Jonathan B Baell (Jonathan Baell)

ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 42

Top Venues

Journal of medicinal chemistry

Nature communications

RSC medicinal chemistry

ChemMedChem

This page only lists publications with an associated author ORCID identifier.

Publications

Bernhard Jandl, Rebecca Zheng, Markus Muttenthaler, Jonathan B Baell
Novel Diacyl-hydrazide Compounds as Potential Therapeutics for Visceral Leishmaniasis. ACS omega 9 (35) (2024)
Jayme L Dahlin, Bruce K Hua, Beth E Zucconi, Shawn D Nelson, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew E Cuellar, Philip A Cole, Jordan L Meier, Tim Thomas, Jonathan B Baell, Peter J Brown, Michael A Walters, Paul A Clemons, Stuart L Schreiber, Bridget K Wagner
Reference compounds for characterizing cellular injury in high-content cellular morphology assays. Nature communications 14 (1) (2023)
Jayme L Dahlin, Bruce K Hua, Beth E Zucconi, Shawn D Nelson, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew E Cuellar, Philip A Cole, Jordan L Meier, Tim Thomas, Jonathan B Baell, Peter J Brown, Michael A Walters, Paul A Clemons, Stuart L Schreiber, Bridget K Wagner
Reference compounds for characterizing cellular injury in high-content cellular morphology assays. Nature communications 14 (1) (2023)
Julia Beveridge, Eric Tran, Girdhar Singh Deora, Fei Huang, Yuzhi Wang, Kieran Stockton, Ignacio Cotillo, Maria Santos Martinez Martinez, Silvia Gonzalez, Pablo Castañeda, Julian Sherman, Ana Rodriguez, Albane Kessler, Jonathan B Baell
Novel Diarylthioether Compounds as Agents for the Treatment of Chagas Disease. Journal of medicinal chemistry 66 (2) (2023)
Julia Beveridge, Eric Tran, Girdhar Singh Deora, Fei Huang, Yuzhi Wang, Kieran Stockton, Ignacio Cotillo, Maria Santos Martinez Martinez, Silvia Gonzalez, Pablo Castañeda, Julian Sherman, Ana Rodriguez, Albane Kessler, Jonathan B Baell
Novel Diarylthioether Compounds as Agents for the Treatment of Chagas Disease. Journal of medicinal chemistry 66 (2) (2023)
Julia Beveridge, Eric Tran, Girdhar Singh Deora, Fei Huang, Yuzhi Wang, Kieran Stockton, Ignacio Cotillo, Maria Santos Martinez Martinez, Silvia Gonzalez, Pablo Castañeda, Julian Sherman, Ana Rodriguez, Albane Kessler, Jonathan B Baell
Novel Diarylthioether Compounds as Agents for the Treatment of Chagas Disease. Journal of medicinal chemistry (2023)
Mingrui Li, Zhiqin He, Wei Zhao, Yang Yu, Fei Huang, Jonathan B Baell
Photocatalytic Benzylic C-H Oxidation/Cyclization of Enaminones to the Synthesis of Polysubstituted Oxazoles. The Journal of organic chemistry (2023)
Jayme L Dahlin, Bruce K Hua, Beth E Zucconi, Shawn D Nelson, Shantanu Singh, Anne E Carpenter, Jonathan H Shrimp, Evelyne Lima-Fernandes, Mathias J Wawer, Lawrence P W Chung, Ayushi Agrawal, Mary O'Reilly, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Fengling Li, Parnian Lak, Matthew E Cuellar, Philip A Cole, Jordan L Meier, Tim Thomas, Jonathan B Baell, Peter J Brown, Michael A Walters, Paul A Clemons, Stuart L Schreiber, Bridget K Wagner
