Stefan Schiesser

ORCID

Publication Activity (10 Years)

Years Active: 2020-2024
Publications (10 Years): 12

Top Venues

Journal of medicinal chemistry

Future medicinal chemistry

ACS medicinal chemistry letters

AstraZeneca

Ludwig-Maximilians-University (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

AstraZeneca Mar 01 2017

Sweden

Associate Principal Scientist :: Department of Medicinal Chemistry

AstraZeneca Jun 01 2016 - Feb 28 2017

Sweden

Senior Research Scientist :: Department of Medicinal Chemistry

Education History

Ludwig-Maximilians-University Sep 01 2009 - Mar 13 2014

Germany

PHD :: Department of Chemistry and Pharmacy

Ludwig-Maximilians University

Germany

MSC :: Department of Chemistry and Pharmacy

Ludwig-Maximilians University

Germany

BSC :: Department of Chemistry and Pharmacy

Publications

Simon C C Lucas, Alexander G Milbradt, J Henry Blackwell, Silvia Bonomo, Andrew Brierley, Doyle J Cassar, Jared Freeman, Thomas E Hadfield, Lucas A Morrill, Rick Riemens, Sunil Sarda, Stefan Schiesser, Daniel Wiktelius, Samiyah Ahmed, Mark J Bostock, Ulf Börjesson, Claudia De Fusco, Carine Guerot, David Hargreaves, Sarah Hewitt, Michelle L Lamb, Nancy Su, Ryan Whatling, Matthew Wheeler, Jason G Kettle
Design of a Lead-Like Cysteine-Targeting Covalent Library and the Identification of Hits to Cys55 of Bfl-1. Journal of medicinal chemistry 67 (13) (2024)
Simon C C Lucas, Alexander G Milbradt, J Henry Blackwell, Silvia Bonomo, Andrew Brierley, Doyle J Cassar, Jared Freeman, Thomas E Hadfield, Lucas A Morrill, Rick Riemens, Sunil Sarda, Stefan Schiesser, Daniel Wiktelius, Samiyah Ahmed, Mark J Bostock, Ulf Börjesson, Claudia De Fusco, Carine Guerot, David Hargreaves, Sarah Hewitt, Michelle L Lamb, Nancy Su, Ryan Whatling, Matthew Wheeler, Jason G Kettle
Design of a Lead-Like Cysteine-Targeting Covalent Library and the Identification of Hits to Cys55 of Bfl-1. Journal of medicinal chemistry 67 (13) (2024)
Simon C C Lucas, Alexander G Milbradt, J Henry Blackwell, Silvia Bonomo, Andrew Brierley, Doyle J Cassar, Jared Freeman, Thomas E Hadfield, Lucas A Morrill, Rick Riemens, Sunil Sarda, Stefan Schiesser, Daniel Wiktelius, Samiyah Ahmed, Mark J Bostock, Ulf Börjesson, Claudia De Fusco, Carine Guerot, David Hargreaves, Sarah Hewitt, Michelle L Lamb, Nancy Su, Ryan Whatling, Matthew Wheeler, Jason G Kettle
Design of a Lead-Like Cysteine-Targeting Covalent Library and the Identification of Hits to Cys55 of Bfl-1. Journal of medicinal chemistry (2024)
Fabio Begnini, Stefan Geschwindner, Patrik Johansson, Lisa Wissler, Richard J Lewis, Emma Danelius, Andreas Luttens, Pierre Matricon, Jens Carlsson, Stijn Lenders, Beate König, Anna Friedel, Peter Sjö, Stefan Schiesser, Jan Kihlberg
Correction to "Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction". Journal of medicinal chemistry (2023)
Fabio Begnini, Stefan Geschwindner, Patrik Johansson, Lisa Wissler, Richard J Lewis, Emma Danelius, Andreas Luttens, Pierre Matricon, Jens Carlsson, Stijn Lenders, Beate König, Anna Friedel, Peter Sjö, Stefan Schiesser, Jan Kihlberg
Correction to "Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction". Journal of medicinal chemistry 66 (3) (2023)
Fabio Begnini, Stefan Geschwindner, Patrik Johansson, Lisa Wissler, Richard J Lewis, Emma Danelius, Andreas Luttens, Pierre Matricon, Jens Carlsson, Stijn Lenders, Beate König, Anna Friedel, Peter Sjö, Stefan Schiesser, Jan Kihlberg
Correction to "Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction". Journal of medicinal chemistry 66 (3) (2023)
Fabio Begnini, Stefan Geschwindner, Patrik Johansson, Lisa Wissler, Richard J Lewis, Emma Danelius, Andreas Luttens, Pierre Matricon, Jens Carlsson, Stijn Lenders, Beate König, Anna Friedel, Peter Sjö, Stefan Schiesser, Jan Kihlberg
Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction. Journal of medicinal chemistry 65 (4) (2022)
Fabio Begnini, Vasanthanathan Poongavanam, Yoseph Atilaw, Máté Erdélyi, Stefan Schiesser, Jan Kihlberg
Cell Permeability of Isomeric Macrocycles: Predictions and NMR Studies. ACS medicinal chemistry letters 12 (6) (2021)
Igor Shamovsky, Lena Ripa, Frank Narjes, Britta Bonn, Stefan Schiesser, Ina Terstiege, Christian Tyrchan
Mechanism-Based Insights into Removing the Mutagenicity of Aromatic Amines by Small Structural Alterations. Journal of medicinal chemistry 64 (12) (2021)
Stefan Schiesser, Rhona J Cox, Werngard Czechtizky
The powerful symbiosis between synthetic and medicinal chemistry. Future medicinal chemistry 13 (11) (2021)
Stefan Schiesser, Hanna Chepliaka, Johanna Kollback, Thibaut Quennesson, Werngard Czechtizky, Rhona J Cox
N-Trifluoromethyl Amines and Azoles: An Underexplored Functional Group in the Medicinal Chemist's Toolbox. Journal of medicinal chemistry 63 (21) (2020)
Fabio Begnini, Vasanthanathan Poongavanam, Björn Over, Marie Castaldo, Stefan Geschwindner, Patrik Johansson, Mohit Tyagi, Christian Tyrchan, Lisa Wissler, Peter Sjö, Stefan Schiesser, Jan Kihlberg
Mining Natural Products for Macrocycles to Drug Difficult Targets. Journal of medicinal chemistry 64 (2) (2020)

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Publication Activity (10 Years)

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Stefan Schiesser