Andrea Ageli (Andrea Angeli)

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2018-2023
Publications (10 Years): 129

Top Venues

Journal of enzyme inhibition and medicinal chemistry

International journal of molecular sciences

Molecules (Basel, Switzerland)

Journal of medicinal chemistry

Institutul de Chimie Macromoleculara Petru Poni

This page only lists publications with an associated author ORCID identifier.

Affiliation History

Institutul de Chimie Macromoleculara Petru Poni Jun 1o 2019

Romania

resercher :: Center of Advanced Research in Bionanoconjugates and Biopolymers

Publications

Marialuigia Fantacuzzi, Ilaria D'Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Mariangela Agamennone, Andrea Ageli, Filomena Sannio, Jean Denis Docquier, Clemente Capasso, Claudiu T Supuran
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris V Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Andrea Ageli, Niccolò Paoletti, Claudiu T Supuran
Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (7) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Moataz A Shaldam, Hadia Almahli, Andrea Ageli, Rehab Mustafa Badi, Eman F Khaleel, Abdelrahman I Zain-Alabdeen, Zainab M Elsayed, Eslam B Elkaeed, Rofaida Salem, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris V Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Lisa Sequeira, Simona Distinto, Rita Meleddu, Marco Gaspari, Andrea Ageli, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Fernanda Borges, Eugenio Uriarte, Stefano Alcaro, Claudiu T Supuran, Elias Maccioni
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Shaimaa M Aboukhatwa, Peter A Sidhom, Andrea Ageli, Claudiu T Supuran, Haytham O Tawfik
Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids. ACS omega 8 (8) (2023)
Andrea Ageli, Claudiu T Supuran
Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Moataz A Shaldam, Hadia Almahli, Andrea Ageli, Rehab Mustafa Badi, Eman F Khaleel, Abdelrahman I Zain-Alabdeen, Zainab M Elsayed, Eslam B Elkaeed, Rofaida Salem, Claudiu T Supuran, Wagdy M Eldehna, Haytham O Tawfik
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Belma Zengin Kurt, Gulsen Celebi, Dilek Ozturk Civelek, Andrea Ageli, Atilla Akdemir, Fatih Sonmez, Claudiu T Supuran
Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS omega 8 (6) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Ageli, Carmen Sanmartin, Claudiu T Supuran
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Jacob Combs, Murat Bozdag, Lochlin D Cravey, Anusha Kota, Robert McKenna, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 28 (2) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Simone Carradori, Andrea Ageli, Patrick Severin Sfragano, Xheila Yzeiri, Massimo Calamante, Damiano Tanini, Antonella Capperucci, Hannah Kunstek, Mihayl Varbanov, Clemente Capasso, Claudiu T Supuran
Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents. International journal of molecular sciences 24 (11) (2023)
Andrea Ageli, Laura Micheli, Fabrizio Carta, Marta Ferraroni, Tracey Pirali, Asia Fernandez Carvajal, Antonio Ferrer Montiel, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Claudiu T Supuran
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. Journal of medicinal chemistry 66 (2) (2023)
Andrea Ageli, Marta Ferraroni, Carlotta Granchi, Filippo Minutolo, Xiaozhuo Chen, Pratik Shriwas, Emilio Russo, Antonio Leo, Silvia Selleri, Fabrizio Carta, Claudiu T Supuran
First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome. Journal of medicinal chemistry (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Maria Giulia Davighi, Francesca Cardona, Andrea Goti, Marta Ferraroni, Andrea Ageli, Claudiu T Supuran, Francesca Cardona
