Andrea Ageli (Andrea Angeli)

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2018-2024
Publications (10 Years): 156

Top Venues

Journal of enzyme inhibition and medicinal chemistry

Journal of medicinal chemistry

International journal of molecular sciences

Molecules (Basel, Switzerland)

Institutul de Chimie Macromoleculara Petru Poni

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Institutul de Chimie Macromoleculara Petru Poni Jun 01 2019

Romania

resercher :: Center of Advanced Research in Bionanoconjugates and Biopolymers

Università degli Studi di Firenze Nov 01 2015 - Nov 01 2018

Italy

dottorando

Publications

Letizia Giampietro, Beatrice Marinacci, Alice Della Valle, Ilaria D'Agostino, Aldo Lauro, Mattia Mori, Simone Carradori, Alessandra Ammazzalorso, Barbara De Filippis, Cristina Maccallini, Andrea Ageli, Clemente Capasso, Santolo Francati, Adriano Mollica, Rossella Grande, Claudiu T Supuran
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies. Pharmaceuticals (Basel, Switzerland) 17 (8) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry 67 (4) (2024)
Bianca Laura Bernardoni, Ilaria D'Agostino, Concettina La Motta, Andrea Ageli
An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans , the pivotal pathogens in the oral cavity. Expert opinion on therapeutic patents 34 (6) (2024)
Bianca Laura Bernardoni, Ilaria D'Agostino, Concettina La Motta, Andrea Ageli
An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans , the pivotal pathogens in the oral cavity. Expert opinion on therapeutic patents (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry 67 (4) (2024)
Muhammed Trawally, Kübra Demir-Yazıcı, Andrea Ageli, Kerem Kaya, Atilla Akdemir, Claudiu T Supuran, Özlen Güzel-Akdemir
Thiosemicarbazone-benzenesulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies. Anti-cancer agents in medicinal chemistry 24 (9) (2024)
Arzu Gumus, Ilaria D'Agostino, Valentina Puca, Valentina Crocetta, Simone Carradori, Luigi Cutarella, Mattia Mori, Fabrizio Carta, Andrea Ageli, Clemente Capasso, Claudiu T Supuran
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α-carbonic anhydrase inhibitors. Archiv der Pharmazie (2024)
Elena Lucarini, Vanessa D'Antogiovanni, Luca Antonioli, Carla Ghelardini, Lorenzo Di Cesare Mannelli, Marta Ferraroni, Maria Locuoco, Antonella Capperucci, Damiano Tanini, Andrea Ageli, Claudiu T Supuran
Study of Chalcogen Aspirin Derivatives with Carbonic Anhydrase Inhibitory Properties for Treating Inflammatory Pain. ACS medicinal chemistry letters 15 (9) (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Davide Moi, Serena Vittorio, Andrea Ageli, Claudiu T Supuran, Valentina Onnis
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (4) (2024)
Bianca Laura Bernardoni, Ilaria D'Agostino, Concettina La Motta, Andrea Ageli
An insight into the last 5-year patents on porphyromonas gingivalis and streptococcus mutans , the pivotal pathogens in the oral cavity. Expert opinion on therapeutic patents (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Davide Moi, Serena Vittorio, Andrea Ageli, Claudiu T Supuran, Valentina Onnis
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (4) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Andrea Ageli, Irene Chelli, Laura Lucarini, Silvia Sgambellone, Silvia Marri, Serafina Villano, Marta Ferraroni, Viviana De Luca, Clemente Capasso, Fabrizio Carta, Claudiu T Supuran
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. Journal of medicinal chemistry (2024)
Viviana De Luca, Andrea Ageli, Alessio Nocentini, Paola Gratteri, Silvia Pratesi, Damiano Tanini, Vincenzo Carginale, Antonella Capperucci, Claudiu T Supuran, Clemente Capasso
