Alessio Nocentini

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 122

Top Venues

Journal of enzyme inhibition and medicinal chemistry

Journal of medicinal chemistry

International journal of molecular sciences

Molecules (Basel, Switzerland)

This page only lists publications with an associated author ORCID identifier.

Publications

Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Silvia Bua, Alessio Nocentini, Alessandro Bonardi, Giuseppe Palma, Giulia Ciampi, Angela Giliberti, Federica Iannelli, Francesca Bruzzese, Claudiu T Supuran, Filomena de Nigris
Harnessing Nitric Oxide-Donating Benzofuroxans for Targeted Inhibition of Carbonic Anhydrase IX in Cancer. Journal of medicinal chemistry (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry 67 (5) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry 67 (11) (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Silvia Bua, Alessandro Bonardi, Georgiana Ramona Mük, Alessio Nocentini, Paola Gratteri, Claudiu T Supuran
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains. International journal of molecular sciences 25 (5) (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry 67 (5) (2024)
Molly S Youse, Nader S Abutaleb, Alessio Nocentini, Abdallah S Abdelsattar, Farman Ali, Claudiu T Supuran, Mohamed N Seleem, Daniel P Flaherty
Optimization of Ethoxzolamide Analogs with Improved Pharmacokinetic Properties for In Vivo Efficacy against Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T Supuran
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction. Journal of medicinal chemistry (2024)
Haytham O Tawfik, Mohamed M Saleh, Andrea Ammara, Eman F Khaleel, Rehab Badi, Yomna T T Khater, Rabab Ahmed Rasheed, Ahmed A Attia, Salma M Hefny, Eslam B Elkaeed, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna, Moataz A Shaldam
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma. Journal of medicinal chemistry 67 (2) (2024)
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, Niccolò Paoletti, Andrea Ammara, Silvia Bua, Nader S Abutaleb, Abdallah S Abdelsattar, Clemente Capasso, Paola Gratteri, Daniel P Flaherty, Mohamed N Seleem, Claudiu T Supuran
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae . Journal of medicinal chemistry (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Haytham O Tawfik, Mohamed M Saleh, Andrea Ammara, Eman F Khaleel, Rehab Badi, Yomna T T Khater, Rabab Ahmed Rasheed, Ahmed A Attia, Salma M Hefny, Eslam B Elkaeed, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna, Moataz A Shaldam
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma. Journal of medicinal chemistry (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Gianluca Bartolucci, Marta Menicatti, Marialessandra Contino, Nicola Antonio Colabufo, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Elisabetta Teodori
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. Molecules (Basel, Switzerland) 29 (14) (2024)
Alessio Nocentini, Alessia Costa, Alessandro Bonardi, Andrea Ammara, Simone Giovannuzzi, Andrea Petreni, Gianluca Bartolucci, Barbara Rani, Manuela Leri, Monica Bucciantini, José G Fernández-Bolaños, Óscar López, Maria Beatrice Passani, Gustavo Provensi, Paola Gratteri, Claudiu T Supuran
Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases. Journal of medicinal chemistry (2024)
Haytham O Tawfik, Mohamed M Saleh, Andrea Ammara, Eman F Khaleel, Rehab Badi, Yomna T T Khater, Rabab Ahmed Rasheed, Ahmed A Attia, Salma M Hefny, Eslam B Elkaeed, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna, Moataz A Shaldam
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma. Journal of medicinal chemistry 67 (2) (2024)
Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Doretta Cuffaro, Riccardo Di Leo, Lidia Ciccone, Alessio Nocentini, Claudiu T Supuran, Elisa Nuti, Armando Rossello
New isoxazolidinyl-based N -alkylethanolamines as new activators of human brain carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Doretta Cuffaro, Riccardo Di Leo, Lidia Ciccone, Alessio Nocentini, Claudiu T Supuran, Elisa Nuti, Armando Rossello
New isoxazolidinyl-based N -alkylethanolamines as new activators of human brain carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Carbonic Anhydrase Inhibitors as Novel Antibacterials in the Era of Antibiotic Resistance: Where Are We Now? Antibiotics (Basel, Switzerland) 12 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T Supuran, Raivis Žalubovskis
Aryl derivatives of 3 H -1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Ashraf K El-Damasy, Hyun Ji Kim, Alessio Nocentini, Seon Hee Seo, Wagdy M Eldehna, Eun-Kyoung Bang, Claudiu T Supuran, Gyochang Keum
Discovery of new 6-ureido/amidocoumarins as highly potent and selective inhibitors for the tumour-relevant carbonic anhydrases IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Mónica Martínez-Montiel, Laura L Romero-Hernández, Simone Giovannuzzi, Paloma Begines, Adrián Puerta, Ana I Ahuja-Casarín, Miguel X Fernandes, Penélope Merino-Montiel, Sara Montiel-Smith, Alessio Nocentini, José Manuel Padrón, Claudiu T Supuran, José G Fernández-Bolaños, Óscar López
Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (11) (2023)
Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T Supuran, Antonello Mai
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T Supuran
Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T Supuran
Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Davide Ialongo, Antonella Messore, Valentina Noemi Madia, Valeria Tudino, Alessio Nocentini, Paola Gratteri, Simone Giovannuzzi, Claudiu T Supuran, Alice Nicolai, Susanna Scarpa, Samanta Taurone, Michele Camarda, Marco Artico, Veronica Papa, Francesco Saccoliti, Luigi Scipione, Roberto Di Santo, Roberta Costi
Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII. Pharmaceuticals (Basel, Switzerland) 16 (2) (2023)
Jekateri Na Ivanova, Alessio Nocentini, Kaspars Tars, Ja Nis Leita Ns, Elviss Dvinskis, Andris Kazaks, Ilona Domračeva, Claudiu T Supuran, Raivis Žalubovskis
Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect. Journal of medicinal chemistry (2023)
Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T Supuran
Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Ahmed E Elsawi, Mostafa M Elbadawi, Alessio Nocentini, Hadia Almahli, Simone Giovannuzzi, Moataz A Shaldam, Rofaida Salem, Tamer M Ibrahim, Hatem A Abdel-Aziz, Claudiu T Supuran, Wagdy M Eldehna
1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory Activities. Journal of medicinal chemistry (2023)
Domiziana Masci, Michela Puxeddu, Laura Di Magno, Michele D'Ambrosio, Anastasia Parisi, Marianna Nalli, Ruoli Bai, Antonio Coluccia, Pietro Sciò, Viviana Orlando, Sara D'Angelo, Stefano Biagioni, Andrea Urbani, Ernest Hamel, Alessio Nocentini, Serena Filiberti, Marta Turati, Roberto Ronca, Joanna Kopecka, Chiara Riganti, Cinzia Fionda, Rosa Bordone, Giorgia Della Rocca, Gianluca Canettieri, Claudiu T Supuran, Romano Silvestri, Giuseppe La Regina
4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1 H -pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activity against Multidrug Resistant Cancer Cells. Journal of medicinal chemistry (2023)
Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Carbonic Anhydrase Inhibitors as Novel Antibacterials in the Era of Antibiotic Resistance: Where Are We Now? Antibiotics (Basel, Switzerland) 12 (1) (2023)