Mono- and three-tailed sugar and iminosugar decorated benzenesulfonamide carbonic anhydrase inhibitors. Organic & biomolecular chemistry (2023)
Francesco Melfi, Simone Carradori, Andrea Ageli, Ilaria D'Agostino
Nature as a source and inspiration for human monoamine oxidase B (Hmao-B) inhibition: A review of the recent advances in chemical modification of natural compounds. Expert opinion on drug discovery (2023)
Shaimaa M Aboukhatwa, Peter A Sidhom, Andrea Ageli, Claudiu T Supuran, Haytham O Tawfik
Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids. ACS omega 8 (8) (2023)
Andrea Ageli, Claudiu T Supuran
Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Andrea Ageli, Petrou Anthi, Victor Kartsev, Boris V Lichitsky, Andrey Nikolaevich Komogortsev, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. International journal of molecular sciences 24 (3) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Susanna Haapanen, Andrea Ageli, Martti Tolvanen, Reza Zolfaghari Emameh, Claudiu T Supuran, Seppo Parkkila
Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni . Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Belma Zengin Kurt, Gulsen Celebi, Dilek Ozturk Civelek, Andrea Ageli, Atilla Akdemir, Fatih Sonmez, Claudiu T Supuran
Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS omega 8 (6) (2023)
Andrea Ageli, Marta Ferraroni, Alessandro Bonardi, Claudiu T Supuran, Alessio Nocentini
Diversely N -substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N -nitrosulfonamides. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Ageli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T Supuran, Srinivas Nanduri
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. Journal of enzyme inhibition and medicinal chemistry 38 (1) (2023)
Kiran Siwach, Amit Kumar, Harish Panchal, Rajiv Kumar, Jitender Kumar Bhardwaj, Andrea Ageli, Claudiu T Supuran, Pawan K Sharma
Selective inhibition of carbonic anhydrase IX by sulphonylated 1,2,3-triazole incorporated benzenesulphonamides capable of inducing apoptosis. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Haytham O Tawfik, Amany Belal, Mohammad A S Abourehab, Andrea Ageli, Alessandro Bonardi, Claudiu T Supuran, Mervat H El-Hamamsy
Dependence on linkers' flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Andrea Ageli, Victor Kartsev, Petrou Anthi, Boris Lichitsky, Andrey Nikolaevich Komogortsev, Mariana Pinteala, Geronikaki Athina, Claudiu T Supuran
Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies. Pharmaceuticals (Basel, Switzerland) 15 (3) (2022)
Andrea Ageli, Linda J Urbański, Clemente Capasso, Seppo Parkkila, Claudiu T Supuran
Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Mariangela Agamennone, Marialuigia Fantacuzzi, Simone Carradori, Anél Petzer, Jacobus P Petzer, Andrea Ageli, Claudiu T Supuran, Grazia Luisi
Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and ( Pseudo )-Dipeptidyl Appendages: In Vitro and Computational Studies. Molecules (Basel, Switzerland) 27 (22) (2022)
Niccolò Chiaramonte, Alessio Gabellini, Andrea Ageli, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T Supuran, Maria Novella Romanelli
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators. Molecules (Basel, Switzerland) 27 (2) (2022)
Francesca Mancuso, Andrea Ageli, Viviana De Luca, Federica Bucolo, Laura De Luca, Clemente Capasso, Claudiu T Supuran, Rosaria Gitto
Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae. Archiv der Pharmazie 355 (10) (2022)
Angelica Artasensi, Andrea Ageli, Carmen Lammi, Carlotta Bollati, Silvia Gervasoni, Giovanna Baron, Rosanna Matucci, Claudiu T Supuran, Vistoli Giulio, Laura Fumagalli
Discovery of a Potent and Highly Selective Dipeptidyl Peptidase IV and Carbonic Anhydrase Inhibitor as "Antidiabesity" Agents Based on Repurposing and Morphing of WB-4101. Journal of medicinal chemistry 65 (20) (2022)
