Sandro Cosconati

Scopus Author ID Loop profile ResearcherID ORCID

Publication Activity (10 Years)

Years Active: 2014-2024
Publications (10 Years): 34

Top Venues

Journal of medicinal chemistry

Journal of chemical information and modeling

ACS medicinal chemistry letters

Journal of enzyme inhibition and medicinal chemistry

University of Campania "Luigi Vanvitelli"

Universita degli Studi di Napoli Federico II (PHD)

This page only lists publications with an associated author ORCID identifier.

Affiliation History

University of Campania "Luigi Vanvitelli" Nov 01 2017

Italy

Associate Professor :: DiSTABiF

University of Campania "Luigi Vanvitelli" Mar 01 2011

Italy

Assistant Professor :: DiSTABiF

Education History

Universita degli Studi di Napoli Federico II Dec 01 2003 - Dec 21 2006

Italy

PHD :: Pharmacy

Publications

Santo Previti, Roberta Ettari, Elsa Calcaterra, Michele Roggia, Benito Natale, Annabelle Carolin Weldert, Christin Müller-Ruttloff, Florian Salisch, Anna Irto, Rosalia Maria Cigala, John Ziebuhr, Tanja Schirmeister, Sandro Cosconati, Maria Zappalà
Identification of Dual Inhibitors Targeting Main Protease (M pro ) and Cathepsin L as Potential Anti-SARS-CoV-2 Agents. ACS medicinal chemistry letters 15 (5) (2024)
Michele Roggia, Benito Natale, Giorgio Amendola, Nicola Grasso, Salvatore Di Maro, Sabrina Taliani, Sabrina Castellano, Serena Concetta Rita Reina, Erica Salvati, Jussara Amato, Sandro Cosconati
Discovering Dually Active Anti-cancer Compounds with a Hybrid AI-structure-based Approach. Journal of chemical information and modeling (2024)
Carla Di Chio, Josè Starvaggi, Noemi Totaro, Santo Previti, Benito Natale, Sandro Cosconati, Marta Bogacz, Tanja Schirmeister, Jenny Legac, Philip J Rosenthal, Maria Zappalà, Roberta Ettari
Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria. International journal of molecular sciences 25 (8) (2024)
Santo Previti, Roberta Ettari, Elsa Calcaterra, Michele Roggia, Benito Natale, Annabelle Carolin Weldert, Christin Müller-Ruttloff, Florian Salisch, Anna Irto, Rosalia Maria Cigala, John Ziebuhr, Tanja Schirmeister, Sandro Cosconati, Maria Zappalà
Identification of Dual Inhibitors Targeting Main Protease (M pro ) and Cathepsin L as Potential Anti-SARS-CoV-2 Agents. ACS medicinal chemistry letters 15 (5) (2024)
Carla Di Chio, Josè Starvaggi, Noemi Totaro, Santo Previti, Benito Natale, Sandro Cosconati, Marta Bogacz, Tanja Schirmeister, Jenny Legac, Philip J Rosenthal, Maria Zappalà, Roberta Ettari
Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria. International journal of molecular sciences 25 (8) (2024)
Carla Di Chio, Josè Starvaggi, Noemi Totaro, Santo Previti, Benito Natale, Sandro Cosconati, Marta Bogacz, Tanja Schirmeister, Jenny Legac, Philip J Rosenthal, Maria Zappalà, Roberta Ettari
Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria. International journal of molecular sciences 25 (8) (2024)
Elisa Patacchini, Valentina Noemi Madia, Aurora Albano, Giuseppe Ruggieri, Antonella Messore, Davide Ialongo, Francesco Saccoliti, Luigi Scipione, Sandro Cosconati, Pratibha C Koneru, Reed Haney, Mamuka Kvaratskhelia, Roberto Di Santo, Roberta Costi
Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions. ACS medicinal chemistry letters 15 (9) (2024)
