Terrence R Burke

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 24

Top Topics

Structural Basis

Men Who Have Sex With Men

Top Venues

ACS infectious diseases

RSC chemical biology

Nature communications

This page only lists publications with an associated author ORCID identifier.

Publications

Xue Zhi Zhao, Idris A Barakat, George T Lountos, Wenjie Wang, Keli Agama, Md Rasel Al Mahmud, Kiall F Suazo, Thorkell Andresson, Yves Pommier, Terrence R Burke
Targeted sulfur(VI) fluoride exchange-mediated covalent modification of a tyrosine residue in the catalytic pocket of tyrosyl-DNA phosphodiesterase 1. Communications chemistry 7 (1) (2024)
Pankaj S Mahajan, Steven J Smith, Min Li, Robert Craigie, Stephen H Hughes, Xue Zhi Zhao, Terrence R Burke
N -Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants. ACS infectious diseases 10 (3) (2024)
Pankaj S Mahajan, Steven J Smith, Min Li, Robert Craigie, Stephen H Hughes, Xue Zhi Zhao, Terrence R Burke
N -Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants. ACS infectious diseases 10 (3) (2024)
Pankaj S Mahajan, Steven J Smith, Min Li, Robert Craigie, Stephen H Hughes, Xue Zhi Zhao, Terrence R Burke
N -Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants. ACS infectious diseases 10 (3) (2024)
Pankaj S Mahajan, Steven J Smith, Min Li, Robert Craigie, Stephen H Hughes, Xue Zhi Zhao, Terrence R Burke
N -Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants. ACS infectious diseases 10 (3) (2024)
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
Affinity enhancement of polo-like kinase 1 polo box domain-binding ligands by a bivalent approach using a covalent kinase-binding component. RSC chemical biology 5 (8) (2024)
Pankaj S Mahajan, Steven J Smith, Min Li, Robert Craigie, Stephen H Hughes, Xue Zhi Zhao, Terrence R Burke
N -Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants. ACS infectious diseases 10 (3) (2024)
Pankaj S Mahajan, Steven J Smith, Min Li, Robert Craigie, Stephen H Hughes, Xue Zhi Zhao, Terrence R Burke
N -Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants. ACS infectious diseases (2024)
Kohei Tsuji, Hirokazu Tamamura, Terrence R Burke
Affinity enhancement of polo-like kinase 1 polo box domain-binding ligands by a bivalent approach using a covalent kinase-binding component. RSC chemical biology 5 (8) (2024)
Xue Zhi Zhao, Wenjie Wang, George T Lountos, Evgeny Kiselev, Joseph E Tropea, Danielle Needle, Yves Pommier, Terrence R Burke
Identification of multidentate tyrosyl-DNA phosphodiesterase 1 (TDP1) inhibitors that simultaneously access the DNA, protein and catalytic-binding sites by oxime diversification. RSC chemical biology 4 (5) (2023)
Xue Zhi Zhao, Wenjie Wang, George T Lountos, Evgeny Kiselev, Joseph E Tropea, Danielle Needle, Yves Pommier, Terrence R Burke
Identification of multidentate tyrosyl-DNA phosphodiesterase 1 (TDP1) inhibitors that simultaneously access the DNA, protein and catalytic-binding sites by oxime diversification. RSC chemical biology 4 (5) (2023)
Min Li, Dario Oliveira Passos, Zelin Shan, Steven J Smith, Qinfang Sun, Avik Biswas, Indrani Choudhuri, Timothy S Strutzenberg, Allan Haldane, Nanjie Deng, Zhaoyang Li, Xue Zhi Zhao, Lorenzo Briganti, Mamuka Kvaratskhelia, Terrence R Burke, Ronald M Levy, Stephen H Hughes, Robert Craigie, Dmitry Lyumkis
Mechanisms of HIV-1 integrase resistance to dolutegravir and potent inhibition of drug-resistant variants. Science advances 9 (29) (2023)
