Ian H Gilbert

Scopus Author ID ORCID

Publication Activity (10 Years)

Years Active: 2017-2023
Publications (10 Years): 52

Top Venues

ACS infectious diseases

Journal of medicinal chemistry

Nature reviews. Chemistry

ACS omega

This page only lists publications with an associated author ORCID identifier.

Publications

Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases 9 (5) (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases 9 (5) (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases 9 (5) (2023)
Simon R Green, Caroline Wilson, Thomas C Eadsforth, Avinash S Punekar, Fabio K Tamaki, Gavin Wood, Nicola Caldwell, Barbara Forte, Neil R Norcross, Michael Kiczun, John M Post, Eva Maria Lopez-Román, Curtis A Engelhart, Iva Lukac, Fabio Zuccotto, Ola Epemolu, Helena I M Boshoff, Dirk Schnappinger, Chris Walpole, Ian H Gilbert, Kevin D Read, Paul G Wyatt, Beatriz Baragaña
Identification and Optimization of Novel Inhibitors of the Polyketide Synthase 13 Thioesterase Domain with Antitubercular Activity. Journal of medicinal chemistry (2023)
Megan Bergkessel, Barbara Forte, Ian H Gilbert
Small-Molecule Antibiotic Drug Development: Need and Challenges. ACS infectious diseases (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases 9 (5) (2023)
Riccardo Guareschi, Iva Lukac, Ian H Gilbert, Fabio Zuccotto
SophosQM: Accurate Binding Affinity Prediction in Compound Optimization. ACS omega 8 (17) (2023)
James S Martin, Claire J Mackenzie, De Lin, Nadine Homeyer, David W Gray, Fabio Zuccotto, Ian H Gilbert
Design and Synthesis of Covalent Inhibitors of FabA. ACS omega 8 (14) (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases 9 (5) (2023)
Laura A T Cleghorn, Richard J Wall, Sébastien Albrecht, Stuart A MacGowan, Suzanne Norval, Manu De Rycker, Andrew Woodland, Daniel Spinks, Stephen Thompson, Stephen Patterson, Victoriano Corpas Lopez, Gourav Dey, Iain T Collie, Irene Hallyburton, Robert Kime, Frederick R C Simeons, Laste Stojanovski, Julie A Frearson, Paul G Wyatt, Kevin D Read, Ian H Gilbert, Susan Wyllie
Development of a 2,4-Diaminothiazole Series for the Treatment of Human African Trypanosomiasis Highlights the Importance of Static-Cidal Screening of Analogues. Journal of medicinal chemistry (2023)
Michael G Thomas, Kate McGonagle, Paul Rowland, David A Robinson, Peter G Dodd, Isabel Camino-Díaz, Lorna Campbell, Juan Cantizani, Pablo Castañeda, Daniel Conn, Peter D Craggs, Darren Edwards, Liam Ferguson, Andrew Fosberry, Laura Frame, Panchali Goswami, Xiao Hu, Justyna Korczynska, Lorna MacLean, J Julio Martin, Nicole Mutter, Maria Osuna-Cabello, Christy Paterson, Imanol Peña, Erika G Pinto, Caterina Pont, Jennifer Riley, Yoko Shishikura, Frederick R C Simeons, Laste Stojanovski, John Thomas, Karolina Wrobel, Robert J Young, Filip Zmuda, Fabio Zuccotto, Kevin D Read, Ian H Gilbert, Maria Marco, Timothy J Miles, Pilar Manzano, Manu De Rycker
Structure-Guided Design and Synthesis of a Pyridazinone Series of Trypanosoma cruzi Proteasome Inhibitors. Journal of medicinal chemistry (2023)
Riccardo Guareschi, Iva Lukac, Ian H Gilbert, Fabio Zuccotto
SophosQM: Accurate Binding Affinity Prediction in Compound Optimization. ACS omega 8 (17) (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases (2023)
