Martyna Szpakowska

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2020-2024
Publications (10 Years): 27

Top Topics

Chronic Lymphocytic Leukemia

Emergency Department

Top Venues

Nature communications

Journal of medicinal chemistry

This page only lists publications with an associated author ORCID identifier.

Publications

Alp Bayrak, Martyna Szpakowska, Valerie Dicenta, Manuel Counson, Alexander Rasch, Anne-Katrin Rohlfing, Andy Chevigné, Meinrad Gawaz, Stefan A Laufer, Thanigaimalai Pillaiyar
Novel Small-Molecule Atypical Chemokine Receptor 3 Agonists: Design, Synthesis, and Pharmacological Evaluation for Antiplatelet Therapy. Journal of medicinal chemistry 67 (16) (2024)
Alp Bayrak, Martyna Szpakowska, Valerie Dicenta, Manuel Counson, Alexander Rasch, Anne-Katrin Rohlfing, Andy Chevigné, Meinrad Gawaz, Stefan A Laufer, Thanigaimalai Pillaiyar
Novel Small-Molecule Atypical Chemokine Receptor 3 Agonists: Design, Synthesis, and Pharmacological Evaluation for Antiplatelet Therapy. Journal of medicinal chemistry (2024)
Alp Bayrak, Martyna Szpakowska, Valerie Dicenta, Manuel Counson, Alexander Rasch, Anne-Katrin Rohlfing, Andy Chevigné, Meinrad Gawaz, Stefan A Laufer, Thanigaimalai Pillaiyar
Novel Small-Molecule Atypical Chemokine Receptor 3 Agonists: Design, Synthesis, and Pharmacological Evaluation for Antiplatelet Therapy. Journal of medicinal chemistry 67 (16) (2024)
Lara Toy, Max E Huber, Minhee Lee, Ana Alonso Bartolomé, Natalia V Ortiz Zacarías, Sherif Nasser, Stephan Scholl, Darius P Zlotos, Yasmine M Mandour, Laura H Heitman, Martyna Szpakowska, Andy Chevigné, Matthias Schiedel
Fluorophore-Labeled Pyrrolones Targeting the Intracellular Allosteric Binding Site of the Chemokine Receptor CCR1. ACS pharmacology & translational science 7 (7) (2024)
Lara Toy, Max E Huber, Minhee Lee, Ana Alonso Bartolomé, Natalia V Ortiz Zacarías, Sherif Nasser, Stephan Scholl, Darius P Zlotos, Yasmine M Mandour, Laura H Heitman, Martyna Szpakowska, Andy Chevigné, Matthias Schiedel
Fluorophore-Labeled Pyrrolones Targeting the Intracellular Allosteric Binding Site of the Chemokine Receptor CCR1. ACS pharmacology & translational science 7 (7) (2024)
Aurelien M Zarca, Ilze Adlere, Cristina P Viciano, Marta Arimont-Segura, Max Meyrath, Icaro A Simon, Jan Paul Bebelman, Dennis Laan, Hans G J Custers, Elwin Janssen, Kobus L Versteegh, Maurice C M L Buzink, Desislava N Nesheva, Reggie Bosma, Iwan J P de Esch, Henry F Vischer, Maikel Wijtmans, Martyna Szpakowska, Andy Chevigné, Carsten Hoffmann, Chris de Graaf, Barbara A Zarzycka, Albert D Windhorst, Martine J Smit, Rob Leurs
Pharmacological Characterization and Radiolabeling of VUF15485, a High-Affinity Small-Molecule Agonist for the Atypical Chemokine Receptor ACKR3. Molecular pharmacology 105 (4) (2024)