Arzu Gumus, Murat Bozdag, Atilla Akdemir, Andrea Ageli, Silvia Selleri, Fabrizio Carta, Claudiu T Supuran
Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII. Molecules (Basel, Switzerland) 27 (14) (2022)
Laura Micheli, Lara Testai, Andrea Ageli, Donatello Carrino, Alessandra Pacini, Francesco Margiotta, Lorenzo Flori, Claudiu T Supuran, Vincenzo Calderone, Carla Ghelardini, Lorenzo Di Cesare Mannelli
Inhibitors of Mitochondrial Human Carbonic Anhydrases VA and VB as a Therapeutic Strategy against Paclitaxel-Induced Neuropathic Pain in Mice. International journal of molecular sciences 23 (11) (2022)
Baijayantimala Swain, Abrar Khan, Priti Singh, Vaibhav S Marde, Andrea Ageli, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Simone Carradori, Claudiu T Supuran, Arifuddin Mohammed
Design, Synthesis and Biological Assessment of Rhodanine-Linked Benzenesulfonamide Derivatives as Selective and Potent Human Carbonic Anhydrase Inhibitors. Molecules (Basel, Switzerland) 27 (22) (2022)
Tatiana Sharonova, Petr Zhmurov, Stanislav Kalinin, Alessio Nocentini, Andrea Ageli, Marta Ferraroni, Mikhail Korsakov, Claudiu T Supuran, Mikhail Krasavin
Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Hossam Nada, Ahmed Elkamhawy, Magda H Abdellatif, Andrea Ageli, Chang Hoon Lee, Claudiu T Supuran, Kyeong Lee
4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro , and in-silico biological studies. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Simone Carradori, Marialuigia Fantacuzzi, Alessandra Ammazzalorso, Andrea Ageli, Barbara De Filippis, Salvatore Galati, Anél Petzer, Jacobus P Petzer, Giulio Poli, Tiziano Tuccinardi, Mariangela Agamennone, Claudiu T Supuran
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases? Molecules (Basel, Switzerland) 27 (22) (2022)
Davide Moi, Alessandro Deplano, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity. Molecules (Basel, Switzerland) 27 (17) (2022)
Ahmed Elkamhawy, Jiyu Woo, Hossam Nada, Andrea Ageli, Dong Keun Han, Claudiu T Supuran, Kyeong Lee
Identification of Novel and Potent Indole-Based Benzenesulfonamides as Selective Human Carbonic Anhydrase II Inhibitors: Design, Synthesis, In Vitro, and In Silico Studies. International journal of molecular sciences 23 (5) (2022)
Andrea Ageli, Alice Velluzzi, Silvia Selleri, Clemente Capasso, Costanza Spadini, Mattia Iannarelli, Clotilde S Cabassi, Fabrizio Carta, Claudiu T Supuran
Seleno Containing Compounds as Potent and Selective Antifungal Agents. ACS infectious diseases 8 (9) (2022)
Viviana De Luca, Andrea Ageli, Valeria Mazzone, Claudia Adelfio, Vincenzo Carginale, Andrea Scaloni, Fabrizio Carta, Silvia Selleri, Claudiu T Supuran, Clemente Capasso
Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis . Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Thor Eysteinsson, Andrea García-Llorca, Andrea Ageli, Claudiu T Supuran, Fabrizio Carta
Vasodilation of Pre-contracted Porcine Retinal Arteries by Carbonic Anhydrase Inhibitors with Enhanced Lipophilicity. Current eye research 47 (12) (2022)
Davide Moi, Serena Vittorio, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. Molecules (Basel, Switzerland) 28 (1) (2022)
Oscar Francesconi, Francisco Corzana, Georgia-Ioanna Kontogianni, Giorgio Pesciullesi, Roberta Gualdani, Claudiu T Supuran, Andrea Ageli, Rafaela Maria Kavasi, Maria Chatzinikolaidou, Cristina Nativi
Lipoyl-Based Antagonists of Transient Receptor Potential Cation A (TRPA1) Downregulate Osteosarcoma Cell Migration and Expression of Pro-Inflammatory Cytokines. ACS pharmacology & translational science 5 (11) (2022)
Andrea Ageli, Marta Ferraroni, Fabrizio Carta, Cécile Häberli, Jennifer Keiser, Gabriele Costantino, Claudiu T Supuran
