Roberto Di Santo (R Di Santo)

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 40

Top Topics

Molecular Dynamics Simulations

Candida Albicans

Arabidopsis Thaliana

Top Venues

Pharmaceuticals (Basel, Switzerland)

Journal of medicinal chemistry

International journal of molecular sciences

Molecules (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Antonella Messore, Paolo Malune, Elisa Patacchini, Valentina Noemi Madia, Davide Ialongo, Merve Arpacioglu, Aurora Albano, Giuseppe Ruggieri, Francesco Saccoliti, Luigi Scipione, Enzo Tramontano, Serena Canton, Angela Corona, Sante Scognamiglio, Annalaura Paulis, Mustapha Suleiman, Helmi Mohammed Al-Maqtari, Fatma Mohamed A Abid, Sarkar Mohammad Abe Kawsar, Sankaranarayanan Murugesan, Roberto Di Santo, Francesca Esposito, Roberta Costi
New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors. Pharmaceuticals (Basel, Switzerland) 17 (5) (2024)
Antonella Messore, Paolo Malune, Elisa Patacchini, Valentina Noemi Madia, Davide Ialongo, Merve Arpacioglu, Aurora Albano, Giuseppe Ruggieri, Francesco Saccoliti, Luigi Scipione, Enzo Tramontano, Serena Canton, Angela Corona, Sante Scognamiglio, Annalaura Paulis, Mustapha Suleiman, Helmi Mohammed Al-Maqtari, Fatma Mohamed A Abid, Sarkar Mohammad Abe Kawsar, Sankaranarayanan Murugesan, Roberto Di Santo, Francesca Esposito, Roberta Costi
New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors. Pharmaceuticals (Basel, Switzerland) 17 (5) (2024)
Elisa Patacchini, Valentina Noemi Madia, Aurora Albano, Giuseppe Ruggieri, Antonella Messore, Davide Ialongo, Francesco Saccoliti, Luigi Scipione, Sandro Cosconati, Pratibha C Koneru, Reed Haney, Mamuka Kvaratskhelia, Roberto Di Santo, Roberta Costi
Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions. ACS medicinal chemistry letters 15 (9) (2024)
Valeria Manganelli, Roberta Misasi, Gloria Riitano, Antonella Capozzi, Vincenzo Mattei, Tuba Rana Caglar, Davide Ialongo, Valentina Noemi Madia, Antonella Messore, Roberta Costi, Roberto Di Santo, Maurizio Sorice, Tina Garofalo
Role of a Novel Heparanase Inhibitor on the Balance between Apoptosis and Autophagy in U87 Human Glioblastoma Cells. Cells 12 (14) (2023)
Valentina Noemi Madia, Davide Ialongo, Elisa Patacchini, Cécile Exertier, Lorenzo Antonelli, Gianni Colotti, Antonella Messore, Valeria Tudino, Francesco Saccoliti, Luigi Scipione, Andrea Ilari, Roberta Costi, Roberto Di Santo
Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site. Molecules (Basel, Switzerland) 28 (1) (2023)
Marco Gasparella, Carola Cenzi, Monica Piccione, Valentina Noemi Madia, Roberto Di Santo, Valeria Tudino, Marco Artico, Samanta Taurone, Chiara De Ponte, Roberta Costi, Rosa Di Liddo
Effects of Modified Glucosamine on the Chondrogenic Potential of Circulating Stem Cells under Experimental Inflammation. International journal of molecular sciences 24 (12) (2023)
Andrea Lepri, C Longo, A Messore, H Kazmi, Valentina Noemi Madia, Roberto Di Santo, R Costi, Paola Vittorioso
Plants and Small Molecules: An Up-and-Coming Synergy. Plants (Basel, Switzerland) 12 (8) (2023)
Andrea Lepri, C Longo, A Messore, H Kazmi, Valentina Noemi Madia, Roberto Di Santo, R Costi, Paola Vittorioso
Plants and Small Molecules: An Up-and-Coming Synergy. Plants (Basel, Switzerland) 12 (8) (2023)
Andrea Lepri, C Longo, A Messore, H Kazmi, Valentina Noemi Madia, Roberto Di Santo, R Costi, Paola Vittorioso
Plants and Small Molecules: An Up-and-Coming Synergy. Plants (Basel, Switzerland) 12 (8) (2023)
Valentina Noemi Madia, Davide Ialongo, Elisa Patacchini, Cécile Exertier, Lorenzo Antonelli, Gianni Colotti, Antonella Messore, Valeria Tudino, Francesco Saccoliti, Luigi Scipione, Andrea Ilari, Roberta Costi, Roberto Di Santo
Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site. Molecules (Basel, Switzerland) 28 (1) (2023)
