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Suresh V Ambudkar

ORCID

Publication Activity (10 Years)

Years Active: 2017-2023
Publications (10 Years): 35

Top Venues

Pharmaceutics

International journal of molecular sciences

Biomolecules

Cancers

Johns Hopkins School of Medicine

Madurai Kamaraj University School of Biological Sciences (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Johns Hopkins School of Medicine Apr 1o 1989 - May 31o 1995

United States

Assistant Professor :: Medicine

Education History

Madurai Kamaraj University School of Biological Sciences Jul 26o 1974 - Mar 4o 1978

India

PHD :: Biochemistry

Publications

Glaucio Valdameri, Diogo Henrique Kita, Julia de Paula Dutra, Diego Lima Gomes, Arun Kumar Tonduru, Thales Kronenberger, Bruno Gavinho, Izadora Volpato Rossi, Mariana Mazetto de Carvalho, Basile Pérès, Ingrid Fatima Zattoni, Fabiane Gomes de Moraes Rego, Geraldo Picheth, Rilton Alves de Freitas, Antti Poso, Suresh V Ambudkar, Marcel I Ramirez, Ahcène Boumendjel, Vivian Rotuno Moure
Characterization of Potent ABCG2 Inhibitor Derived from Chromone: From the Mechanism of Inhibition to Human Extracellular Vesicles for Drug Delivery. Pharmaceutics 15 (4) (2023)
Chao-Yun Cai, Qiu-Xu Teng, Megumi Murakami, Suresh V Ambudkar, Zhe-Sheng Chen, Vijaya L Korlipara
Design, Synthesis and Biological Evaluation of Quinazolinamine Derivatives as Breast Cancer Resistance Protein and P-Glycoprotein Inhibitors with Improved Metabolic Stability. Biomolecules 13 (2) (2023)
Chung-Pu Wu, Cheng-Yu Hung, Ya-Ju Hsieh, Megumi Murakami, Yang-Hui Huang, Tsung-Yao Su, Tai-Ho Hung, Jau-Song Yu, Yu-Shan Wu, Suresh V Ambudkar
ABCB1 and ABCG2 Overexpression Mediates Resistance to the Phosphatidylinositol 3-Kinase Inhibitor HS-173 in Cancer Cell Lines. Cells 12 (7) (2023)
Chung-Pu Wu, Yen-Ching Li, Megumi Murakami, Sung-Han Hsiao, Yun-Chieh Lee, Yang-Hui Huang, Yu-Tzu Chang, Tai-Ho Hung, Yu-Shan Wu, Suresh V Ambudkar
Furmonertinib, a Third-Generation EGFR Tyrosine Kinase Inhibitor, Overcomes Multidrug Resistance through Inhibiting ABCB1 and ABCG2 in Cancer Cells. International journal of molecular sciences 24 (18) (2023)
Dong-Mei Zhang, Chang Shu, Jun-Jiang Chen, Kamlesh Sodani, Jiao Wang, Jaya Bhatnagar, Ping Lan, Zhi-Xiong Ruan, Zhi-Jie Xiao, Suresh V Ambudkar, Wei-Min Chen, Zhe-Sheng Chen, Wen-Cai Ye
Correction to "BBA, a Derivative of 23-Hydroxybetulinic Acid, Potently Reverses ABCB1-Mediated Drug Resistance in Vitro and in Vivo ". Molecular pharmaceutics (2023)
Glaucio Valdameri, Diogo Henrique Kita, Julia de Paula Dutra, Diego Lima Gomes, Arun Kumar Tonduru, Thales Kronenberger, Bruno Gavinho, Izadora Volpato Rossi, Mariana Mazetto de Carvalho, Basile Pérès, Ingrid Fatima Zattoni, Fabiane Gomes de Moraes Rego, Geraldo Picheth, Rilton Alves de Freitas, Antti Poso, Suresh V Ambudkar, Marcel I Ramirez, Ahcène Boumendjel, Vivian Rotuno Moure
Characterization of Potent ABCG2 Inhibitor Derived from Chromone: From the Mechanism of Inhibition to Human Extracellular Vesicles for Drug Delivery. Pharmaceutics 15 (4) (2023)