Development of Praziquantel sulphonamide derivatives as antischistosomal drugs. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Davide Moi, Serena Vittorio, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. Molecules (Basel, Switzerland) 28 (1) (2022)
Ilaria D'Agostino, Githa Elizabeth Mathew, Paola Angelini, Roberto Venanzoni, Giancarlo Angeles Flores, Andrea Ageli, Simone Carradori, Beatrice Marinacci, Luigi Menghini, Mohamed A Abdelgawad, Mohammed M Ghoneim, Bijo Mathew, Claudiu T Supuran
Biological investigation of N -methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors. Journal of enzyme inhibition and medicinal chemistry 37 (1) (2022)
Virginia Pontecorvi, Mattia Mori, Francesca Picarazzi, Susi Zara, Simone Carradori, Amelia Cataldi, Andrea Ageli, Emanuela Berrino, Paola Chimenti, Alessia Ciogli, Daniela Secci, Paolo Guglielmi, Claudiu T Supuran
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies. International journal of molecular sciences 23 (14) (2022)
Melisa E Gantner, Denis N Prada Gori, Manuel A Llanos, Alan Talevi, Andrea Ageli, Daniela Vullo, Claudiu T Supuran, Luciana Gavernet
Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening. Journal of chemical information and modeling 62 (19) (2022)
Davide Moi, Serena Vittorio, Andrea Ageli, Gianfranco Balboni, Claudiu T Supuran, Valentina Onnis
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. Molecules (Basel, Switzerland) 28 (1) (2022)
Gioele Vannozzi, Daniela Vullo, Andrea Ageli, Marta Ferraroni, Jacob Combs, Carrie Lomelino, Jacob T Andring, Robert Mckenna, Gianluca Bartolucci, Marco Pallecchi, Laura Lucarini, Silvia Sgambellone, Emanuela Masini, Fabrizio Carta, Claudiu T Supuran
One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. Journal of medicinal chemistry 65 (1) (2021)
Alessio Nocentini, Andrea Ageli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A Donald, Claudiu T Supuran
Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Andrea Ageli, Victor Kartsev, Petrou Anthi, Mariana Pinteala, Volodymyr Brovarets, Roman Vydzhak, Svitlana Y Panchishin, Geronikaki Athina, Claudiu T Supuran
Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors. Molecules (Basel, Switzerland) 26 (22) (2021)
Giacomo Biagiotti, Andrea Ageli, Arianna Giacomini, Gianluca Toniolo, Luca Landini, Gianluca Salerno, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Tommaso Mello, Silvia Mussi, Cosetta Ravelli, Marcello Marelli, Stefano Cicchi, Enzo Menna, Roberto Ronca, Claudiu T Supuran, Barbara Richichi
Glyco-Coated CdSe/ZnS Quantum Dots as Nanoprobes for Carbonic Anhydrase IX Imaging in Cancer Cells. ACS applied nano materials 4 (12) (2021)
Niccolò Chiaramonte, Soumia Maach, Caterina Biliotti, Andrea Ageli, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T Supuran, Maria Novella Romanelli
Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine1. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Charikleia Paloukopoulou, Sofia Govari, Athina Soulioti, Ilias Stefanis, Andrea Ageli, An Matheeussen, Clemente Capasso, Paul Cos, Claudiu T Supuran, Anastasia Karioti
Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase. Natural product research (2021)
Rita Meleddu, Serenella Deplano, Elias Maccioni, Francesco Ortuso, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Andrea Ageli, Rossella Angius, Stefano Alcaro, Claudiu T Supuran, Simona Distinto
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Andrea Ageli, Victor Kartsev, Petrou Anthi, Mariana Pinteala, Roman M Vydzhak, Svitlana Y Panchishin, Volodymyr Brovarets, Viviana De Luca, Clemente Capasso, Geronikaki Athina, Claudiu T Supuran
New Sulfanilamide Derivatives Incorporating Heterocyclic Carboxamide Moieties as Carbonic Anhydrase Inhibitors. Pharmaceuticals (Basel, Switzerland) 14 (8) (2021)