Aurelien M Zarca, Ilze Adlere, Cristina P Viciano, Marta Arimont-Segura, Max Meyrath, Icaro A Simon, Jan Paul Bebelman, Dennis Laan, Hans G J Custers, Elwin Janssen, Kobus L Versteegh, Maurice C M L Buzink, Desislava N Nesheva, Reggie Bosma, Iwan J P de Esch, Henry F Vischer, Maikel Wijtmans, Martyna Szpakowska, Andy Chevigné, Carsten Hoffmann, Chris de Graaf, Barbara A Zarzycka, Albert D Windhorst, Martine J Smit, Rob Leurs
Pharmacological Characterization and Radiolabeling of VUF15485, a High-Affinity Small-Molecule Agonist for the Atypical Chemokine Receptor ACKR3. Molecular pharmacology 105 (4) (2024)
Nathan Vanalken, Katrijn Boon, Martyna Szpakowska, Andy Chevigné, Dominique Schols, Tom Van Loy
Systematic Assessment of Human CCR7 Signalling Using NanoBRET Biosensors Points towards the Importance of the Cellular Context. Biosensors 14 (3) (2024)
Nathan Vanalken, Katrijn Boon, Martyna Szpakowska, Andy Chevigné, Dominique Schols, Tom Van Loy
Systematic Assessment of Human CCR7 Signalling Using NanoBRET Biosensors Points towards the Importance of the Cellular Context. Biosensors 14 (3) (2024)
Aurelien Zarca, Ilze Adlere, Cristina P Viciano, Marta Arimont-Segura, Max Meyrath, Icaro A Simon, Jan Paul Bebelman, Dennis Laan, Hans G J Custers, Elwin Janssen, Kobus L K Versteegh, Maurice Buzink, Desislava Nesheva, Reggie Bosma, Iwan J P de Esch, Henry Vischer, Maikel Wijtmans, Martyna Szpakowska, Andy Chevigné, Carsten Hoffmann, Chris de Graaf, Barbara A Zarzycka, Albert D Windhorst, Martine J Smit, Rob Leurs
Pharmacological characterization and radiolabeling of VUF15485, a high-affinity small-molecule agonist for the atypical chemokine receptor ACKR3. Molecular pharmacology (2024)
Max E Huber, Silas L Wurnig, Aurélien F A Moumbock, Lara Toy, Evi Kostenis, Ana Alonso Bartolomé, Martyna Szpakowska, Andy Chevigné, Stefan Günther, Finn K Hansen, Matthias Schiedel
Development of a NanoBRET Assay Platform to Detect Intracellular Ligands for the Chemokine Receptors CCR6 and CXCR1. ChemMedChem (2024)
Nathan Vanalken, Katrijn Boon, Martyna Szpakowska, Andy Chevigné, Dominique Schols, Tom Van Loy
Systematic Assessment of Human CCR7 Signalling Using NanoBRET Biosensors Points towards the Importance of the Cellular Context. Biosensors 14 (3) (2024)
Anne Largeot, Vanessa Klapp, Elodie Viry, Susanne Gonder, Iria Fernandez Botana, Arnaud Blomme, Mohaned Benzarti, Sandrine Pierson, Chloé Duculty, Petra Marttila, Marina Wierz, Ernesto Gargiulo, Giulia Pagano, Ning An, Najla El Hachem, Daniel Perez-Hernandez, Supriya Chakraborty, Loïc Ysebaert, Jean-Hugues François, Susan Denisse Cortez Clemente, Guy Berchem, Dimitar G Efremov, Gunnar Dittmar, Martyna Szpakowska, Andy Chevigné, Petr V Nazarov, Thomas Helleday, Pierre Close, Johannes Meiser, Basile Stamatopoulos, Laurent Désaubry, Jérôme Paggetti, Etienne Moussay
Inhibition of MYC translation through targeting of the newly identified PHB-eIF4F complex as therapeutic strategy in CLL. Blood (2023)