Yamuna Devi Bakthavatchalam, Divyaa Elangovan, Subha Vajjiravelu Jaganathan, Nivedhana Subburaju, Abirami Shankar, Yuvasri Manokaran, Sudarsana J, Rema Devi, Sujata Baveja, Sheela Devi, Jayakumar S, Sanjay Bhattacharya, Rudresh S M, Bineshlal Yesudhason, Vignesh Shetty, Ankur Mutreja, Abi Manesh, George M Varghese, Charis A Marwick, Benjamin J Parcell, Ian H Gilbert, Veeraraghavan Balaji
In Vitro Activity of Two Cefepime-Based Novel Combinations, Cefepime/Taniborbactam and Cefepime/Zidebactam, against Carbapenemase-Expressing Enterobacterales Collected in India. Microbiology spectrum (2023)
Nicola Caldwell, Rana Afshar, Beatriz Baragaña, Amaya L Bustinduy, Conor R Caffrey, James J Collins, Daniela Fusco, Amadou Garba, Mark Gardner, Mireille Gomes, Karl F Hoffmann, Michael Hsieh, Nathan C Lo, Case W MacNamara, Justin Komguep Nono, Gilda Padalino, Kevin D Read, Meta Roestenberg, Thomas Spangenberg, Sabine Specht, Ian H Gilbert
Perspective on Schistosomiasis Drug Discovery: Highlights from a Schistosomiasis Drug Discovery Workshop at Wellcome Collection, London, September 2022. ACS infectious diseases (2023)
Lauren A Webster, Susan E Farrell, Ian H Gilbert, Kevin D Read
Bespoke Drug Discovery Training for Low-Middle Income Countries. ACS medicinal chemistry letters 14 (8) (2023)
Lauren A Webster, Susan E Farrell, Ian H Gilbert, Paul G Wyatt, Kevin D Read
Correction to "Bespoke Drug Discovery Training for Low-Middle Income Countries". ACS medicinal chemistry letters 14 (11) (2023)
Fabio Tamaki, Fabio Fisher, Rachel Milne, Fernando Sánchez-Román Terán, Natalie Wiedemar, Karolina Wrobel, Darren Edwards, Hella Baumann, Ian H Gilbert, Beatriz Baragana, Jake Baum, Susan Wyllie
High-Throughput Screening Platform To Identify Inhibitors of Protein Synthesis with Potential for the Treatment of Malaria. Antimicrobial agents and chemotherapy 66 (6) (2022)
Simon R Green, Susan H Davis, Sebastian Damerow, Curtis A Engelhart, Michael Mathieson, Beatriz Baragaña, David A Robinson, Jevgenia Tamjar, Alice Dawson, Fabio K Tamaki, Kirsteen I Buchanan, John Post, Karen Dowers, Sharon M Shepherd, Chimed Jansen, Fabio Zuccotto, Ian H Gilbert, Ola Epemolu, Jennifer Riley, Laste Stojanovski, Maria Osuna-Cabello, Esther Pérez-Herrán, María José Rebollo, Laura Guijarro López, Patricia Casado Castro, Isabel Camino, Heather C Kim, James M Bean, Navid Nahiyaan, Kyu Y Rhee, Qinglan Wang, Vee Y Tan, Helena I M Boshoff, Paul J Converse, Si-Yang Li, Yong S Chang, Nader Fotouhi, Anna M Upton, Eric L Nuermberger, Dirk Schnappinger, Kevin D Read, Lourdes Encinas, Robert H Bates, Paul G Wyatt, Laura A T Cleghorn
Lysyl-tRNA synthetase, a target for urgently needed M. tuberculosis drugs. Nature communications 13 (1) (2022)
Alasdair Smith, Richard J Wall, Stephen Patterson, Tim Rowan, Eva Rico Vidal, Laste Stojanovski, Margaret Huggett, Shahienaz E Hampton, Michael G Thomas, Victoriano Corpas Lopez, Kirsten Gillingwater, Jeff Duke, Grant Napier, Rose Peter, Hervé S Vitouley, Justin R Harrison, Rachel Milne, Laura Jeacock, Nicola Baker, Susan H Davis, Frederick Simeons, Jennifer Riley, David Horn, Reto Brun, Fabio Zuccotto, Michael J Witty, Susan Wyllie, Kevin D Read, Ian H Gilbert
Repositioning of a Diaminothiazole Series Confirmed to Target the Cyclin-Dependent Kinase CRK12 for Use in the Treatment of African Animal Trypanosomiasis. Journal of medicinal chemistry 65 (7) (2022)