Chao-Yun Cai, Qiu-Xu Teng, Megumi Murakami, Suresh V Ambudkar, Zhe-Sheng Chen, Vijaya L Korlipara
Design, Synthesis and Biological Evaluation of Quinazolinamine Derivatives as Breast Cancer Resistance Protein and P-Glycoprotein Inhibitors with Improved Metabolic Stability. Biomolecules 13 (2) (2023)
Glaucio Valdameri, Diogo Henrique Kita, Julia de Paula Dutra, Diego Lima Gomes, Arun Kumar Tonduru, Thales Kronenberger, Bruno Gavinho, Izadora Volpato Rossi, Mariana Mazetto de Carvalho, Basile Pérès, Ingrid Fatima Zattoni, Fabiane Gomes de Moraes Rego, Geraldo Picheth, Rilton Alves de Freitas, Antti Poso, Suresh V Ambudkar, Marcel I Ramirez, Ahcène Boumendjel, Vivian Rotuno Moure
Characterization of Potent ABCG2 Inhibitor Derived from Chromone: From the Mechanism of Inhibition to Human Extracellular Vesicles for Drug Delivery. Pharmaceutics 15 (4) (2023)
Chao-Yun Cai, Qiu-Xu Teng, Megumi Murakami, Suresh V Ambudkar, Zhe-Sheng Chen, Vijaya L Korlipara
Design, Synthesis and Biological Evaluation of Quinazolinamine Derivatives as Breast Cancer Resistance Protein and P-Glycoprotein Inhibitors with Improved Metabolic Stability. Biomolecules 13 (2) (2023)
Andaleeb Sajid, Hadiar Rahman, Suresh V Ambudkar
Advances in the structure, mechanism and targeting of chemoresistance-linked ABC transporters. Nature reviews. Cancer (2023)
Maria João Moreno, Hugo A L Filipe, Susana V P Cunha, Cristiana V Ramos, Patrícia A T Martins, Biebele Abel, Luís M S Loura, Suresh V Ambudkar
Interaction of a Homologous Series of Amphiphiles with P-glycoprotein in a Membrane Environment-Contributions of Polar and Non-Polar Interactions. Pharmaceutics 15 (1) (2023)
Chung-Pu Wu, Megumi Murakami, Yen-Ching Li, Yang-Hui Huang, Yu-Tzu Chang, Tai-Ho Hung, Yu-Shan Wu, Suresh V Ambudkar
Imperatorin Restores Chemosensitivity of Multidrug-Resistant Cancer Cells by Antagonizing ABCG2-Mediated Drug Transport. Pharmaceuticals (Basel, Switzerland) 16 (11) (2023)
Chao-Yun Cai, Qiu-Xu Teng, Megumi Murakami, Suresh V Ambudkar, Zhe-Sheng Chen, Vijaya L Korlipara
Design, Synthesis and Biological Evaluation of Quinazolinamine Derivatives as Breast Cancer Resistance Protein and P-Glycoprotein Inhibitors with Improved Metabolic Stability. Biomolecules 13 (2) (2023)
Hadiar Rahman, Mark J Ware, Andaleeb Sajid, Sabrina Lusvarghi, Stewart R Durell, Suresh V Ambudkar
Residues from Homologous Transmembrane Helices 4 and 10 Are Critical for P-Glycoprotein (ABCB1)-Mediated Drug Transport. Cancers 15 (13) (2023)
Glaucio Valdameri, Diogo Henrique Kita, Julia de Paula Dutra, Diego Lima Gomes, Arun Kumar Tonduru, Thales Kronenberger, Bruno Gavinho, Izadora Volpato Rossi, Mariana Mazetto de Carvalho, Basile Pérès, Ingrid Fatima Zattoni, Fabiane Gomes de Moraes Rego, Geraldo Picheth, Rilton Alves de Freitas, Antti Poso, Suresh V Ambudkar, Marcel I Ramirez, Ahcène Boumendjel, Vivian Rotuno Moure
Characterization of Potent ABCG2 Inhibitor Derived from Chromone: From the Mechanism of Inhibition to Human Extracellular Vesicles for Drug Delivery. Pharmaceutics 15 (4) (2023)
