Michael Kassiou (M Kassiou)

Loop profile Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 43

Top Topics

Oxide Nanoparticles

Molecularly Imprinted

Structure Activity Relationship

Top Venues

ACS chemical neuroscience

Journal of medicinal chemistry

International journal of molecular sciences

This page only lists publications with an associated author ORCID identifier.

Publications

Eric Sparkes, Callan J Maloney, Jack W Markham, Chianna Dane, Rochelle Boyd, Jayson Gilchrist, Michael Moir, Rebecca Gordon, Jia Lin Luo, Edward Pike, Katelyn A Walker, Michael Kassiou, Iain S McGregor, Richard C Kevin, David E Hibbs, William T Jorgensen, Samuel D Banister, Elizabeth A Cairns, Adam Ametovski
Structure-Activity Relationships, Deuteration, and Fluorination of Synthetic Cannabinoid Receptor Agonists Related to AKB48, 5F-AKB-48, and AFUBIATA. ACS chemical neuroscience (2024)
Eric Sparkes, Callan J Maloney, Jack W Markham, Chianna Dane, Rochelle Boyd, Jayson Gilchrist, Michael Moir, Rebecca Gordon, Jia Lin Luo, Edward Pike, Katelyn A Walker, Michael Kassiou, Iain S McGregor, Richard C Kevin, David E Hibbs, William T Jorgensen, Samuel D Banister, Elizabeth A Cairns, Adam Ametovski
Structure-Activity Relationships, Deuteration, and Fluorination of Synthetic Cannabinoid Receptor Agonists Related to AKB48, 5F-AKB-48, and AFUBIATA. ACS chemical neuroscience 15 (11) (2024)
Taylor R Garrett, Jayson Gilchrist, Andre D J McKenzie, Fayaz Ali Larik, Jonathan J Danon, Eryn L Werry, Michael Kassiou
An Investigation on Linker Modifications of Cyanoguanidine-Based P2X7 Receptor Antagonists. ChemMedChem 19 (17) (2024)
Taylor R Garrett, Jayson Gilchrist, Andre D J McKenzie, Fayaz Ali Larik, Jonathan J Danon, Eryn L Werry, Michael Kassiou
An Investigation on Linker Modifications of Cyanoguanidine-Based P2X7 Receptor Antagonists. ChemMedChem (2024)
Taylor R Garrett, Jayson Gilchrist, Andre D J McKenzie, Fayaz Ali Larik, Jonathan J Danon, Eryn L Werry, Michael Kassiou
An Investigation on Linker Modifications of Cyanoguanidine-Based P2X7 Receptor Antagonists. ChemMedChem 19 (17) (2024)
Eric Sparkes, Callan J Maloney, Jack W Markham, Chianna Dane, Rochelle Boyd, Jayson Gilchrist, Michael Moir, Rebecca Gordon, Jia Lin Luo, Edward Pike, Katelyn A Walker, Michael Kassiou, Iain S McGregor, Richard C Kevin, David E Hibbs, William T Jorgensen, Samuel D Banister, Elizabeth A Cairns, Adam Ametovski
Structure-Activity Relationships, Deuteration, and Fluorination of Synthetic Cannabinoid Receptor Agonists Related to AKB48, 5F-AKB-48, and AFUBIATA. ACS chemical neuroscience 15 (11) (2024)
Eric Sparkes, Callan J Maloney, Jack W Markham, Chianna Dane, Rochelle Boyd, Jayson Gilchrist, Michael Moir, Rebecca Gordon, Jia Lin Luo, Edward Pike, Katelyn A Walker, Michael Kassiou, Iain S McGregor, Richard C Kevin, David E Hibbs, William T Jorgensen, Samuel D Banister, Elizabeth A Cairns, Adam Ametovski
Structure-Activity Relationships, Deuteration, and Fluorination of Synthetic Cannabinoid Receptor Agonists Related to AKB48, 5F-AKB-48, and AFUBIATA. ACS chemical neuroscience 15 (11) (2024)
Nathan J Castellino, Andrew P Montgomery, Jonathan J Danon, Michael Kassiou