Anne Largeot, Vanessa Klapp, Elodie Viry, Susanne Gonder, Iria Fernandez Botana, Arnaud Blomme, Mohaned Benzarti, Sandrine Pierson, Chloé Duculty, Petra Marttila, Marina Wierz, Ernesto Gargiulo, Giulia Pagano, Ning An, Najla El Hachem, Daniel Perez-Hernandez, Supriya Chakraborty, Loïc Ysebaert, Jean-Hugues François, Susan Denisse Cortez Clemente, Guy Berchem, Dimitar G Efremov, Gunnar Dittmar, Martyna Szpakowska, Andy Chevigné, Petr V Nazarov, Thomas Helleday, Pierre Close, Johannes Meiser, Basile Stamatopoulos, Laurent Désaubry, Jérôme Paggetti, Etienne Moussay
Inhibition of MYC translation through targeting of the newly identified PHB-eIF4F complex as therapeutic strategy in CLL. Blood (2023)
Evi Kostenis, Jesús Gomeza, Elke Miess-Tanneberg, Nina Kathleen Blum, Tobias Benkel, Andy Chevigné, Carsten Hoffmann, Peter Kolb, Viacheslav O Nikolaev, Maria Waldhoer, Martyna Szpakowska, Asuka Inoue, Stefan Schulz
Reply to: How carvedilol does not activate β 2 -adrenoceptors. Nature communications 14 (1) (2023)
Anne Largeot, Vanessa Klapp, Elodie Viry, Susanne Gonder, Iria Fernandez Botana, Arnaud Blomme, Mohaned Benzarti, Sandrine Pierson, Chloé Duculty, Petra Marttila, Marina Wierz, Ernesto Gargiulo, Giulia Pagano, Ning An, Najla El Hachem, Daniel Perez-Hernandez, Supriya Chakraborty, Loïc Ysebaert, Jean-Hugues François, Susan Denisse Cortez Clemente, Guy Berchem, Dimitar G Efremov, Gunnar Dittmar, Martyna Szpakowska, Andy Chevigné, Petr V Nazarov, Thomas Helleday, Pierre Close, Johannes Meiser, Basile Stamatopoulos, Laurent Désaubry, Jérôme Paggetti, Etienne Moussay
Inhibition of MYC translation through targeting of the newly identified PHB-eIF4F complex as therapeutic strategy in CLL. Blood (2023)
Anne Largeot, Vanessa Klapp, Elodie Viry, Susanne Gonder, Iria Fernandez Botana, Arnaud Blomme, Mohaned Benzarti, Sandrine Pierson, Chloé Duculty, Petra Marttila, Marina Wierz, Ernesto Gargiulo, Giulia Pagano, Ning An, Najla El Hachem, Daniel Perez-Hernandez, Supriya Chakraborty, Loïc Ysebaert, Jean-Hugues François, Susan Denisse Cortez Clemente, Guy Berchem, Dimitar G Efremov, Gunnar Dittmar, Martyna Szpakowska, Andy Chevigné, Petr V Nazarov, Thomas Helleday, Pierre Close, Johannes Meiser, Basile Stamatopoulos, Laurent Désaubry, Jérôme Paggetti, Etienne Moussay
Inhibition of MYC translation through targeting of the newly identified PHB-eIF4F complex as therapeutic strategy in CLL. Blood (2023)
Tobias Benkel, Mirjam Zimmermann, Julian Zeiner, Sergi Bravo, Nicole Merten, Victor Jun Yu Lim, Edda Sofie Fabienne Matthees, Julia Drube, Elke Miess-Tanneberg, Daniela Malan, Martyna Szpakowska, Stefania Monteleone, Jak Grimes, Zsombor Koszegi, Yann Lanoiselée, Shannon O'Brien, Nikoleta Pavlaki, Nadine Dobberstein, Asuka Inoue, Viacheslav O Nikolaev, Davide Calebiro, Andy Chevigné, Philipp Sasse, Stefan Schulz, Carsten Hoffmann, Peter Kolb, Maria Waldhoer, Katharina Simon, Jesus Gomeza, Evi Kostenis
How Carvedilol activates β 2 -adrenoceptors. Nature communications 13 (1) (2022)
Andrew B Kleist, Shawn Jenjak, Andrija Sente, Lauren J Laskowski, Martyna Szpakowska, Maggie M Calkins, Emilie I Anderson, Lisa M McNally, Raimond Heukers, Vladimir Bobkov, Francis C Peterson, Monica A Thomas, Andy Chevigné, Martine J Smit, John D McCorvy, M Madan Babu, Brian F Volkman
