Ewgenij Proschak

ORCID

Publication Activity (10 Years)

Years Active: 2017-2024
Publications (10 Years): 55

Top Venues

Journal of medicinal chemistry

Advanced science (Weinheim, Baden-Wurttemberg, Germany)

ChemistryOpen

ChemMedChem

This page only lists publications with an associated author ORCID identifier.

Publications

Victor Hernandez-Olmos, Jan Heering, Beatrice Marinescu, Tina Weiß, Vladimir V Ivanov, Yurii S Moroz, Sheila Nevermann, Marius Mathes, Johanna H M Ehrler, Mohamad Wessam Alnouri, Markus Wolf, Alicia S Haydo, Tessa Schmachtel, Andrea Zaliani, Georg Höfner, Astrid Kaiser, Manfred Schubert-Zsilavecz, Annette G Beck-Sickinger, Stefan Offermanns, Philipp Gribbon, Michael A Rieger, Daniel Merk, Marco Sisignano, Dieter Steinhilber, Ewgenij Proschak
Development of a Potent and Selective G2A (GPR132) Agonist. Journal of medicinal chemistry 67 (13) (2024)
Christian J Muñoz Sosa, Christopher Lenz, Anton Hamann, Frederic Farges, Johannes Dopfer, Andreas Krämer, Veronika Cherkashyna, Andrey Tarnovskiy, Yurii S Moroz, Ewgenij Proschak, Václav Němec, Susanne Müller, Krishna Saxena, Stefan Knapp
A C-Degron Structure-Based Approach for the Development of Ligands Targeting the E3 Ligase TRIM7. ACS chemical biology (2024)
Annika Balzulat, W Felix Zhu, Cathrin Flauaus, Victor Hernandez-Olmos, Jan Heering, Sunesh Sethumadhavan, Mariam Dubiel, Annika Frank, Amelie Menge, Maureen Hebchen, Katharina Metzner, Ruirui Lu, Robert Lukowski, Peter Ruth, Stefan Knapp, Susanne Müller, Dieter Steinhilber, Inga Hänelt, Holger Stark, Ewgenij Proschak, Achim Schmidtko
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch. Advanced science (Weinheim, Baden-Wurttemberg, Germany) (2024)
Lara Dötsch, Caitlin Davies, Elisabeth Hennes, Julia Schönfeld, Adarsh Kumar, Celine Da Cruz Lopes Guita, Johanna H M Ehrler, Kerstin Hiesinger, Sasikala Thavam, Petra Janning, Sonja Sievers, Stefan Knapp, Ewgenij Proschak, Slava Ziegler, Herbert Waldmann
Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator. Journal of medicinal chemistry 67 (6) (2024)
Victor Hernandez-Olmos, Jan Heering, Beatrice Marinescu, Tina Weiß, Vladimir V Ivanov, Yurii S Moroz, Sheila Nevermann, Marius Mathes, Johanna H M Ehrler, Mohamad Wessam Alnouri, Markus Wolf, Alicia S Haydo, Tessa Schmachtel, Andrea Zaliani, Georg Höfner, Astrid Kaiser, Manfred Schubert-Zsilavecz, Annette G Beck-Sickinger, Stefan Offermanns, Philipp Gribbon, Michael A Rieger, Daniel Merk, Marco Sisignano, Dieter Steinhilber, Ewgenij Proschak
Development of a Potent and Selective G2A (GPR132) Agonist. Journal of medicinal chemistry 67 (13) (2024)
Sabine Willems, Romy Busch, Felix Nawa, Marco Ballarotto, Felix F Lillich, Till Kasch, Úrsula López-García, Julian A Marschner, Lorena A Rüger, Beatrice Renelt, Julia Ohrndorf, Silvia Arifi, Daniel Zaienne, Ewgenij Proschak, Jörg Pabel, Daniel Merk
Structural Optimization of Oxaprozin for Selective Inverse Nurr1 Agonism. Journal of medicinal chemistry 67 (15) (2024)
