Dimitrios-Ilias Balourdas

Publication Activity (10 Years)

Years Active: 2022-2024
Publications (10 Years): 21

Top Topics

Transcription Factor

Photodynamic Therapy

Top Venues

Journal of medicinal chemistry

ACS chemical biology

Cell death & disease

Bioconjugate chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Marcel Rak, Amelie Menge, Roberta Tesch, Lena M Berger, Dimitrios-Ilias Balourdas, Ekaterina Shevchenko, Andreas Krämer, Lewis Elson, Benedict-Tilmann Berger, Ismahan Abdi, Laurenz M Wahl, Antti Poso, Astrid Kaiser, Thomas Hanke, Thales Kronenberger, Andreas C Joerger, Susanne Müller, Stefan Knapp
Development of Selective Pyrido[2,3- d ]pyrimidin-7(8 H )-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors. Journal of medicinal chemistry 67 (5) (2024)
Fernando H de Souza Gama, Luiz A Dutra, Michael Hawgood, Caio Vinícius Dos Reis, Ricardo A M Serafim, Marcos A Ferreira, Bruno V M Teodoro, Jéssica Emi Takarada, André da Silva Santiago, Dimitrios-Ilias Balourdas, Ann-Sofie Nilsson, Bruno Urien, Vitor M Almeida, Carina Gileadi, Priscila Z Ramos, Anita Salmazo, Stanley N S Vasconcelos, Micael Rodrigues Cunha, Susanne Müller, Stefan Knapp, Katlin Brauer Massirer, Jonathan M Elkins, Opher Gileadi, Alessandra Mascarello, Bennie B L G Lemmens, Cristiano R W Guimarães, Hatylas Azevedo, Rafael Miguez Couñago
Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1δ/ε. Journal of medicinal chemistry 67 (11) (2024)
Marcel Rak, Amelie Menge, Roberta Tesch, Lena M Berger, Dimitrios-Ilias Balourdas, Ekaterina Shevchenko, Andreas Krämer, Lewis Elson, Benedict-Tilmann Berger, Ismahan Abdi, Laurenz M Wahl, Antti Poso, Astrid Kaiser, Thomas Hanke, Thales Kronenberger, Andreas C Joerger, Susanne Müller, Stefan Knapp
Development of Selective Pyrido[2,3- d ]pyrimidin-7(8 H )-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors. Journal of medicinal chemistry (2024)
Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R Schneider, Xin Zhang, Lena Marie Berger, Benedict-Tilmann Berger, Martin Peter Schwalm, Nick A Klopp, Jens T Siveke, Stefan Knapp, Andreas C Joerger
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization. ACS chemical biology (2024)
Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R Schneider, Xin Zhang, Lena Marie Berger, Benedict-Tilmann Berger, Martin Peter Schwalm, Nick A Klopp, Jens T Siveke, Stefan Knapp, Andreas C Joerger
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization. ACS chemical biology 19 (2) (2024)
Dimitrios-Ilias Balourdas, Anja M Markl, Andreas Krämer, Giovanni Settanni, Andreas C Joerger
Structural basis of p53 inactivation by cavity-creating cancer mutations and its implications for the development of mutant p53 reactivators. Cell death & disease 15 (6) (2024)
Fernando H de Souza Gama, Luiz A Dutra, Michael Hawgood, Caio Vinícius Dos Reis, Ricardo A M Serafim, Marcos A Ferreira, Bruno V M Teodoro, Jéssica Emi Takarada, André da Silva Santiago, Dimitrios-Ilias Balourdas, Ann-Sofie Nilsson, Bruno Urien, Vitor M Almeida, Carina Gileadi, Priscila Z Ramos, Anita Salmazo, Stanley N S Vasconcelos, Micael Rodrigues Cunha, Susanne Müller, Stefan Knapp, Katlin Brauer Massirer, Jonathan M Elkins, Opher Gileadi, Alessandra Mascarello, Bennie B L G Lemmens, Cristiano R W Guimarães, Hatylas Azevedo, Rafael Miguez Couñago
Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1δ/ε. Journal of medicinal chemistry (2024)
Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R Schneider, Xin Zhang, Lena Marie Berger, Benedict-Tilmann Berger, Martin Peter Schwalm, Nick A Klopp, Jens T Siveke, Stefan Knapp, Andreas C Joerger
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization. ACS chemical biology 19 (2) (2024)
Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R Schneider, Xin Zhang, Lena Marie Berger, Benedict-Tilmann Berger, Martin Peter Schwalm, Nick A Klopp, Jens T Siveke, Stefan Knapp, Andreas C Joerger
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization. ACS chemical biology 19 (2) (2024)