Davide Ialongo, Antonella Messore, Valentina Noemi Madia, Valeria Tudino, Alessio Nocentini, Paola Gratteri, Simone Giovannuzzi, Claudiu T Supuran, Alice Nicolai, Susanna Scarpa, Samanta Taurone, Michele Camarda, Marco Artico, Veronica Papa, Francesco Saccoliti, Luigi Scipione, Roberto Di Santo, Roberta Costi
Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII. Pharmaceuticals (Basel, Switzerland) 16 (2) (2023)
Davide Ialongo, Valeria Tudino, Merve Arpacioglu, Antonella Messore, Elisa Patacchini, Roberta Costi, Roberto Di Santo, Valentina Noemi Madia
Synergistic Effects of Caffeine in Combination with Conventional Drugs: Perspectives of a Drug That Never Ages. Pharmaceuticals (Basel, Switzerland) 16 (5) (2023)
Marco Gasparella, Carola Cenzi, Monica Piccione, Valentina Noemi Madia, Roberto Di Santo, Valeria Tudino, Marco Artico, Samanta Taurone, Chiara De Ponte, Roberta Costi, Rosa Di Liddo
Effects of Modified Glucosamine on the Chondrogenic Potential of Circulating Stem Cells under Experimental Inflammation. International journal of molecular sciences 24 (12) (2023)
Vandna Sharma, Valentina Noemi Madia, Valeria Tudino, Jennifer V Nguyen, Anjan Debnath, Antonella Messore, Davide Ialongo, Elisa Patacchini, Irene Palenca, Silvia Basili Franzin, Luisa Seguella, Giuseppe Esposito, Rita Petrucci, Paola Di Matteo, Martina Bortolami, Francesco Saccoliti, Roberto Di Santo, Luigi Scipione, Roberta Costi, Larissa M Podust
Miconazole-like Scaffold is a Promising Lead for Naegleria fowleri -Specific CYP51 Inhibitors. Journal of medicinal chemistry (2023)
Valentina Noemi Madia, Davide Ialongo, Elisa Patacchini, Cécile Exertier, Lorenzo Antonelli, Gianni Colotti, Antonella Messore, Valeria Tudino, Francesco Saccoliti, Luigi Scipione, Andrea Ilari, Roberta Costi, Roberto Di Santo
Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site. Molecules (Basel, Switzerland) 28 (1) (2023)
Marco Gasparella, Carola Cenzi, Monica Piccione, Valentina Noemi Madia, Roberto Di Santo, Valeria Tudino, Marco Artico, Samanta Taurone, Chiara De Ponte, Roberta Costi, Rosa Di Liddo
Effects of Modified Glucosamine on the Chondrogenic Potential of Circulating Stem Cells under Experimental Inflammation. International journal of molecular sciences 24 (12) (2023)
Andrea Lepri, C Longo, A Messore, H Kazmi, Valentina Noemi Madia, Roberto Di Santo, R Costi, Paola Vittorioso
Plants and Small Molecules: An Up-and-Coming Synergy. Plants (Basel, Switzerland) 12 (8) (2023)
Martina Bortolami, Fabiana Pandolfi, Valeria Tudino, Antonella Messore, Valentina Noemi Madia, Daniela De Vita, Roberto Di Santo, Roberta Costi, Isabella Romeo, Stefano Alcaro, Marisa Colone, Annarita Stringaro, Alba Espargaró, Raimon Sabatè, Luigi Scipione
Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors. Pharmaceuticals (Basel, Switzerland) 15 (6) (2022)
Valentina Noemi Madia, Walter Toscanelli, Daniela De Vita, Marta De Angelis, Antonella Messore, Davide Ialongo, Luigi Scipione, Valeria Tudino, Felicia Diodata D'Auria, Roberto Di Santo, Stefania Garzoli, Annarita Stringaro, Marisa Colone, Magda Marchetti, Fabiana Superti, Lucia Nencioni, Roberta Costi
Ultrastructural Damages to H1N1 Influenza Virus Caused by Vapor Essential Oils. Molecules (Basel, Switzerland) 27 (12) (2022)
Carolina Orlando Vaso, Níura Madalena Bila, Fabiana Pandolfi, Daniela De Vita, Martina Bortolami, Jean Lucas Carvalho Bonatti, Rosângela Aparecida De Moraes Silva, Larissa Naiara Carvalho Gonçalves, Valeria Tudino, Roberta Costi, Roberto Di Santo, Maria José Soares Mendes-Giannini, Caroline Barcelos Costa-Orlandi, Luigi Scipione, Ana Marisa Fusco-Almeida
Evaluation of the Anti- Histoplasma capsulatum Activity of Indole and Nitrofuran Derivatives and Their Pharmacological Safety in Three-Dimensional Cell Cultures. Pharmaceutics 14 (5) (2022)