Annika Balzulat, W Felix Zhu, Cathrin Flauaus, Victor Hernandez-Olmos, Jan Heering, Sunesh Sethumadhavan, Mariam Dubiel, Annika Frank, Amelie Menge, Maureen Hebchen, Katharina Metzner, Ruirui Lu, Robert Lukowski, Peter Ruth, Stefan Knapp, Susanne Müller, Dieter Steinhilber, Inga Hänelt, Holger Stark, Ewgenij Proschak, Achim Schmidtko
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch. Advanced science (Weinheim, Baden-Wurttemberg, Germany) 11 (15) (2024)
Christian J Muñoz Sosa, Christopher Lenz, Anton Hamann, Frederic Farges, Johannes Dopfer, Andreas Krämer, Veronika Cherkashyna, Andrey Tarnovskiy, Yurii S Moroz, Ewgenij Proschak, Václav Němec, Susanne Müller, Krishna Saxena, Stefan Knapp
A C-Degron Structure-Based Approach for the Development of Ligands Targeting the E3 Ligase TRIM7. ACS chemical biology 19 (7) (2024)
Lara Dötsch, Caitlin Davies, Elisabeth Hennes, Julia Schönfeld, Adarsh Kumar, Celine Da Cruz Lopes Guita, Johanna H M Ehrler, Kerstin Hiesinger, Sasikala Thavam, Petra Janning, Sonja Sievers, Stefan Knapp, Ewgenij Proschak, Slava Ziegler, Herbert Waldmann
Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator. Journal of medicinal chemistry 67 (6) (2024)
Annika Balzulat, W Felix Zhu, Cathrin Flauaus, Victor Hernandez-Olmos, Jan Heering, Sunesh Sethumadhavan, Mariam Dubiel, Annika Frank, Amelie Menge, Maureen Hebchen, Katharina Metzner, Ruirui Lu, Robert Lukowski, Peter Ruth, Stefan Knapp, Susanne Müller, Dieter Steinhilber, Inga Hänelt, Holger Stark, Ewgenij Proschak, Achim Schmidtko
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch. Advanced science (Weinheim, Baden-Wurttemberg, Germany) 11 (15) (2024)
Annika Balzulat, W Felix Zhu, Cathrin Flauaus, Victor Hernandez-Olmos, Jan Heering, Sunesh Sethumadhavan, Mariam Dubiel, Annika Frank, Amelie Menge, Maureen Hebchen, Katharina Metzner, Ruirui Lu, Robert Lukowski, Peter Ruth, Stefan Knapp, Susanne Müller, Dieter Steinhilber, Inga Hänelt, Holger Stark, Ewgenij Proschak, Achim Schmidtko
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch. Advanced science (Weinheim, Baden-Wurttemberg, Germany) 11 (15) (2024)
Victor Hernandez-Olmos, Jan Heering, Beatrice Marinescu, Tina Weiß, Vladimir V Ivanov, Yurii S Moroz, Sheila Nevermann, Marius Mathes, Johanna H M Ehrler, Mohamad Wessam Alnouri, Markus Wolf, Alicia S Haydo, Tessa Schmachtel, Andrea Zaliani, Georg Höfner, Astrid Kaiser, Manfred Schubert-Zsilavecz, Annette G Beck-Sickinger, Stefan Offermanns, Philipp Gribbon, Michael A Rieger, Daniel Merk, Marco Sisignano, Dieter Steinhilber, Ewgenij Proschak
Development of a Potent and Selective G2A (GPR132) Agonist. Journal of medicinal chemistry 67 (13) (2024)
Victor Hernandez-Olmos, Jan Heering, Beatrice Marinescu, Tina Weiß, Vladimir V Ivanov, Yurii S Moroz, Sheila Nevermann, Marius Mathes, Johanna H M Ehrler, Mohamad Wessam Alnouri, Markus Wolf, Alicia S Haydo, Tessa Schmachtel, Andrea Zaliani, Georg Höfner, Astrid Kaiser, Manfred Schubert-Zsilavecz, Annette G Beck-Sickinger, Stefan Offermanns, Philipp Gribbon, Michael A Rieger, Daniel Merk, Marco Sisignano, Dieter Steinhilber, Ewgenij Proschak
