Elisabetta Chiarparin

ORCID

Publication Activity (10 Years)

Years Active: 2019-2024
Publications (10 Years): 14

Top Venues

Journal of medicinal chemistry

The Journal of organic chemistry

Journal of the American Chemical Society

This page only lists publications with an associated author ORCID identifier.

Publications

Markus Schade, James S Scott, Thomas G Hayhow, Andy Pike, Ina Terstiege, Marie Ahlqvist, Johan R Johansson, Coura R Diene, Charlene Fallan, Amber Y S Balazs, Elisabetta Chiarparin, David Wilson
Structural and Physicochemical Features of Oral PROTACs. Journal of medicinal chemistry 67 (15) (2024)
James M Smith, Bernard Barlaam, David Beattie, Lauren Bradshaw, Ho Man Chan, Elisabetta Chiarparin, Olga Collingwood, Sophie L Cooke, Anna Cronin, Iain Cumming, Emma Dean, Judit É Debreczeni, Iván Del Barco Barrantes, Coura R Diene, Davide Gianni, Carine Guerot, Xiaoxiao Guo, Sinem Guven, Thomas G Hayhow, Ted Hong, Paul D Kemmitt, Gillian M Lamont, Scott Lamont, James T Lynch, Lisa McWilliams, Shaun Moore, Piotr Raubo, Graeme R Robb, James Robinson, James S Scott, Bharath Srinivasan, Oliver Steward, Christopher J Stubbs, Karl Syson, Lixiang Tan, Oliver Turner, Elizabeth Underwood, Jelena Urosevic, Mercedes Vazquez-Chantada, Amy L Whittaker, David M Wilson, Jon J Winter-Holt
Discovery and In Vivo Efficacy of AZ-PRMT5i-1, a Novel PRMT5 Inhibitor with High MTA Cooperativity. Journal of medicinal chemistry 67 (16) (2024)
Markus Schade, James S Scott, Thomas G Hayhow, Andy Pike, Ina Terstiege, Marie Ahlqvist, Johan R Johansson, Coura R Diene, Charlene Fallan, Amber Y S Balazs, Elisabetta Chiarparin, David Wilson
Structural and Physicochemical Features of Oral PROTACs. Journal of medicinal chemistry 67 (15) (2024)
James M Smith, Bernard Barlaam, David Beattie, Lauren Bradshaw, Ho Man Chan, Elisabetta Chiarparin, Olga Collingwood, Sophie L Cooke, Anna Cronin, Iain Cumming, Emma Dean, Judit É Debreczeni, Iván Del Barco Barrantes, Coura R Diene, Davide Gianni, Carine Guerot, Xiaoxiao Guo, Sinem Guven, Thomas G Hayhow, Ted Hong, Paul D Kemmitt, Gillian M Lamont, Scott Lamont, James T Lynch, Lisa McWilliams, Shaun Moore, Piotr Raubo, Graeme R Robb, James Robinson, James S Scott, Bharath Srinivasan, Oliver Steward, Christopher J Stubbs, Karl Syson, Lixiang Tan, Oliver Turner, Elizabeth Underwood, Jelena Urosevic, Mercedes Vazquez-Chantada, Amy L Whittaker, David M Wilson, Jon J Winter-Holt
Discovery and In Vivo Efficacy of AZ-PRMT5i-1, a Novel PRMT5 Inhibitor with High MTA Cooperativity. Journal of medicinal chemistry 67 (16) (2024)
James M Smith, Bernard Barlaam, David Beattie, Lauren Bradshaw, Ho Man Chan, Elisabetta Chiarparin, Olga Collingwood, Sophie L Cooke, Anna Cronin, Iain Cumming, Emma Dean, Judit É Debreczeni, Iván Del Barco Barrantes, Coura R Diene, Davide Gianni, Carine Guerot, Xiaoxiao Guo, Sinem Guven, Thomas G Hayhow, Ted Hong, Paul D Kemmitt, Gillian M Lamont, Scott Lamont, James T Lynch, Lisa McWilliams, Shaun Moore, Piotr Raubo, Graeme R Robb, James Robinson, James S Scott, Bharath Srinivasan, Oliver Steward, Christopher J Stubbs, Karl Syson, Lixiang Tan, Oliver Turner, Elizabeth Underwood, Jelena Urosevic, Mercedes Vazquez-Chantada, Amy L Whittaker, David M Wilson, Jon J Winter-Holt
Discovery and In Vivo Efficacy of AZ-PRMT5i-1, a Novel PRMT5 Inhibitor with High MTA Cooperativity. Journal of medicinal chemistry (2024)
Markus Schade, James S Scott, Thomas G Hayhow, Andy Pike, Ina Terstiege, Marie Ahlqvist, Johan R Johansson, Coura R Diene, Charlene Fallan, Amber Y S Balazs, Elisabetta Chiarparin, David Wilson
Structural and Physicochemical Features of Oral PROTACs. Journal of medicinal chemistry (2024)
