Ganesha Rai

ORCID

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 21

Top Venues

ACS pharmacology & translational science

Journal of medicinal chemistry

ACS chemical biology

Assay and drug development technologies

National Institutes of Health (PHD)

This page only lists publications with an associated author ORCID identifier.

Education History

National Institutes of Health Aug 02 2006

United States

PHD :: NCATS

Publications

Kalyan Golla, Adam Yasgar, Voddarahally N Manjuprasanna, Meghna U Naik, Bolormaa Baljinnyam, Alexey V Zakharov, Sankalp Jain, Ganesha Rai, Ajit Jadhav, Anton Simeonov, Ulhas P Naik
Small-Molecule Disruptors of the Interaction between Calcium- and Integrin-Binding Protein 1 and Integrin α IIb β 3 as Novel Antiplatelet Agents. ACS pharmacology & translational science 7 (7) (2024)
Megan N Doleschal, Jenna Miller, Sankalp Jain, Alexey V Zakharov, Ganesha Rai, Anton Simeonov, Bolormaa Baljinnyam, Zhihao Zhuang
Cell-Based Covalent-Capture Deubiquitinase Assay for Inhibitor Discovery. ACS pharmacology & translational science 7 (9) (2024)
Kalyan Golla, Adam Yasgar, Voddarahally N Manjuprasanna, Meghna U Naik, Bolormaa Baljinnyam, Alexey V Zakharov, Sankalp Jain, Ganesha Rai, Ajit Jadhav, Anton Simeonov, Ulhas P Naik
Small-Molecule Disruptors of the Interaction between Calcium- and Integrin-Binding Protein 1 and Integrin α IIb β 3 as Novel Antiplatelet Agents. ACS pharmacology & translational science 7 (7) (2024)
Vinicius M Alves, Adam Yasgar, James Wellnitz, Ganesha Rai, Marielle Rath, Rodolpho C Braga, Stephen J Capuzzi, Anton Simeonov, Eugene N Muratov, Alexey V Zakharov, Alexander Trospsha
Lies and Liabilities: Computational Assessment of High-Throughput Screening Hits to Identify Artifact Compounds. Journal of medicinal chemistry (2023)
Jung-Eun Park, Hobin Lee, Paola Oliva, Klara Kirsch, Bora Kim, Jong Il Ahn, Celeste N Alverez, Snehal Gaikwad, Kristopher W Krausz, Robert O'Connor, Ganesha Rai, Anton Simeonov, Beverly A Mock, Frank J Gonzalez, Kyung S Lee, Kenneth A Jacobson
Structural Optimization and Anticancer Activity of Polo-like Kinase 1 (Plk1) Polo-Box Domain (PBD) Inhibitors and Their Prodrugs. ACS pharmacology & translational science 6 (3) (2023)
Quinlin M Hanson, Nate Hoxie, Min Shen, Hui Guo, Ig-Jun Cho, Ipsita Chakraborty, Brooklyn M Aragon, Ganesha Rai, Samarjit Patnaik, John S Janiszewski, Matthew D Hall
Target Class Profiling of Small-Molecule Methyltransferases. ACS chemical biology (2023)
Haider H Dar, Karolina Mikulska-Ruminska, Yulia Y Tyurina, Diane K Luci, Adam Yasgar, Svetlana N Samovich, Alexander A Kapralov, Austin B Souryavong, Vladimir A Tyurin, Andrew A Amoscato, Michael W Epperly, Galina V Shurin, Melissa Standley, Theodore R Holman, Claudette M St Croix, Simon C Watkins, Andrew P VanDemark, Sandeep Rana, Alexey V Zakharov, Anton Simeonov, Juan Jose Marugan, Rama K Mallampalli, Sally E Wentzel, Joel S Greenberger, Ganesha Rai, Hülya Bayir, Ivet Bahar, Valerian E Kagan
