Zlatko Janeba

Loop profile ORCID

Publication Activity (10 Years)

Years Active: 2016-2024
Publications (10 Years): 28

Top Venues

Journal of medicinal chemistry

ChemMedChem

Antiviral chemistry & chemotherapy

The Journal of organic chemistry

Institute of Organic Chemistry and Biochemistry AS CR

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Institute of Organic Chemistry and Biochemistry AS CR Jan 01 2016

Czechia

Senior Group Leader :: Bioorganic & Medicinal Chemistry

Institute of Organic Chemistry and Biochemistry AS CR, v.v.i. Jan 01 2010 - Dec 31 2015

Czechia

Junior group leader :: Bioorganic & medicinal chemistry

Publications

Artem Chayka, Michal Česnek, Erika Kužmová, Jaroslav Kozák, Eva Tloušt'ová, Alexandra Dvořáková, Timotej Strmeň, Břetislav Brož, Zuzana Osifová, Martin Dračínský, Helena Mertlíková-Kaiserová, Zlatko Janeba
Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine. Journal of medicinal chemistry 67 (12) (2024)
Artem Chayka, Michal Česnek, Erika Kužmová, Jaroslav Kozák, Eva Tloušt'ová, Alexandra Dvořáková, Timotej Strmeň, Břetislav Brož, Zuzana Osifová, Martin Dračínský, Helena Mertlíková-Kaiserová, Zlatko Janeba
Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine. Journal of medicinal chemistry 67 (12) (2024)
Jitendra Kumar Meena, Jarey H Wang, Nicholas J Neill, Dianne Keough, Nagireddy Putluri, Panagiostis Katsonis, Amanda M Koire, Hyemin Lee, Elizabeth A Bowling, Siddhartha Tyagi, Mayra Orellana, Rocio Dominguez-Vidana, Heyuan Li, Kenneth Eagle, Charles H Danan, Hsiang-Ching Chung, Andrew D Yang, William Wu, Sarah J Kurley, Brian M Ho, Joseph R Zoeller, Calla M Olson, Kristen L Meerbrey, Olivier Lichtarge, Arun Sreekumar, Clifford C Dacso, Luke W Guddat, Dominik Rejman, Dana Hocková, Zlatko Janeba, Lukas M Simon, Charles Y Lin, Monica C Pillon, Thomas F Westbrook
MYC Induces Oncogenic Stress through RNA Decay and Ribonucleotide Catabolism in Breast Cancer. Cancer discovery (2024)
Artem Chayka, Michal Česnek, Erika Kužmová, Jaroslav Kozák, Eva Tloušt'ová, Alexandra Dvořáková, Timotej Strmeň, Břetislav Brož, Zuzana Osifová, Martin Dračínský, Helena Mertlíková-Kaiserová, Zlatko Janeba
Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine. Journal of medicinal chemistry 67 (12) (2024)
Artem Chayka, Michal Česnek, Erika Kužmová, Jaroslav Kozák, Eva Tloušt'ová, Alexandra Dvořáková, Timotej Strmeň, Břetislav Brož, Zuzana Osifová, Martin Dračínský, Helena Mertlíková-Kaiserová, Zlatko Janeba
Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine. Journal of medicinal chemistry 67 (12) (2024)
Artem Chayka, Michal Česnek, Erika Kužmová, Jaroslav Kozák, Eva Tloušt'ová, Alexandra Dvořáková, Timotej Strmeň, Břetislav Brož, Zuzana Osifová, Martin Dračínský, Helena Mertlíková-Kaiserová, Zlatko Janeba
Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine. Journal of medicinal chemistry (2024)
Ladislav Prener, Ondřej Baszczyňski, Martin M Kaiser, Martin Dračínský, George Stepan, Yu-Jen Lee, Boris Brumshtein, Helen Yu, Petr Jansa, Eric B Lansdon, Zlatko Janeba
Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of medicinal chemistry 66 (3) (2023)