Development of a Potent and Selective G2A (GPR132) Agonist. Journal of medicinal chemistry (2024)
Sabine Willems, Romy Busch, Felix Nawa, Marco Ballarotto, Felix F Lillich, Till Kasch, Úrsula López-García, Julian A Marschner, Lorena A Rüger, Beatrice Renelt, Julia Ohrndorf, Silvia Arifi, Daniel Zaienne, Ewgenij Proschak, Jörg Pabel, Daniel Merk
Structural Optimization of Oxaprozin for Selective Inverse Nurr1 Agonism. Journal of medicinal chemistry 67 (15) (2024)
W Felix Zhu, Claire Empel, Sveva Pelliccia, René M Koenigs, Ewgenij Proschak, Victor Hernandez-Olmos
Photochemistry in Medicinal Chemistry and Chemical Biology. Journal of medicinal chemistry 67 (6) (2024)
Lara Dötsch, Caitlin Davies, Elisabeth Hennes, Julia Schönfeld, Adarsh Kumar, Celine Da Cruz Lopes Guita, Johanna H M Ehrler, Kerstin Hiesinger, Sasikala Thavam, Petra Janning, Sonja Sievers, Stefan Knapp, Ewgenij Proschak, Slava Ziegler, Herbert Waldmann
Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator. Journal of medicinal chemistry 67 (6) (2024)
Lara Dötsch, Caitlin Davies, Elisabeth Hennes, Julia Schönfeld, Adarsh Kumar, Celine Da Cruz Lopes Guita, Johanna H M Ehrler, Kerstin Hiesinger, Sasikala Thavam, Petra Janning, Sonja Sievers, Stefan Knapp, Ewgenij Proschak, Slava Ziegler, Herbert Waldmann
Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator. Journal of medicinal chemistry (2024)
W Felix Zhu, Claire Empel, Sveva Pelliccia, René M Koenigs, Ewgenij Proschak, Victor Hernandez-Olmos
Photochemistry in Medicinal Chemistry and Chemical Biology. Journal of medicinal chemistry (2024)
Annika Balzulat, W Felix Zhu, Cathrin Flauaus, Victor Hernandez-Olmos, Jan Heering, Sunesh Sethumadhavan, Mariam Dubiel, Annika Frank, Amelie Menge, Maureen Hebchen, Katharina Metzner, Ruirui Lu, Robert Lukowski, Peter Ruth, Stefan Knapp, Susanne Müller, Dieter Steinhilber, Inga Hänelt, Holger Stark, Ewgenij Proschak, Achim Schmidtko
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch. Advanced science (Weinheim, Baden-Wurttemberg, Germany) 11 (15) (2024)
Annika Balzulat, W Felix Zhu, Cathrin Flauaus, Victor Hernandez-Olmos, Jan Heering, Sunesh Sethumadhavan, Mariam Dubiel, Annika Frank, Amelie Menge, Maureen Hebchen, Katharina Metzner, Ruirui Lu, Robert Lukowski, Peter Ruth, Stefan Knapp, Susanne Müller, Dieter Steinhilber, Inga Hänelt, Holger Stark, Ewgenij Proschak, Achim Schmidtko
Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch. Advanced science (Weinheim, Baden-Wurttemberg, Germany) 11 (15) (2024)
W Felix Zhu, Claire Empel, Sveva Pelliccia, René M Koenigs, Ewgenij Proschak, Victor Hernandez-Olmos
Photochemistry in Medicinal Chemistry and Chemical Biology. Journal of medicinal chemistry 67 (6) (2024)