Discovering selective antiferroptotic inhibitors of the 15LOX/PEBP1 complex noninterfering with biosynthesis of lipid mediators. Proceedings of the National Academy of Sciences of the United States of America 120 (25) (2023)
Pengfei Yu, Shuwen Cao, Shyh-Ming Yang, Ganesha Rai, Natalia J Martinez, Adam Yasgar, Alexey V Zakharov, Anton Simeonov, William A Molina-Arocho, Graham P Lobel, Hesham Mohei, Alexis L Scott, Li Zhai, Emma E Furth, M Celeste Simon, Malay Haldar
RALDH1 inhibition shows immunotherapeutic efficacy in hepatocellular carcinoma. Cancer immunology research (2023)
Jung-Eun Park, Hobin Lee, Paola Oliva, Klara Kirsch, Bora Kim, Jong Il Ahn, Celeste N Alverez, Snehal Gaikwad, Kristopher W Krausz, Robert O'Connor, Ganesha Rai, Anton Simeonov, Beverly A Mock, Frank J Gonzalez, Kyung S Lee, Kenneth A Jacobson
Structural Optimization and Anticancer Activity of Polo-like Kinase 1 (Plk1) Polo-Box Domain (PBD) Inhibitors and Their Prodrugs. ACS pharmacology & translational science 6 (3) (2023)
Joshua E Hochuli, Sankalp Jain, Cleber Melo-Filho, Zoe L Sessions, Tesia Bobrowski, Jun Choe, Johnny Zheng, Richard T Eastman, Daniel C Talley, Ganesha Rai, Anton Simeonov, Alexander Trospsha, Eugene N Muratov, Bolormaa Baljinnyam, Alexey V Zakharov
Allosteric Binders of ACE2 Are Promising Anti-SARS-CoV-2 Agents. ACS pharmacology & translational science 5 (7) (2022)
Guangping Dong, Youchao Deng, Adam Yasgar, Ravi Yadav, Daniel Talley, Alexey V Zakharov, Sankalp Jain, Ganesha Rai, Nicholas Noinaj, Anton Simeonov, Rong Huang
Venglustat Inhibits Protein N-Terminal Methyltransferase 1 in a Substrate-Competitive Manner. Journal of medicinal chemistry 65 (18) (2022)
Tino W Sanchez, Michael H Ronzetti, Ashley E Owens, Maria Antony, Ty Voss, Eric Wallgren, Daniel Talley, Krishna Balakrishnan, Sebastian E Leyes Porello, Ganesha Rai, Juan Jose Marugan, Samuel G Michael, Bolormaa Baljinnyam, Noel T Southall, Anton Simeonov, Mark J Henderson
Real-Time Cellular Thermal Shift Assay to Monitor Target Engagement. ACS chemical biology 17 (9) (2022)
Sankalp Jain, Daniel C Talley, Bolormaa Baljinnyam, Jun Choe, Quinlin Hanson, Wei Zhu, Miao Xu, Catherine Z Chen, Wei Zheng, Xin Hu, Min Shen, Ganesha Rai, Matthew D Hall, Anton Simeonov, Alexey V Zakharov
Hybrid In Silico Approach Reveals Novel Inhibitors of Multiple SARS-CoV-2 Variants. ACS pharmacology & translational science 4 (5) (2021)
Juan Alvarez-Gonzalez, Adam Yasgar, Robert W Maul, Amanda E Rieffer, Daniel J Crawford, Daniel J Salamango, Dorjbal Dorjsuren, Alexey V Zakharov, Daniel J Jansen, Ganesha Rai, Juan Jose Marugan, Anton Simeonov, Reuben S Harris, Rahul M Kohli, Patricia J Gearhart
Small Molecule Inhibitors of Activation-Induced Deaminase Decrease Class Switch Recombination in B Cells. ACS pharmacology & translational science 4 (3) (2021)
Hunter G Larson, Alexey V Zakharov, Sukumar Sarkar, Shyh-Ming Yang, Ganesha Rai, James M Larner, Anton Simeonov, Natalia J Martinez
A Genome-Edited ERα-HiBiT Fusion Reporter Cell Line for the Identification of ERα Modulators Via High-Throughput Screening and CETSA. Assay and drug development technologies 19 (8) (2021)
