Santiago Vázquez

ResearcherID Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 33

Top Topics

Mycobacterium Tuberculosis

Molecular Docking

Plasmodium Falciparum

Multidrug Resistant

Top Venues

ACS infectious diseases

Journal of medicinal chemistry

Molecules (Basel, Switzerland)

Microbiology spectrum

This page only lists publications with an associated author ORCID identifier.

Publications

Ali Pormohammad, Melika Moradi, Josefien W Hommes, Eugènia Pujol, Lieve Naesens, Santiago Vázquez, Bas G J Surewaard, Mohammad Zarei, Manuel Vazquez-Carrera, Raymond Joseph Turner
Novel pentafluorosulfanyl-containing triclocarban analogs selectively kill Gram-positive bacteria. Microbiology spectrum 12 (6) (2024)
Savannah J Watson, Mariëtte E van der Watt, Anjo Theron, Janette Reader, Sizwe Tshabalala, Erica Erlank, Lizette L Koekemoer, Mariska Naude, Marianna Stampolaki, Feyisola Adewole, Katie Sadowska, Pilar Pérez-Lozano, Andreea L Turcu, Santiago Vázquez, Jihee Ko, Ben Mazurek, Davinder Singh, Satish R Malwal, Mathew Njoroge, Kelly Chibale, Oluseye K Onajole, Antonios D Kolocouris, Eric Oldfield, Lyn-Marié Birkholtz
The Tuberculosis Drug Candidate SQ109 and Its Analogs Have Multistage Activity against Plasmodium falciparum . ACS infectious diseases (2024)
Ali Pormohammad, Melika Moradi, Josefien W Hommes, Eugènia Pujol, Lieve Naesens, Santiago Vázquez, Bas G J Surewaard, Mohammad Zarei, Manuel Vazquez-Carrera, Raymond Joseph Turner
Novel pentafluorosulfanyl-containing triclocarban analogs selectively kill Gram-positive bacteria. Microbiology spectrum (2024)
Ali Pormohammad, Melika Moradi, Josefien W Hommes, Eugènia Pujol, Lieve Naesens, Santiago Vázquez, Bas G J Surewaard, Mohammad Zarei, Manuel Vazquez-Carrera, Raymond Joseph Turner
Novel pentafluorosulfanyl-containing triclocarban analogs selectively kill Gram-positive bacteria. Microbiology spectrum 12 (6) (2024)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases 9 (2) (2023)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases 9 (2) (2023)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases 9 (2) (2023)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases (2023)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases 9 (2) (2023)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases (2023)
Marianna Stampolaki, Satish R Malwal, Nadine Alvarez-Cabrera, Zijun Gao, Mohammad Moniruzzaman, Svitlana O Babii, Nikolaos Naziris, André Rey-Cibati, Mariana Valladares-Delgado, Andreea L Turcu, Kyung-Hwa Baek, Trong-Nhat Phan, Hyeryon Lee, Mattheo Alcaraz, Savannah Watson, Mariette van der Watt, Dina Coertzen, Natasa Efstathiou, Maria Chountoulesi, Carolyn M Shoen, Ioannis P Papanastasiou, Jose Brea, Michael H Cynamon, Lyn-Marié Birkholtz, Laurent Kremer, Joo Hwan No, Santiago Vázquez, Gustavo Benaim, Costas Demetzos, Helen I Zgurskaya, Thomas Dick, Eric Oldfield, Antonios D Kolocouris
Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria Parasites. ACS infectious diseases (2023)
Meijian Zhang, Andrea Bagán, Donna Martínez, Emma Barroso, Xavier Palomer, Santiago Vázquez, Carmen Escolano, Manuel Vázquez-Carrera
Design and Synthesis of AMPK Activators and GDF15 Inducers. Molecules (Basel, Switzerland) 28 (14) (2023)
Sandra Codony, Caterina Pont, Christian Griñán-Ferré, Ania Di Pede-Mattatelli, Carla Calvó-Tusell, Ferran Feixas, Sílvia Osuna, Júlia Jarné-Ferrer, Marina Naldi, Manuela Bartolini, Maria Isabel Loza, José Brea, Belén Pérez, Clara Bartra, Coral Sanfeliu, Jordi Juárez-Jiménez, Christophe Morisseau, Bruce D Hammock, Mercé Pallàs, Santiago Vázquez, Diego Muñoz-Torrero
Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's Disease. Journal of medicinal chemistry 65 (6) (2022)
Sandra Codony, José M Entrena, Carla Calvó-Tusell, Beatrice Jora, Rafael González-Cano, Sílvia Osuna, Rubén Corpas, Christophe Morisseau, Belén Pérez, Marta Barniol-Xicota, Christian Griñán-Ferré, Concepción Pérez, María Isabel Rodríguez-Franco, Antón L Martínez, Maria Isabel Loza, Mercé Pallàs, Steven H L Verhelst, Coral Sanfeliu, Ferran Feixas, Bruce D Hammock, Jose Brea, Enrique J Cobos, Santiago Vázquez
Synthesis, In Vitro Profiling, and In Vivo Evaluation of Benzohomoadamantane-Based Ureas for Visceral Pain: A New Indication for Soluble Epoxide Hydrolase Inhibitors. Journal of medicinal chemistry 65 (20) (2022)
Júlia Jarne-Ferrer, Christian Griñán-Ferré, Aina Bellver-Sanchis, Santiago Vázquez, Diego Muñoz-Torrero, Mercé Pallàs
A Combined Chronic Low-Dose Soluble Epoxide Hydrolase and Acetylcholinesterase Pharmacological Inhibition Promotes Memory Reinstatement in Alzheimer's Disease Mice Models. Pharmaceuticals (Basel, Switzerland) 15 (8) (2022)
Madeleine R Wilcox, Aparna Nigam, Nathan G Glasgow, Chamali Narangoda, Matthew B Phillips, Dhilon S Patel, Samaneh Mesbahi-Vasey, Andreea L Turcu, Santiago Vázquez, Maria G Kurnikova, Jon W Johnson
Inhibition of NMDA receptors through a membrane-to-channel path. Nature communications 13 (1) (2022)
Sandra Codony, Carla Calvó-Tusell, Elena Valverde, Sílvia Osuna, Christophe Morisseau, M Isabel Loza, José Brea, Concepción Pérez, María Isabel Rodríguez-Franco, Javier Pizarro-Delgado, Rubén Corpas, Christian Griñán-Ferré, Mercé Pallàs, Coral Sanfeliu, Manuel Vázquez-Carrera, Bruce D Hammock, Ferran Feixas, Santiago Vázquez
From the Design to the In Vivo Evaluation of Benzohomoadamantane-Derived Soluble Epoxide Hydrolase Inhibitors for the Treatment of Acute Pancreatitis. Journal of medicinal chemistry 64 (9) (2021)
Sergio Rodriguez-Arevalo, Eugènia Pujol, Sònia Abás, Carles Galdeano, Carmen Escolano, Santiago Vázquez
Synthesis, Characterization and HPLC Analysis of the (1S,2S,5R)-Diastereomer and the Enantiomer of the Clinical Candidate AR-15512. Molecules (Basel, Switzerland) 26 (4) (2021)
Dolors Puigoriol-Illamola, Júlia Companys-Alemany, Kris McGuire, Natalie Z M Homer, Rosana Leiva, Santiago Vázquez, Damian J Mole, Christian Griñán-Ferré, Mercé Pallàs
Inhibition of 11β-HSD1 Ameliorates Cognition and Molecular Detrimental Changes after Chronic Mild Stress in SAMP8 Mice. Pharmaceuticals (Basel, Switzerland) 14 (10) (2021)
Christian Griñán-Ferré, Júlia Companys-Alemany, Júlia Jarné-Ferrer, Sandra Codony, Celia González-Castillo, Daniel Ortuño-Sahagún, Lluïsa Vilageliu, Daniel Grinberg, Santiago Vázquez, Mercé Pallàs
Inhibition of Soluble Epoxide Hydrolase Ameliorates Phenotype and Cognitive Abilities in a Murine Model of Niemann Pick Type C Disease. International journal of molecular sciences 22 (7) (2021)
Alexandra Probst, Eugènia Pujol, Cécile Häberli, Jennifer Keiser, Santiago Vázquez
In Vitro, In Vivo, and Absorption, Distribution, Metabolism, and Excretion Evaluation of SF5-Containing N,N'-Diarylureas as Antischistosomal Agents. Antimicrobial agents and chemotherapy 65 (10) (2021)
Juan Martín-López, Sandra Codony, Clara Bartra, Christophe Morisseau, María Isabel Loza, Coral Sanfeliu, Bruce D Hammock, Jose Brea, Santiago Vázquez