Victor Hernandez-Olmos, Jan Heering, Beatrice Marinescu, Tina Weiß, Vladimir V Ivanov, Yurii S Moroz, Sheila Nevermann, Marius Mathes, Johanna H M Ehrler, Mohamad Wessam Alnouri, Markus Wolf, Alicia S Haydo, Tessa Schmachtel, Andrea Zaliani, Georg Höfner, Astrid Kaiser, Manfred Schubert-Zsilavecz, Annette G Beck-Sickinger, Stefan Offermanns, Philipp Gribbon, Michael A Rieger, Daniel Merk, Marco Sisignano, Dieter Steinhilber, Ewgenij Proschak
Development of a Potent and Selective G2A (GPR132) Agonist. Journal of medicinal chemistry 67 (13) (2024)
Lara Dötsch, Caitlin Davies, Elisabeth Hennes, Julia Schönfeld, Adarsh Kumar, Celine Da Cruz Lopes Guita, Johanna H M Ehrler, Kerstin Hiesinger, Sasikala Thavam, Petra Janning, Sonja Sievers, Stefan Knapp, Ewgenij Proschak, Slava Ziegler, Herbert Waldmann
Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator. Journal of medicinal chemistry 67 (6) (2024)
Sabine Willems, Romy Busch, Felix Nawa, Marco Ballarotto, Felix F Lillich, Till Kasch, Úrsula López-García, Julian A Marschner, Lorena A Rüger, Beatrice Renelt, Julia Ohrndorf, Silvia Arifi, Daniel Zaienne, Ewgenij Proschak, Jörg Pabel, Daniel Merk
Structural Optimization of Oxaprozin for Selective Inverse Nurr1 Agonism. Journal of medicinal chemistry (2024)
Silvia Arifi, Julian A Marschner, Julius Pollinger, Laura Isigkeit, Pascal Heitel, Astrid Kaiser, Lennart Obeser, Georg Höfner, Ewgenij Proschak, Stefan Knapp, Apirat Chaikuad, Jan Heering, Daniel Merk
Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation. Journal of the American Chemical Society (2023)
W Felix Zhu, Andreas Krämer, Stefan Knapp, Ewgenij Proschak, Victor Hernandez-Olmos
Cascade Synthesis of Kinase-Privileged 3-Aminoindazoles via Intramolecular N-N Bond Formation. The Journal of organic chemistry 87 (5) (2022)
Steffen Brunst, Julia Schönfeld, Peter Breunig, Luisa D Burgers, Murphy DeMeglio, Johanna H M Ehrler, Felix F Lillich, Lilia Weizel, Jasmin K Hefendehl, Robert Fürst, Ewgenij Proschak, Kerstin Hiesinger
Designing a Small Fluorescent Inhibitor to Investigate Soluble Epoxide Hydrolase Engagement in Living Cells. ACS medicinal chemistry letters 13 (7) (2022)
Benedikt Hufnagel, W Felix Zhu, Hanna M Franz, Ewgenij Proschak, Victor Hernandez-Olmos
Phenolate-Induced N-O Bond Formation versus TiemannType Rearrangement for the Synthesis of 3-Aminobenzisoxazoles and 2-Aminobenzoxazoles. ChemistryOpen 11 (12) (2022)
Jan Heering, Victor Hernandez-Olmos, Niklas Ildefeld, Ting Liu, Anja Kaiser, Zumer Naeem, Timo Frömel, Ingrid Fleming, Dieter Steinhilber, Ewgenij Proschak
Development and Characterization of a Fluorescent Ligand for Leukotriene B4 Receptor 2 in Cells and Tissues. Journal of medicinal chemistry 65 (3) (2022)
Benedikt Hufnagel, W Felix Zhu, Hanna M Franz, Ewgenij Proschak, Victor Hernandez-Olmos
Phenolate-Induced N-O Bond Formation versus TiemannType Rearrangement for the Synthesis of 3-Aminobenzisoxazoles and 2-Aminobenzoxazoles. ChemistryOpen 11 (12) (2022)
Benedikt Hufnagel, W Felix Zhu, Hanna M Franz, Ewgenij Proschak, Victor Hernandez-Olmos