Alessio Nocentini, Alessandro Bonardi, Carla Bazzicalupi, Vincenzo Alterio, Davide Esposito, Simona Maria Monti, Michael Smietana, Giuseppina De Simone, Claudiu T Supuran, Paola Gratteri, Jean-Yves Winum
6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography. Journal of medicinal chemistry (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Alma Fuentes-Aguilar, Penélope Merino-Montiel, Sara Montiel-Smith, Socorro Meza-Reyes, José Luis Vega-Báez, Adrián Puerta, Miguel X Fernandes, José M Padrón, Andrea Petreni, Alessio Nocentini, Claudiu T Supuran, Óscar López, José G Fernández-Bolaños
2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Anil Kumar Marapaka, Alessio Nocentini, Molly S Youse, Weiwei An, Katrina J Holly, Chittaranjan Das, Ravi Yadav, Mohamed N Seleem, Claudiu T Supuran, Daniel P Flaherty
Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to Neisseria gonorrhoeae α-Carbonic Anhydrase. ACS medicinal chemistry letters 14 (1) (2022)
Simone Giovannuzzi, Chad S Hewitt, Alessio Nocentini, Clemente Capasso, Daniel P Flaherty, Claudiu T Supuran
Coumarins effectively inhibit bacterial α-carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Alessio Nocentini, Alessandro Bonardi, Simone Pratesi, Paola Gratteri, Carlo Dani, Claudiu T Supuran
Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubin. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Tarfah Al-Warhi, Mostafa M Elbadawi, Alessandro Bonardi, Alessio Nocentini, Ahmed Ali Al-Karmalawy, Nada Aljaeed, Ohoud J Alotaibi, Hatem A Abdel-Aziz, Claudiu T Supuran, Wagdy M Eldehna
Design and synthesis of benzothiazole-based SLC-0111 analogues as new inhibitors for the cancer-associated carbonic anhydrase isoforms IX and XII. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Silvia Mussi, Sara Rezzola, Paola Chiodelli, Alessio Nocentini, Claudiu T Supuran, Roberto Ronca
Antiproliferative effects of sulphonamide carbonic anhydrase inhibitors C18, SLC-0111 and acetazolamide on bladder, glioblastoma and pancreatic cancer cell lines. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Adel S El-Azab, Alaa A-M Abdel-Aziz, Hazem A Ghabbour, Silvia Bua, Alessio Nocentini, Hamad M Al Kahtani, Nawaf A Alsaif, Mohamed H M Al-Agamy, Claudiu T Supuran
Carbonic Anhydrase Inhibition Activities of Schiff's Bases Based on Quinazoline-Linked Benzenesulfonamide. Molecules (Basel, Switzerland) 27 (22) (2022)
Simone Giovannuzzi, Clemente Capasso, Alessio Nocentini, Claudiu T Supuran
Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII. Molecules (Basel, Switzerland) 27 (13) (2022)
Aleksandrs Pustenko, Anastasija Balašova, Alessio Nocentini, Claudiu T Supuran, Raivis Žalubovskis
3 H -1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2022)
Simone Giovannuzzi, Nader S Abutaleb, Chad S Hewitt, Fabrizio Carta, Alessio Nocentini, Mohamed N Seleem, Daniel P Flaherty, Claudiu T Supuran
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae . Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Nader S Abutaleb, Ahmed E M Elhassanny, Alessio Nocentini, Chad S Hewitt, Ahmed Elkashif, Bruce R Cooper, Claudiu T Supuran, Mohamed N Seleem, Daniel P Flaherty
Repurposing FDA-approved sulphonamide carbonic anhydrase inhibitors for treatment of Neisseria gonorrhoeae . Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Alessandro Bonardi, Laura Micheli, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Paola Gratteri, Alessio Nocentini, Claudiu T Supuran
Development of Hydrogen Sulfide-Releasing Carbonic Anhydrases IX- and XII-Selective Inhibitors with Enhanced Antihyperalgesic Action in a Rat Model of Arthritis. Journal of medicinal chemistry 65 (19) (2022)