Chiara Longo, Andrea Lepri, Andrea Paciolla, Antonella Messore, Daniela De Vita, Maria Carmela Bonaccorsi di Patti, Matteo Amadei, Valentina Noemi Madia, Davide Ialongo, Roberto Di Santo, Roberta Costi, Paola Vittorioso
New Inhibitors of the Human p300/CBP Acetyltransferase Are Selectively Active against the Arabidopsis HAC Proteins. International journal of molecular sciences 23 (18) (2022)
Martina Bortolami, Fabiana Pandolfi, Valeria Tudino, Antonella Messore, Valentina Noemi Madia, Daniela De Vita, Roberto Di Santo, Roberta Costi, Isabella Romeo, Stefano Alcaro, Marisa Colone, Annarita Stringaro, Alba Espargaró, Raimon Sabatè, Luigi Scipione
New Pyrimidine and Pyridine Derivatives as Multitarget Cholinesterase Inhibitors: Design, Synthesis, and In Vitro and In Cellulo Evaluation. ACS chemical neuroscience 12 (21) (2021)
Serena Ammendola, Valerio Secli, Francesca Pacello, Martina Bortolami, Fabiana Pandolfi, Antonella Messore, Roberto Di Santo, Luigi Scipione, Andrea Battistoni
Salmonella Typhimurium and Pseudomonas aeruginosa Respond Differently to the Fe Chelator Deferiprone and to Some Novel Deferiprone Derivatives. International journal of molecular sciences 22 (19) (2021)
Valentina Noemi Madia, Daniela De Vita, Antonella Messore, Chiara Toniolo, Valeria Tudino, Alessandro De Leo, Ivano Pindinello, Davide Ialongo, Francesco Saccoliti, Anna Maria D'Ursi, Manuela Grimaldi, Pietro Ceccobelli, Luigi Scipione, Roberto Di Santo, Roberta Costi
Analytical Characterization of an Inulin-Type Fructooligosaccharide from Root-Tubers of Asphodelusramosus L. Pharmaceuticals (Basel, Switzerland) 14 (3) (2021)
Valentina Noemi Madia, Daniela De Vita, Davide Ialongo, Valeria Tudino, Alessandro De Leo, Luigi Scipione, Roberto Di Santo, Roberta Costi, Antonella Messore
Recent Advances in Recovery of Lycopene from Tomato Waste: A Potent Antioxidant with Endless Benefits. Molecules (Basel, Switzerland) 26 (15) (2021)
Martina Bortolami, Daniele Rocco, Antonella Messore, Roberto Di Santo, Roberta Costi, Valentina Noemi Madia, Luigi Scipione, Fabiana Pandolfi
Acetylcholinesterase inhibitors for the treatment of Alzheimer's disease - a patent review (2016-present). Expert opinion on therapeutic patents 31 (5) (2021)
Dalila Boi, Fani Souvalidou, Davide Capelli, Federica Polverino, Grazia Marini, Roberta Montanari, Giorgio Pochetti, Angela Tramonti, Roberto Contestabile, Daniela Trisciuoglio, Patrizia Carpinelli, Camilla Ascanelli, Catherine Lindon, Alessandro De Leo, Alessandro Tossi, Roberto Di Santo, Roberta Costi, Giulia Guarguaglini, Alessandro Paiardini
PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc. International journal of molecular sciences 22 (23) (2021)
Alice Nicolai, Valentina Noemi Madia, Antonella Messore, Daniela De Vita, Alessandro De Leo, Davide Ialongo, Valeria Tudino, Elisabetta Tortorella, Luigi Scipione, Samanta Taurone, Tiziano Pergolizzi, Marco Artico, Roberto Di Santo, Roberta Costi, Susanna Scarpa
Anti-Tumoral Effects of a (1H-Pyrrol-1-yl)Methyl-1H-Benzoimidazole Carbamate Ester Derivative on Head and Neck Squamous Carcinoma Cell Lines. Pharmaceuticals (Basel, Switzerland) 14 (6) (2021)
Valentina Noemi Madia, Marta De Angelis, Daniela De Vita, Antonella Messore, Alessandro De Leo, Davide Ialongo, Valeria Tudino, Francesco Saccoliti, Giovanna De Chiara, Stefania Garzoli, Luigi Scipione, Anna Teresa Palamara, Roberto Di Santo, Lucia Nencioni, Roberta Costi
Investigation of Commiphora myrrha (Nees) Engl. Oil and Its Main Components for Antiviral Activity. Pharmaceuticals (Basel, Switzerland) 14 (3) (2021)
Antonella Messore, Angela Corona, Valentina Noemi Madia, Francesco Saccoliti, Valeria Tudino, Alessandro De Leo, Davide Ialongo, Luigi Scipione, Daniela De Vita, Giorgio Amendola, Ettore Novellino, Sandro Cosconati, Mathieu Métifiot, Marie-Line Andreola, Francesca Esposito, Nicole Grandi, Enzo Tramontano, Roberta Costi, Roberto Di Santo
Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase. Journal of medicinal chemistry 64 (12) (2021)
Francesco Saccoliti, Roberto Di Santo, Roberta Costi
Recent Advancement in the Search of Innovative Antiprotozoal Agents Targeting Trypanothione Metabolism. ChemMedChem 15 (24) (2020)
Daniela De Vita, Antonella Messore, Chiara Toniolo, Claudio Frezza, Luigi Scipione, Cinzia Margherita Bertea, Marco Micera, Veronica Di Sarno, Valentina Noemi Madia, Ivano Pindinello, Patrizia Roscilli, Alfonso Botto, Giovanna Simonetti, Anastasia Orekhova, Stefano Manfredini, Roberta Costi, Roberto Di Santo
Towards a new application of amaranth seed oil as an agent against Candida albicans. Natural product research 35 (22) (2019)
Daniela De Vita, Valentina Noemi Madia, Valeria Tudino, Francesco Saccoliti, Alessandro De Leo, Antonella Messore, Patrizia Roscilli, Alfonso Botto, Ivano Pindinello, Gianluigi Santilli, Luigi Scipione, Roberta Costi, Roberto Di Santo
Comparison of different methods for the extraction of cannabinoids from cannabis. Natural product research 34 (20) (2019)
Francesco Saccoliti, Valentina Noemi Madia, Valeria Tudino, Alessandro De Leo, Luca Pescatori, Antonella Messore, Daniela De Vita, Luigi Scipione, Reto Brun, Marcel Kaiser, Pascal Mäser, Claudia M Calvet, Gareth K Jennings, Larissa M Podust, Giacomo Pepe, Roberto Cirilli, Cristina Faggi, Annalise Di Marco, Maria Rosaria Battista, Vincenzo Summa, Roberta Costi, Roberto Di Santo
Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents. Journal of medicinal chemistry 62 (3) (2019)
Vasanthanathan Poongavanam, Angela Corona, Casper Steinmann, Luigi Scipione, Nicole Grandi, Fabiana Pandolfi, Roberto Di Santo, Roberta Costi, Francesca Esposito, Enzo Tramontano, Jacob Kongsted
Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studies. MedChemComm 9 (3) (2018)
Valentina Noemi Madia, Antonella Messore, Luca Pescatori, Francesco Saccoliti, Valeria Tudino, Alessandro De Leo, Martina Bortolami, Luigi Scipione, Roberta Costi, Silvia Rivara, Laura Scalvini, Marco Mor, Fabiana Fosca Ferrara, Emiliano Pavoni, Giuseppe Roscilli, Giuliana Cassinelli, Ferdinando M Milazzo, Gianfranco Battistuzzi, Roberto Di Santo, Giuseppe Giannini
Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity. Journal of medicinal chemistry 61 (15) (2018)
Antonella Messore, Valentina Noemi Madia, Luca Pescatori, Francesco Saccoliti, Valeria Tudino, Alessandro De Leo, Martina Bortolami, Daniela De Vita, Luigi Scipione, Federico Pepi, Roberta Costi, Silvia Rivara, Laura Scalvini, Marco Mor, Fabiana Fosca Ferrara, Emiliano Pavoni, Giuseppe Roscilli, Giuliana Cassinelli, Ferdinando M Milazzo, Gianfranco Battistuzzi, Roberto Di Santo, Giuseppe Giannini
Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity. Journal of medicinal chemistry 61 (23) (2018)
Valentina Noemi Madia, Antonella Messore, Luca Pescatori, Francesco Saccoliti, Valeria Tudino, Alessandro De Leo, Luigi Scipione, Lucia Fiore, Eric Rhoden, Fabrizio Manetti, M Steven Oberste, Roberto Di Santo, Roberta Costi
In Vitro Antiviral Activity of New Oxazoline Derivatives as Potent Poliovirus Inhibitors. Journal of medicinal chemistry 62 (2) (2018)
Valentina Noemi Madia, Rosaria Benedetti, Maria Letizia Barreca, Liza Ngo, Luca Pescatori, Antonella Messore, Giovanni Pupo, Francesco Saccoliti, Sergio Valente, Antonello Mai, Luigi Scipione, Yujun George Zheng, Cristina Tintori, Maurizio Botta, Violetta Cecchetti, Lucia Altucci, Roberto Di Santo, Roberta Costi
Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase. ChemMedChem 12 (16) (2017)
Daniela De Vita, Andrea Angeli, Fabiana Pandolfi, Martina Bortolami, Roberta Costi, Roberto Di Santo, Elisabetta Suffredini, Mariangela Ceruso, Sonia Del Prete, Clemente Capasso, Luigi Scipione, Claudiu T Supuran
Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties. Journal of enzyme inhibition and medicinal chemistry 32 (1) (2017)