Andrea Bertarello, Pierrick Berruyer, Markus Artelsmair, Charles S Elmore, Sepideh Heydarkhan-Hagvall, Markus Schade, Elisabetta Chiarparin, Staffan Schantz, Lyndon Emsley
In-Cell Quantification of Drugs by Magic-Angle Spinning Dynamic Nuclear Polarization NMR. Journal of the American Chemical Society 144 (15) (2022)
Jon J Winter-Holt, Catherine Bardelle, Elisabetta Chiarparin, Ian L Dale, Paul R J Davey, Nichola L Davies, Christopher Denz, Shaun M Fillery, Carine M Guérot, Fujin Han, Samantha J Hughes, Meghana Kulkarni, Zhaoqun Liu, Alexander Milbradt, Thomas A Moss, Huijun Niu, Joe Patel, Alfred A Rabow, Marianne Schimpl, Junjie Shi, Dongqing Sun, Dejian Yang, Sylvie Guichard
Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models. Journal of medicinal chemistry 65 (4) (2022)
Amber Y S Balazs, Rodrigo J Carbajo, Nichola L Davies, Yu Dong, Alexander W Hird, Jeffrey W Johannes, Michelle L Lamb, William McCoull, Piotr Raubo, Graeme R Robb, Martin J Packer, Elisabetta Chiarparin
Correction to "Free Ligand 1D NMR Conformational Signatures To Enhance Structure Based Drug Design of a Mcl-1 Inhibitor (AZD5991) and Other Synthetic Macrocycles". Journal of medicinal chemistry 64 (5) (2021)
Robert I Troup, Benjamin Jeffries, Raphael El-Bekri Saudain, Eleni Georgiou, Johanna Fish, James S Scott, Elisabetta Chiarparin, Charlene Fallan, Bruno Linclau
Skipped Fluorination Motifs: Synthesis of Building Blocks and Comparison of Lipophilicity Trends with Vicinal and Isolated Fluorination Motifs. The Journal of organic chemistry 86 (2) (2021)
Claudia De Fusco, Marianne Schimpl, Ulf Börjesson, Tony Cheung, Iain Collie, Laura Evans, Priyanka Narasimhan, Christopher Stubbs, Mercedes Vazquez-Chantada, David J Wagner, Michael Grondine, Matthew G Sanders, Sharon Tentarelli, Elizabeth Underwood, Argyrides Argyrou, James M Smith, James T Lynch, Elisabetta Chiarparin, Graeme R Robb, Sharan K Bagal, James S Scott
Fragment-Based Design of a Potent MAT2a Inhibitor and in Vivo Evaluation in an MTAP Null Xenograft Model. Journal of medicinal chemistry 64 (10) (2021)
James S Scott, Thomas A Moss, Amber Balazs, Bernard Barlaam, Jason Breed, Rodrigo J Carbajo, Elisabetta Chiarparin, Paul R J Davey, Oona Delpuech, Stephen Fawell, David I Fisher, Sladjana Gagrica, Eric T Gangl, Tyler Grebe, Ryan D Greenwood, Sudhir Hande, Holia Hatoum-Mokdad, Kara Herlihy, Samantha Hughes, Thomas A Hunt, Hoan Huynh, Sophie L M Janbon, Tony Johnson, Stefan Kavanagh, Teresa Klinowska, Mandy Lawson, Andrew S Lister, Stacey Marden, Dermot F McGinnity, Christopher J Morrow, J Willem M Nissink, Daniel H O' Donovan, Bo Peng, Radoslaw Polanski, Darren S Stead, Stephen Stokes, Kumar Thakur, Scott R Throner, Michael J Tucker, Jeffrey Varnes, Haixia Wang, David M Wilson, Dedong Wu, Ye Wu, Bin Yang, Wenzhan Yang
Discovery of AZD9833, a Potent and Orally Bioavailable Selective Estrogen Receptor Degrader and Antagonist. Journal of medicinal chemistry 63 (23) (2020)
Benjamin Jeffries, Zhong Wang, Hannah R Felstead, Jean-Yves Le Questel, James S Scott, Elisabetta Chiarparin, Jérôme Graton, Bruno Linclau
Systematic Investigation of Lipophilicity Modulation by Aliphatic Fluorination Motifs. Journal of medicinal chemistry 63 (3) (2020)
Amber Y S Balazs, Rodrigo J Carbajo, Nichola L Davies, Yu Dong, Alexander W Hird, Jeffrey W Johannes, Michelle L Lamb, William McCoull, Piotr Raubo, Graeme R Robb, Martin J Packer, Elisabetta Chiarparin
Free Ligand 1D NMR Conformational Signatures To Enhance Structure Based Drug Design of a Mcl-1 Inhibitor (AZD5991) and Other Synthetic Macrocycles. Journal of medicinal chemistry 62 (21) (2019)

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Publication Activity (10 Years)

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Elisabetta Chiarparin