomas Nehls, Christian Meyners, Satish Gandhesiri, Sebastian J Pomplun, Bradley L Pentelute, Frederik Lermyte, Felix Hausch
Automated Flow Peptide Synthesis Enables Engineering of Proteins with Stabilized Transient Binding Pockets. ACS central science 10 (3) (2024)
Jiayuan Miao, Arghya Pratim Ghosh, Minh Ngoc Ho, Chengxi Li, Xuejian Huang, Bradley L Pentelute, James D Baleja, Yu-Shan Lin
Assessing the Performance of Peptide Force Fields for Modeling the Solution Structural Ensembles of Cyclic Peptides. The journal of physical chemistry. B (2024)
Bin Liu, Jacob Rodriguez, Landon J Kilgallon, Wencong Wang, Yuyan Wang, Aiden Wang, Yutong Dai, Hung V-T Nguyen, Bradley L Pentelute, Jeremiah A Johnson
An organometallic swap strategy for bottlebrush polymer-protein conjugate synthesis. Chemical communications (Cambridge, England) 60 (31) (2024)
Jiayuan Miao, Arghya Pratim Ghosh, Minh Ngoc Ho, Chengxi Li, Xuejian Huang, Bradley L Pentelute, James D Baleja, Yu-Shan Lin
Assessing the Performance of Peptide Force Fields for Modeling the Solution Structural Ensembles of Cyclic Peptides. The journal of physical chemistry. B 128 (22) (2024)
Carly K Schissel, Charlotte E Farquhar, Andrei Loas, Annika B Malmberg, Bradley L Pentelute
In-Cell Penetration Selection-Mass Spectrometry Produces Noncanonical Peptides for Antisense Delivery. ACS chemical biology 18 (3) (2023)
Azin Saebi, Joseph S Brown, Victoria M Marando, Nina Hartrampf, Nicole M Chumbler, Stephanie Hanna, Mackenzie Poskus, Andrei Loas, Laura L Kiessling, Deborah T Hung, Bradley L Pentelute
Rapid Single-Shot Synthesis of the 214 Amino Acid-Long N-Terminal Domain of Pyocin S2. ACS chemical biology (2023)
Xiyun Ye, Peiyuan Zhang, Jason Tao, John C K Wang, Amirhossein Mafi, Nathalie M Grob, Anthony J Quartararo, Hannah T Baddock, Leanne J G Chan, Fiona E McAllister, Ian Foe, Andrei Loas, Dan L Eaton, Qi Hao, Aaron H Nile, Bradley L Pentelute
Discovery of reactive peptide inhibitors of human papillomavirus oncoprotein E6. Chemical science 14 (44) (2023)
Carly K Schissel, Charlotte E Farquhar, Andrei Loas, Annika B Malmberg, Bradley L Pentelute
In-Cell Penetration Selection-Mass Spectrometry Produces Noncanonical Peptides for Antisense Delivery. ACS chemical biology (2023)
Simon L Rössler, Nathalie M Grob, Stephen L Buchwald, Bradley L Pentelute
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis. Science (New York, N.Y.) 379 (6635) (2023)
Nathalie M Grob, Clint Remarcik, Simon L Rössler, Jeffrey Y K Wong, John C K Wang, Jason Tao, Corey L Smith, Andrei Loas, Stephen L Buchwald, Dan L Eaton, Magdalena Preciado López, Bradley L Pentelute
Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders. ACS chemical biology (2023)
Kohei Sato, Charlotte E Farquhar, Jacob Rodriguez, Bradley L Pentelute
Automated Fast-Flow Synthesis of Chromosome 9 Open Reading Frame 72 Dipeptide Repeat Proteins. Journal of the American Chemical Society (2023)
Simon L Rössler, Nathalie M Grob, Stephen L Buchwald, Bradley L Pentelute
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis. Science (New York, N.Y.) 379 (6635) (2023)
Nicholas L Truex, Aurélie Rondon, Simon L Rössler, Cameron C Hanna, Yehlin Cho, Bin-You Wang, Coralie M Backlund, Emi A Lutz, Darrell J Irvine, Bradley L Pentelute
Enhanced Vaccine Immunogenicity Enabled by Targeted Cytosolic Delivery of Tumor Antigens into Dendritic Cells. ACS central science 9 (9) (2023)
Azin Saebi, Joseph S Brown, Victoria M Marando, Nina Hartrampf, Nicole M Chumbler, Stephanie Hanna, Mackenzie Poskus, Andrei Loas, Laura L Kiessling, Deborah T Hung, Bradley L Pentelute