Alessandra Feoli, Giulia Iannelli, Alessandra Cipriano, Ciro Milite, Lei Shen, Zhihao Wang, Andrea Hadjikyriacou, Troy L Lowe, Cyrus Safaeipour, Monica Viviano, Giuliana Sarno, Elva Morretta, Maria Chiara Monti, Yanzhong Yang, Steven G Clarke, Sandro Cosconati, Sabrina Castellano, Gianluca Sbardella
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor. Journal of medicinal chemistry (2023)
Michele Roggia, Benito Natale, Giorgio Amendola, Salvatore Di Maro, Sandro Cosconati
Streamlining Large Chemical Library Docking with Artificial Intelligence: the PyRMD2Dock Approach. Journal of chemical information and modeling (2023)
Stefano Tomassi, Marilisa Pia Dimmito, Minying Cai, Antonia D'Aniello, Alessandra Del Bene, Anna Messere, Zekun Liu, Tingyi Zhu, Victor J Hruby, Azzurra Stefanucci, Sandro Cosconati, Adriano Mollica, Salvatore Di Maro
CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists. Journal of medicinal chemistry 65 (5) (2022)
Santo Previti, Roberta Ettari, Carla Di Chio, Rahul Ravichandran, Marta Bogacz, Ute A Hellmich, Tanja Schirmeister, Sandro Cosconati, Maria Zappalà
Development of Reduced Peptide Bond Pseudopeptide Michael Acceptors for the Treatment of Human African Trypanosomiasis. Molecules (Basel, Switzerland) 27 (12) (2022)
Santo Previti, Roberta Ettari, Elsa Calcaterra, Carla Di Chio, Rahul Ravichandran, Collin Zimmer, Stefan Hammerschmidt, Annika Wagner, Marta Bogacz, Sandro Cosconati, Tanja Schirmeister, Maria Zappalà
Development of Urea-Bond-Containing Michael Acceptors as Antitrypanosomal Agents Targeting Rhodesain. ACS medicinal chemistry letters 13 (7) (2022)
Valentina Albanese, Chiara Ruzza, Erika Marzola, Tatiana Bernardi, Martina Fabbri, Anna Fantinati, Claudio Trapella, Rainer K Reinscheid, Federica Ferrari, Chiara Sturaro, Girolamo Calò, Giorgio Amendola, Sandro Cosconati, Salvatore Pacifico, Remo Guerrini, Delia Preti
Structure-Activity Relationship Studies on Oxazolo[3,4-a]pyrazine Derivatives Leading to the Discovery of a Novel Neuropeptide S Receptor Antagonist with Potent In Vivo Activity. Journal of medicinal chemistry 64 (7) (2021)
Giorgio Amendola, Sandro Cosconati
PyRMD: A New Fully Automated AI-Powered Ligand-Based Virtual Screening Tool. Journal of chemical information and modeling 61 (8) (2021)
Giorgio Amendola, Roberta Ettari, Santo Previti, Carla Di Chio, Anna Messere, Salvatore Di Maro, Stefan J Hammerschmidt, Collin Zimmer, Robert A Zimmermann, Tanja Schirmeister, Maria Zappalà, Sandro Cosconati
Lead Discovery of SARS-CoV-2 Main Protease Inhibitors through Covalent Docking-Based Virtual Screening. Journal of chemical information and modeling 61 (4) (2021)
Antonella Messore, Angela Corona, Valentina Noemi Madia, Francesco Saccoliti, Valeria Tudino, Alessandro De Leo, Davide Ialongo, Luigi Scipione, Daniela De Vita, Giorgio Amendola, Ettore Novellino, Sandro Cosconati, Mathieu Métifiot, Marie-Line Andreola, Francesca Esposito, Nicole Grandi, Enzo Tramontano, Roberta Costi, Roberto Di Santo
Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase. Journal of medicinal chemistry 64 (12) (2021)
Emma Baglini, Rahul Ravichandran, Emanuela Berrino, Silvia Salerno, Elisabetta Barresi, Anna Maria Marini, Monica Viviano, Sabrina Castellano, Federico Da Settimo, Claudiu T Supuran, Sandro Cosconati, Sabrina Taliani
Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Elisabetta Barresi, Rahul Ravichandran, Lorenzo Germelli, Andrea Ageli, Emma Baglini, Silvia Salerno, Anna Maria Marini, Barbara Costa, Eleonora Da Pozzo, Claudia Martini, Federico Da Settimo, Claudiu T Supuran, Sandro Cosconati, Sabrina Taliani
Carbonic anhydrase activation profile of indole-based derivatives. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Stamatia Zavitsanou, Alexandros Tsengenes, Michail Papadourakis, Giorgio Amendola, Alexios Chatzigoulas, Dimitris Dellis, Sandro Cosconati, Zoe Cournia
FEPrepare: A Web-Based Tool for Automating the Setup of Relative Binding Free Energy Calculations. Journal of chemical information and modeling 61 (9) (2021)
Agostino Bruno, Elisabetta Barresi, Nicola Simola, Eleonora Da Pozzo, Barbara Costa, Ettore Novellino, Federico Da Settimo, Claudia Martini, Sabrina Taliani, Sandro Cosconati
Unbinding of Translocator Protein 18 kDa (TSPO) Ligands: From in Vitro Residence Time to in Vivo Efficacy via in Silico Simulations. ACS chemical neuroscience 10 (8) (2019)
Rosaria Benedetti, Carmela Dell'Aversana, Tommaso De Marchi, Dante Rotili, Ning Qing Liu, Boris Novakovic, Serena Boccella, Salvatore Di Maro, Sandro Cosconati, Alfonso Baldi, Emma Niméus, Johan Schultz, Urban Höglund, Sabatino Maione, Chiara Papulino, Ugo Chianese, Francesco Iovino, Antonio Federico, Antonello Mai, Hendrik G Stunnenberg, Angela Nebbioso, Lucia Altucci
Inhibition of Histone Demethylases LSD1 and UTX Regulates ERα Signaling in Breast Cancer. Cancers 11 (12) (2019)
Ciro Milite, Giorgio Amendola, Alessio Nocentini, Silvia Bua, Alessandra Cipriano, Elisabetta Barresi, Alessandra Feoli, Ettore Novellino, Federico Da Settimo, Claudiu T Supuran, Sabrina Castellano, Sandro Cosconati, Sabrina Taliani
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies. Journal of enzyme inhibition and medicinal chemistry 34 (1) (2019)
Ciro Milite, Alessandra Feoli, John R Horton, Donatella Rescigno, Alessandra Cipriano, Vincenzo Pisapia, Monica Viviano, Giacomo Pepe, Giorgio Amendola, Ettore Novellino, Sandro Cosconati, Xiaodong Cheng, Sabrina Castellano, Gianluca Sbardella
Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1/2 (GLP/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal Structure. Journal of medicinal chemistry 62 (5) (2019)
Roberta Ettari, Santo Previti, Santina Maiorana, Giorgio Amendola, Annika Wagner, Sandro Cosconati, Tanja Schirmeister, Ute A Hellmich, Maria Zappalà
Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis. Journal of medicinal chemistry 62 (23) (2019)
Francesco Merlino, Stefano Tomassi, Ali M Yousif, Anna Messere, Luciana Marinelli, Paolo Grieco, Ettore Novellino, Sandro Cosconati, Salvatore Di Maro
Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication. Organic letters 21 (16) (2019)
Silvia Salerno, Elisabetta Barresi, Giorgio Amendola, Emanuela Berrino, Ciro Milite, Anna Maria Marini, Federico Da Settimo, Ettore Novellino, Claudiu T Supuran, Sandro Cosconati, Sabrina Taliani
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors. Journal of medicinal chemistry 61 (13) (2018)
Barbara Cosimelli, Giovanni Greco, Sonia Laneri, Ettore Novellino, Antonia Sacchi, Simona Collina, Daniela Rossi, Sandro Cosconati, Elisabetta Barresi, Sabrina Taliani, Maria Letizia Trincavelli, Claudia Martini
