Alexandros Makriyannis (A Makriyannis)

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 21

Top Topics

Molecular Dynamics Simulations

Diabetic Nephropathy

Top Venues

ACS chemical biology

Journal of medicinal chemistry

Journal of natural products

British journal of pharmacology

This page only lists publications with an associated author ORCID identifier.

Publications

Katharina Grotsch, Anastasiia V Sadybekov, Sydney Hiller, Saheem Zaidi, Dmitry B Eremin, Austen Le, Yong-Feng Liu, Evan Carlton Smith, Christos Illiopoulis-Tsoutsouvas, Joice Thomas, Shubhangi Aggarwal, Julie E Pickett, Cesar Reyes, Elias Picazo, Bryan L Roth, Alexandros Makriyannis, Vsevolod Katritch, Valery V Fokin
Virtual Screening of a Chemically Diverse "Superscaffold" Library Enables Ligand Discovery for a Key GPCR Target. ACS chemical biology 19 (4) (2024)
Spyros P Nikas, Lipin Ji, Yingpeng Liu, Markos-Orestis Georgiadis, Amey Dopeshwarkar, Alex Straiker, Shalley N Kudalkar, Anastasiia V Sadybekov, Michaela Dvorakova, Vsevolod Katritch, Ken Mackie, Lawrence J Marnett, Alexandros Makriyannis
Chiral Me-2-arachidonoyl Glycerols: The First Potent Endocannabinoid Glyceride Templates with Stability to COX-2. ACS medicinal chemistry letters 15 (6) (2024)
Katharina Grotsch, Anastasiia V Sadybekov, Sydney Hiller, Saheem Zaidi, Dmitry B Eremin, Austen Le, Yong-Feng Liu, Evan Carlton Smith, Christos Illiopoulis-Tsoutsouvas, Joice Thomas, Shubhangi Aggarwal, Julie E Pickett, Cesar Reyes, Elias Picazo, Bryan L Roth, Alexandros Makriyannis, Vsevolod Katritch, Valery V Fokin
Virtual Screening of a Chemically Diverse "Superscaffold" Library Enables Ligand Discovery for a Key GPCR Target. ACS chemical biology 19 (4) (2024)
Spyros P Nikas, Lipin Ji, Yingpeng Liu, Markos-Orestis Georgiadis, Amey Dopeshwarkar, Alex Straiker, Shalley N Kudalkar, Anastasiia V Sadybekov, Michaela Dvorakova, Vsevolod Katritch, Ken Mackie, Lawrence J Marnett, Alexandros Makriyannis
Chiral Me-2-arachidonoyl Glycerols: The First Potent Endocannabinoid Glyceride Templates with Stability to COX-2. ACS medicinal chemistry letters 15 (6) (2024)
Katharina Grotsch, Anastasiia V Sadybekov, Sydney Hiller, Saheem Zaidi, Dmitry B Eremin, Austen Le, Yong-Feng Liu, Evan Carlton Smith, Christos Illiopoulis-Tsoutsouvas, Joice Thomas, Shubhangi Aggarwal, Julie E Pickett, Cesar Reyes, Elias Picazo, Bryan L Roth, Alexandros Makriyannis, Vsevolod Katritch, Valery V Fokin
Virtual Screening of a Chemically Diverse "Superscaffold" Library Enables Ligand Discovery for a Key GPCR Target. ACS chemical biology 19 (4) (2024)
Katharina Grotsch, Anastasiia V Sadybekov, Sydney Hiller, Saheem Zaidi, Dmitry B Eremin, Austen Le, Yong-Feng Liu, Evan Carlton Smith, Christos Illiopoulis-Tsoutsouvas, Joice Thomas, Shubhangi Aggarwal, Julie E Pickett, Cesar Reyes, Elias Picazo, Bryan L Roth, Alexandros Makriyannis, Vsevolod Katritch, Valery V Fokin
Virtual Screening of a Chemically Diverse "Superscaffold" Library Enables Ligand Discovery for a Key GPCR Target. ACS chemical biology 19 (4) (2024)
Katharina Grotsch, Anastasiia V Sadybekov, Sydney Hiller, Saheem Zaidi, Dmitry B Eremin, Austen Le, Yong-Feng Liu, Evan Carlton Smith, Christos Illiopoulis-Tsoutsouvas, Joice Thomas, Shubhangi Aggarwal, Julie E Pickett, Cesar Reyes, Elias Picazo, Bryan L Roth, Alexandros Makriyannis, Vsevolod Katritch, Valery V Fokin
Virtual Screening of a Chemically Diverse "Superscaffold" Library Enables Ligand Discovery for a Key GPCR Target. ACS chemical biology (2024)
Evangelos Dadiotis, Meng Cui, Maria Gerasi, Vangelis Mitsis, Eleni Melliou, Alexandros Makriyannis, Diomedes E Logothetis, Prokopios Magiatis
A Simple Chiral 1 H NMR Method for the Discrimination of ( R )- and ( S )-Cannabichromene in Complex Natural Mixtures and Their Effects on TRPA1 Activity. Journal of natural products (2023)
Evangelos Dadiotis, Meng Cui, Maria Gerasi, Vangelis Mitsis, Eleni Melliou, Alexandros Makriyannis, Diomedes E Logothetis, Prokopios Magiatis
A Simple Chiral 1 H NMR Method for the Discrimination of ( R )- and ( S )-Cannabichromene in Complex Natural Mixtures and Their Effects on TRPA1 Activity. Journal of natural products 87 (1) (2023)