Conformational selection guides β-arrestin recruitment at a biased G protein-coupled receptor. Science (New York, N.Y.) 377 (6602) (2022)
Justine S Paradis, Xiang Feng, Brigitte Murat, Jefferson Roberts, Badr Sokrat, Martyna Szpakowska, Mireille Hogue, Nick D Bergkamp, Franziska M Heydenreich, Martine J Smit, Andy Chevigné, Michel Bouvier, Patrick Barth
Computationally designed GPCR quaternary structures bias signaling pathway activation. Nature communications 13 (1) (2022)
Alp Bayrak, Florian Mohr, Kyra Kolb, Martyna Szpakowska, Ekaterina Shevchenko, Valerie Dicenta, Anne-Katrin Rohlfing, Mark Kudolo, Tatu Pantsar, Marcel Günther, Agnieszka A Kaczor, Antti Poso, Andy Chevigné, Thanigaimalai Pillaiyar, Meinrad Gawaz, Stefan A Laufer
Discovery and Development of First-in-Class ACKR3/CXCR7 Superagonists for Platelet Degranulation Modulation. Journal of medicinal chemistry 65 (19) (2022)
Damla Isci, Giulia D'Uonnolo, May Wantz, Bernard Rogister, Arnaud Lombard, Andy Chevigné, Martyna Szpakowska, Virginie Neirinckx
Patient-Oriented Perspective on Chemokine Receptor Expression and Function in Glioma. Cancers 14 (1) (2021)
Andy Chevigné, Bassam Janji, Max Meyrath, Nathan Reynders, Giulia D'Uonnolo, Tomasz Uchański, Malina Xiao, Guy Berchem, Markus Ollert, Yong-Jun Kwon, Muhammad Zaeem Noman, Martyna Szpakowska
CXCL10 Is an Agonist of the CC Family Chemokine Scavenger Receptor ACKR2/D6. Cancers 13 (5) (2021)
Martyna Szpakowska, Ann M Decker, Max Meyrath, Christie B Palmer, Bruce E Blough, Ojas A Namjoshi, Andy Chevigné
The natural analgesic conolidine targets the newly identified opioid scavenger ACKR3/CXCR7. Signal transduction and targeted therapy 6 (1) (2021)
Adam M Passman, Robyn P Strauss, Sarah B McSpadden, Megan Finch-Edmondson, Neil Andrewartha, Ken H Woo, Luke A Diepeveen, Weihao Zhao, Joaquín Fernández-Irigoyen, Enrique Santamaria, Laura Medina-Ruiz, Martyna Szpakowska, Andy Chevigné, Hyerin Park, Rodrigo Carlessi, Janina E E Tirnitz-Parker, José-Ramon Blanco, Roslyn London, Bernard A Callus, Caryn L Elsegood, Murray V Baker, Alfredo Martínez, George C T Yeoh, Laura Ochoa-Callejero
Maraviroc Prevents HCC Development by Suppressing Macrophages and the Liver Progenitor Cell Response in a Murine Chronic Liver Disease Model. Cancers 13 (19) (2021)
Max Meyrath, Nathan Reynders, Tomasz Uchański, Andy Chevigné, Martyna Szpakowska
Systematic reassessment of chemokine-receptor pairings confirms CCL20 but not CXCL13 and extends the spectrum of ACKR4 agonists to CCL22. Journal of leukocyte biology 109 (2) (2020)
Max Meyrath, Martyna Szpakowska, Julian Zeiner, Laurent Massotte, Myriam P Merz, Tobias Benkel, Katharina Simon, Jochen Ohnmacht, Jonathan David Turner, Rejko Krüger, Vincent Seutin, Markus Ollert, Evi Kostenis, Andy Chevigné
The atypical chemokine receptor ACKR3/CXCR7 is a broad-spectrum scavenger for opioid peptides. Nature communications 11 (1) (2020)