Chandra Bhushan Mishra, Shikha Kumari, Andrea Ageli, Silvia Bua, Raj Kumar Mongre, Manisha Tiwari, Claudiu T Supuran
Discovery of Potent Carbonic Anhydrase Inhibitors as Effective Anticonvulsant Agents: Drug Design, Synthesis, and In Vitro and In Vivo Investigations. Journal of medicinal chemistry 64 (6) (2021)
Murat Bozdag, Claudiu T Supuran, Davide Esposito, Andrea Ageli, Fabrizio Carta, Simona Maria Monti, Giuseppina De Simone, Vincenzo Alterio
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site. Chemical communications (Cambridge, England) 56 (59) (2021)
Emanuela Berrino, Simone Carradori, Andrea Ageli, Fabrizio Carta, Claudiu T Supuran, Paolo Guglielmi, Cecilia Coletti, Roberto Paciotti, Helmut Schweikl, Francesca Maestrelli, Elisabetta Cerbai, Marialucia Gallorini
Dual Carbonic Anhydrase IX/XII Inhibitors and Carbon Monoxide Releasing Molecules Modulate LPS-Mediated Inflammation in Mouse Macrophages. Antioxidants (Basel, Switzerland) 10 (1) (2021)
Linda J Urbański, Andrea Ageli, Vesa P Hytönen, Anna Di Fiore, Giuseppina De Simone, Seppo Parkkila, Claudiu T Supuran
Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Andrea Ageli, Marta Ferraroni, Akram A Da'dara, Silvia Selleri, Mariana Pinteala, Fabrizio Carta, Patrick J Skelly, Claudiu T Supuran
Structural Insights into Schistosoma mansoni Carbonic Anhydrase (SmCA) Inhibition by Selenoureido-Substituted Benzenesulfonamides. Journal of medicinal chemistry 64 (14) (2021)
Andrea Ageli, Emanuela Berrino, Simone Carradori, Claudiu T Supuran, Marzia Cirri, Fabrizio Carta, Gabriele Costantino
Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators. Molecules (Basel, Switzerland) 26 (23) (2021)
Linda J Urbański, Anna Di Fiore, Latifeh Azizi, Vesa P Hytönen, Marianne Kuuslahti, Martina Buonanno, Simona M Monti, Andrea Ageli, Reza Zolfaghari Emameh, Claudiu T Supuran, Giuseppina De Simone, Seppo Parkkila
Biochemical and structural characterisation of a protozoan beta-carbonic anhydrase from Trichomonas vaginalis. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Francesca Mancuso, Laura De Luca, Andrea Ageli, Sonia Del Prete, Clemente Capasso, Claudiu T Supuran, Rosaria Gitto
Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Linda J Urbanski, Silvia Bua, Andrea Ageli, Marianne Kuuslahti, Vesa P Hytönen, Claudiu T Supuran, Seppo Parkkila
Sulphonamide inhibition profile of Staphylococcus aureus β-carbonic anhydrase. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Pavitra S Thacker, Prerna L Tiwari, Andrea Ageli, Danaboina Srikanth, Baijayantimala Swain, Arifuddin Mohammed, Claudiu T Supuran
Synthesis and Biological Evaluation of Coumarin-Linked 4-Anilinomethyl-1,2,3-Triazoles as Potent Inhibitors of Carbonic Anhydrases IX and XIII Involved in Tumorigenesis. Metabolites 11 (4) (2021)
Francesca Mancuso, Laura De Luca, Federica Bucolo, Milan Vrabel, Andrea Ageli, Clemente Capasso, Claudiu T Supuran, Rosaria Gitto
4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae. ChemMedChem (2021)
Rossella Grande, Simone Carradori, Valentina Puca, Irene Vitale, Andrea Ageli, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Paola Lanuti, Giuseppina Bologna, Pasquale Simeone, Clemente Capasso, Viviana De Luca, Claudiu T Supuran
Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles. International journal of molecular sciences 22 (21) (2021)
Paolo Guglielmi, Giulia Rotondi, Daniela Secci, Andrea Ageli, Paola Chimenti, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Simone Carradori, Claudiu T Supuran
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2021)
Andrea Ageli, Victor Kartsev, Petrou Anthi, Mariana Pinteala, Volodymyr Brovarets, Sergii Slyvchuk, Stepan Pilyo, Geronikaki Athina, Claudiu T Supuran