Studies on enantioselectivity of chiral 4-acetylamino-6-alkyloxy-2-alkylthiopyrimidines acting as antagonists of the human A3 adenosine receptor. MedChemComm 9 (1) (2017)
Mariateresa Giustiniano, Simona Daniele, Sveva Pelliccia, Valeria La Pietra, Deborah Pietrobono, Diego Brancaccio, Sandro Cosconati, Anna Messere, Stefano Giuntini, Linda Cerofolini, Marco Fragai, Claudio Luchinat, Sabrina Taliani, Giuseppe La Regina, Federico Da Settimo, Romano Silvestri, Claudia Martini, Ettore Novellino, Luciana Marinelli
Computer-Aided Identification and Lead Optimization of Dual Murine Double Minute 2 and 4 Binders: Structure-Activity Relationship Studies and Pharmacological Activity. Journal of medicinal chemistry 60 (19) (2017)
Erica Salvati, Lorenzo Botta, Jussara Amato, Francesco Saverio Di Leva, Pasquale Zizza, Antimo Gioiello, Bruno Pagano, Grazia Graziani, Madalena Tarsounas, Antonio Randazzo, Ettore Novellino, Annamaria Biroccio, Sandro Cosconati
Lead Discovery of Dual G-Quadruplex Stabilizers and Poly(ADP-ribose) Polymerases (PARPs) Inhibitors: A New Avenue in Anticancer Treatment. Journal of medicinal chemistry 60 (9) (2017)
Ciro Milite, Elisabetta Barresi, Eleonora Da Pozzo, Barbara Costa, Monica Viviano, Amalia Porta, Anna Messere, Gianluca Sbardella, Federico Da Settimo, Ettore Novellino, Sandro Cosconati, Sabrina Castellano, Sabrina Taliani, Claudia Martini
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO). Journal of medicinal chemistry 60 (18) (2017)
Santo Previti, Roberta Ettari, Sandro Cosconati, Giorgio Amendola, Khawla Chouchene, Annika Wagner, Ute A Hellmich, Kathrin Ulrich, R Luise Krauth-Siegel, Peter Richard Wich, Ira Schmid, Tanja Schirmeister, Jiri Gut, Philip J Rosenthal, Silvana Grasso, Maria Zappalà
Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs). Journal of medicinal chemistry 60 (16) (2017)
Floriana Morgillo, Giorgio Amendola, Carminia Maria Della Corte, Chiara Giacomelli, Lorenzo Botta, Salvatore Di Maro, Anna Messere, Vincenza Ciaramella, Sabrina Taliani, Luciana Marinelli, Maria Letizia Trincavelli, Claudia Martini, Ettore Novellino, Fortunato Ciardiello, Sandro Cosconati
Dual MET and SMO Negative Modulators Overcome Resistance to EGFR Inhibitors in Human Nonsmall Cell Lung Cancer. Journal of medicinal chemistry 60 (17) (2017)
Antonio Laezza, Angela Casillo, Sandro Cosconati, Caroline I Biggs, Antonio Fabozzi, Luigi Paduano, Alfonso Iadonisi, Ettore Novellino, Matthew I Gibson, Antonio Randazzo, Maria M Corsaro, Emiliano Bedini
Decoration of Chondroitin Polysaccharide with Threonine: Synthesis, Conformational Study, and Ice-Recrystallization Inhibition Activity. Biomacromolecules 18 (8) (2017)
Teresa Rivera, Candy Haggblom, Sandro Cosconati, Jan Karlseder
A balance between elongation and trimming regulates telomere stability in stem cells. Nature structural & molecular biology 24 (1) (2016)
Maria Gaglione, M Emilia Mercurio, Nicoletta Potenza, Nicola Mosca, Aniello Russo, Ettore Novellino, Sandro Cosconati, Anna Messere
Synthesis and gene silencing properties of siRNAs containing terminal amide linkages. BioMed research international 2014 (2014)

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Publication Activity (10 Years)

Top Topics

Top Venues

Sandro Cosconati