Paola Gratteri (P Gratteri)

ResearcherID Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2016-2024
Publications (10 Years): 68

Top Venues

Journal of enzyme inhibition and medicinal chemistry

Journal of medicinal chemistry

International journal of molecular sciences

Molecules (Basel, Switzerland)

University of Firenze

This page only lists publications with an associated author ORCID identifier.

Affiliation History

University of Firenze

Italy

Associate Professor :: NEUROFARBA

Publications

Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry 67 (5) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry 67 (11) (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry 67 (5) (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T Supuran, Antonio Randazzo, Paola Gratteri
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Alessio Nocentini, Alessia Costa, Alessandro Bonardi, Andrea Ammara, Simone Giovannuzzi, Andrea Petreni, Gianluca Bartolucci, Barbara Rani, Manuela Leri, Monica Bucciantini, José G Fernández-Bolaños, Óscar López, Maria Beatrice Passani, Gustavo Provensi, Paola Gratteri, Claudiu T Supuran
Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases. Journal of medicinal chemistry (2024)
Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids. Journal of enzyme inhibition and medicinal chemistry 39 (1) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Morteza Abdoli, Alessandro Bonardi, Niccolò Paoletti, Ashok Aspatwar, Seppo Parkkila, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N -((4-Sulfamoylphenyl)carbamothioyl) Amides. Molecules (Basel, Switzerland) 28 (10) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Mudasir Nabi Peerzada, Daniela Vullo, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Amir Azam
Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors. ACS medicinal chemistry letters 14 (6) (2023)
Marjan Sobati, Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T Supuran, Raivis Žalubovskis
Inhibition Profiles of Some Novel Sulfonamide-Incorporated α-Aminophosphonates on Human Carbonic Anhydrases. ACS medicinal chemistry letters 14 (8) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Davide Ialongo, Antonella Messore, Valentina Noemi Madia, Valeria Tudino, Alessio Nocentini, Paola Gratteri, Simone Giovannuzzi, Claudiu T Supuran, Alice Nicolai, Susanna Scarpa, Samanta Taurone, Michele Camarda, Marco Artico, Veronica Papa, Francesco Saccoliti, Luigi Scipione, Roberto Di Santo, Roberta Costi
Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII. Pharmaceuticals (Basel, Switzerland) 16 (2) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Alessio Nocentini, Alessandro Bonardi, Carla Bazzicalupi, Vincenzo Alterio, Davide Esposito, Simona Maria Monti, Michael Smietana, Giuseppina De Simone, Claudiu T Supuran, Paola Gratteri, Jean-Yves Winum
6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography. Journal of medicinal chemistry (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Alessandro Bonardi, Laura Micheli, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Development of Hydrogen Sulfide-Releasing Carbonic Anhydrases IX- and XII-Selective Inhibitors with Enhanced Antihyperalgesic Action in a Rat Model of Arthritis. Journal of medicinal chemistry 65 (19) (2022)
Carla Bazzicalupi, Alessandro Bonardi, Tarita Biver, Marta Ferraroni, Francesco Papi, Matteo Savastano, Paolo Lombardi, Paola Gratteri
Probing the Efficiency of 13-Pyridylalkyl Berberine Derivatives to Human Telomeric G-Quadruplexes Binding: Spectroscopic, Solid State and In Silico Analysis. International journal of molecular sciences 23 (22) (2022)
Alessandro Bonardi, Alessio Nocentini, Sameh Mohamed Osman, Fatmah Ali Alasmary, Tahani Mazyad Almutairi, Dalal Saied Abdullah, Paola Gratteri, Claudiu T Supuran
Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs - a joint docking/molecular dynamics study. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Rossella Grande, Simone Carradori, Valentina Puca, Irene Vitale, Andrea Ageli, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Paola Lanuti, Giuseppina Bologna, Pasquale Simeone, Clemente Capasso, Viviana De Luca, Claudiu T Supuran
Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles. International journal of molecular sciences 22 (21) (2021)
Matteo Savastano, Matteo Fiaschi, Giovanni Ferraro, Paola Gratteri, Palma Mariani, Antonio Bianchi, Carla Bazzicalupi
Sensing Zn2+ in Aqueous Solution with a Fluorescent Scorpiand Macrocyclic Ligand Decorated with an Anthracene Bearing Tail. Molecules (Basel, Switzerland) 25 (6) (2020)
Giang Thi Huong Nguyen, Alessio Nocentini, Andrea Ageli, Paola Gratteri, Claudiu T Supuran, W Alexander Donald
Perfluoroalkyl Substances of Significant Environmental Concern Can Strongly Inhibit Human Carbonic Anhydrase Isozymes. Analytical chemistry 92 (6) (2020)
Giacomo Picci, Carla Bazzicalupi, Simon J Coles, Paola Gratteri, Francesco Isaia, Vito Lippolis, Riccardo Montis, Sergio Murgia, Alessio Nocentini, James B Orton, Claudia Caltagirone
Halogenated isophthalamides and dipicolineamides: the role of the halogen substituents in the anion binding properties. Dalton transactions (Cambridge, England : 2003) 49 (27) (2020)