Reference compounds for characterizing cellular injury in high-content cellular morphology assays. Nature communications 14 (1) (2023)
Shuwei Liang, Eric Tran, Xin Du, Jiajun Dong, Harrison Sudholz, Hao Chen, Zihan Qu, Nicholas D Huntington, Jeffrey J Babon, Nadia J Kershaw, Zhong-Yin Zhang, Jonathan B Baell, Florian Wiede, Tony Tiganis
A small molecule inhibitor of PTP1B and PTPN2 enhances T cell anti-tumor immunity. Nature communications 14 (1) (2023)
Julia Beveridge, Eric Tran, Girdhar Singh Deora, Fei Huang, Yuzhi Wang, Kieran Stockton, Ignacio Cotillo, Maria Santos Martinez Martinez, Silvia Gonzalez, Pablo Castañeda, Julian Sherman, Ana Rodriguez, Albane Kessler, Jonathan B Baell
Novel Diarylthioether Compounds as Agents for the Treatment of Chagas Disease. Journal of medicinal chemistry 66 (2) (2023)
Melanie Heinlein, Luke C Gandolfo, Kelin Zhao, Charis E Teh, Nghi Nguyen, Jonathan B Baell, Yael Goldfarb, Jakub Abramson, Johannes Wichmann, Anne K Voss, Andreas Strasser, Aaron T L Lun, Tim Thomas, Daniel H D Gray
The acetyltransferase KAT7 is required for thymic epithelial cell expansion, expression of AIRE target genes, and thymic tolerance. Science immunology 7 (67) (2022)
Susanne Müller, Stephen V Frye, Jonathan B Baell
The future of chemical probes is diversity. RSC medicinal chemistry 13 (12) (2022)
Noel P Pitcher, Jitendra R Harjani, Yichao Zhao, Jianwen Jin, Daniel R Knight, Lucy Li, Papanin Putsathit, Thomas V Riley, Glen P Carter, Jonathan B Baell
Development of 1,2,4-Oxadiazole Antimicrobial Agents to Treat Enteric Pathogens within the Gastrointestinal Tract. ACS omega 7 (8) (2022)
Jiajun Feng, Yuzhi Wang, Luoyu Gao, Yang Yu, Jonathan B Baell, Fei Huang
Electrochemical Synthesis of Polysubstituted Sulfonated Pyrazoles via Cascade Intermolecular Condensation, Radical-Radical Cross Coupling Sulfonylation, and Pyrazole Annulation. The Journal of organic chemistry 87 (19) (2022)
Lisa Barbaro, Gayathri Nagalingam, James A Triccas, Lendl Tan, Nicholas P West, Daniel L Priebbenow, Jonathan B Baell
Discovery of Anti-tubercular Analogues of Bedaquiline with Modified A-, B- and C-Ring Subunits. ChemMedChem (2022)
Jiajun Feng, Tiantong He, Yuxing Xie, Yang Yu, Jonathan B Baell, Fei Huang
I2-Promoted [4 + 2] cycloaddition of in situ generated azoalkenes with enaminones: facile and efficient synthesis of 1,4-dihydropyridazines and pyridazines. Organic & biomolecular chemistry 18 (46) (2022)
Michael J Roy, Amelia Vom, Toru Okamoto, Brian J Smith, Richard W Birkinshaw, Hong Yang, Houda Abdo, Christine A White, David Segal, David C S Huang, Jonathan B Baell, Peter M Colman, Peter E Czabotar, Guillaume L Lessene
Structure-Guided Development of Potent Benzoylurea Inhibitors of BCL-XL and BCL-2. Journal of medicinal chemistry 64 (9) (2021)
Yufei Xue, Hua Bai, Bo Peng, Bin Fang, Jonathan B Baell, Lin Li, Wei Huang, Nicolas Hans Voelcker
Stimulus-cleavable chemistry in the field of controlled drug delivery. Chemical Society reviews 50 (8) (2021)