Natalia J Martinez, John C Braisted, Patricia K Dranchak, John J Moran, Hunter Larson, Bryan Queme, Evgenia Pak, Amalia Dutra, Ganesha Rai, Ken Chih-Chien Cheng, John Svaren, James Inglese
Genome-Edited Coincidence and PMP22-HiBiT Fusion Reporter Cell Lines Enable an Artifact-Suppressive Quantitative High-Throughput Screening Strategy for PMP22 Gene-Dosage Disorder Drug Discovery. ACS pharmacology & translational science 4 (4) (2021)
Celeste N Alverez, Jung-Eun Park, Kiran S Toti, Yangliu Xia, Kristopher W Krausz, Ganesha Rai, Jeong Kyu Bang, Frank J Gonzalez, Kenneth A Jacobson, Kyung S Lee
Identification of a New Heterocyclic Scaffold for Inhibitors of the Polo-Box Domain of Polo-like Kinase 1. Journal of medicinal chemistry 63 (22) (2020)
Ganesha Rai, Daniel J Urban, Bryan T Mott, Xin Hu, Shyh-Ming Yang, Gloria A Benavides, Michelle S Johnson, Giuseppe L Squadrito, Kyle R Brimacombe, Tobie D Lee, Dorian M Cheff, Hu Zhu, Mark J Henderson, Katherine Pohida, Gary A Sulikowski, David M Dranow, Md Kabir, Pranav Shah, Elias Padilha, Dingyin Tao, Yuhong Fang, Plamen P Christov, Kwangho Kim, Somnath Jana, Pavan Muttil, Tamara Anderson, Nitesh K Kunda, Helen J Hathaway, Donna F Kusewitt, Nobu Oshima, Murali Cherukuri, Douglas R Davies, Jeffrey P Norenberg, Larry A Sklar, William J Moore, Chi V Dang, Gordon M Stott, Leonard Neckers, Andrew J Flint, Victor M Darley-Usmar, Anton Simeonov, Alex G Waterson, Ajit Jadhav, Matthew D Hall, David J Maloney
Pyrazole-Based Lactate Dehydrogenase Inhibitors with Optimized Cell Activity and Pharmacokinetic Properties. Journal of medicinal chemistry 63 (19) (2020)
Vinicius M Alves, Stephen J Capuzzi, Rodolpho C Braga, Daniel Korn, Joshua E Hochuli, Kyle H Bowler, Adam Yasgar, Ganesha Rai, Anton Simeonov, Eugene N Muratov, Alexey V Zakharov, Alexander Trospsha
SCAM Detective: Accurate Predictor of Small, Colloidally Aggregating Molecules. Journal of chemical information and modeling 60 (8) (2020)
John R Horton, Clayton B Woodcock, Qin Chen, Xu Liu, Xing Zhang, John Shanks, Ganesha Rai, Bryan T Mott, Daniel J Jansen, Stephen C Kales, Mark J Henderson, Matthew Cyr, Katherine Pohida, Xin Hu, Pranav Shah, Xin Xu, Ajit Jadhav, David J Maloney, Matthew D Hall, Anton Simeonov, Haian Fu, Paula M Vertino, Xiaodong Cheng
Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A. Journal of medicinal chemistry 61 (23) (2018)
John R Horton, Xu Liu, Lizhen Wu, Kai Zhang, John Shanks, Xing Zhang, Ganesha Rai, Bryan T Mott, Daniel J Jansen, Stephen C Kales, Mark J Henderson, Katherine Pohida, Yuhong Fang, Xin Hu, Ajit Jadhav, David J Maloney, Matthew D Hall, Anton Simeonov, Haian Fu, Paula M Vertino, Qin Yan, Xiaodong Cheng
Insights into the Action of Inhibitor Enantiomers against Histone Lysine Demethylase 5A. Journal of medicinal chemistry 61 (7) (2018)

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Publication Activity (10 Years)

Top Topics

Top Venues

Ganesha Rai