Maria João Moreno, Hugo A L Filipe, Susana V P Cunha, Cristiana V Ramos, Patrícia A T Martins, Biebele Abel, Luís M S Loura, Suresh V Ambudkar
Interaction of a Homologous Series of Amphiphiles with P-glycoprotein in a Membrane Environment-Contributions of Polar and Non-Polar Interactions. Pharmaceutics 15 (1) (2023)
Maria João Moreno, Hugo A L Filipe, Susana V P Cunha, Cristiana V Ramos, Patrícia A T Martins, Biebele Abel, Luís M S Loura, Suresh V Ambudkar
Interaction of a Homologous Series of Amphiphiles with P-glycoprotein in a Membrane Environment-Contributions of Polar and Non-Polar Interactions. Pharmaceutics 15 (1) (2023)
Yan-Qing Li, Megumi Murakami, Yang-Hui Huang, Tai-Ho Hung, Shun-Ping Wang, Yu-Shan Wu, Suresh V Ambudkar, Chung-Pu Wu
Hydroxygenkwanin Improves the Efficacy of Cytotoxic Drugs in ABCG2-Overexpressing Multidrug-Resistant Cancer Cells. International journal of molecular sciences 23 (21) (2022)
Chung-Pu Wu, Cheng-Yu Hung, Megumi Murakami, Yu-Shan Wu, Chun-Ling Lin, Yang-Hui Huang, Tai-Ho Hung, Jau-Song Yu, Suresh V Ambudkar
P-glycoprotein Mediates Resistance to the Anaplastic Lymphoma Kinase Inhiitor Ensartinib in Cancer Cells. Cancers 14 (9) (2022)
Priya Yadav, Suresh V Ambudkar, Nagarajan Rajendra Prasad
Emerging nanotechnology-based therapeutics to combat multidrug-resistant cancer. Journal of nanobiotechnology 20 (1) (2022)
Shoji Kokubo, Shinobu Ohnuma, Megumi Murakami, Haruhisa Kikuchi, Shota Funayama, Hideyuki Suzuki, Taiki Kajiwara, Akihiro Yamamura, Hideaki Karasawa, Norihiko Sugisawa, Kosuke Ohsawa, Kuniyuki Kano, Junken Aoki, Takayuki Doi, Takeshi Naitoh, Suresh V Ambudkar, Michiaki Unno
A Phenylfurocoumarin Derivative Reverses ABCG2-Mediated Multidrug Resistance In Vitro and In Vivo. International journal of molecular sciences 22 (22) (2021)
Chung-Pu Wu, Cheng-Yu Hung, Sabrina Lusvarghi, Yen-Fu Chang, Sung-Han Hsiao, Yang-Hui Huang, Tai-Ho Hung, Jau-Song Yu, Suresh V Ambudkar
Overexpression of Human ABCB1 and ABCG2 Reduces the Susceptibility of Cancer Cells to the Histone Deacetylase 6-Specific Inhibitor Citarinostat. International journal of molecular sciences 22 (5) (2021)
Sabrina Lusvarghi, Stewart R Durell, Suresh V Ambudkar
Does the ATP-bound EQ mutant reflect the pre- or post-ATP hydrolysis state in the catalytic cycle of human P-glycoprotein (ABCB1)? FEBS letters 595 (6) (2021)
Diogo Henrique Kita, Nathalie Guragossian, Ingrid Fatima Zattoni, Vivian Rotuno Moure, Fabiane Gomes de Moraes Rego, Sabrina Lusvarghi, Thomas Moulenat, Billel Belhani, Fabiane Gomes de Moraes Rego, Sofiane Bouacida, Zouhair Bouaziz, Christelle Marminon, Malika Berredjem, Joachim Jose, Marcos Brown Gonçalves, Suresh V Ambudkar, Glaucio Valdameri, Marc Le Borgne
Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles. Scientific reports 11 (1) (2021)
Diogo Henrique Kita, Gisele Alves de Andrade, Juliana Morais Missina, Kahoana Postal, Viktor Kalbermatter Boell, Francielli Sousa Santana, Ingrid Fatima Zattoni, Isadora da Silva Zanzarini, Vivian Rotuno Moure, Fabiane Gomes de Moraes Rego, Geraldo Picheth, Emanuel Maltempi de Souza, David A Mitchell, Suresh V Ambudkar, Giovana Gioppo Nunes, Glaucio Valdameri
