Steffen Pockes

Publication Activity (10 Years)

Years Active: 2019-2024
Publications (10 Years): 30

Top Topics

Structural Basis

Angiotensin Converting Enzyme

Top Venues

Journal of medicinal chemistry

ACS applied materials & interfaces

Nature communications

ACS pharmacology & translational science

This page only lists publications with an associated author ORCID identifier.

Publications

Melanie Walter, Merlin Bresinsky, Oliver Zimmer, Steffen Pockes, Achim M Goepferich
Conditional Cell-Penetrating Peptide Exposure as Selective Nanoparticle Uptake Signal. ACS applied materials & interfaces (2024)
Melanie Walter, Merlin Bresinsky, Oliver Zimmer, Steffen Pockes, Achim M Goepferich
Conditional Cell-Penetrating Peptide Exposure as Selective Nanoparticle Uptake Signal. ACS applied materials & interfaces 16 (29) (2024)
Melanie Walter, Merlin Bresinsky, Oliver Zimmer, Steffen Pockes, Achim M Goepferich
Conditional Cell-Penetrating Peptide Exposure as Selective Nanoparticle Uptake Signal. ACS applied materials & interfaces 16 (29) (2024)
Zoe Köck, Kilian Schnelle, Margherita Persechino, Simon Umbach, Hannes Schihada, Dovile Januliene, Kristian Parey, Steffen Pockes, Peter Kolb, Volker Dötsch, Arne Möller, Daniel Hilger, Frank Bernhard
Cryo-EM structure of cell-free synthesized human histamine 2 receptor/G s complex in nanodisc environment. Nature communications 15 (1) (2024)
Melanie Walter, Merlin Bresinsky, Oliver Zimmer, Steffen Pockes, Achim M Goepferich
Conditional Cell-Penetrating Peptide Exposure as Selective Nanoparticle Uptake Signal. ACS applied materials & interfaces 16 (29) (2024)
Melanie Walter, Merlin Bresinsky, Oliver Zimmer, Steffen Pockes, Achim M Goepferich
Conditional Cell-Penetrating Peptide Exposure as Selective Nanoparticle Uptake Signal. ACS applied materials & interfaces 16 (29) (2024)
Denise Mönnich, Laura J Humphrys, Carina Höring, Bradley L Hoare, Lisa Forster, Steffen Pockes
Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology. ACS pharmacology & translational science 7 (3) (2024)
Denise Mönnich, Laura J Humphrys, Carina Höring, Bradley L Hoare, Lisa Forster, Steffen Pockes
Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology. ACS pharmacology & translational science 7 (3) (2024)
Zoe Köck, Kilian Schnelle, Margherita Persechino, Simon Umbach, Hannes Schihada, Dovile Januliene, Kristian Parey, Steffen Pockes, Peter Kolb, Volker Dötsch, Arne Möller, Daniel Hilger, Frank Bernhard
Cryo-EM structure of cell-free synthesized human histamine 2 receptor/G s complex in nanodisc environment. Nature communications 15 (1) (2024)
Zoe Köck, Kilian Schnelle, Margherita Persechino, Simon Umbach, Hannes Schihada, Dovile Januliene, Kristian Parey, Steffen Pockes, Peter Kolb, Volker Dötsch, Arne Möller, Daniel Hilger, Frank Bernhard
Cryo-EM structure of cell-free synthesized human histamine 2 receptor/G s complex in nanodisc environment. Nature communications 15 (1) (2024)
Katarzyna Szczepańska, Tadeusz Karcz, Maria Dichiara, Szczepan Mogilski, Justyna Kalinowska-Tłuścik, Bogusław Pilarski, Arkadiusz Leniak, Wojciech Pietruś, Sabina Podlewska, Katarzyna Popiołek-Barczyk, Laura J Humphrys, Ma Carmen Ruiz Cantero, David Reiner-Link, Luisa Leitzbach, Dorota Łażewska, Steffen Pockes, Michał Górka, Adam Zmysłowski, Thierry Calmels, Enrique J Cobos, Agostino Marrazzo, Holger Stark, Andrzej J Bojarski, Emanuele Amata, Katarzyna Kieć-Kononowicz
Dual Piperidine-Based Histamine H 3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain. Journal of medicinal chemistry (2023)
Niklas Rosier, Denise Mönnich, Martin Nagl, Hannes Schihada, Alexei Sirbu, Nergis Konar, Irene Reyes-Resina, Gemma Navarro, Rafael Franco, Peter Kolb, Paolo Annibale, Steffen Pockes
Shedding Light on the D 1 -Like Receptors: A Fluorescence-Based Toolbox for Visualization of the D 1 and D 5 Receptors. Chembiochem : a European journal of chemical biology (2023)
Merlin Bresinsky, Aida Shahraki, Peter Kolb, Steffen Pockes, Hannes Schihada
Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3. Journal of medicinal chemistry (2023)
Denise Mönnich, Martin Nagl, Lisa Forster, Niklas Rosier, Patrick Igel, Steffen Pockes