Late-stage Functionalization for Improving Drug-like Molecular Properties. Chemical reviews (2023)
Weiqian E Lee, Marie Besnier, Elijah Genetzakis, Owen Tang, Katharine A Kott, Stephen T Vernon, Michael P Gray, Stuart M Grieve, Michael Kassiou, Gemma A Figtree
High-Throughput Measure of Mitochondrial Superoxide Levels as a Marker of Coronary Artery Disease to Accelerate Drug Translation in Patient-Derived Endothelial Cells Using Opera Phenix ® Technology. International journal of molecular sciences 25 (1) (2023)
Annukka Kallinen, Karine Mardon, Samuel Lane, Andrew P Montgomery, Rajiv Bhalla, Damion H R Stimson, Muneer Ahamed, Gary J Cowin, David E Hibbs, Eryn L Werry, Roger R Fulton, Mark Connor, Michael Kassiou
Synthesis and Preclinical Evaluation of Fluorinated 5-Azaindoles as CB2 PET Radioligands. ACS chemical neuroscience (2023)
Weiqian E Lee, Marie Besnier, Elijah Genetzakis, Owen Tang, Katharine A Kott, Stephen T Vernon, Michael P Gray, Stuart M Grieve, Michael Kassiou, Gemma A Figtree
High-Throughput Measure of Mitochondrial Superoxide Levels as a Marker of Coronary Artery Disease to Accelerate Drug Translation in Patient-Derived Endothelial Cells Using Opera Phenix ® Technology. International journal of molecular sciences 25 (1) (2023)
Weiqian E Lee, Marie Besnier, Elijah Genetzakis, Owen Tang, Katharine A Kott, Stephen T Vernon, Michael P Gray, Stuart M Grieve, Michael Kassiou, Gemma A Figtree
High-Throughput Measure of Mitochondrial Superoxide Levels as a Marker of Coronary Artery Disease to Accelerate Drug Translation in Patient-Derived Endothelial Cells Using Opera Phenix ® Technology. International journal of molecular sciences 25 (1) (2023)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience 14 (1) (2022)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience (2022)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience 14 (1) (2022)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience 14 (1) (2022)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience 14 (1) (2022)
Timothy B Callis, Taylor R Garrett, Andrew P Montgomery, Jonathan J Danon, Michael Kassiou
Recent Scaffold Hopping Applications in Central Nervous System Drug Discovery. Journal of medicinal chemistry 65 (20) (2022)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience 14 (1) (2022)
André D J Mckenzie, Taylor R Garrett, Eryn L Werry, Michael Kassiou
Purinergic P2X 7 Receptor: A Therapeutic Target in Amyotrophic Lateral Sclerosis. ACS chemical neuroscience 13 (10) (2022)
Prita R Asih, Anne Poljak, Michael Kassiou, Yazi D Ke, Lars M Ittner
Differential mitochondrial protein interaction profile between human translocator protein and its A147T polymorphism variant. PloS one 17 (5) (2022)
Sarah R Ball, Julius S P Adamson, Michael A Sullivan, Manuela R Zimmermann, Victor Lo, Maximo Sanz-Hernandez, Xiaofan Jiang, Ann H Kwan, André D J Mckenzie, Eryn L Werry, Tuomas P J Knowles, Michael Kassiou, Georg Meisl, Matthew H Todd, Peter J Rutledge, Margaret Sunde
Perphenazine-Macrocycle Conjugates Rapidly Sequester the Aβ42 Monomer and Prevent Formation of Toxic Oligomers and Amyloid. ACS chemical neuroscience 14 (1) (2022)