Rapid Single-Shot Synthesis of the 214 Amino Acid-Long N-Terminal Domain of Pyocin S2. ACS chemical biology 18 (3) (2023)
Carly K Schissel, Charlotte E Farquhar, Andrei Loas, Annika B Malmberg, Bradley L Pentelute
In-Cell Penetration Selection-Mass Spectrometry Produces Noncanonical Peptides for Antisense Delivery. ACS chemical biology 18 (3) (2023)
Simon L Rössler, Nathalie M Grob, Stephen L Buchwald, Bradley L Pentelute
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis. Science (New York, N.Y.) 379 (6635) (2023)
Azin Saebi, Joseph S Brown, Victoria M Marando, Nina Hartrampf, Nicole M Chumbler, Stephanie Hanna, Mackenzie Poskus, Andrei Loas, Laura L Kiessling, Deborah T Hung, Bradley L Pentelute
Rapid Single-Shot Synthesis of the 214 Amino Acid-Long N-Terminal Domain of Pyocin S2. ACS chemical biology 18 (3) (2023)
Xiyun Ye, Yen-Chun Lee, Zachary P Gates, Yingjie Ling, Jennifer C Mortensen, Fan-Shen Yang, Yu-Shan Lin, Bradley L Pentelute
Binary combinatorial scanning reveals potent poly-alanine-substituted inhibitors of protein-protein interactions. Communications chemistry 5 (1) (2022)
Martin Gazvoda, Heemal H Dhanjee, Jacob Rodriguez, Joseph S Brown, Charlotte E Farquhar, Nicholas L Truex, Andrei Loas, Stephen L Buchwald, Bradley L Pentelute
Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins. Journal of the American Chemical Society 144 (17) (2022)
Carly K Schissel, Charlotte E Farquhar, Annika B Malmberg, Andrei Loas, Bradley L Pentelute
Cell-Penetrating d-Peptides Retain Antisense Morpholino Oligomer Delivery Activity. ACS bio & med chem Au 2 (2) (2022)
Kyan A D'Angelo, Carly K Schissel, Bradley L Pentelute, Mohammad Movassaghi
Total synthesis of himastatin. Science (New York, N.Y.) 375 (6583) (2022)
Chengxi Li, Genwei Zhang, Somesh Mohapatra, Alex J Callahan, Andrei Loas, Rafael Gomez-Bombarelli, Bradley L Pentelute
Machine Learning Guides Peptide Nucleic Acid Flow Synthesis and Sequence Design. Advanced science (Weinheim, Baden-Wurttemberg, Germany) (2022)
Genwei Zhang, Joseph S Brown, Anthony J Quartararo, Chengxi Li, Xuyu Tan, Stephanie Hanna, Sarah Antilla, Amanda E Cowfer, Andrei Loas, Bradley L Pentelute
Rapid de novo discovery of peptidomimetic affinity reagents for human angiotensin converting enzyme 2. Communications chemistry 5 (1) (2022)
Xiyun Ye, Yen-Chun Lee, Zachary P Gates, Yingjie Ling, Jennifer C Mortensen, Fan-Shen Yang, Yu-Shan Lin, Bradley L Pentelute
Binary combinatorial scanning reveals potent poly-alanine-substituted inhibitors of protein-protein interactions. Communications chemistry 5 (1) (2022)
Genwei Zhang, Joseph S Brown, Anthony J Quartararo, Chengxi Li, Xuyu Tan, Stephanie Hanna, Sarah Antilla, Amanda E Cowfer, Andrei Loas, Bradley L Pentelute
Rapid de novo discovery of peptidomimetic affinity reagents for human angiotensin converting enzyme 2. Communications chemistry 5 (1) (2022)
Anthony J Rojas, Justin M Wolfe, Heemal H Dhanjee, Ivan Buslov, Nicholas L Truex, Richard Y Liu, Walter Massefski, Bradley L Pentelute, Stephen L Buchwald
Palladium-peptide oxidative addition complexes for bioconjugation. Chemical science 13 (40) (2022)
Carly K Schissel, Charlotte E Farquhar, Annika B Malmberg, Andrei Loas, Bradley L Pentelute
Cell-Penetrating d-Peptides Retain Antisense Morpholino Oligomer Delivery Activity. ACS bio & med chem Au 2 (2) (2022)