Laura Braconi, Elisabetta Teodori, Chiara Riganti, Marcella Coronnello, Alessio Nocentini, Gianluca Bartolucci, Marco Pallecchi, Marialessandra Contino, Dina Manetti, Maria Novella Romanelli, Claudiu T Supuran, Silvia Dei
New Dual P-Glycoprotein (P-gp) and Human Carbonic Anhydrase XII (hCA XII) Inhibitors as Multidrug Resistance (MDR) Reversers in Cancer Cells. Journal of medicinal chemistry 65 (21) (2022)
Haytham O Tawfik, Moataz A Shaldam, Alessio Nocentini, Rofaida Salem, Hadia Almahli, Sara T Al-Rashood, Claudiu T Supuran, Wagdy M Eldehna
Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activity. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Karol Biernacki, Olga Ciupak, Mateusz Daśko, Janusz Rachon, Witold Kozak, Janusz Rak, Konrad Kubiński, Maciej Masłyk, Aleksandra Martyna, Magdalena Śliwka-Kaszyńska, Joanna Wietrzyk, Marta Świtalska, Alessio Nocentini, Claudiu T Supuran, Sebastian Demkowicz
Development of Sulfamoylated 4-(1-Phenyl-1 H -1,2,3-triazol-4-yl)phenol Derivatives as Potent Steroid Sulfatase Inhibitors for Efficient Treatment of Breast Cancer. Journal of medicinal chemistry 65 (6) (2022)
Giulia Arrighi, Adrián Puerta, Andrea Petrini, Francisco J Hicke, Alessio Nocentini, Miguel X Fernandes, José Manuel Padrón, Claudiu T Supuran, José G Fernández-Bolaños, Óscar López
Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations. International journal of molecular sciences 23 (14) (2022)
Anil Kumar Marapaka, Alessio Nocentini, Molly S Youse, Weiwei An, Katrina J Holly, Chittaranjan Das, Ravi Yadav, Mohamed N Seleem, Claudiu T Supuran, Daniel P Flaherty
Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to Neisseria gonorrhoeae α-Carbonic Anhydrase. ACS medicinal chemistry letters 14 (1) (2022)
Tatiana Sharonova, Petr Zhmurov, Stanislav Kalinin, Alessio Nocentini, Andrea Ageli, Marta Ferraroni, Mikhail Korsakov, Claudiu T Supuran, Mikhail Krasavin
Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Mahmoud F Abo-Ashour, Hadia Almahli, Alessandro Bonardia, Amira Khalil, Tarfah Al-Warhi, Sara T Al-Rashood, Hatem A Abdel-Aziz, Alessio Nocentini, Claudiu T Supuran, Wagdy M Eldehna
Enaminone-based carboxylic acids as novel non-classical carbonic anhydrases inhibitors: design, synthesis and in vitro biological assessment. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Simone Giovannuzzi, Chad S Hewitt, Alessio Nocentini, Clemente Capasso, Gabriele Costantino, Daniel P Flaherty, Claudiu T Supuran
Inhibition studies of bacterial α-carbonic anhydrases with phenols. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T Supuran
1,2,3-Benzoxathiazine-2,2-dioxides - effective inhibitors of human carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2022)
Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Perspectives on the design and discovery of α-ketoamide inhibitors for the treatment of novel coronavirus: where do we stand and where do we go? Expert opinion on drug discovery 17 (6) (2022)
Weiwei An, Katrina J Holly, Alessio Nocentini, Ryan D Imhoff, Chad S Hewitt, Nader S Abutaleb, Xufeng Cao, Mohamed N Seleem, Claudiu T Supuran, Daniel P Flaherty
Structure-activity relationship studies for inhibitors for vancomycin-resistant Enterococcus and human carbonic anhydrases. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Wagdy M Eldehna, Mohammed S Taghour, Tarfah Al-Warhi, Alessio Nocentini, Mostafa M Elbadawi, Hazem A Mahdy, Mohamed A Abdelrahman, Ohoud J Alotaibi, Nada Aljaeed, Diaaeldin M Elimam, Kamyar Afarinkia, Hatem A Abdel-Aziz, Claudiu T Supuran
Discovery of 2,4-thiazolidinedione-tethered coumarins as novel selective inhibitors for carbonic anhydrase IX and XII isoforms. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Stanislav Kalinin, Alexander Kovalenko, Annika Valtari, Alessio Nocentini, Maxim A Gureev, Arto Urtti, Mikhail Korsakov, Claudiu T Supuran, Mikhail Yu Krasavin