Polyoxovanadates as new P-glycoprotein inhibitors: insights into the mechanism of inhibition. FEBS letters 596 (3) (2021)
Barry J Liang, Sabrina Lusvarghi, Suresh V Ambudkar, Huang-Chiao Huang
Use of photoimmunoconjugates to characterize ABCB1 in cancer cells. Nanophotonics 10 (12) (2021)
Sabrina Lusvarghi, Robert W Robey, Michael M Gottesman, Suresh V Ambudkar
Multidrug transporters: recent insights from cryo-electron microscopy-derived atomic structures and animal models. F1000Research 9 (2020)
Andaleeb Sajid, Sabrina Lusvarghi, Megumi Murakami, Eduardo E Chufan, Biebele Abel, Michael M Gottesman, Stewart R Durell, Suresh V Ambudkar
Reversing the direction of drug transport mediated by the human multidrug transporter P-glycoprotein. Proceedings of the National Academy of Sciences of the United States of America 117 (47) (2020)
Hadiar Rahman, Andrew Rudrow, Joshua Carneglia, Sister Stephen Patrick Joly, Dante Nicotera, Michael Naldrett, John Choy, Suresh V Ambudkar, John Golin
Nonsynonymous Mutations in Linker-2 of the Pdr5 Multidrug Transporter Identify a New RNA Stability Element. G3 (Bethesda, Md.) 10 (1) (2020)
Zhuo-Xun Wu, Yuqi Yang, Qiu-Xu Teng, Jing-Quan Wang, Zi-Ning Lei, Jing-Qiu Wang, Sabrina Lusvarghi, Suresh V Ambudkar, Dong-Hua Yang, Zhe-Sheng Chen
Tivantinib, A c-Met Inhibitor in Clinical Trials, Is Susceptible to ABCG2-Mediated Drug Resistance. Cancers 12 (1) (2020)
Georgina P Sava, Hailing Fan, Rosemary A Fisher, Sabrina Lusvarghi, Sunil Pancholi, Suresh V Ambudkar, Lesley-Ann Martin, R Charles Coombes, Lakjaya Buluwela, Simak Ali
ABC-transporter upregulation mediates resistance to the CDK7 inhibitors THZ1 and ICEC0942. Oncogene 39 (3) (2019)
Shahrooz Vahedi, Sabrina Lusvarghi, Kristen Pluchino, Yinon Shafrir, Stewart R Durell, Michael M Gottesman, Suresh V Ambudkar
Mapping discontinuous epitopes for MRK-16, UIC2 and 4E3 antibodies to extracellular loops 1 and 4 of human P-glycoprotein. Scientific reports 8 (1) (2018)
Andaleeb Sajid, Sabrina Lusvarghi, Eduardo E Chufan, Suresh V Ambudkar
Evidence for the critical role of transmembrane helices 1 and 7 in substrate transport by human P-glycoprotein (ABCB1). PloS one 13 (9) (2018)
Bhargav A Patel, Biebele Abel, Anna Maria Barbuti, Uday Kiran Velagapudi, Zhe-Sheng Chen, Suresh V Ambudkar, Tanaji T Talele
Comprehensive Synthesis of Amino Acid-Derived Thiazole Peptidomimetic Analogues to Understand the Enigmatic Drug/Substrate-Binding Site of P-Glycoprotein. Journal of medicinal chemistry 61 (3) (2018)
Megumi Murakami, Shinobu Ohnuma, Michihiro Fukuda, Eduardo E Chufan, Katsuyoshi Kudoh, Keigo Kanehara, Norihiko Sugisawa, Masaharu Ishida, Takeshi Naitoh, Hiroyuki Shibata, Yoshiharu Iwabuchi, Suresh V Ambudkar, Michiaki Unno
Synthetic Analogs of Curcumin Modulate the Function of Multidrug Resistance-Linked ATP-Binding Cassette Transporter ABCG2. Drug metabolism and disposition: the biological fate of chemicals 45 (11) (2017)

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Publication Activity (10 Years)

Top Topics

Top Venues

Suresh V Ambudkar