Alessio Nocentini, Vincenzo Alterio, Silvia Bua, Laura Micheli, Davide Esposito, Martina Buonanno, Gianluca Bartolucci, Sameh M Osman, Zeid Abdullah ALOthman, Roberto Cirilli, Marco Pierini, Simona Maria Monti, Lorenzo Di Cesare Mannelli, Paola Gratteri, Carla Ghelardini, Giuseppina De Simone, Claudiu T Supuran
Phenyl(thio)phosphon(amid)ate Benzenesulfonamides as Potent and Selective Inhibitors of Human Carbonic Anhydrases II and VII Counteract Allodynia in a Mouse Model of Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 63 (10) (2020)
Alessandro Bonardi, Alessio Nocentini, Silvia Bua, Jacob Combs, Carrie L Lomelino, Jacob T Andring, Laura Lucarini, Silvia Sgambellone, Emanuela Masini, Robert McKenna, Paola Gratteri, Claudiu T Supuran
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of Action. Journal of medicinal chemistry 63 (13) (2020)
Matteo Savastano, Celeste García-Gallarín, Claudia Giorgi, Paola Gratteri, Maria Dolores López de la Torre, Carla Bazzicalupi, Antonio Bianchi, Beatriz Sánchez-Calvo
Solid State and Solution Study on the Formation of Inorganic Anion Complexes with a Series of Tetrazine-Based Ligands. Molecules (Basel, Switzerland) 24 (12) (2019)
Dina Manetti, Alexandra Garifulina, Gianluca Bartolucci, Carla Bazzicalupi, Cristina Bellucci, Niccolò Chiaramonte, Silvia Dei, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Paola Gratteri, Ekaterina Spirova, Irina Shelukhina, Elisabetta Teodori, Katia Varani, Victor Tsetlin, Maria Novella Romanelli
New Rigid Nicotine Analogues, Carrying a Norbornane Moiety, Are Potent Agonists of α7 and α3* Nicotinic Receptors. Journal of medicinal chemistry 62 (4) (2019)
Mohamed A Abdelrahman, Wagdy M Eldehna, Alessio Nocentini, Silvia Bua, Sara T Al-Rashood, Ghada S Hassan, Alessandro Bonardi, Abdulrahman A Al-Mehizia, Hamad M Alkahtani, Amal Alharbi, Paola Gratteri, Claudiu T Supuran
Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights. International journal of molecular sciences 20 (10) (2019)
Silvia Bua, Laura Lucarini, Laura Micheli, Marta Menicatti, Gianluca Bartolucci, Silvia Selleri, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Emanuela Masini, Fabrizio Carta, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Bioisosteric Development of Multitarget Nonsteroidal Anti-Inflammatory Drug-Carbonic Anhydrases Inhibitor Hybrids for the Management of Rheumatoid Arthritis. Journal of medicinal chemistry 63 (5) (2019)
Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide-Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors. Chemistry (Weinheim an der Bergstrasse, Germany) 25 (5) (2018)
Alessio Nocentini, Elena Trallori, Srishti Singh, Carrie L Lomelino, Gianluca Bartolucci, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Robert McKenna, Paola Gratteri, Claudiu T Supuran
4-Hydroxy-3-nitro-5-ureido-benzenesulfonamides Selectively Target the Tumor-Associated Carbonic Anhydrase Isoforms IX and XII Showing Hypoxia-Enhanced Antiproliferative Profiles. Journal of medicinal chemistry 61 (23) (2018)
Alessio Nocentini, Mariangela Ceruso, Silvia Bua, Carrie L Lomelino, Jacob T Andring, Robert McKenna, Cecilia Lanzi, Silvia Sgambellone, Riccardo Pecori, Rosanna Matucci, Luca Filippi, Paola Gratteri, Fabrizio Carta, Emanuela Masini, Silvia Selleri, Claudiu T Supuran
Discovery of β-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy. Journal of medicinal chemistry 61 (12) (2018)
Alessio Nocentini, Fabrizio Carta, Muhammet Tanc, Silvia Selleri, Claudiu T Supuran, Carla Bazzicalupi, Paola Gratteri
Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies. Chemistry (Weinheim an der Bergstrasse, Germany) 24 (31) (2018)
Marco Fragai, Giuseppina Comito, Lorenzo Di Cesare Mannelli, Roberta Gualdani, Vito Calderone, Alexandra Louka, Barbara Richichi, Oscar Francesconi, Andrea Angeli, Alessio Nocentini, Paola Gratteri, Paola Chiarugi, Carla Ghelardini, Francesco Tadini-Buoninsegni, Claudiu T Supuran, Cristina Nativi
Lipoyl-Homotaurine Derivative (ADM_12) Reverts Oxaliplatin-Induced Neuropathy and Reduces Cancer Cells Malignancy by Inhibiting Carbonic Anhydrase IX (CAIX). Journal of medicinal chemistry 60 (21) (2017)
Julia Wirmer-Bartoschek, Lars Erik Bendel, Hendrik R A Jonker, J Tassilo Grün, Francesco Papi, Carla Bazzicalupi, Luigi Messori, Paola Gratteri, Harald Schwalbe
Solution NMR Structure of a Ligand/Hybrid-2-G-Quadruplex Complex Reveals Rearrangements that Affect Ligand Binding. Angewandte Chemie (International ed. in English) 56 (25) (2017)
F Papi, M Ferraroni, R Rigo, S Da Ros, C Bazzicalupi, Claudia Sissi, Paola Gratteri
Role of the Benzodioxole Group in the Interactions between the Natural Alkaloids Chelerythrine and Coptisine and the Human Telomeric G-Quadruplex DNA. A Multiapproach Investigation. Journal of natural products 80 (12) (2017)
Marta Ferraroni, Carla Bazzicalupi, Francesco Papi, Gaetano Fiorillo, Luis Miguel Guamán-Ortiz, Alessio Nocentini, Anna Ivana Scovassi, Paolo Lombardi, Paola Gratteri
Solution and Solid-State Analysis of Binding of 13-Substituted Berberine Analogues to Human Telomeric G-quadruplexes. Chemistry, an Asian journal 11 (7) (2016)

Paola Gratteri.css-eqlu8i{font-size:small;padding-left:4px;} (P Gratteri)

Publication Activity (10 Years)

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Paola Gratteri (P Gratteri)