Martin Gazvoda, Heemal H Dhanjee, Jacob Rodriguez, Joseph S Brown, Charlotte E Farquhar, Nicholas L Truex, Andrei Loas, Stephen L Buchwald, Bradley L Pentelute
Correction to "Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins". Journal of the American Chemical Society 144 (22) (2022)
Chengxi Li, Alex J Callahan, Mark D Simon, Kyle A Totaro, Alexander J Mijalis, Kruttika-Suhas Phadke, Genwei Zhang, Nina Hartrampf, Carly K Schissel, Ming Zhou, Hong Zong, Gunnar J Hanson, Andrei Loas, Nicola L B Pohl, David E Verhoeven, Bradley L Pentelute
Fully automated fast-flow synthesis of antisense phosphorodiamidate morpholino oligomers. Nature communications 12 (1) (2021)
Muhammad Jbara, Jacob Rodriguez, Heemal H Dhanjee, Andrei Loas, Stephen L Buchwald, Bradley L Pentelute
Oligonucleotide Bioconjugation with Bifunctional Palladium Reagents. Angewandte Chemie (International ed. in English) 60 (21) (2021)
Sebastian Pomplun, Muhammad Jbara, Carly K Schissel, Susana Wilson Hawken, Ann Boija, Charles Li, Isaac Klein, Bradley L Pentelute
Parallel Automated Flow Synthesis of Covalent Protein Complexes That Can Inhibit MYC-Driven Transcription. ACS central science 7 (8) (2021)
Zhuting Hu, Donna E Leet, Rosa L Allesøe, Giacomo Oliveira, Shuqiang Li, Adrienne M Luoma, Jinyan Liu, Juliet Forman, Teddy Huang, J Bryan Iorgulescu, Rebecca Holden, Siranush Sarkizova, Satyen H Gohil, Robert A Redd, Jing Sun, Liudmila Elagina, Anita Giobbie-Hurder, Wandi Zhang, Lauren Peter, Zoe Ciantra, Scott Rodig, Oriol Olive, Keerthi Shetty, Jason Pyrdol, Mohamed Uduman, Patrick C Lee, Pavan Bachireddy, Elizabeth I Buchbinder, Charles H Yoon, Donna Neuberg, Bradley L Pentelute, Nir Hacohen, Kenneth J Livak, Sachet A Shukla, Lars Rønn Olsen, Dan H Barouch, Kai W Wucherpfennig, Edward F Fritsch, Derin B Keskin, Catherine J Wu, Patrick A Ott
Personal neoantigen vaccines induce persistent memory T cell responses and epitope spreading in patients with melanoma. Nature medicine 27 (3) (2021)
Carly K Schissel, Somesh Mohapatra, Justin M Wolfe, Colin M Fadzen, Kamela Bellovoda, Chia-Ling Wu, Jenna A Wood, Annika B Malmberg, Andrei Loas, Rafael Gomez-Bombarelli, Bradley L Pentelute
Deep learning to design nuclear-targeting abiotic miniproteins. Nature chemistry 13 (10) (2021)
Genwei Zhang, Chengxi Li, Anthony J Quartararo, Andrei Loas, Bradley L Pentelute
Automated affinity selection for rapid discovery of peptide binders. Chemical science 12 (32) (2021)
Muhammad Jbara, Sebastian Pomplun, Carly K Schissel, Susana Wilson Hawken, Ann Boija, Isaac Klein, Jacob Rodriguez, Stephen L Buchwald, Bradley L Pentelute
Engineering Bioactive Dimeric Transcription Factor Analogs via Palladium Rebound Reagents. Journal of the American Chemical Society 143 (30) (2021)
Chengxi Li, Alex J Callahan, Kruttika S Phadke, Bryan H Bellaire, Charlotte E Farquhar, Genwei Zhang, Carly K Schissel, Alexander J Mijalis, Nina Hartrampf, Andrei Loas, David E Verhoeven, Bradley L Pentelute
Automated Flow Synthesis of Peptide-PNA Conjugates. ACS central science 8 (2) (2021)
Nicole J Yang, Joerg Isensee, Dylan V Neel, Andreza U Quadros, Han-Xiong Bear Zhang, Justas Lauzadis, Sai Man Liu, Stephanie Shiers, Andreea Belu, Shilpa Palan, Sandra Marlin, Jacquie Maignel, Angela Kennedy-Curran, Victoria S Tong, Mahtab Moayeri, Pascal Röderer, Anja Nitzsche, Mike Lu, Bradley L Pentelute, Oliver Brüstle, Vineeta Tripathi, Keith A Foster, Theodore John Price, R John Collier, Stephen H Leppla, Michelino Puopolo, Bruce P Bean, Thiago M Cunha, Tim Hucho, Isaac M Chiu