C Glenn Begley, Mark Ashton, Jonathan B Baell, Michael Bettess, Michael P Brown, Brett Carter, William N Charman, Christopher Davis, Simon Fisher, Ian Hector Frazer, Anand Gautam, Michael P Jennings, Philip Kearney, Eloise Keeffe, Darren Kelly, Angel F Lopez, Michael A McGuckin, Michael W Parker, Craig Rayner, Brett Roberts, James S Rush, Mark Sullivan
Drug repurposing: Misconceptions, challenges, and opportunities for academic researchers. Science translational medicine 13 (612) (2021)
Daniel L Priebbenow, Mitch Mathiew, Da-Hua Shi, Jitendra R Harjani, Julia G Beveridge, Marina Chavchich, Michael D Edstein, Sandra Duffy, Vicky M Avery, Robert T Jacobs, Stephen Brand, David M Shackleford, Wen Wang, Longjin Zhong, Given Lee, Erin Tay, Helena Barker, Elly Crighton, Karen L White, Susan A Charman, Amanda De Paoli, Darren John Creek, Jonathan B Baell
Discovery of Potent and Fast-Acting Antimalarial Bis-1,2,4-triazines. Journal of medicinal chemistry 64 (7) (2021)
Lisa Barbaro, Gayathri Nagalingam, James A Triccas, Lendl Tan, Nicholas P West, Jonathan B Baell, Daniel L Priebbenow
Synthesis and evaluation of pyridine-derived bedaquiline analogues containing modifications at the A-ring subunit. RSC medicinal chemistry 12 (6) (2021)
Jonathan B Baell
Early career research in medicinal chemistry. Future medicinal chemistry 13 (2) (2021)
Susanne Müller, Suzanne Ackloo, Arij Al Chawaf, Bissan Al-Lazikani, Albert Antolin, Jonathan B Baell, Hartmut Beck, Shaunna Beedie, Ulrich A K Betz, Gustavo Arruda Bezerra, Paul E Brennan, David Brown, Peter J Brown, Alex N Bullock, Adrian J Carter, Apirat Chaikuad, Mathilde Chaineau, Alessio Ciulli, Ian Collins, Jan Dreher, David Drewry, Kristina Edfeldt, Aled M Edwards, Ursula Egner, Stephen V Frye, Stephen M Fuchs, Matthew D Hall, Ingo V Hartung, Alexander Hillisch, Stephen H Hitchcock, Evert Homan, Natarajan Kannan, James R Kiefer, Stefan Knapp, Milka Kostic, Stefan Kubicek, Andrew R Leach, Sven Lindemann, Brian D Marsden, Hisanori Matsui, Jordan L Meier, Daniel Merk, Maurice Michel, Maxwell Robert Morgan, Anke Mueller-Fahrnow, Dafydd R Owen, Benjamin G Perry, Saul H Rosenberg, Kumar Singh Saikatendu, Matthieu Schapira, Cora Scholten, Sujata Sharma, Anton Simeonov, Michael Sundström, Giulio Superti-Furga, Matthew H Todd, Claudia Tredup, Masoud Vedadi, Frank von Delft, Timothy M Willson, Georg E Winter, Paul Workman, Cheryl H Arrowsmith
Target 2035 - update on the quest for a probe for every protein. RSC medicinal chemistry 13 (1) (2021)
Yiyue Xie, Padmaja Tummala, Aaron J Oakley, Girdhar Singh Deora, Yuji Nakano, Melissa Rooke, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Marco G Casarotto, Philip G Board, Jonathan B Baell
Development of Benzenesulfonamide Derivatives as Potent Glutathione Transferase Omega-1 Inhibitors. Journal of medicinal chemistry 63 (6) (2020)
Ronald W Brown, Ashraf M Abdel-Megeed, Paul A Keller, Amy J Jones, Melissa Louise Sykes, Marcel Kaiser, Jonathan B Baell, Vicky Marie Avery, Christopher J T Hyland
Investigation of thiazolyl-benzothiophenamides as potential agents for African sleeping sickness. RSC medicinal chemistry 11 (12) (2020)
Nicole McNamara, Raphael Rahmani, Melissa Louise Sykes, Vicky Marie Avery, Jonathan B Baell