Kohei Tsuji, David Hymel, Buyong Ma, Hirokazu Tamamura, Ruth Nussinov, Terrence R Burke
Development of ultra-high affinity bivalent ligands targeting the polo-like kinase 1. RSC chemical biology 3 (9) (2022)
Michal S Barski, Teresa Vanzo, Xue Zhi Zhao, Steven J Smith, Allison Ballandras-Colas, Nora B Cronin, Valerie E Pye, Stephen H Hughes, Terrence R Burke, Peter Cherepanov, Goedele N Maertens
Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures. Nature communications 12 (1) (2021)
Steven J Smith, Andrea Ferris, Xue Zhi Zhao, Gary Pauly, Joel P Schneider, Terrence R Burke, Stephen H Hughes
INSTIs and NNRTIs Potently Inhibit HIV-1 Polypurine Tract Mutants in a Single Round Infection Assay. Viruses 13 (12) (2021)
Steven J Smith, Xue Zhi Zhao, Dario Oliveira Passos, Valerie E Pye, Peter Cherepanov, Dmitry Lyumkis, Terrence R Burke, Stephen H Hughes
HIV-1 Integrase Inhibitors with Modifications That Affect Their Potencies against Drug Resistant Integrase Mutants. ACS infectious diseases 7 (6) (2021)
David Hymel, Kohei Tsuji, Robert A Grant, Ramesh M Chingle, Dominique L Kunciw, Micheal B Yaffe, Terrence R Burke
Design and synthesis of a new orthogonally protected glutamic acid analog and its use in the preparation of high affinity polo-like kinase 1 polo-box domain - binding peptide macrocycles. Organic & biomolecular chemistry 19 (36) (2021)
Steven J Smith, Xue Zhi Zhao, Dario Oliveira Passos, Dmitry Lyumkis, Terrence R Burke, Stephen H Hughes
Integrase Strand Transfer Inhibitors Are Effective Anti-HIV Drugs. Viruses 13 (2) (2021)
Michal S Barski, Teresa Vanzo, Xue Zhi Zhao, Steven J Smith, Allison Ballandras-Colas, Nora B Cronin, Valerie E Pye, Stephen H Hughes, Terrence R Burke, Peter Cherepanov, Goedele N Maertens
Publisher Correction: Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures. Nature communications 12 (1) (2021)
Xue Zhi Zhao, Evgeny Kiselev, George T Lountos, Wenjie Wang, Joseph E Tropea, Danielle Needle, Thomas A Hilimire, John S Schneekloth, David S Waugh, Yves Pommier, Terrence R Burke
Small molecule microarray identifies inhibitors of tyrosyl-DNA phosphodiesterase 1 that simultaneously access the catalytic pocket and two substrate binding sites. Chemical science 12 (11) (2021)
Stephen E Miller, Kohei Tsuji, Rachel P M Abrams, Terrence R Burke, Joel P Schneider
Uncoupling the Folding-Function Paradigm of Lytic Peptides to Deliver Impermeable Inhibitors of Intracellular Protein-Protein Interactions. Journal of the American Chemical Society 142 (47) (2020)
Dario Oliveira Passos, Min Li, Ilona K Jóźwik, Xue Zhi Zhao, Diogo Santos-Martins, Renbin Yang, Steven J Smith, Youngmin Jeon, Stefano Forli, Stephen H Hughes, Terrence R Burke, Robert Craigie, Dmitry Lyumkis
Structural basis for strand-transfer inhibitor binding to HIV intasomes. Science (New York, N.Y.) 367 (6479) (2020)
Dobeen Hwang, Kohei Tsuji, HaJeung Park, Terrence R Burke, Christoph Rader
Site-Specific Lysine Arylation as an Alternative Bioconjugation Strategy for Chemically Programmed Antibodies and Antibody-Drug Conjugates. Bioconjugate chemistry 30 (11) (2019)
Xue Zhi Zhao, Steven J Smith, Daniel P Maskell, Mathieu Métifiot, Valerie E Pye, Katherine Fesen, Christophe Marchand, Yves Pommier, Peter Cherepanov, Stephen H Hughes, Terrence R Burke
Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors. Journal of medicinal chemistry 60 (17) (2017)