2-(Piperidin-4-yl)acetamides as Potent Inhibitors of Soluble Epoxide Hydrolase with Anti-Inflammatory Activity. Pharmaceuticals (Basel, Switzerland) 14 (12) (2021)
Sandra Codony, Eugènia Pujol, Javier Pizarro, Ferran Feixas, Elena Valverde, M Isabel Loza, José M Brea, Elena Saez, Julen Oyarzábal, Antonio Pineda-Lucena, Belén Pérez, Concepción Pérez, María Isabel Rodríguez-Franco, Rosana Leiva, Sílvia Osuna, Christophe Morisseau, Bruce D Hammock, Manuel Vázquez-Carrera, Santiago Vázquez
2-Oxaadamant-1-yl Ureas as Soluble Epoxide Hydrolase Inhibitors: In Vivo Evaluation in a Murine Model of Acute Pancreatitis. Journal of medicinal chemistry 63 (17) (2020)
Mercé Pallàs, Santiago Vázquez, Coral Sanfeliu, Carles Galdeano, Christian Griñán-Ferré
Soluble Epoxide Hydrolase Inhibition to Face Neuroinflammation in Parkinson's Disease: A New Therapeutic Strategy. Biomolecules 10 (5) (2020)
Júlia Companys-Alemany, Andreea L Turcu, Aina Bellver-Sanchis, Maria I Loza, José M Brea, Anna M Canudas, Rosana Leiva, Santiago Vázquez, Mercé Pallàs, Christian Griñán-Ferré
A Novel NMDA Receptor Antagonist Protects against Cognitive Decline Presented by Senescent Mice. Pharmaceutics 12 (3) (2020)
Christina Tzitzoglaki, Kelly McGuire, Panagiotis Lagarias, Athina Konstantinidi, Anja Hoffmann, Natalie A Fokina, Chulong Ma, Ioannis P Papanastasiou, Peter Richard Schreiner, Santiago Vázquez, Michaela Schmidtke, Jun Wang, David D Busath, Antonios D Kolocouris
Chemical Probes for Blocking of Influenza A M2 Wild-type and S31N Channels. ACS chemical biology 15 (9) (2020)
Liam Hudson, James Mui, Santiago Vázquez, Diana M Carvalho, Eleanor Williams, Chris Jones, Alex N Bullock, Swen Hoelder
Novel Quinazolinone Inhibitors of ALK2 Flip between Alternate Binding Modes: Structure-Activity Relationship, Structural Characterization, Kinase Profiling, and Cellular Proof of Concept. Journal of medicinal chemistry 61 (16) (2018)
Eugènia Pujol, Núria Blanco-Cabra, Esther Julián, Rosana Leiva, Eduard Torrents, Santiago Vázquez
Pentafluorosulfanyl-containing Triclocarban Analogs with Potent Antimicrobial Activity. Molecules (Basel, Switzerland) 23 (11) (2018)
Rosana Leiva, Andrew McBride, Margaret Binnie, Scott P Webster, Santiago Vázquez
Exploring N-acyl-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-enes as 11β-HSD1 Inhibitors. Molecules (Basel, Switzerland) 23 (3) (2018)
Rosana Leiva, Matthew B Phillips, Andreea L Turcu, Esther Gratacòs-Batlle, Lara León-García, Francesc X Sureda, David Soto, Jon W Johnson, Santiago Vázquez
Pharmacological and Electrophysiological Characterization of Novel NMDA Receptor Antagonists. ACS chemical neuroscience 9 (11) (2018)
Olga Karoutzou, Seung-Hwa Kwak, So-Deok Lee, Daina Martínez-Falguera, Francesc X Sureda, Santiago Vázquez, Yong-Chul Kim, Marta Barniol-Xicota
Towards a Novel Class of Multitarget-Directed Ligands: Dual P2X7-NMDA Receptor Antagonists. Molecules (Basel, Switzerland) 23 (1) (2018)
Marta Barniol-Xicota, Sabrina Gazzarrini, Eva Torres, Yanmei Hu, Jun Wang, Lieve Naesens, Anna Moroni, Santiago Vázquez
Slow but Steady Wins the Race: Dissimilarities among New Dual Inhibitors of the Wild-Type and the V27A Mutant M2 Channels of Influenza A Virus. Journal of medicinal chemistry 60 (9) (2017)
Rosana Leiva, Marta Barniol-Xicota, Sandra Codony, Tiziana Ginex, Evelien Vanderlinden, Marta Montes, Michael Caffrey, Francisco Javier Luque, Lieve Naesens, Santiago Vázquez
Aniline-Based Inhibitors of Influenza H1N1 Virus Acting on Hemagglutinin-Mediated Fusion. Journal of medicinal chemistry 61 (1) (2017)