Hit-to-lead optimization of novel benzimidazole phenylacetamides as broad spectrum trypanosomacides. RSC medicinal chemistry 11 (6) (2020)
Daniel L Priebbenow, David J Leaver, Nghi Nguyen, Benjamin Cleary, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, David M Shackleford, Kasiram Katneni, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Ian P Street, Brendon J Monahan, Kate E Jarman, Helene Jousset Sabroux, Hendrik Falk, Matthew C Chung, Stefan J Hermans, Natalie L Downer, Michael W Parker, Anne K Voss, Tim Thomas, Jonathan B Baell
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents. Journal of medicinal chemistry 63 (9) (2020)
Xiangyan Yi, Lian Xue, Tim Thomas, Jonathan B Baell
Action plan for hit identification (APHID): KAT6A as a case study. Future medicinal chemistry 12 (5) (2020)
Sarah Preston, Jose F Garcia-Bustos, Liam G Hall, Sheree D Martin, Thuy G Le, Abhijit Kundu, Atanu Ghoshal, Nghi H Nguyen, Yaqing Jiao, Banfeng Ruan, Lian Xue, Fei Huang, Bill C H Chang, Sean L McGee, Timothy N C Wells, Michael J Palmer, Abdul Jabbar, Robin B Gasser, Jonathan B Baell
1-Methyl-1H-pyrazole-5-carboxamide Derivatives Exhibit Unexpected Acute Mammalian Toxicity. Journal of medicinal chemistry 64 (1) (2020)
Swapna Varghese, Raphaël Rahmani, Damien R Drew, James G Beeson, Jake Baum, Brian J Smith, Jonathan B Baell
Structure-Activity Studies of Truncated Latrunculin Analogues with Antimalarial Activity. ChemMedChem 16 (4) (2020)
Thuy G Le, Abhijit Kundu, Atanu Ghoshal, Nghi H Nguyen, Sarah Preston, Yaqing Jiao, Banfeng Ruan, Lian Xue, Fei Huang, Jennifer Keiser, Andreas Hofmann, Bill C H Chang, Jose Garcia-Bustos, Timothy N C Wells, Michael J Palmer, Abdul Jabbar, Robin B Gasser, Jonathan B Baell
Novel 1-Methyl-1 H-pyrazole-5-carboxamide Derivatives with Potent Anthelmintic Activity. Journal of medicinal chemistry 62 (7) (2019)
Thuy G Le, Abhijit Kundu, Atanu Ghoshal, Nghi H Nguyen, Sarah Preston, Yaqing Jiao, Banfeng Ruan, Lian Xue, Fei Huang, Jennifer Keiser, Andreas Hofmann, Bill C H Chang, Jose Garcia-Bustos, Timothy N C Wells, Michael J Palmer, Abdul Jabbar, Robin B Gasser, Jonathan B Baell
Structure-Activity Relationship Studies of Tolfenpyrad Reveal Subnanomolar Inhibitors of Haemonchus contortus Development. Journal of medicinal chemistry 62 (2) (2019)
Lian Xue, Da-Hua Shi, Jitendra R Harjani, Fei Huang, Julia G Beveridge, Tamir Dingjan, Kung Ban, Sarah Diab, Sandra Duffy, Leonardo Lucantoni, Sabine Fletcher, Francis C K Chiu, Scott Blundell, Katherine Ellis, Stuart A Ralph, Grennady Wirjanata, Silvia Teguh, Rintis Noviyanti, Marina Chavchich, Darren John Creek, Ric N Price, Jutta Marfurt, Susan A Charman, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Michael D Edstein, Vicky M Avery, Jonathan B Baell
3,3'-Disubstituted 5,5'-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity. Journal of medicinal chemistry 62 (5) (2019)
Girdhar Singh Deora, Chengxue Helena Qin, Elizabeth A Vecchio, Aaron J Debono, Daniel L Priebbenow, Ryan M Brady, Julia Beveridge, Silvia C Teguh, Minh Deo, Lauren T May, Guy Krippner, Rebecca H Ritchie, Jonathan B Baell