Phenolate-Induced N-O Bond Formation versus TiemannType Rearrangement for the Synthesis of 3-Aminobenzisoxazoles and 2-Aminobenzoxazoles. ChemistryOpen 11 (12) (2022)
Cansu Kaya, Jelena Konstantinović, Andreas M Kany, Anastasia Andreas, Jan S Kramer, Steffen Brunst, Lilia Weizel, Marco J Rotter, Denia Frank, Samir Yahiaoui, Daniel Krug, Rolf Wolfgang Hartmann, Jörg Haupenthal, Ewgenij Proschak, Thomas A Wichelhaus, Anna Katharina Herta Hirsch
N -Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases. Journal of medicinal chemistry 65 (5) (2022)
Markus Hartmann, Jessica Huber, Jan S Kramer, Jan Heering, Larissa Pietsch, Holger Stark, Dalibor Odadzic, Iris Bischoff, Robert Fürst, Martin Schröder, Masato Akutsu, Apirat Chaikuad, Volker Dötsch, Stefan Knapp, Ricardo M Biondi, Vladimir V Rogov, Ewgenij Proschak
Demonstrating Ligandability of the LC3A and LC3B Adapter Interface. Journal of medicinal chemistry 64 (7) (2021)
Felix F Lillich, Sabine Willems, Xiaomin Ni, Whitney Kilu, Carmen Borkowsky, Mirko Brodsky, Jan S Kramer, Steffen Brunst, Victor Hernandez-Olmos, Jan Heering, Simone Schierle, Roxane-I Kestner, Franziska M Mayser, Moritz Helmstädter, Tamara Göbel, Lilia Weizel, Dmitry Namgaladze, Astrid Kaiser, Dieter Steinhilber, Waltraud Pfeilschifter, Astrid S Kahnt, Anna Proschak, Apirat Chaikuad, Stefan Knapp, Daniel Merk, Ewgenij Proschak
Structure-Based Design of Dual Partial Peroxisome Proliferator-Activated Receptor γ Agonists/Soluble Epoxide Hydrolase Inhibitors. Journal of medicinal chemistry 64 (23) (2021)
Mikhail Krasavin, Daniil Zhukovsky, Igor Solovyev, Darina Barkhatova, Dmitry Dar'in, Denia Frank, Giada Martinelli, Lilia Weizel, Anna Proschak, Marco Rotter, Jan S Kramer, Steffen Brunst, Thomas A Wichelhaus, Ewgenij Proschak
RhII -Catalyzed De-symmetrization of Ethane-1,2-dithiol and Propane-1,3-dithiol Yields Metallo-β-lactamase Inhibitors. ChemMedChem 16 (22) (2021)
Moritz Helmstädter, Astrid Kaiser, Steffen Brunst, Jurema Schmidt, Riccardo Ronchetti, Lilia Weizel, Ewgenij Proschak, Daniel Merk
Second-Generation Dual FXR/sEH Modulators with Optimized Pharmacokinetics. Journal of medicinal chemistry 64 (13) (2021)
Steffen Brunst, Jan S Kramer, Whitney Kilu, Jan Heering, Julius Pollinger, Kerstin Hiesinger, Sven George, Dieter Steinhilber, Daniel Merk, Ewgenij Proschak
Systematic Assessment of Fragment Identification for Multitarget Drug Design. ChemMedChem 16 (7) (2021)
Simone Schierle, Apirat Chaikuad, Felix F Lillich, Xiaomin Ni, Stefano Woltersdorf, Espen Schallmayer, Beatrice Renelt, Riccardo Ronchetti, Stefan Knapp, Ewgenij Proschak, Daniel Merk
Oxaprozin Analogues as Selective RXR Agonists with Superior Properties and Pharmacokinetics. Journal of medicinal chemistry 64 (8) (2021)
Markus Hartmann, Sofia-Iris Bibli, Daniel Tews, Xiaomin Ni, Theresa Kircher, Jan S Kramer, Whitney Kilu, Jan Heering, Victor Hernandez-Olmos, Lilia Weizel, Gerhard K E Scriba, Sulaiman Krait, Stefan Knapp, Apirat Chaikuad, Daniel Merk, Ingrid Fleming, Pamela Fischer-Posovszky, Ewgenij Proschak