Evangelos Dadiotis, Meng Cui, Maria Gerasi, Vangelis Mitsis, Eleni Melliou, Alexandros Makriyannis, Diomedes E Logothetis, Prokopios Magiatis
A Simple Chiral 1 H NMR Method for the Discrimination of ( R )- and ( S )-Cannabichromene in Complex Natural Mixtures and Their Effects on TRPA1 Activity. Journal of natural products 87 (1) (2023)
Evangelos Dadiotis, Meng Cui, Maria Gerasi, Vangelis Mitsis, Eleni Melliou, Alexandros Makriyannis, Diomedes E Logothetis, Prokopios Magiatis
A Simple Chiral 1 H NMR Method for the Discrimination of ( R )- and ( S )-Cannabichromene in Complex Natural Mixtures and Their Effects on TRPA1 Activity. Journal of natural products 87 (1) (2023)
Arman A Sadybekov, Anastasiia V Sadybekov, Yong-Feng Liu, Christos Iliopoulos-Tsoutsouvas, Xi-Ping Huang, Julie E Pickett, Blake Houser, Nilkanth Patel, Ngan K Tran, Fei Tong, Nikolai Zvonok, Manish Kumar Jain, Olena Savych, Dmytro S Radchenko, Spyros P Nikas, Nicos A Petasis, Yurii S Moroz, Bryan L Roth, Alexandros Makriyannis, Vsevolod Katritch
Synthon-based ligand discovery in virtual libraries of over 11 billion compounds. Nature 601 (7893) (2021)
Tao Hu, Guoxun Zheng, Dongxiang Xue, Simeng Zhao, Fei Li, Fang Zhou, Fei Zhao, Linshan Xie, Cuiping Tian, Tian Hua, Suwen Zhao, Yueming Xu, Guisheng Zhong, Zhi-Jie Liu, Alexandros Makriyannis, Raymond C Stevens, Houchao Tao
Rational Remodeling of Atypical Scaffolds for the Design of Photoswitchable Cannabinoid Receptor Tools. Journal of medicinal chemistry 64 (18) (2021)
Shan Jiang, Christos Iliopoulos-Tsoutsouvas, Fei Tong, Christina A Brust, Catherine M Keenan, Jimit Girish Raghav, Tian Hua, Simiao Wu, Jo-Hao Ho, Yiran Wu, Travis W Grim, Nikolai Zvonok, Ganesh A Thakur, Zhi-Jie Liu, Keith A Sharkey, Laura M Bohn, Spyros P Nikas, Alexandros Makriyannis
Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists. Journal of medicinal chemistry 64 (7) (2021)
Xiaoyan Wang, Dongsheng Liu, Ling Shen, Fahui Li, Yongze Li, Lingyun Yang, Tiandan Xu, Houchao Tao, Deqiang Yao, Lijie Wu, Kunio Hirata, Laura M Bohn, Alexandros Makriyannis, Xiaohong Liu, Tian Hua, Zhi-Jie Liu, Jiangyun Wang
A Genetically Encoded F-19 NMR Probe Reveals the Allosteric Modulation Mechanism of Cannabinoid Receptor 1. Journal of the American Chemical Society 143 (40) (2021)
Sean B Ogden, Michael S Malamas, Alexandros Makriyannis, Lisa A Eckel
The novel cannabinoid CB1 receptor agonist AM11101 increases food intake in female rats. British journal of pharmacology 176 (20) (2019)
Shivani Sachdev, V Kiran Vemuri, Samuel D Banister, Mitchell Longworth, Michael Kassiou, Marina J Santiago, Alexandros Makriyannis, Mark Connor
In vitro determination of the efficacy of illicit synthetic cannabinoids at CB1 receptors. British journal of pharmacology 176 (24) (2019)
Yingpeng Liu, Lipin Ji, Marsha Eno, Shalley Kudalkar, Ai-Ling Li, Marion Schimpgen, Othman Benchama, Paula Morales, Shu Xu, Dow Hurst, Simiao Wu, Khadijah A Mohammad, JodiAnne T Wood, Nikolai Zvonok, Demetris P Papahatjis, Han Zhou, Chandrashekhar Honrao, Ken Mackie, Patricia Reggio, Andrea G Hohmann, Lawrence J Marnett, Alexandros Makriyannis, Spyros P Nikas
( R)- N-(1-Methyl-2-hydroxyethyl)-13-( S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes. Journal of medicinal chemistry 61 (19) (2018)
Dennis Szymanski, Malvina Papanastasiou, Lakshmipathi Pandarinathan, Nikolai Zvonok, David R Janero, Spiro Pavlopoulos, Paul Vouros, Alexandros Makriyannis
Aliphatic Azides as Selective Cysteine Labeling Reagents for Integral Membrane Proteins. Journal of medicinal chemistry 61 (24) (2018)
Federica Barutta, Stefania Bellini, Raffaella Mastrocola, R Gambino, Fabiana Piscitelli, Vincenzo Di Marzo, Beatrice Corbetta, V Kiran Vemuri, Alexandros Makriyannis, Laura Annaratone, Graziella Bruno, Gabriella Gruden
Reversal of albuminuria by combined AM6545 and perindopril therapy in experimental diabetic nephropathy. British journal of pharmacology 175 (23) (2018)
Thanh C Ho, Naoyuki Shimada, Marcus A Tius, Spyros P Nikas, Wen Zhang, Alexandros Makriyannis
C1'-Azacycloalkyl Hexahydrocannabinols. The Journal of organic chemistry 82 (15) (2017)