5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Alessandro Bonardi, Silvia Bua, Jacob Combs, Carrie Lomelino, Jacob Andring, Sameh Mohamed Osman, Alessandra Toti, Di Cesare Mannelli Lorenzo, Paola Gratteri, Carla Ghelardini, Robert McKenna, Alessio Nocentini, Claudiu T Supuran
The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Zainab Saad Yusuf, Tugba Kevser Uysal, Ender Simsek, Alessio Nocentini, Sameh Mohamed Osman, Claudiu T Supuran, Özen Özensoy Güler
The inhibitory effect of boric acid on hypoxia-regulated tumour-associated carbonic anhydrase IX. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Alane Beatriz Vermelho, Giseli Capaci Rodrigues, Alessio Nocentini, Felipe R P Mansoldo, Claudiu T Supuran
Discovery of novel drugs for Chagas disease: is carbonic anhydrase a target for antiprotozoal drugs? Expert opinion on drug discovery 17 (10) (2022)
Simone Giovannuzzi, Viviana De Luca, Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum . Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Viviana De Luca, Andrea Petreni, Alessio Nocentini, Andrea Scaloni, Claudiu T Supuran, Clemente Capasso
Effect of Sulfonamides and Their Structurally Related Derivatives on the Activity of ι-Carbonic Anhydrase from Burkholderia territorii International journal of molecular sciences 22 (2) (2021)
Alessio Nocentini, Sonia Del Prete, Margaret D Mastrolorenzo, William A Donald, Clemente Capasso, Claudiu T Supuran
Activation studies of the β-carbonic anhydrases from Escherichia coli with amino acids and amines. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Small-molecule CD73 inhibitors for the immunotherapy of cancer: a patent and literature review (2017-present). Expert opinion on therapeutic patents 31 (10) (2021)
Alessio Nocentini, Andrea Ageli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A Donald, Claudiu T Supuran
Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Claudiu T Supuran, Alessio Nocentini, Elena Yakubova, Nikolay Savchuk, Stanislav Kalinin, Mikhail Krasavin
Biochemical profiling of anti-HIV prodrug Elsulfavirine (Elpida®) and its active form VM1500A against a panel of twelve human carbonic anhydrase isoforms. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Alessio Nocentini, Chad S Hewitt, Margaret D Mastrolorenzo, Daniel P Flaherty, Claudiu T Supuran
Anion inhibition studies of the α-carbonic anhydrases from Neisseria gonorrhoeae. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Alessandro Bonardi, Alessio Nocentini, Sameh Mohamed Osman, Fatmah Ali Alasmary, Tahani Mazyad Almutairi, Dalal Saied Abdullah, Paola Gratteri, Claudiu T Supuran
Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs - a joint docking/molecular dynamics study. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Sarah L Mueller, Panagiotis K Chrysanthopoulos, Maria A Halili, Caryn Hepburn, Tom Nebl, Claudiu T Supuran, Alessio Nocentini, Thomas S Peat, Sally-Ann Poulsen
The Glitazone Class of Drugs as Carbonic Anhydrase Inhibitors-A Spin-Off Discovery from Fragment Screening. Molecules (Basel, Switzerland) 26 (10) (2021)
Ilaria Dettori, Irene Fusco, Irene Bulli, Lisa Gaviano, Elisabetta Coppi, Federica Cherchi, Martina Venturini, Di Cesare Mannelli Lorenzo, Carla Ghelardini, Alessio Nocentini, Claudiu T Supuran, Anna Maria Pugliese, Felicita Pedata
Protective effects of carbonic anhydrase inhibition in brain ischaemia in vitro and in vivo models. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Chiraz Ismail, Alessio Nocentini, Claudiu T Supuran, Jean-Yves Winum, Rafik Gharbi