Combined Cardioprotective and Adipocyte Browning Effects Promoted by the Eutomer of Dual sEH/PPARγ Modulator. Journal of medicinal chemistry 64 (5) (2021)
Victor Hernandez-Olmos, Jan Heering, Iris Bischoff-Kont, Alexander Kaps, Rinusha Rajkumar, Ting Liu, Robert Fürst, Dieter Steinhilber, Ewgenij Proschak
Discovery of Irbesartan Derivatives as BLT2 Agonists by Virtual Screening. ACS medicinal chemistry letters 12 (8) (2021)
Victor Hernandez-Olmos, Jan Heering, Viktoria Planz, Ting Liu, Alexander Kaps, Rinusha Rajkumar, Matthias Gramzow, Astrid Kaiser, Manfred Schubert-Zsilavecz, Michael J Parnham, Maike Windbergs, Dieter Steinhilber, Ewgenij Proschak
First Structure-Activity Relationship Study of Potent BLT2 Agonists as Potential Wound-Healing Promoters. Journal of medicinal chemistry 63 (20) (2020)
Leonie Gellrich, Pascal Heitel, Jan Heering, Whitney Kilu, Julius Pollinger, Tamara Goebel, Astrid Kahnt, Silvia Arifi, Werner Pogoda, Alexander Paulke, Dieter Steinhilber, Ewgenij Proschak, Mario Wurglics, Manfred Schubert-Zsilavecz, Apirat Chaikuad, Stefan Knapp, Iris Bischoff, Robert Fürst, Daniel Merk
l-Thyroxin and the Nonclassical Thyroid Hormone TETRAC Are Potent Activators of PPARγ. Journal of medicinal chemistry 63 (13) (2020)
Thomas Hanke, Sun-Yee Cheung, Whitney Kilu, Jan Heering, Xiaomin Ni, Viktoria Planz, Simone Schierle, Giuseppe Faudone, Marius Friedrich, Marek Wanior, Oliver Werz, Maike Windbergs, Ewgenij Proschak, Manfred Schubert-Zsilavecz, Apirat Chaikuad, Stefan Knapp, Daniel Merk
A Selective Modulator of Peroxisome Proliferator-Activated Receptor γ with an Unprecedented Binding Mode. Journal of medicinal chemistry 63 (9) (2020)
Kerstin Hiesinger, Dmitry Dar'in, Ewgenij Proschak, Mikhail Krasavin
Spirocyclic Scaffolds in Medicinal Chemistry. Journal of medicinal chemistry 64 (1) (2020)
Kerstin Hiesinger, Jan S Kramer, Sandra Beyer, Timon Eckes, Steffen Brunst, Cathrin Flauaus, Sandra K Wittmann, Lilia Weizel, Astrid Kaiser, Simon B M Kretschmer, Sven George, Carlo Angioni, Jan Heering, Gerd Geisslinger, Manfred Schubert-Zsilavecz, Achim Schmidtko, Denys Pogoryelov, Josef Pfeilschifter, Bettina Hofmann, Dieter Steinhilber, Stephanie Schwalm, Ewgenij Proschak
Design, Synthesis, and Structure-Activity Relationship Studies of Dual Inhibitors of Soluble Epoxide Hydrolase and 5-Lipoxygenase. Journal of medicinal chemistry 63 (20) (2020)
Julius Pollinger, Leonie Gellrich, Simone Schierle, Whitney Kilu, Jurema Schmidt, Lena Kalinowsky, Julia Ohrndorf, Astrid Kaiser, Jan Heering, Ewgenij Proschak, Daniel Merk
Tuning Nuclear Receptor Selectivity of Wy14,643 towards Selective Retinoid X Receptor Modulation. Journal of medicinal chemistry 62 (4) (2019)
Jan S Kramer, Stefano Woltersdorf, Thomas Duflot, Kerstin Hiesinger, Felix F Lillich, Felix Knöll, Sandra K Wittmann, Franca-M Klingler, Steffen Brunst, Apirat Chaikuad, Christophe Morisseau, Bruce D Hammock, Carola Buccellati, Angelo Sala, G Enrico Rovati, Matthieu Leuillier, Sylvain Fraineau, Julie Rondeaux, Victor Hernandez-Olmos, Jan Heering, Daniel Merk, Denys Pogoryelov, Dieter Steinhilber, Stefan Knapp, Jeremy Bellien, Ewgenij Proschak