Dimitrios-Ilias Balourdas, Anja M Markl, Andreas Krämer, Giovanni Settanni, Andreas C Joerger
Structural basis of p53 inactivation by cavity-creating cancer mutations and its implications for the development of mutant p53 reactivators. Cell death & disease 15 (6) (2024)
Dimitrios-Ilias Balourdas, Anja M Markl, Andreas Krämer, Giovanni Settanni, Andreas C Joerger
Structural basis of p53 inactivation by cavity-creating cancer mutations and its implications for the development of mutant p53 reactivators. Cell death & disease 15 (6) (2024)
Marcel Rak, Amelie Menge, Roberta Tesch, Lena M Berger, Dimitrios-Ilias Balourdas, Ekaterina Shevchenko, Andreas Krämer, Lewis Elson, Benedict-Tilmann Berger, Ismahan Abdi, Laurenz M Wahl, Antti Poso, Astrid Kaiser, Thomas Hanke, Thales Kronenberger, Andreas C Joerger, Susanne Müller, Stefan Knapp
Development of Selective Pyrido[2,3- d ]pyrimidin-7(8 H )-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors. Journal of medicinal chemistry 67 (5) (2024)
Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R Schneider, Xin Zhang, Lena Marie Berger, Benedict-Tilmann Berger, Martin Peter Schwalm, Nick A Klopp, Jens T Siveke, Stefan Knapp, Andreas C Joerger
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization. ACS chemical biology 19 (2) (2024)
Dimitrios-Ilias Balourdas, Anja M Markl, Andreas Krämer, Giovanni Settanni, Andreas C Joerger
Structural basis of p53 inactivation by cavity-creating cancer mutations and its implications for the development of mutant p53 reactivators. Cell death & disease 15 (6) (2024)
Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R Schneider, Xin Zhang, Lena Marie Berger, Benedict-Tilmann Berger, Martin Peter Schwalm, Nick A Klopp, Jens T Siveke, Stefan Knapp, Andreas C Joerger
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization. ACS chemical biology 19 (2) (2024)
Jennifer Alisa Amrhein, Lena Marie Berger, Dimitrios-Ilias Balourdas, Andreas C Joerger, Amelie Menge, Andreas Krämer, Julia Marie Frischkorn, Benedict-Tilmann Berger, Lewis Elson, Astrid Kaiser, Manfred Schubert-Zsilavecz, Susanne Müller, Stefan Knapp, Thomas Hanke
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3. Journal of medicinal chemistry (2023)
Jennifer Alisa Amrhein, Lena Marie Berger, Dimitrios-Ilias Balourdas, Andreas C Joerger, Amelie Menge, Andreas Krämer, Julia Marie Frischkorn, Benedict-Tilmann Berger, Lewis Elson, Astrid Kaiser, Manfred Schubert-Zsilavecz, Susanne Müller, Stefan Knapp, Thomas Hanke
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3. Journal of medicinal chemistry 67 (1) (2023)
Jennifer Alisa Amrhein, Lena Marie Berger, Dimitrios-Ilias Balourdas, Andreas C Joerger, Amelie Menge, Andreas Krämer, Julia Marie Frischkorn, Benedict-Tilmann Berger, Lewis Elson, Astrid Kaiser, Manfred Schubert-Zsilavecz, Susanne Müller, Stefan Knapp, Thomas Hanke
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3. Journal of medicinal chemistry 67 (1) (2023)
Maëva M Pichon, Dawid Drelinkiewicz, David Lozano, Ruxandra Moraru, Laura J Hayward, Megan Jones, Michael A McCoy, Samuel Allstrum-Graves, Dimitrios-Ilias Balourdas, Andreas C Joerger, Richard J Whitby, Stephen Michael Goldup, Neil Wells, Graham J Langley, Julie M Herniman, Matthias G J Baud
Structure-Reactivity Studies of 2-Sulfonylpyrimidines Allow Selective Protein Arylation. Bioconjugate chemistry (2023)
Jennifer Alisa Amrhein, Lena Marie Berger, Dimitrios-Ilias Balourdas, Andreas C Joerger, Amelie Menge, Andreas Krämer, Julia Marie Frischkorn, Benedict-Tilmann Berger, Lewis Elson, Astrid Kaiser, Manfred Schubert-Zsilavecz, Susanne Müller, Stefan Knapp, Thomas Hanke
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3. Journal of medicinal chemistry 67 (1) (2023)
Qiang Zhang, Dimitrios-Ilias Balourdas, Bruno Baron, Alon Senitzki, Tali E Haran, Klas G Wiman, Thierry Soussi, Andreas C Joerger
Evolutionary history of the p53 family DNA-binding domain: insights from an Alvinella pompejana homolog. Cell death & disease 13 (3) (2022)