Michael A Walters

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 24

Top Topics

Plasmodium Falciparum

Lipopolysaccharide Induced

Top Venues

Journal of medicinal chemistry

Nature communications

ACS chemical neuroscience

Scientific reports

This page only lists publications with an associated author ORCID identifier.

Publications

Deepti Mudaliar, Rachel H Mansky, Angel White, Grace Baudhuin, Jon E Hawkinson, Henry L Wong, Michael A Walters, Rocio Gomez-Pastor
Identification of CK2α' selective inhibitors by the screening of an allosteric-kinase-inhibitor-like compound library. bioRxiv : the preprint server for biology (2024)
Deepti Mudaliar, Rachel H Mansky, Angel White, Grace Baudhuin, Jon E Hawkinson, Henry L Wong, Michael A Walters, Rocio Gomez-Pastor
Discovery of a CK2α'-Biased ATP-Competitive Inhibitor from a High-Throughput Screen of an Allosteric-Inhibitor-Like Compound Library. ACS chemical neuroscience 15 (15) (2024)
Deepti Mudaliar, Rachel H Mansky, Angel White, Grace Baudhuin, Jon E Hawkinson, Henry L Wong, Michael A Walters, Rocio Gomez-Pastor
Discovery of a CK2α'-Biased ATP-Competitive Inhibitor from a High-Throughput Screen of an Allosteric-Inhibitor-Like Compound Library. ACS chemical neuroscience (2024)
Deepti Mudaliar, Rachel H Mansky, Angel White, Grace Baudhuin, Jon E Hawkinson, Henry L Wong, Michael A Walters, Rocio Gomez-Pastor
Identification of CK2α' selective inhibitors by the screening of an allosteric-kinase-inhibitor-like compound library. bioRxiv : the preprint server for biology (2024)
Jayme L Dahlin, Bruce K Hua, Beth E Zucconi, Shawn D Nelson, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew E Cuellar, Philip A Cole, Jordan L Meier, Tim Thomas, Jonathan B Baell, Peter J Brown, Michael A Walters, Paul A Clemons, Stuart L Schreiber, Bridget K Wagner
Reference compounds for characterizing cellular injury in high-content cellular morphology assays. Nature communications 14 (1) (2023)
Jayme L Dahlin, Bruce K Hua, Beth E Zucconi, Shawn D Nelson, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew E Cuellar, Philip A Cole, Jordan L Meier, Tim Thomas, Jonathan B Baell, Peter J Brown, Michael A Walters, Paul A Clemons, Stuart L Schreiber, Bridget K Wagner
Reference compounds for characterizing cellular injury in high-content cellular morphology assays. Nature communications 14 (1) (2023)
Jayme L Dahlin, Bruce K Hua, Beth E Zucconi, Shawn D Nelson, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew E Cuellar, Philip A Cole, Jordan L Meier, Tim Thomas, Jonathan B Baell, Peter J Brown, Michael A Walters, Paul A Clemons, Stuart L Schreiber, Bridget K Wagner
Reference compounds for characterizing cellular injury in high-content cellular morphology assays. Nature communications 14 (1) (2023)
Gurpreet Singh, Peng Liu, Katherine R Yao, Jessica M Strasser, Chris Hlynialuk, Kailee Leinonen-Wright, Peter J Teravskis, Jessica M Choquette, Junaid Ikramuddin, Merlin Bresinsky, Kathryn M Nelson, Dezhi Liao, Karen H Ashe, Michael A Walters, Steffen Pockes
Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy. ACS chemical neuroscience 13 (10) (2022)
Merlin Bresinsky, Jessica M Strasser, Bernadette Vallaster, Peng Liu, William M McCue, Jessica L Fuller, Alexander Hubmann, Gurpreet Singh, Kathryn M Nelson, Matthew E Cuellar, Carrie M Wilmot, Barry C Finzel, Karen H Ashe, Michael A Walters, Steffen Pockes
Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314. ACS pharmacology & translational science 5 (1) (2022)
Noah Nathan Kochen, Vivek Vasandani, Darren Seaney, Anil K Pandey, Michael A Walters, Anthony R Braun, Jonathan N Sachs
Threonine Cavities Are Targetable Motifs That Control Alpha-Synuclein Fibril Growth. ACS chemical neuroscience 13 (17) (2022)
Kathryn M Nelson, Michael A Walters
The Communication of Hit Quality Using Natural History Visualizations (NHVs). SLAS discovery : advancing life sciences R & D 26 (7) (2021)
Yiyue Xie, Padmaja Tummala, Aaron J Oakley, Girdhar Singh Deora, Yuji Nakano, Melissa Rooke, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Marco G Casarotto, Philip G Board, Jonathan B Baell
Development of Benzenesulfonamide Derivatives as Potent Glutathione Transferase Omega-1 Inhibitors. Journal of medicinal chemistry 63 (6) (2020)
Daniel L Priebbenow, David J Leaver, Nghi Nguyen, Benjamin Cleary, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, David M Shackleford, Kasiram Katneni, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Ian P Street, Brendon J Monahan, Kate E Jarman, Helene Jousset Sabroux, Hendrik Falk, Matthew C Chung, Stefan J Hermans, Natalie L Downer, Michael W Parker, Anne K Voss, Tim Thomas, Jonathan B Baell
