Janez Ilaš

Scopus Author ID ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2019-2024
Publications (10 Years): 33

Top Venues

Journal of medicinal chemistry

Pharmaceuticals (Basel, Switzerland)

Journal of chemical information and modeling

RSC advances

University of Ljubljana

University of Ljubljana (MSC)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

University of Ljubljana Oct 01 2003

Slovenia

Professor :: Faculty of Pharmacy

Education History

University of Ljubljana Oct 01 1998 - Sep 05 2003

Slovenia

MSC :: Faculty of Pharmacy

Publications

Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Andrej Emanuel Cotman, Federica Fulgheri, Martina Piga, Peter Peršolja, Davide Benedetto Tiz, Žiga Skok, Martina Durcik, Maša Sterle, Jaka Dernovšek, Cristina D Cruz, Päivi Tammela, Petra Éva Szili, Lejla Daruka, Csaba Pál, Anamarija Zega, Lucija Peterlin Mašič, Janez Ilaš, Tihomir Tomašič, Danijel Kikelj, Nace Zidar
New N -phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity. RSC advances 14 (39) (2024)
Martina Durcik, Cristina D Cruz, Mariano Andrea Scorciapino, Janez Ilaš, Päivi Tammela, Matteo Ceccarelli, Lucija Peterlin Mašič, Tihomir Tomašič
Benzothiazole DNA gyrase inhibitors and their conjugates with siderophore mimics: design, synthesis and evaluation. RSC advances 14 (5) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 64 (12) (2024)
Martina Durcik, Cristina D Cruz, Mariano Andrea Scorciapino, Janez Ilaš, Päivi Tammela, Matteo Ceccarelli, Lucija Peterlin Mašič, Tihomir Tomašič
Benzothiazole DNA gyrase inhibitors and their conjugates with siderophore mimics: design, synthesis and evaluation. RSC advances 14 (5) (2024)
Martina Piga, Zoltan Varga, Adam Feher, Ferenc Papp, Eva Korpos, Kavya C Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar
Identification of a Novel Structural Class of H V 1 Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling (2024)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A Pardo, Diarmaid Hughes, Douglas L Huseby, Talía Berruga Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus . Journal of medicinal chemistry 66 (6) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A Pardo, Diarmaid Hughes, Douglas L Huseby, Talía Berruga Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus . Journal of medicinal chemistry 66 (6) (2023)
Maša Sterle, Martina Durcik, Clare E M Stevenson, Sara R Henderson, Petra Eva Szili, Marton Czikkely, David M Lawson, Anthony Maxwell, Dominique Cahard, Danijel Kikelj, Nace Zidar, Csaba Pal, Lucija Peterlin Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega
Exploring the 5-Substituted 2-Aminobenzothiazole-Based DNA Gyrase B Inhibitors Active against ESKAPE Pathogens. ACS omega 8 (27) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry (2023)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A Pardo, Diarmaid Hughes, Douglas L Huseby, Talía Berruga Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus . Journal of medicinal chemistry (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V Korol, Zhe Jin, Francisca Vicente, Maria C Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R Henderson, Julia E A Mundy, Anthony Maxwell, Clare E M Stevenson, David M Lawson, Guido V Janssen, Geert Jan Sterk, Danijel Kikelj
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa . Journal of medicinal chemistry 66 (2) (2023)
Péter Ábrányi-Balogh, Aaron Keeley, György G Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast Rambaher, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Miklós Keserű
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors. Pharmaceuticals (Basel, Switzerland) 15 (12) (2022)
Péter Ábrányi-Balogh, Aaron Keeley, György G Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast Rambaher, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Miklós Keserű