Chromene-Containing Aromatic Sulfonamides with Carbonic Anhydrase Inhibitory Properties. International journal of molecular sciences 22 (10) (2021)
Andrea Ageli, Linda J Urbański, Vesa P Hytönen, Seppo Parkkila, Claudiu T Supuran
Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Elisabetta Barresi, Rahul Ravichandran, Lorenzo Germelli, Andrea Ageli, Emma Baglini, Silvia Salerno, Anna Maria Marini, Barbara Costa, Eleonora Da Pozzo, Claudia Martini, Federico Da Settimo, Claudiu T Supuran, Sandro Cosconati, Sabrina Taliani
Carbonic anhydrase activation profile of indole-based derivatives. Journal of enzyme inhibition and medicinal chemistry 36 (1) (2021)
Eva Havránková, Vladimír Garaj, Šárka Mascaretti, Andrea Ageli, Zuzana Soldánová, Miroslav Kemka, Jozef Motyčka, Marie Brázdová, Jozef Csöllei, Josef Jampilek, Claudiu T Supuran
Novel 1,3,5-Triazinyl Aminobenzenesulfonamides Incorporating Aminoalcohol, Aminochalcone and Aminostilbene Structural Motifs as Potent Anti-VRE Agents, and Carbonic Anhydrases I, II, VII, IX, and XII Inhibitors. International journal of molecular sciences 23 (1) (2021)
Anna A Plyasova, Emanuela Berrino, Irina I Khan, Alexander V Veselovsky, Vadim S Pokrovsky, Andrea Ageli, Marta Ferraroni, Claudiu T Supuran, Marina V Pokrovskaya, Svetlana S Alexandrova, Yulia A Gladilina, Nikolay N Sokolov, Abdullah Hilal, Fabrizio Carta, Dmitry D Zhdanov
Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors. Journal of medicinal chemistry 64 (15) (2021)
Viviana De Luca, Andrea Ageli, Valeria Mazzone, Claudia Adelfio, Fabrizio Carta, Silvia Selleri, Vincenzo Carginale, Andrea Scaloni, Claudiu T Supuran, Clemente Capasso
Inhibitory Effects of Sulfonamide Derivatives on the β-Carbonic Anhydrase (MpaCA) from Malassezia pachydermatis, a Commensal, Pathogenic Fungus Present in Domestic Animals. International journal of molecular sciences 22 (22) (2021)
Andrea Ageli, Bogdan-Florin Craciun, Stelian Sergiu Maier, Bogdan C Simionescu, Akram A Da'dara, Patrick J Skelly, Claudiu T Supuran
Sulfonamide Inhibition Studies of an α-Carbonic Anhydrase from Schistosoma mansoni, a Platyhelminth Parasite Responsible for Schistosomiasis. International journal of molecular sciences 21 (5) (2020)
Felipe Raposo Passos Mansoldo, Fabrizio Carta, Andrea Ageli, Verônica da Silva Cardoso, Claudiu T Supuran, Alane Beatriz Vermelho
Chagas Disease: Perspectives on the Past and Present and Challenges in Drug Discovery. Molecules (Basel, Switzerland) 25 (22) (2020)
Majid Ali, Murat Bozdag, Umar Farooq, Andrea Ageli, Fabrizio Carta, Paola Berto, Giuseppe Zanotti, Claudiu T Supuran
Benzylaminoethyureido-Tailed Benzenesulfonamides: Design, Synthesis, Kinetic and X-ray Investigations on Human Carbonic Anhydrases. International journal of molecular sciences 21 (7) (2020)
Kübra Demir-Yazıcı, Özlen Güzel-Akdemir, Andrea Ageli, Claudiu T Supuran, Atilla Akdemir
Novel Indole-Based Hydrazones as Potent Inhibitors of the α-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae. International journal of molecular sciences 21 (9) (2020)
Barbara Kaproń, Robert Czarnomysy, Mariusz Wysokiński, Rudolf Andrys, Kamil Musilek, Andrea Ageli, Claudiu T Supuran, Tomasz Plech
1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2020)
Mikhail Krasavin, Stanislav Kalinin, Sergey Zozulya, Anastasia Griniukova, Petro Borysko, Andrea Ageli, Claudiu T Supuran
Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scanning fluorimetry leads to chemotype refinement. Journal of enzyme inhibition and medicinal chemistry 35 (1) (2020)

Andrea Ageli.css-eqlu8i{font-size:small;padding-left:4px;} (Andrea Angeli)

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Andrea Ageli (Andrea Angeli)