Substituted Pyridazin-3(2 H)-ones as Highly Potent and Biased Formyl Peptide Receptor Agonists. Journal of medicinal chemistry 62 (10) (2019)
David J Leaver, Benjamin Cleary, Nghi Nguyen, Daniel L Priebbenow, H Rachel Lagiakos, Julie Sanchez, Lian Xue, Fei Huang, Yuxin Sun, Prashant Mujumdar, Ramesh Mudududdla, Swapna Varghese, Silvia Teguh, Susan A Charman, Karen L White, Kasiram Katneni, Matthew Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Ian P Street, Brendon J Monahan, Kate E Jarman, Helene Jousset Sabroux, Hendrik Falk, Matthew C Chung, Stefan J Hermans, Michael W Parker, Tim Thomas, Jonathan B Baell
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A. Journal of medicinal chemistry 62 (15) (2019)
Cheng Xue Qin, Lauren T May, Patrick M Sexton, Aaron J DeBono, Jonathan B Baell, Arthur Christopoulos, Rebecca H Ritchie
Correspondence: Reply to 'Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury'. Nature communications 9 (1) (2018)
Yiyue Xie, Jayme L Dahlin, Aaron J Oakley, Marco G Casarotto, Philip G Board, Jonathan B Baell
Reviewing Hit Discovery Literature for Difficult Targets: Glutathione Transferase Omega-1 as an Example. Journal of medicinal chemistry 61 (17) (2018)
Thuy G Le, Abhijit Kundu, Atanu Ghoshal, Nghi H Nguyen, Sarah Preston, Yaqing Jiao, Banfeng Ruan, Lian Xue, Fei Huang, Jennifer Keiser, Andreas Hofmann, Bill C H Chang, Jose Garcia-Bustos, Abdul Jabbar, Timothy N C Wells, Michael J Palmer, Robin B Gasser, Jonathan B Baell
Optimization of Novel 1-Methyl-1 H-Pyrazole-5-carboxamides Leads to High Potency Larval Development Inhibitors of the Barber's Pole Worm. Journal of medicinal chemistry 61 (23) (2018)
Elena K Schneider, Daniel Hoyer, Alexander A Khromykh, Jonathan B Baell, Glenn A Marsh, Mark A Baker, Jian Li, Xukai Jiang
Contemporary Anti-Ebola Drug Discovery Approaches and Platforms. ACS infectious diseases 5 (1) (2018)
Jayme L Dahlin, Kathryn M Nelson, Jessica M Strasser, Dalia Barsyte-Lovejoy, Magdalena M Szewczyk, Shawna Organ, Matthew E Cuellar, Gurpreet Singh, Jonathan H Shrimp, Nghi Nguyen, Jordan L Meier, Cheryl H Arrowsmith, Peter J Brown, Jonathan B Baell, Michael A Walters
Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors. Nature communications 8 (1) (2017)
Jonathan B Baell, J Willem M Nissink
Seven Year Itch: Pan-Assay Interference Compounds (PAINS) in 2017-Utility and Limitations. ACS chemical biology 13 (1) (2017)
Deepthi Menon, Ashlee Innes, Aaron J Oakley, Jane E Dahlstrom, Lora M Jensen, Anne Brüstle, Padmaja Tummala, Melissa Rooke, Marco G Casarotto, Jonathan B Baell, Nghi Nguyen, Yiyue Xie, Matthew E Cuellar, Jessica M Strasser, Jayme L Dahlin, Michael A Walters, Gaetan Burgio, Luke A J O'Neill, Philip G Board
GSTO1-1 plays a pro-inflammatory role in models of inflammation, colitis and obesity. Scientific reports 7 (1) (2017)

Jonathan B Baell.css-eqlu8i{font-size:small;padding-left:4px;} (Jonathan Baell)

Publication Activity (10 Years)

Top Topics

Top Venues

Jonathan B Baell (Jonathan Baell)