Discovery of a Tritiated Radioligand with High Affinity and Selectivity for the Histamine H 3 Receptor. ACS medicinal chemistry letters 14 (11) (2023)
Gurpreet Singh, Peng Liu, Katherine R Yao, Jessica M Strasser, Chris Hlynialuk, Kailee Leinonen-Wright, Peter J Teravskis, Jessica M Choquette, Junaid Ikramuddin, Merlin Bresinsky, Kathryn M Nelson, Dezhi Liao, Karen H Ashe, Michael A Walters, Steffen Pockes
Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy. ACS chemical neuroscience 13 (10) (2022)
Merlin Bresinsky, Jessica M Strasser, Alexander Hubmann, Bernadette Vallaster, William M McCue, Jessica Fuller, Gurpreet Singh, Kathryn M Nelson, Matthew E Cuellar, Barry C Finzel, Karen H Ashe, Michael A Walters, Steffen Pockes
Characterization of caspase-2 inhibitors based on specific sites of caspase-2-mediated proteolysis. Archiv der Pharmazie 355 (9) (2022)
Merlin Bresinsky, Jessica M Strasser, Bernadette Vallaster, Peng Liu, William M McCue, Jessica L Fuller, Alexander Hubmann, Gurpreet Singh, Kathryn M Nelson, Matthew E Cuellar, Carrie M Wilmot, Barry C Finzel, Karen H Ashe, Michael A Walters, Steffen Pockes
Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314. ACS pharmacology & translational science 5 (1) (2022)
Katharina Tropmann, Merlin Bresinsky, Lisa Forster, Denise Mönnich, Armin Buschauer, Hans-Joachim Wittmann, Harald Hübner, Peter Gmeiner, Steffen Pockes, Andrea Strasser
Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists. Journal of medicinal chemistry 64 (12) (2021)
Lukas Grätz, Katharina Tropmann, Merlin Bresinsky, Christoph Müller, Guenther Bernhardt, Steffen Pockes
Author Correction: NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells. Scientific reports 11 (1) (2021)
Lukas Grätz, Katharina Tropmann, Merlin Bresinsky, Christoph Müller, Guenther Bernhardt, Steffen Pockes
Author Correction: NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells. Scientific reports 11 (1) (2021)
Steffen Pockes, Katharina Tropmann
Histamine H2 receptor radioligands: triumphs and challenges. Future medicinal chemistry 13 (12) (2021)
Katarzyna Szczepańska, Sabina Podlewska, Maria Dichiara, Davide Gentile, Vincenzo Patamia, Niklas Rosier, Denise Mönnich, Ma Carmen Ruiz Cantero, Tadeusz Karcz, Dorota Łażewska, Agata Siwek, Steffen Pockes, Enrique J Cobos, Agostino Marrazzo, Holger Stark, Antonio Rescifina, Andrzej J Bojarski, Emanuele Amata, Katarzyna Kieć-Kononowicz
Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H 3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties. ACS chemical neuroscience 13 (1) (2021)
Niklas Rosier, Lukas Grätz, Hannes Schihada, Jan Möller, Ali Işbilir, Laura J Humphrys, Martin Nagl, Ulla Seibel, Martin J Lohse, Steffen Pockes
A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor. Journal of medicinal chemistry 64 (15) (2021)
Carina Höring, Ulla Seibel-Ehlert, Katharina Tropmann, Lukas Grätz, Denise Mönnich, Sebastian Pitzl, Guenther Bernhardt, Steffen Pockes, Andrea Strasser
A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes. International journal of molecular sciences 21 (22) (2020)
Katharina Tropmann, Carina Höring, Nicole Plank, Steffen Pockes
Discovery of a G Protein-Biased Radioligand for the Histamine H2 Receptor with Reversible Binding Properties. Journal of medicinal chemistry 63 (21) (2020)
Lukas Grätz, Katharina Tropmann, Merlin Bresinsky, Christoph Müller, Guenther Bernhardt, Steffen Pockes
NanoBRET binding assay for histamine H2 receptor ligands using live recombinant HEK293T cells. Scientific reports 10 (1) (2020)
Lisa Forster, Lukas Grätz, Denise Mönnich, Günther Bernhardt, Steffen Pockes
A Split Luciferase Complementation Assay for the Quantification of β-Arrestin2 Recruitment to Dopamine D2-Like Receptors. International journal of molecular sciences 21 (17) (2020)
Beatrice Soliman, Ning Wang, Giuseppe Zagotto, Steffen Pockes
Synthesis and biological evaluation of heteroalicyclic cyanoguanidines at histamine receptors. Archiv der Pharmazie 352 (9) (2019)
Karin Rustler, Steffen Pockes, Burkhard König
Light-Switchable Antagonists for the Histamine H1 Receptor at the Isolated Guinea Pig Ileum. ChemMedChem 14 (6) (2019)
Steffen Pockes, David Wifling, Armin Buschauer, Sigurd Elz
Structure-Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands†. ChemistryOpen 8 (3) (2019)