Discovery of the First in Vivo Active Inhibitors of the Soluble Epoxide Hydrolase Phosphatase Domain. Journal of medicinal chemistry 62 (18) (2019)
Andreas Martin Kany, Asfandyar Sikandar, Jörg Haupenthal, Samir Yahiaoui, Christine K Maurer, Ewgenij Proschak, Jesko Koehnke, Rolf Wolfgang Hartmann
Binding Mode Characterization and Early in Vivo Evaluation of Fragment-Like Thiols as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa. ACS infectious diseases 4 (6) (2018)
Ewgenij Proschak, Holger Stark, Daniel Merk
Polypharmacology by Design: A Medicinal Chemist's Perspective on Multitargeting Compounds. Journal of medicinal chemistry 62 (2) (2018)
Simone Schierle, Cathrin Flauaus, Pascal Heitel, Sabine Willems, Jurema Schmidt, Astrid Kaiser, Lilia Weizel, Tamara Goebel, Astrid S Kahnt, Gerd Geisslinger, Dieter Steinhilber, Mario Wurglics, G Enrico Rovati, Achim Schmidtko, Ewgenij Proschak, Daniel Merk
Boosting Anti-Inflammatory Potency of Zafirlukast by Designed Polypharmacology. Journal of medicinal chemistry 61 (13) (2018)
René Blöcher, Karen M Wagner, Raghavender R Gopireddy, Todd R Harris, Hao Wu, Bogdan Barnych, Sung Hee Hwang, Yang K Xiang, Ewgenij Proschak, Christophe Morisseau, Bruce D Hammock
Orally Available Soluble Epoxide Hydrolase/Phosphodiesterase 4 Dual Inhibitor Treats Inflammatory Pain. Journal of medicinal chemistry 61 (8) (2018)
Jurema Schmidt, Marco Rotter, Tim Weiser, Sandra Wittmann, Lilia Weizel, Astrid Kaiser, Jan Heering, Tamara Goebel, Carlo Angioni, Mario Wurglics, Alexander Paulke, Gerd Geisslinger, Astrid Kahnt, Dieter Steinhilber, Ewgenij Proschak, Daniel Merk
A Dual Modulator of Farnesoid X Receptor and Soluble Epoxide Hydrolase To Counter Nonalcoholic Steatohepatitis. Journal of medicinal chemistry 60 (18) (2017)
Dominik Büttner, Jan S Kramer, Franca-M Klingler, Sandra K Wittmann, Markus R Hartmann, Christian G Kurz, Daniel Kohnhäuser, Lilia Weizel, Astrid Brüggerhoff, Denia Frank, Dieter Steinhilber, Thomas A Wichelhaus, Denys Pogoryelov, Ewgenij Proschak
Challenges in the Development of a Thiol-Based Broad-Spectrum Inhibitor for Metallo-β-Lactamases. ACS infectious diseases 4 (3) (2017)
Daniel Flesch, Sun-Yee Cheung, Jurema Schmidt, Matthias Gabler, Pascal Heitel, Jan Kramer, Astrid Kaiser, Markus Hartmann, Mara Lindner, Kerstin Lüddens-Dämgen, Jan Heering, Christina Lamers, Hartmut Lüddens, Mario Wurglics, Ewgenij Proschak, Manfred Schubert-Zsilavecz, Daniel Merk
Nonacidic Farnesoid X Receptor Modulators. Journal of medicinal chemistry 60 (16) (2017)
Ewgenij Proschak, Pascal Heitel, Lena Kalinowsky, Daniel Merk
Opportunities and Challenges for Fatty Acid Mimetics in Drug Discovery. Journal of medicinal chemistry 60 (13) (2017)

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Publication Activity (10 Years)

Top Topics

Top Venues

Ewgenij Proschak