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents. Journal of medicinal chemistry 63 (9) (2020)
Paul A Jackson, Henry A M Schares, Katherine F M Jones, John C Widen, Daniel P Dempe, Francois Grillet, Matthew E Cuellar, Michael A Walters, Daniel A Harki, Kay M Brummond
Synthesis of Guaianolide Analogues with a Tunable α-Methylene-γ-lactam Electrophile and Correlating Bioactivity with Thiol Reactivity. Journal of medicinal chemistry 63 (23) (2020)
Trinh A D Holth, Michael A Walters, Oliver E Hutt, Gunda I Georg
Diversity-Oriented Library Synthesis from Steviol and Isosteviol-Derived Scaffolds. ACS combinatorial science 22 (3) (2020)
Jonathan H Shrimp, Yihang Jing, Supuni Thalalla Gamage, Kathryn M Nelson, Joseph Han, Keri M Bryson, David C Montgomery, Justin M Thomas, Kellie D Nance, Sunny Sharma, Stephen D Fox, Thorkell Andressen, Wilson R Sinclair, Hong Wu, Abdellah Allali-Hassani, Guillermo Senisterra, Masoud Vedadi, Denis Lafontaine, Jayme L Dahlin, Ronen Marmorstein, Michael A Walters, Jordan L Meier
Remodelin Is a Cryptic Assay Interference Chemotype That Does Not Inhibit NAT10-Dependent Cytidine Acetylation. ACS medicinal chemistry letters 12 (6) (2020)
Kathryn M Nelson, Jonathan Bisson, Gurpreet Singh, James G Graham, Shao-Nong Chen, John Brent Friesen, Jayme L Dahlin, Matthias Niemitz, Michael A Walters, Guido F Pauli
The Essential Medicinal Chemistry of Cannabidiol (CBD). Journal of medicinal chemistry 63 (21) (2020)
Karthik Selvaraju, Arjan Mofers, Paola Pellegrini, Johannes Salomonsson, Alexandra Ahlner, Vivian Morad, Ellin-Kristina Hillert, Belen Espinosa, Elias S J Arnér, Lasse Jensen, Jonas Malmström, Maria V Turkina, Padraig D'Arcy, Michael A Walters, Maria Sunnerhagen, Stig Linder
Cytotoxic unsaturated electrophilic compounds commonly target the ubiquitin proteasome system. Scientific reports 9 (1) (2019)
Lian Xue, Da-Hua Shi, Jitendra R Harjani, Fei Huang, Julia G Beveridge, Tamir Dingjan, Kung Ban, Sarah Diab, Sandra Duffy, Leonardo Lucantoni, Sabine Fletcher, Francis C K Chiu, Scott Blundell, Katherine Ellis, Stuart A Ralph, Grennady Wirjanata, Silvia Teguh, Rintis Noviyanti, Marina Chavchich, Darren John Creek, Ric N Price, Jutta Marfurt, Susan A Charman, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Michael D Edstein, Vicky M Avery, Jonathan B Baell
3,3'-Disubstituted 5,5'-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity. Journal of medicinal chemistry 62 (5) (2019)
Darko Bosnakovski, Meiricris T da Silva, Sithara T Sunny, Elizabeth T Ener, Erik A Toso, Ce Yuan, Ziyou Cui, Michael A Walters, Ajit Jadhav, Michael Kyba
A novel P300 inhibitor reverses DUX4-mediated global histone H3 hyperacetylation, target gene expression, and cell death. Science advances 5 (9) (2019)
David J Leaver, Benjamin Cleary, Nghi Nguyen, Daniel L Priebbenow, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, Kasiram Katneni, Matthew Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Ian P Street, Brendon J Monahan, Kate E Jarman, Helene Jousset Sabroux, Hendrik Falk, Matthew C Chung, Stefan J Hermans, Michael W Parker, Tim Thomas, Jonathan B Baell
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A. Journal of medicinal chemistry 62 (15) (2019)
Karthik Selvaraju, Arjan Mofers, Paola Pellegrini, Johannes Salomonsson, Alexandra Ahlner, Vivian Morad, Ellin-Kristina Hillert, Belen Espinosa, Elias S J Arnér, Lasse Jensen, Jonas Malmström, Maria V Turkina, Padraig D'Arcy, Michael A Walters, Maria Sunnerhagen, Stig Linder
Author Correction: Cytotoxic unsaturated electrophilic compounds commonly target the ubiquitin proteasome system. Scientific reports 9 (1) (2019)
Jayme L Dahlin, Kathryn M Nelson, Jessica M Strasser, Dalia Barsyte-Lovejoy, Magdalena M Szewczyk, Shawna Organ, Matthew E Cuellar, Gurpreet Singh, Jonathan H Shrimp, Nghi Nguyen, Jordan L Meier, Cheryl H Arrowsmith, Peter J Brown, Jonathan B Baell, Michael A Walters
Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors. Nature communications 8 (1) (2017)
Deepthi Menon, Ashlee Innes, Aaron J Oakley, Jane E Dahlstrom, Lora M Jensen, Anne Brüstle, Padmaja Tummala, Melissa Rooke, Marco G Casarotto, Jonathan B Baell, Nghi Nguyen, Yiyue Xie, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Gaetan Burgio, Luke A J O'Neill, Philip G Board
GSTO1-1 plays a pro-inflammatory role in models of inflammation, colitis and obesity. Scientific reports 7 (1) (2017)