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors. Pharmaceuticals (Basel, Switzerland) 15 (12) (2022)
Péter Ábrányi-Balogh, Aaron Keeley, György G Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast Rambaher, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Miklós Keserű
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors. Pharmaceuticals (Basel, Switzerland) 15 (12) (2022)
Péter Ábrányi-Balogh, Aaron Keeley, György G Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast Rambaher, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Miklós Keserű
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors. Pharmaceuticals (Basel, Switzerland) 15 (12) (2022)
Oussama Moussaoui, Rajendra Bhadane, Riham Sghyar, Janez Ilaš, El Mestafa El Hadrami, Said Chakroune, Outi M H Salo-Ahen
Design, Synthesis, in vitro and in silico Characterization of 2-Quinolone-L-alaninate-1,2,3-triazoles as Antimicrobial Agents. ChemMedChem 17 (5) (2022)
Tihomir Tomašič, Asta Zubrienė, Žiga Skok, Riccardo Martini, Stane Pajk, Gobec Izidor Sosič, Janez Ilaš, Daumantas Matulis, Sharon D Bryant
Selective DNA Gyrase Inhibitors: Multi-Target in Silico Profiling with 3D-Pharmacophores. Pharmaceuticals (Basel, Switzerland) 14 (8) (2021)
Dávid Bajusz, Warren S Wade, Grzegorz Satała, Andrzej J Bojarski, Janez Ilaš, Jessica Ebner, Florian Grebien, Henrietta Papp, Ferenc Jakab, Alice Douangamath, Daren Fearon, Frank von Delft, Marion Schuller, Ivan Ahel, Amanda Wakefield, Sándor Vajda, János Gerencsér, Péter Pallai, György Miklós Keserű
Exploring protein hotspots by optimized fragment pharmacophores. Nature communications 12 (1) (2021)
Petra Dunkel, Janez Ilaš
Targeted Cancer Therapy Using Compounds Activated by Light. Cancers 13 (13) (2021)
Martina Durcik, Žiga Skok, Janez Ilaš, Nace Zidar, Anamarija Zega, Petra Éva Szili, Gábor Draskovits, Tamás Révész, Danijel Kikelj, Akos Nyerges, Csaba Pál, Lucija Peterlin Mašič, Tihomir Tomašič
Hybrid Inhibitors of DNA Gyrase A and B: Design, Synthesis and Evaluation. Pharmaceutics 13 (1) (2020)
Nina Žigart, Martin Črnugelj, Janez Ilaš, Zdenko Časar
On the Stability and Degradation Pathways of Venetoclax under Stress Conditions. Pharmaceutics 12 (7) (2020)
Akos Nyerges, Tihomir Tomašič, Martina Durcik, Tamas Revesz, Petra Szili, Gabor Draskovits, Ferenc Bogar, Žiga Skok, Nace Zidar, Janez Ilaš, Anamarija Zega, Danijel Kikelj, Lejla Daruka, Balint Kintses, Balint Vasarhelyi, Imre Foldesi, Diána Kata, Martin Welin, Yengo Raymond Kimbung, Dorota Focht, Lucija Peterlin Mašič, Csaba Pál
Rational design of balanced dual-targeting antibiotics with limited resistance. PLoS biology 18 (10) (2020)
Jelena Rupar, Vladimir Dobričić, Jelena Grahovac, Siniša Radulović, Žiga Skok, Janez Ilaš, Mara Aleksić, Jasmina Brborić, Olivera Čudina
Synthesis and evaluation of anticancer activity of new 9-acridinyl amino acid derivatives. RSC medicinal chemistry 11 (3) (2020)
Martina Durcik, Tihomir Tomašič, Nace Zidar, Anamarija Zega, Danijel Kikelj, Lucija Peterlin Mašič, Janez Ilaš
ATP-competitive DNA gyrase and topoisomerase IV inhibitors as antibacterial agents. Expert opinion on therapeutic patents 29 (3) (2019)
Žiga Skok, Nace Zidar, Danijel Kikelj, Janez Ilaš
Dual Inhibitors of Human DNA Topoisomerase II and Other Cancer-Related Targets. Journal of medicinal chemistry 63 (3) (2019)
Nace Zidar, Helena Macut, Tihomir Tomašič, Lucija Peterlin Mašič, Janez Ilaš, Anamarija Zega, Päivi Tammela, Danijel Kikelj
New N-phenyl-4,5-dibromopyrrolamides as DNA gyrase B inhibitors. MedChemComm 10 (6) (2019)

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Publication Activity (10 Years)

Top Topics

Top Venues

Janez Ilaš