Ariadna Recasens, Sean J Humphrey, Michael Ellis, Monira Hoque, Ramzi H Abbassi, Brianna Chen, Mitchell Longworth, Elise J Needham, David E James, Terrance G Johns, Bryan W Day, Michael Kassiou, Pengyi Yang, Lenka Munoz
Global phosphoproteomics reveals DYRK1A regulates CDK1 activity in glioblastoma cells. Cell death discovery 7 (1) (2021)
Shahinda S R Alsayed, Amreena Suri, Anders W Bailey, Samuel Lane, Eryn L Werry, Chiang-Ching Huang, Li-Fang Yu, Michael Kassiou, Simone Treiger Sredni, Hendra Gunosewoyo
Synthesis and antitumour evaluation of indole-2-carboxamides against paediatric brain cancer cells. RSC medicinal chemistry 12 (11) (2021)
Philip Ryan, Ming-Ming Xu, Kousar Jahan, Andrew K Davey, Prasad V Bharatam, Shailendra Anoopkumar-Dukie, Michael Kassiou, George D Mellick, Santosh Rudrawar
Novel Furan-2-yl-1H-pyrazoles Possess Inhibitory Activity against α-Synuclein Aggregation. ACS chemical neuroscience 11 (15) (2020)
Sophie V Vo, Samuel D Banister, Isaac Freelander, Eryn L Werry, Tristan A Reekie, Lars M Ittner, Michael Kassiou
Reversing binding sensitivity to A147T translocator protein. RSC medicinal chemistry 11 (4) (2020)
Alexander Gillis, Arisbel B Gondin, Andrea Kliewer, Julie Sanchez, Herman D Lim, Claudia Alamein, Preeti Manandhar, Marina J Santiago, Sebastian Fritzwanker, Frank Schmiedel, Timothy A Katte, Tristan A Reekie, Natasha L Grimsey, Michael Kassiou, Barrie Kellam, Cornelius Krasel, Michelle L Halls, Mark Connor, J Robert Lane, Stefan Schulz, Macdonald J Christie, Meritxell Canals
Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists. Science signaling 13 (625) (2020)
Agnieszka Pyrczak-Felczykowska, Rajeshwar Narlawar, Anna Pawlik, Beata Guzow-Krzemińska, Damian Artymiuk, Aleksandra Hać, Kamil Ryś, Louis M Rendina, Tristan A Reekie, Anna Herman-Antosiewicz, Michael Kassiou
Correction to Synthesis of Usnic Acid Derivatives and Evaluation of Their Antiproliferative Activity against Cancer Cells. Journal of natural products 83 (2) (2020)
Natalie B Vinh, Nyssa Drinkwater, Tess R Malcolm, Michael Kassiou, Leonardo Lucantoni, Peter M Grin, Georgina S Butler, Sandra Duffy, Christopher M Overall, Vicky M Avery, Peter J Scammells, Sheena McGowan
Hydroxamic Acid Inhibitors Provide Cross-Species Inhibition of Plasmodium M1 and M17 Aminopeptidases. Journal of medicinal chemistry 62 (2) (2019)
Shivani Sachdev, V Kiran Vemuri, Samuel D Banister, Mitchell Longworth, Michael Kassiou, Marina J Santiago, Alexandros Makriyannis, Mark Connor
In vitro determination of the efficacy of illicit synthetic cannabinoids at CB1 receptors. British journal of pharmacology 176 (24) (2019)
Agnieszka Pyrczak-Felczykowska, Rajeshwar Narlawar, Anna Pawlik, Beata Guzow-Krzemińska, Damian Artymiuk, Aleksandra Hać, Kamil Ryś, Louis M Rendina, Tristan A Reekie, Anna Herman-Antosiewicz, Michael Kassiou
Synthesis of Usnic Acid Derivatives and Evaluation of Their Antiproliferative Activity against Cancer Cells. Journal of natural products 82 (7) (2019)
Philip Ryan, Ming-Ming Xu, Andrew K Davey, Jonathan J Danon, George D Mellick, Michael Kassiou, Santosh Rudrawar
O-GlcNAc Modification Protects against Protein Misfolding and Aggregation in Neurodegenerative Disease. ACS chemical neuroscience 10 (5) (2019)