Leveraging SARS-CoV-2 Main Protease (M pro ) for COVID-19 Mitigation with Selenium-Based Inhibitors. International journal of molecular sciences 25 (2) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry (2024)
Letizia Giampietro, Beatrice Marinacci, Alice Della Valle, Ilaria D'Agostino, Aldo Lauro, Mattia Mori, Simone Carradori, Alessandra Ammazzalorso, Barbara De Filippis, Cristina Maccallini, Andrea Ageli, Clemente Capasso, Santolo Francati, Adriano Mollica, Rossella Grande, Claudiu T Supuran
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies. Pharmaceuticals (Basel, Switzerland) 17 (8) (2024)
Hakan Aslan, Gioele Renzi, Andrea Ageli, Ilaria D'Agostino, Roberto Ronca, Maria Luisa Massardi, Camilla Tavani, Simone Carradori, Marta Ferraroni, Paolo Governa, Fabrizio Manetti, Fabrizio Carta, Claudiu T Supuran
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC medicinal chemistry 15 (6) (2024)
Muhammed Trawally, Kübra Demir-Yazıcı, Andrea Ageli, Kerem Kaya, Atilla Akdemir, Claudiu T Supuran, Özlen Güzel-Akdemir
Thiosemicarbazone-benzene Sulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies. Anti-cancer agents in medicinal chemistry (2024)
Davide Moi, Serena Vittorio, Andrea Ageli, Claudiu T Supuran, Valentina Onnis
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS medicinal chemistry letters 15 (4) (2024)
Hakan Aslan, Gioele Renzi, Andrea Ageli, Ilaria D'Agostino, Roberto Ronca, Maria Luisa Massardi, Camilla Tavani, Simone Carradori, Marta Ferraroni, Paolo Governa, Fabrizio Manetti, Fabrizio Carta, Claudiu T Supuran
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC medicinal chemistry 15 (6) (2024)
Cristina-Maria Al Matarneh, Mariana Pinteala, Alina Nicolescu, Mihaela Silion, Francesca Mocci, Razvan Puf, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Susi Zara, Simone Carradori, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. Journal of medicinal chemistry 67 (4) (2024)
Marialuigia Fantacuzzi, Ilaria D'Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Mariangela Agamennone, Andrea Ageli, Filomena Sannio, Jean Denis Docquier, Clemente Capasso, Claudiu T Supuran
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris Valerievich Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Andrea Ageli, Niccolò Paoletti, Claudiu T Supuran
Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (7) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Moataz A Shaldam, Hadia Almahli, Andrea Ageli, Rehab Mustafa Badi, Eman F Khaleel, Abdelrahman I Zain-Alabdeen, Zainab M Elsayed, Eslam B Elkaeed, Rofaida Salem, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris Valerievich Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Lisa Sequeira, Simona Distinto, Rita Meleddu, Marco Gaspari, Andrea Ageli, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Fernanda Borges, Eugenio Uriarte, Stefano Alcaro, Claudiu T Supuran, Elias Maccioni
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Shaimaa M Aboukhatwa, Peter A Sidhom, Andrea Ageli, Claudiu T Supuran, Haytham O Tawfik
Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids. ACS omega 8 (8) (2023)
Andrea Ageli, Claudiu T Supuran
Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Moataz A Shaldam, Hadia Almahli, Andrea Ageli, Rehab Mustafa Badi, Eman F Khaleel, Abdelrahman I Zain-Alabdeen, Zainab M Elsayed, Eslam B Elkaeed, Rofaida Salem, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Belma Zengin Kurt, Gulsen Celebi, Dilek Öztürk Civelek, Andrea Ageli, Atilla Akdemir, Fatih Sonmez, Claudiu T Supuran
Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS omega 8 (6) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Simone Carradori, Andrea Ageli, Patrick Severin Sfragano, Xheila Yzeiri, Massimo Calamante, Damiano Tanini, Antonella Capperucci, Hannah Kunstek, Mihayl Varbanov, Clemente Capasso, Claudiu T Supuran
Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents. International journal of molecular sciences 24 (11) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Andrea Ageli, Marta Ferraroni, Carlotta Granchi, Filippo Minutolo, Xiaozhuo Chen, Pratik Shriwas, Emilio Russo, Antonio Leo, Silvia Selleri, Fabrizio Carta, Claudiu T Supuran
First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome. Journal of medicinal chemistry (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Maria Giulia Davighi, Francesca Cardona, Andrea Goti, Marta Ferraroni, Andrea Ageli, Claudiu T Supuran, Francesca Cardona
Mono- and three-tailed sugar and iminosugar decorated benzenesulfonamide carbonic anhydrase inhibitors. Organic & biomolecular chemistry (2023)
Francesco Melfi, Simone Carradori, Andrea Ageli, Ilaria D'Agostino
Nature as a source and inspiration for human monoamine oxidase B (Hmao-B) inhibition: A review of the recent advances in chemical modification of natural compounds. Expert opinion on drug discovery (2023)
Shaimaa M Aboukhatwa, Peter A Sidhom, Andrea Ageli, Claudiu T Supuran, Haytham O Tawfik
Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids. ACS omega 8 (8) (2023)
Andrea Ageli, Claudiu T Supuran
Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris Valerievich Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Toni C Denner, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Rene Csuk
Ureidobenzenesulfonamides as Selective Carbonic Anhydrase I, IX, and XII Inhibitors. Molecules (Basel, Switzerland) 28 (23) (2023)
Belma Zengin Kurt, Gulsen Celebi, Dilek Öztürk Civelek, Andrea Ageli, Atilla Akdemir, Fatih Sonmez, Claudiu T Supuran
Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS omega 8 (6) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Kiran Siwach, Amit Kumar, Harish Panchal, Rajiv Kumar, Jitender Kumar Bhardwaj, Andrea Ageli, Claudiu T Supuran, Pawan K Sharma
Selective inhibition of carbonic anhydrase IX by sulphonylated 1,2,3-triazole incorporated benzenesulphonamides capable of inducing apoptosis. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Haytham O Tawfik, Amany Belal, Mohammad A S Abourehab, Andrea Ageli, Alessandro Bonardi, Claudiu T Supuran, Mervat H El-Hamamsy
Dependence on linkers' flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Andrea Ageli, Victor Kartsev, Petrou Anthi, Boris Lichitsky, Andrey Nikolaevich Komogortsev, Mariana Pinteală, Geronikaki Athina, Claudiu T Supuran
Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies. Pharmaceuticals (Basel, Switzerland) 15 (3) (2022)
Andrea Ageli, Linda J Urbański, Clemente Capasso, Seppo Parkkila, Claudiu T Supuran
Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Mariangela Agamennone, Marialuigia Fantacuzzi, Simone Carradori, Anél Petzer, Jacobus P Petzer, Andrea Ageli, Claudiu T Supuran, Grazia Luisi
Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and ( Pseudo )-Dipeptidyl Appendages: In Vitro and Computational Studies. Molecules (Basel, Switzerland) 27 (22) (2022)
Niccolò Chiaramonte, Alessio Gabellini, Andrea Ageli, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T Supuran, Maria Novella Romanelli
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators. Molecules (Basel, Switzerland) 27 (2) (2022)
Francesca Mancuso, Andrea Ageli, Viviana De Luca, Federica Bucolo, Laura De Luca, Clemente Capasso, Claudiu T Supuran, Rosaria Gitto
Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae. Archiv der Pharmazie 355 (10) (2022)
Angelica Artasensi, Andrea Ageli, Carmen Lammi, Carlotta Bollati, Silvia Gervasoni, Giovanna Baron, Rosanna Matucci, Claudiu T Supuran, Vistoli Giulio, Laura Fumagalli
Discovery of a Potent and Highly Selective Dipeptidyl Peptidase IV and Carbonic Anhydrase Inhibitor as "Antidiabesity" Agents Based on Repurposing and Morphing of WB-4101. Journal of medicinal chemistry 65 (20) (2022)
Arzu Gumus, Murat Bozdag, Atilla Akdemir, Andrea Ageli, Silvia Selleri, Fabrizio Carta, Claudiu T Supuran
Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII. Molecules (Basel, Switzerland) 27 (14) (2022)
Micheli Laura, Lara Testai, Andrea Ageli, Donatello Carrino, Alessandra Pacini, Francesco Margiotta, Lorenzo Flori, Claudiu T Supuran, Vincenzo Calderone, Carla Ghelardini, Di Cesare Mannelli Lorenzo
Inhibitors of Mitochondrial Human Carbonic Anhydrases VA and VB as a Therapeutic Strategy against Paclitaxel-Induced Neuropathic Pain in Mice. International journal of molecular sciences 23 (11) (2022)
Baijayantimala Swain, Abrar Khan, Priti Singh, Vaibhav S Marde, Andrea Ageli, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Simone Carradori, Claudiu T Supuran, Arifuddin Mohammed
Design, Synthesis and Biological Assessment of Rhodanine-Linked Benzenesulfonamide Derivatives as Selective and Potent Human Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 27 (22) (2022)
Tatiana Sharonova, Petr Zhmurov, Stanislav Kalinin, Alessio Nocentini, Andrea Ageli, Marta Ferraroni, Mikhail Korsakov, Claudiu T Supuran, Mikhail Krasavin
Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Hossam Nada, Ahmed Elkamhawy, Magda H Abdellatif, Andrea Ageli, Chang Hoon Lee, Claudiu T Supuran, Kyeong Lee
4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro , and in-silico biological studies. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Simone Carradori, Marialuigia Fantacuzzi, Alessandra Ammazzalorso, Andrea Ageli, Barbara De Filippis, Salvatore Galati, Anél Petzer, Jacobus P Petzer, Giulio Poli, Tiziano Tuccinardi, Mariangela Agamennone, Claudiu T Supuran
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases? Molecules (Basel, Switzerland) 27 (22) (2022)
Davide Moi, Alessandro Deplano, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity. Molecules (Basel, Switzerland) 27 (17) (2022)
Ahmed Elkamhawy, Jiyu Woo, Hossam Nada, Andrea Ageli, Dong Keun Han, Claudiu T Supuran, Kyeong Lee
Identification of Novel and Potent Indole-Based Benzenesulfonamides as Selective Human Carbonic Anhydrase II Inhibitors: Design, Synthesis, In Vitro, and In Silico Studies. International journal of molecular sciences 23 (5) (2022)
Andrea Ageli, Alice Velluzzi, Silvia Selleri, Clemente Capasso, Costanza Spadini, Mattia Iannarelli, Clotilde S Cabassi, Fabrizio Carta, Claudiu T Supuran
Seleno Containing Compounds as Potent and Selective Antifungal Agents. ACS infectious diseases 8 (9) (2022)
Viviana De Luca, Andrea Ageli, Valeria Mazzone, Claudia Adelfio, Vincenzo Carginale, Andrea Scaloni, Fabrizio Carta, Silvia Selleri, Claudiu T Supuran, Clemente Capasso
Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis . Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Thor Eysteinsson, Andrea García-Llorca, Andrea Ageli, Claudiu T Supuran, Fabrizio Carta
Vasodilation of Pre-contracted Porcine Retinal Arteries by Carbonic Anhydrase Inhibitors with Enhanced Lipophilicity. Current eye research 47 (12) (2022)
Davide Moi, Serena Vittorio, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. Molecules (Basel, Switzerland) 28 (1) (2022)