Ladislav Prener, Ondřej Baszczyňski, Martin M Kaiser, Martin Dračínský, George Stepan, Yu-Jen Lee, Boris Brumshtein, Helen Yu, Petr Jansa, Eric B Lansdon, Zlatko Janeba
Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of medicinal chemistry 66 (3) (2023)
Ladislav Prener, Ondřej Baszczyňski, Martin M Kaiser, Martin Dračínský, George Stepan, Yu-Jen Lee, Boris Brumshtein, Helen Yu, Petr Jansa, Eric B Lansdon, Zlatko Janeba
Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of medicinal chemistry 66 (3) (2023)
Ladislav Prener, Ondřej Baszczyňski, Martin M Kaiser, Martin Dračínský, George Stepan, Yu-Jen Lee, Boris Brumshtein, Helen Yu, Petr Jansa, Eric B Lansdon, Zlatko Janeba
Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of medicinal chemistry 66 (3) (2023)
Ladislav Prener, Ondřej Baszczyňski, Martin M Kaiser, Martin Dračínský, George Stepan, Yu-Jen Lee, Boris Brumshtein, Helen Yu, Petr Jansa, Eric B Lansdon, Zlatko Janeba
Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of medicinal chemistry (2023)
Jan Skácel, Stefan Djukic, Ondřej Baszczyňski, Filip Kalčic, Tadeáš Bílek, Karel Chalupský, Jaroslav Kozák, Alexandra Dvořáková, Eva Tloušt'ová, Zuzana Král'ová, Markéta Šmídková, Jan Voldřich, Michaela Rumlová, Petr Pachl, Jiří Brynda, Tereza Vučková, Milan Fábry, Jan Snášel, Iva Pichová, Pavlína Řezáčová, Helena Mertlíková-Kaiserová, Zlatko Janeba
Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of medicinal chemistry (2023)
Tomáš Klejch, Dianne T Keough, Gordon King, Eva Doleželová, Michal Česnek, Miloš Buděšínský, Alena Zíková, Zlatko Janeba, Luke W Guddat, Dana Hocková
Stereo-Defined Acyclic Nucleoside Phosphonates are Selective and Potent Inhibitors of Parasite 6-Oxopurine Phosphoribosyltransferases. Journal of medicinal chemistry 65 (5) (2022)
Filip Kalčic, Viktor Kolman, Zdeněk Zídek, Zlatko Janeba
Polysubstituted Pyrimidines as Potent Inhibitors of Prostaglandin E2 Production: Increasing Aqueous Solubility. ChemMedChem 16 (18) (2021)
Filip Kalčic, Michala Zgarbová, Jan Hodek, Karel Chalupský, Martin Dračínský, Alexandra Dvořáková, Timotej Strmeň, Jaroslav Šebestík, Ondřej Baszczyňski, Jan Weber, Helena Mertlíková-Kaiserová, Zlatko Janeba
Discovery of Modified Amidate (ProTide) Prodrugs of Tenofovir with Enhanced Antiviral Properties. Journal of medicinal chemistry 64 (22) (2021)
Michal Česnek, Michal Šafránek, Martin Dračínský, Eva Tloušťová, Helena Mertlíková-Kaiserová, Michael P Hayes, Val J Watts, Zlatko Janeba
Halogen-Dance-Based Synthesis of Phosphonomethoxyethyl (PME) Substituted 2-Aminothiazoles as Potent Inhibitors of Bacterial Adenylate Cyclases. ChemMedChem (2021)
Markéta Pimková Polidarová, Petra Břehová, Martin Maxmilian Kaiser, Miroslav Smola, Martin Dračínský, Joshua Smith, Aleš Marek, Milan Dejmek, Michal Šála, Ondrej Gutten, Lubomír Rulíšek, Barbora Novotná, Andrea Brázdová, Zlatko Janeba, Radim Nencka, Evzen Boura, Ondřej Páv, Gabriel Birkuš
Synthesis and Biological Evaluation of Phosphoester and Phosphorothioate Prodrugs of STING Agonist 3',3'-c-Di(2'F,2'dAMP). Journal of medicinal chemistry 64 (11) (2021)
Lucie Čechová, Juraj Filo, Martin Dračínský, Chavdar Slavov, Dazhong Sun, Zlatko Janeba, Tomáš Slanina, Josef Wachtveitl, Eliška Procházková, Marek Cigáň