Anthrax toxins regulate pain signaling and can deliver molecular cargoes into ANTXR2 + DRG sensory neurons. Nature neuroscience 25 (2) (2021)
Eva M López-Vidal, Carly K Schissel, Somesh Mohapatra, Kamela Bellovoda, Chia-Ling Wu, Jenna A Wood, Annika B Malmberg, Andrei Loas, Rafael Gomez-Bombarelli, Bradley L Pentelute
Deep Learning Enables Discovery of a Short Nuclear Targeting Peptide for Efficient Delivery of Antisense Oligomers. JACS Au 1 (11) (2021)
Zeyu Lu, Brenton R Paolella, Nicholas L Truex, Alexander R Loftis, Xiaoli Liao, Amy E Rabideau, Meredith S Brown, John Busanovich, Rameen Beroukhim, Bradley L Pentelute
Targeting Cancer Gene Dependencies with Anthrax-Mediated Delivery of Peptide Nucleic Acids. ACS chemical biology 15 (6) (2020)
Alexander R Loftis, Michael S Santos, Nicholas L Truex, Marco Biancucci, Karla J F Satchell, Bradley L Pentelute
Anthrax Protective Antigen Retargeted with Single-Chain Variable Fragments Delivers Enzymes to Pancreatic Cancer Cells. Chembiochem : a European journal of chemical biology 21 (19) (2020)
Heemal H Dhanjee, Azin Saebi, Ivan Buslov, Alexander R Loftis, Stephen L Buchwald, Bradley L Pentelute
Correction to "Protein-Protein Cross-Coupling via Palladium-Protein Oxidative Addition Complexes from Cysteine Residues". Journal of the American Chemical Society 142 (28) (2020)
Chelsea K Longwell, Stephanie Hanna, Nina Hartrampf, R Andres Parra Sperberg, Po-Ssu Huang, Bradley L Pentelute, Jennifer R Cochran
Identification of N-Terminally Diversified GLP-1R Agonists Using Saturation Mutagenesis and Chemical Design. ACS chemical biology 16 (1) (2020)
Colin M Fadzen, Justin M Wolfe, Wen Zhou, Choi-Fong Cho, Niklas von Spreckelsen, Kathryn T Hutchinson, Yen-Chun Lee, E Antonio Chiocca, Sean E Lawler, Omer H Yilmaz, Stephen J Lippard, Bradley L Pentelute
A Platinum(IV) Prodrug-Perfluoroaryl Macrocyclic Peptide Conjugate Enhances Platinum Uptake in the Brain. Journal of medicinal chemistry 63 (13) (2020)
Anthony J Quartararo, Zachary P Gates, Bente A Somsen, Nina Hartrampf, Xiyun Ye, Arisa Shimada, Yasuhiro Kajihara, Christian Ottmann, Bradley L Pentelute
Ultra-large chemical libraries for the discovery of high-affinity peptide binders. Nature communications 11 (1) (2020)
Heemal H Dhanjee, Azin Saebi, Ivan Buslov, Alexander R Loftis, Stephen L Buchwald, Bradley L Pentelute
Protein-Protein Cross-Coupling via Palladium-Protein Oxidative Addition Complexes from Cysteine Residues. Journal of the American Chemical Society 142 (20) (2020)
Sebastian J Pomplun, Christopher R Shugrue, Adeline Marie Schmitt, Carly K Schissel, Charlotte E Farquhar, Bradley L Pentelute
Secondary Amino Alcohols: Traceless Cleavable Linkers for Use in Affinity Capture and Release. Angewandte Chemie (International ed. in English) 59 (28) (2020)
Sebastian Pomplun, Zachary P Gates, Genwei Zhang, Anthony J Quartararo, Bradley L Pentelute
Discovery of Nucleic Acid Binding Molecules from Combinatorial Biohybrid Nucleobase Peptide Libraries. Journal of the American Chemical Society 142 (46) (2020)
William R Lindemann, Alexander J Mijalis, José L Alonso, Peter P Borbat, Jack H Freed, M Amin Arnaout, Bradley L Pentelute, Julia H Ortony
Conformational Dynamics in Extended RGD-Containing Peptides. Biomacromolecules 21 (7) (2020)
Heemal H Dhanjee, Ivan Buslov, Ian W Windsor, Ronald T Raines, Bradley L Pentelute, Stephen L Buchwald
Palladium-Protein Oxidative Addition Complexes by Amine-Selective Acylation. Journal of the American Chemical Society 142 (51) (2020)