Oscar Francesconi, Francisco Corzana, Georgia-Ioanna Kontogianni, Giorgio Pesciullesi, Roberta Gualdani, Claudiu T Supuran, Andrea Ageli, Rafaela Maria Kavasi, Maria Chatzinikolaidou, Cristina Nativi
Lipoyl-Based Antagonists of Transient Receptor Potential Cation A (TRPA1) Downregulate Osteosarcoma Cell Migration and Expression of Pro-Inflammatory Cytokines. ACS pharmacology & translational science 5 (11) (2022)
Andrea Ageli, Marta Ferraroni, Fabrizio Carta, Cécile Häberli, Jennifer Keiser, Gabriele Costantino, Claudiu T Supuran
Development of Praziquantel sulphonamide derivatives as antischistosomal drugs. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Davide Moi, Serena Vittorio, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. Molecules (Basel, Switzerland) 28 (1) (2022)
Ilaria D'Agostino, Githa Elizabeth Mathew, Paola Angelini, Roberto Venanzoni, Giancarlo Angeles Flores, Andrea Ageli, Simone Carradori, Beatrice Marinacci, Luigi Menghini, Mohamed A Abdelgawad, Mohammed M Ghoneim, Bijo Mathew, Claudiu T Supuran
Biological investigation of N -methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Virginia Pontecorvi, Mattia Mori, Francesca Picarazzi, Susi Zara, Simone Carradori, Amelia Cataldi, Andrea Ageli, Emanuela Berrino, Paola Chimenti, Alessia Ciogli, Daniela Secci, Paolo Guglielmi, Claudiu T Supuran
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies. International journal of molecular sciences 23 (14) (2022)
Melisa E Gantner, Denis N Prada Gori, Manuel A Llanos, Alan Talevi, Andrea Ageli, Daniela Vullo, Claudiu T Supuran, Luciana Gavernet
Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 62 (19) (2022)
Davide Moi, Serena Vittorio, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. Molecules (Basel, Switzerland) 28 (1) (2022)
Gioele Vannozzi, Daniela Vullo, Andrea Ageli, Marta Ferraroni, Jacob Combs, Carrie Lomelino, Jacob T Andring, Robert Mckenna, Gianluca Bartolucci, Marco Pallecchi, Laura Lucarini, Silvia Sgambellone, Emanuela Masini, Fabrizio Carta, Claudiu T Supuran
One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. Journal of medicinal chemistry 65 (1) (2021)
Alessio Nocentini, Andrea Ageli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A Donald, Claudiu T Supuran
Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Andrea Ageli, Victor Kartsev, Petrou Anthi, Mariana Pinteală, Volodymyr Brovarets, Roman Vydzhak, Svitlana Y Panchishin, Geronikaki Athina, Claudiu T Supuran
Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors. Molecules (Basel, Switzerland) 26 (22) (2021)
Giacomo Biagiotti, Andrea Ageli, Arianna Giacomini, Gianluca Toniolo, Luca Landini, Gianluca Salerno, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Tommaso Mello, Silvia Mussi, Cosetta Ravelli, Marcello Marelli, Stefano Cicchi, Enzo Menna, Roberto Ronca, Claudiu T Supuran, Barbara Richichi
Glyco-Coated CdSe/ZnS Quantum Dots as Nanoprobes for Carbonic Anhydrase IX Imaging in Cancer Cells. ACS applied nano materials 4 (12) (2021)
Niccolò Chiaramonte, Soumia Maach, Caterina Biliotti, Andrea Ageli, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T Supuran, Maria Novella Romanelli
Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine1. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Charikleia Paloukopoulou, Sofia Govari, Athina Soulioti, Ilias Stefanis, Andrea Ageli, An Matheeussen, Clemente Capasso, Paul Cos, Claudiu T Supuran, Anastasia Karioti
Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase. Natural product research (2021)

Andrea Ageli.css-eqlu8i{font-size:small;padding-left:4px;} (Andrea Angeli)

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Andrea Ageli (Andrea Angeli)