Hei Wun Alison Cheng, Renee Sokias, Eryn L Werry, Lars M Ittner, Tristan A Reekie, Jonathan J Du, Quanqing Gao, David E Hibbs, Michael Kassiou
First Nondiscriminating Translocator Protein Ligands Produced from a Carbazole Scaffold. Journal of medicinal chemistry 62 (17) (2019)
Annukka Kallinen, Rochelle Boyd, Samuel Lane, Rajiv Bhalla, Karine Mardon, Damion H R Stimson, Eryn L Werry, Roger Fulton, Mark Connor, Michael Kassiou
Synthesis and in vitro evaluation of fluorine-18 benzimidazole sulfones as CB2 PET-radioligands. Organic & biomolecular chemistry 17 (20) (2019)
Tristan A Reekie, Craig M Williams, Louis M Rendina, Michael Kassiou
Cubanes in Medicinal Chemistry. Journal of medicinal chemistry 62 (3) (2018)
Philip Ryan, Bhautikkumar Patel, Vivek Makwana, Hemant R Jadhav, Milton Kiefel, Andrew Davey, Tristan A Reekie, Santosh Rudrawar, Michael Kassiou
Peptides, Peptidomimetics, and Carbohydrate-Peptide Conjugates as Amyloidogenic Aggregation Inhibitors for Alzheimer's Disease. ACS chemical neuroscience 9 (7) (2018)
Tristan A Reekie, Shane M Wilkinson, Vivian Law, David E Hibbs, Jennifer A Ong, Michael Kassiou
Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores. Organic & biomolecular chemistry 15 (3) (2018)
Sook Wern Chua, Alberto Cornejo, Janet van Eersel, Claire H Stevens, Inmaculada Vaca, Mercedes Cueto, Michael Kassiou, Amadeus Gladbach, Alex Macmillan, Lev Lewis, Renee Whan, Lars M Ittner
The Polyphenol Altenusin Inhibits in Vitro Fibrillization of Tau and Reduces Induced Tau Pathology in Primary Neurons. ACS chemical neuroscience 8 (4) (2017)
Shane M Wilkinson, Melissa L Barron, James O'Brien-Brown, Bieneke Janssen, Leanne Stokes, Eryn L Werry, Mansoor Chishty, Kristen K Skarratt, Jennifer A Ong, David E Hibbs, Danielle J Vugts, Stephen Fuller, Albert D Windhorst, Michael Kassiou
Pharmacological Evaluation of Novel Bioisosteres of an Adamantanyl Benzamide P2X7 Receptor Antagonist. ACS chemical neuroscience 8 (11) (2017)
Mitchell Longworth, Mark Connor, Samuel D Banister, Michael Kassiou
Synthesis and Pharmacological Profiling of the Metabolites of Synthetic Cannabinoid Drugs APICA, STS-135, ADB-PINACA, and 5F-ADB-PINACA. ACS chemical neuroscience 8 (8) (2017)
Mitchell Longworth, Samuel D Banister, Rochelle Boyd, Richard C Kevin, Mark Connor, Iain S McGregor, Michael Kassiou
Pharmacology of Cumyl-Carboxamide Synthetic Cannabinoid New Psychoactive Substances (NPS) CUMYL-BICA, CUMYL-PICA, CUMYL-5F-PICA, CUMYL-5F-PINACA, and Their Analogues. ACS chemical neuroscience 8 (10) (2017)
Qingqing Zhou, Athena F Phoa, Ramzi H Abbassi, Monira Hoque, Tristan A Reekie, Josep S Font, Renae M Ryan, Brett W Stringer, Bryan W Day, Terrance G Johns, Lenka Munoz, Michael Kassiou
Structural Optimization and Pharmacological Evaluation of Inhibitors Targeting Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases (DYRK) and CDC-like kinases (CLK) in Glioblastoma. Journal of medicinal chemistry 60 (5) (2017)
M Moir, S W Chua, T Reekie, Adam D Martin, A Ittner, L M Ittner, Michael Kassiou
Ring-opened aminothienopyridazines as novel tau aggregation inhibitors. MedChemComm 8 (6) (2017)