Nina Hartrampf, Azin Saebi, M Poskus, Z P Gates, Alex J Callahan, A E Cowfer, S Hanna, Sarah Antilla, Carly K Schissel, Anthony J Quartararo, X Ye, A J Mijalis, M D Simon, Andrei Loas, S Liu, Carsten Jessen, T E Nielsen, Bradley L Pentelute
Synthesis of proteins by automated flow chemistry. Science (New York, N.Y.) 368 (6494) (2020)
Andrei Loas, Bradley L Pentelute
Introduction: Peptide Chemistry. Chemical reviews 120 (6) (2020)
Colin M Fadzen, Rebecca L Holden, Justin M Wolfe, Zi-Ning Choo, Carly K Schissel, Monica Yao, Gunnar J Hanson, Bradley L Pentelute
Chimeras of Cell-Penetrating Peptides Demonstrate Synergistic Improvement in Antisense Efficacy. Biochemistry 58 (38) (2019)
Ethan D Evans, Zachary P Gates, Zhen-Yu J Sun, Alexander J Mijalis, Bradley L Pentelute
Conformational Stabilization and Rapid Labeling of a 29-Residue Peptide by a Small Molecule Reaction Partner. Biochemistry 58 (10) (2019)
Chi Zhang, Ekaterina V Vinogradova, Alexander M Spokoyny, Stephen L Buchwald, Bradley L Pentelute
Arylation Chemistry for Bioconjugation. Angewandte Chemie (International ed. in English) 58 (15) (2019)
Diana P Slough, Sean M McHugh, Ashleigh E Cummings, Peng Dai, Bradley L Pentelute, Joshua A Kritzer, Yu-Shan Lin
Designing Well-Structured Cyclic Pentapeptides Based on Sequence-Structure Relationships. The journal of physical chemistry. B 122 (14) (2018)
Fayçal Touti, Guillaume Lautrette, Kenneth D Johnson, James C Delaney, Andrew Wollacott, Hamid Tissire, Karthik Viswanathan, Zachary Shriver, Surin K Mong, Alexander J Mijalis, Obadiah J Plante, Bradley L Pentelute
Antibody-Bactericidal Macrocyclic Peptide Conjugates To Target Gram-Negative Bacteria. Chembiochem : a European journal of chemical biology 19 (19) (2018)
Chi Zhang, Peng Dai, Alexander A Vinogradov, Zachary P Gates, Bradley L Pentelute
Site-Selective Cysteine-Cyclooctyne Conjugation. Angewandte Chemie (International ed. in English) 57 (22) (2018)
Justin M Wolfe, Colin M Fadzen, Rebecca L Holden, Monica Yao, Gunnar J Hanson, Bradley L Pentelute
Perfluoroaryl Bicyclic Cell-Penetrating Peptides for Delivery of Antisense Oligonucleotides. Angewandte Chemie (International ed. in English) 57 (17) (2018)
Stella Hartmann, Renae Lopez Cruz, Saleem Alameh, Chi-Lee C Ho, Amy Rabideau, Bradley L Pentelute, Kenneth A Bradley, Mikhail Martchenko Shilman
Characterization of Novel Piperidine-Based Inhibitor of Cathepsin B-Dependent Bacterial Toxins and Viruses. ACS infectious diseases 4 (8) (2018)
Ethan D Evans, Bradley L Pentelute
Discovery of a 29-Amino-Acid Reactive Abiotic Peptide for Selective Cysteine Arylation. ACS chemical biology 13 (3) (2018)
Koji Kubota, Peng Dai, Bradley L Pentelute, Stephen L Buchwald
Palladium Oxidative Addition Complexes for Peptide and Protein Cross-linking. Journal of the American Chemical Society 140 (8) (2018)
Anthony J Rojas, Chi Zhang, Ekaterina V Vinogradova, Nathan H Buchwald, John Reilly, Bradley L Pentelute, Stephen L Buchwald
Divergent unprotected peptide macrocyclisation by palladium-mediated cysteine arylation. Chemical science 8 (6) (2017)
Colin M Fadzen, Justin M Wolfe, Choi-Fong Cho, E Antonio Chiocca, Sean E Lawler, Bradley L Pentelute
Perfluoroarene-Based Peptide Macrocycles to Enhance Penetration Across the Blood-Brain Barrier. Journal of the American Chemical Society 139 (44) (2017)
Surin K Mong, Frank V Cochran, Hongtao Yu, Zachary Graziano, Yu-Shan Lin, Jennifer R Cochran, Bradley L Pentelute
Heterochiral Knottin Protein: Folding and Solution Structure. Biochemistry 56 (43) (2017)