Polysubstituted 5-Phenylazopyrimidines: Extremely Fast Non-ionic Photochromic Oscillators. Angewandte Chemie (International ed. in English) 59 (36) (2020)
Jan Skácel, Martin Dračínský, Zlatko Janeba
Synthesis of Tetrasubstituted Thiophenes via Direct Metalation. The Journal of organic chemistry 85 (2) (2020)
Filip Kalčic, Viktor Kolman, Haresh Ajani, Zdeněk Zídek, Zlatko Janeba
Polysubstituted Pyrimidines as mPGES-1 Inhibitors: Discovery of Potent Inhibitors of PGE2 Production with Strong Anti-inflammatory Effects in Carrageenan-Induced Rat Paw Edema. ChemMedChem 15 (15) (2020)
Jan Frydrych, Lenka Poštová Slavětínská, Martin Dračínský, Zlatko Janeba
Efficient Synthesis of α-Branched Purine-Based Acyclic Nucleosides: Scopes and Limitations of the Method. Molecules (Basel, Switzerland) 25 (18) (2020)
Ondřej Baszczyňski, Martin Maxmilian Kaiser, Michal Česnek, Petra Břehová, Petr Jansa, Eliška Procházková, Martin Dračínský, Robert Snoeck, Graciela Andrei, Zlatko Janeba
Xanthine-based acyclic nucleoside phosphonates with potent antiviral activity against varicella-zoster virus and human cytomegalovirus. Antiviral chemistry & chemotherapy 26 (2019)
Lucie Čechová, Milan Dejmek, Ondřej Baszczyňski, David Šaman, Liping Gao, Eric Hu, George Stepan, Petr Jansa, Zlatko Janeba, Petr Šimon
Synthesis and anti-human immunodeficiency virus activity of substituted ( o,o-difluorophenyl)-linked-pyrimidines as potent non-nucleoside reverse transcriptase inhibitors. Antiviral chemistry & chemotherapy 27 (2019)
Lucie Čechová, Jonas Kind, Martin Dračínský, Juraj Filo, Zlatko Janeba, Christina Marie Thiele, Marek Cigáň, Eliška Procházková
Photoswitching Behavior of 5-Phenylazopyrimidines: In Situ Irradiation NMR and Optical Spectroscopy Combined with Theoretical Methods. The Journal of organic chemistry 83 (11) (2018)
Jan Frydrych, Jan Skácel, Markéta Šmídková, Helena Mertlíková-Kaiserová, Martin Dračínský, Ramachandran Gnanasekaran, Martin Lepšík, Monica Soto-Velasquez, Val J Watts, Zlatko Janeba
Synthesis of α-Branched Acyclic Nucleoside Phosphonates as Potential Inhibitors of Bacterial Adenylate Cyclases. ChemMedChem 13 (2) (2018)
Michal Česnek, Jan Skácel, Petr Jansa, Martin Dračínský, Markéta Šmídková, Helena Mertlíková-Kaiserová, Monica P Soto-Velasquez, Val J Watts, Zlatko Janeba
Nucleobase Modified Adefovir (PMEA) Analogues as Potent and Selective Inhibitors of Adenylate Cyclases from Bordetella pertussis and Bacillus anthracis. ChemMedChem 13 (17) (2018)
Martin Maxmilian Kaiser, Ondřej Baszczyňski, Dana Hocková, Lenka Poštová-Slavětínská, Martin Dračínský, Dianne T Keough, Luke W Guddat, Zlatko Janeba
Acyclic Nucleoside Phosphonates Containing 9-Deazahypoxanthine and a Five-Membered Heterocycle as Selective Inhibitors of Plasmodial 6-Oxopurine Phosphoribosyltransferases. ChemMedChem 12 (14) (2017)
Petra Břehová, Markéta Šmídková, Jan Skácel, Martin Dračínský, Helena Mertlíková-Kaiserová, Monica P Soto Velasquez, Val J Watts, Zlatko Janeba
Design and Synthesis of Fluorescent Acyclic Nucleoside Phosphonates as Potent Inhibitors of Bacterial Adenylate Cyclases. ChemMedChem 11 (22) (2016)

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Publication Activity (10 Years)

Top Topics

Top Venues

Zlatko Janeba