Alison J-A Woolford

ORCID

Publication Activity (10 Years)

Years Active: 2018-2022
Publications (10 Years): 8

Top Venues

Journal of medicinal chemistry

RSC medicinal chemistry

Molecular cancer therapeutics

ACS medicinal chemistry letters

Astex Pharmaceuticals European Corporate and Research Headquarters

University of Cambridge (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Astex Pharmaceuticals European Corporate and Research Headquarters Oct 01 2001

United Kingdom

Director :: Chemistry

Education History

University of Cambridge Oct 01 1997 - Nov 01 2000

United Kingdom

PHD :: Chemistry

Publications

S Paul Jones, James D Firth, Mary C Wheldon, Masakazu Atobe, Roderick Eliot Hubbard, David C Blakemore, Claudia De Fusco, Simon C C Lucas, Stephen D Roughley, Lewis R Vidler, Maria Ann Whatton, Alison J-A Woolford, Gail L Wrigley, Peter O'Brien
Exploration of piperidine 3D fragment chemical space: synthesis and 3D shape analysis of fragments derived from 20 regio- and diastereoisomers of methyl substituted pipecolinates. RSC medicinal chemistry 13 (12) (2022)
S Paul Jones, James D Firth, Mary C Wheldon, Masakazu Atobe, Roderick Eliot Hubbard, David C Blakemore, Claudia De Fusco, Simon C C Lucas, Stephen D Roughley, Lewis R Vidler, Maria Ann Whatton, Alison J-A Woolford, Gail L Wrigley, Peter O'Brien
Exploration of piperidine 3D fragment chemical space: synthesis and 3D shape analysis of fragments derived from 20 regio- and diastereoisomers of methyl substituted pipecolinates. RSC medicinal chemistry 13 (12) (2022)
Emiliano Tamanini, Shin Miyamura, Ildiko M Buck, Benjamin D Cons, Lee Dawson, Charlotte East, Takashi Futamura, Shintaro Goto, Charlotte Griffiths-Jones, Tetsuya Hashimoto, Tom D Heightman, Shunpei Ishikawa, Hideki Ito, Yosuke Kaneko, Tatsuya Kawato, Kazumi Kondo, Naoki Kurihara, James M McCarthy, Yukiko Mori, Tsuyoshi Nagase, Yuichiro Nakaishi, Judith Reeks, Akimasa Sato, Patrick Schöpf, Kuninori Tai, Taichi Tamai, Dominic Tisi, Alison J-A Woolford
Fragment-Based Discovery of a Novel, Brain Penetrant, Orally Active HDAC2 Inhibitor. ACS medicinal chemistry letters 13 (10) (2022)
Tom D Heightman, Valerio Berdini, Luke Bevan, Ildiko M Buck, Maria G Carr, Aurélie Courtin, Joseph E Coyle, James E H Day, Charlotte East, Lynsey Fazal, Charlotte M Griffiths-Jones, Steven Howard, Justyna Kucia-Tran, Vanessa Martins, Sandra Muench, Joanne M Munck, David Norton, Marc O'Reilly, Nicholas Palmer, Puja Pathuri, Torren M Peakman, Michael Reader, David C Rees, Sharna J Rich, Alpesh Shah, Nicola G Wallis, Hugh Walton, Nicola E Wilsher, Alison J-A Woolford, Michael Cooke, David Cousin, Stuart Onions, Jonathan Shannon, John Watts, Christopher W Murray
Discovery of ASTX029, A Clinical Candidate Which Modulates the Phosphorylation and Catalytic Activity of ERK1/2. Journal of medicinal chemistry 64 (16) (2021)
Joanne M Munck, Valerio Berdini, Luke Bevan, Jessica L Brothwood, Juan Castro, Aurélie Courtin, Charlotte East, Roberta Ferraldeschi, Tom D Heightman, Christopher J Hindley, Justyna Kucia-Tran, John F Lyons, Vanessa Martins, Sandra Muench, Christopher W Murray, David Norton, Marc O'Reilly, Michael Reader, David C Rees, Sharna J Rich, Caroline J Richardson, Alpesh D Shah, Lukas Stanczuk, Neil T Thompson, Nicola E Wilsher, Alison J-A Woolford, Nicola G Wallis
ASTX029, a Novel Dual-mechanism ERK Inhibitor, Modulates Both the Phosphorylation and Catalytic Activity of ERK. Molecular cancer therapeutics 20 (10) (2021)
David Norton, William G Bonnette, James F Callahan, Maria G Carr, Charlotte M Griffiths-Jones, Tom D Heightman, Jeffrey K Kerns, Hong Nie, Sharna J Rich, Caroline Richardson, William Rumsey, Yolanda Sanchez, Marcel L Verdonk, Henriëtte M G Willems, William E Wixted, Lawrence Wolfe, Alison J-A Woolford, Zining Wu, Thomas G Davies
Fragment-Guided Discovery of Pyrazole Carboxylic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2 Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction. Journal of medicinal chemistry 64 (21) (2021)
Tom D Heightman, James F Callahan, Elisabetta Chiarparin, Joseph E Coyle, Charlotte Griffiths-Jones, Ami S Lakdawala, Rachel McMenamin, Paul N Mortenson, David Norton, Torren M Peakman, Sharna J Rich, Caroline Richardson, William L Rumsey, Yolanda Sanchez, Gordon Saxty, Henriëtte M G Willems, Lawrence Wolfe, Alison J-A Woolford, Zining Wu, Hongxing Yan, Jeffrey K Kerns, Thomas G Davies
Structure-Activity and Structure-Conformation Relationships of Aryl Propionic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1/Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1/NRF2) Protein-Protein Interaction. Journal of medicinal chemistry 62 (9) (2019)
Tom D Heightman, Valerio Berdini, Hannah Braithwaite, Ildiko M Buck, Megan Cassidy, Juan Castro, Aurélie Courtin, James E H Day, Charlotte East, Lynsey Fazal, Brent Graham, Charlotte M Griffiths-Jones, John F Lyons, Vanessa Martins, Sandra Muench, Joanne M Munck, David Norton, Marc O'Reilly, Nick Palmer, Puja Pathuri, Michael Reader, David C Rees, Sharna J Rich, Caroline Richardson, Harpreet Saini, Neil T Thompson, Nicola G Wallis, Hugh Walton, Nicola E Wilsher, Alison J-A Woolford, Michael Cooke, David Cousin, Stuart Onions, Jonathan Shannon, John Watts, Christopher W Murray
Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2. Journal of medicinal chemistry 61 (11) (2018)

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Publication Activity (10 Years)

Top Topics

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Alison J-A Woolford