1,5-Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors. Archiv der Pharmazie (2021)
Andrea Petreni, Viviana De Luca, Andrea Scaloni, Alessio Nocentini, Clemente Capasso, Claudiu T Supuran
Anion inhibition studies of the Zn(II)-bound ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Francesco Mincione, Alessio Nocentini, Claudiu T Supuran
Advances in the discovery of novel agents for the treatment of glaucoma. Expert opinion on drug discovery 16 (10) (2021)
Simone Giovannuzzi, Mario D'Ambrosio, Cristina Luceri, Sameh Mohamed Osman, Marco Pallecchi, Gianluca Bartolucci, Alessio Nocentini, Claudiu T Supuran
Aromatic Sulfonamides including a Sulfonic Acid Tail: New Membrane Impermeant Carbonic Anhydrase Inhibitors for Targeting Selectively the Cancer-Associated Isoforms. International journal of molecular sciences 23 (1) (2021)
Rossella Grande, Simone Carradori, Valentina Puca, Irene Vitale, Andrea Ageli, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Paola Lanuti, Giuseppina Bologna, Pasquale Simeone, Clemente Capasso, Viviana De Luca, Claudiu T Supuran
Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles. International journal of molecular sciences 22 (21) (2021)
Paolo Guglielmi, Giulia Rotondi, Daniela Secci, Andrea Ageli, Paola Chimenti, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Simone Carradori, Claudiu T Supuran
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Mehmet Oguz, Erbay Kalay, Suleyman Akocak, Alessio Nocentini, Nebih Lolak, Mehmet Boga, Mustafa Yilmaz, Claudiu T Supuran
Synthesis of calix[4]azacrown substituted sulphonamides with antioxidant, acetylcholinesterase, butyrylcholinesterase, tyrosinase and carbonic anhydrase inhibitory action. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Elena Lucarini, Alessio Nocentini, Alessandro Bonardi, Niccolò Chiaramonte, Carmen Parisio, Micheli Laura, Alessandra Toti, Valentina Ferrara, Donatello Carrino, Alessandra Pacini, Maria Novella Romanelli, Claudiu T Supuran, Carla Ghelardini, Di Cesare Mannelli Lorenzo
Carbonic Anhydrase IV Selective Inhibitors Counteract the Development of Colitis-Associated Visceral Pain in Rats. Cells 10 (10) (2021)
Alessio Nocentini, Doretta Cuffaro, Lidia Ciccone, Elisabetta Orlandini, Susanna Nencetti, Elisa Nuti, Armando Rossello, Claudiu T Supuran
Activation of carbonic anhydrases from human brain by amino alcohol oxime ethers: towards human carbonic anhydrase VII selective activators. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Gustavo Provensi, Alessio Nocentini, Maria Beatrice Passani, Patrizio Blandina, Claudiu T Supuran
Activation of carbonic anhydrase isoforms involved in modulation of emotional memory and cognitive disorders with histamine agonists, antagonists and derivatives. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Irene Bulli, Ilaria Dettori, Elisabetta Coppi, Federica Cherchi, Martina Venturini, Di Cesare Mannelli Lorenzo, Carla Ghelardini, Alessio Nocentini, Claudiu T Supuran, Anna Maria Pugliese, Felicita Pedata
Role of Carbonic Anhydrase in Cerebral Ischemia and Carbonic Anhydrase Inhibitors as Putative Protective Agents. International journal of molecular sciences 22 (9) (2021)
Chad S Hewitt, Nader S Abutaleb, Ahmed E M Elhassanny, Alessio Nocentini, Xufeng Cao, Devon P Amos, Molly S Youse, Katrina J Holly, Anil Kumar Marapaka, Weiwei An, Jatinder Kaur, Aaron D Krabill, Ahmed Elkashif, Yehia Elgammal, Amanda L Graboski, Claudiu T Supuran, Mohamed N Seleem, Daniel P Flaherty
Structure-Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against Neisseria gonorrhoeae. ACS infectious diseases 7 (7) (2021)

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Alessio Nocentini