Franz S Gruber, Zoe C Johnston, Neil R Norcross, Irene Georgiou, Caroline Wilson, Kevin D Read, Ian H Gilbert, Jason R Swedlow, Sarah Martins Da Silva, Christopher L R Barratt
Compounds enhancing human sperm motility identified using a high-throughput phenotypic screening platform. Human reproduction (Oxford, England) 37 (3) (2022)
Manu De Rycker, Susan Wyllie, David Horn, Kevin D Read, Ian H Gilbert
Anti-trypanosomatid drug discovery: progress and challenges. Nature reviews. Microbiology (2022)
Rachel Milne, Natalie Wiedemar, Victoriano Corpas-Lopez, Eoin Moynihan, Richard J Wall, Alice Dawson, David A Robinson, Sharon M Shepherd, Robert J Smith, Irene Hallyburton, John M Post, Karen Dowers, Leah S Torrie, Ian H Gilbert, Beatriz Baragaña, Stephen Patterson, Susan Wyllie
Toolkit of Approaches To Support Target-Focused Drug Discovery for Plasmodium falciparum Lysyl tRNA Synthetase. ACS infectious diseases 8 (9) (2022)
Marcus Miethke, Marco Pieroni, Tilmann Weber, Mark Brönstrup, Peter Hammann, Ludovic Halby, Paola B Arimondo, Philippe Glaser, Bertrand Aigle, Helge B Bode, Rui Moreira, Yanyan Li, Andriy Luzhetskyy, Marnix H Medema, Jean-Luc Pernodet, Marc Stadler, José Rubén Tormo, Olga Genilloud, Andrew W Truman, Kira J Weissman, Eriko Takano, Stefano Sabatini, Evi Stegmann, Heike Brötz-Oesterhelt, Wolfgang Wohlleben, Myriam Seemann, Martin Empting, Anna K H Hirsch, Brigitta Loretz, Claus-Michael Lehr, Alexander Titz, Jennifer Herrmann, Timo Jaeger, Silke Alt, Thomas Hesterkamp, Mathias Winterhalter, Andrea Schiefer, Kenneth M Pfarr, Achim Hoerauf, Heather Graz, Michael Graz, Mika Lindvall, Savithri Ramurthy, Anders Karlén, Maarten van Dongen, Hrvoje Petkovic, Andreas Keller, Frédéric Peyrane, Stefano Donadio, Laurent Fraisse, Laura J V Piddock, Ian H Gilbert, Heinz E Moser, Daniel Krug
Towards the sustainable discovery and development of new antibiotics. Nature reviews. Chemistry 5 (10) (2021)
James S Martin, Claire J Mackenzie, Ian H Gilbert
Synthesis of a Series of Diaminoindoles. The Journal of organic chemistry 86 (17) (2021)
Marcus Miethke, Marco Pieroni, Tilmann Weber, Mark Brönstrup, Peter Hammann, Ludovic Halby, Paola B Arimondo, Philippe Glaser, Bertrand Aigle, Helge B Bode, Rui Moreira, Yanyan Li, Andriy Luzhetskyy, Marnix H Medema, Jean-Luc Pernodet, Marc Stadler, José Rubén Tormo, Olga Genilloud, Andrew W Truman, Kira J Weissman, Eriko Takano, Stefano Sabatini, Evi Stegmann, Heike Brötz-Oesterhelt, Wolfgang Wohlleben, Myriam Seemann, Martin Empting, Anna K H Hirsch, Brigitta Loretz, Claus-Michael Lehr, Alexander Titz, Jennifer Herrmann, Timo Jaeger, Silke Alt, Thomas Hesterkamp, Mathias Winterhalter, Andrea Schiefer, Kenneth M Pfarr, Achim Hoerauf, Heather Graz, Michael Graz, Mika Lindvall, Savithri Ramurthy, Anders Karlén, Maarten van Dongen, Hrvoje Petkovic, Andreas Keller, Frédéric Peyrane, Stefano Donadio, Laurent Fraisse, Laura J V Piddock, Ian H Gilbert, Heinz E Moser, Daniel Krug
Towards the sustainable discovery and development of new antibiotics. Nature reviews. Chemistry 5 (10) (2021)
Charles E Mowbray, Stéphanie Braillard, Paul A Glossop, Gavin A Whitlock, Robert T Jacobs, Jason Speake, Bharathi Pandi, Bakela Nare, Louis Maes, Vanessa Yardley, Yvonne Freund, Richard J Wall, Sandra Carvalho, Davide Bello, Magali Van den Kerkhof, Guy Caljon, Ian H Gilbert, Victoriano Corpas-Lopez, Iva Lukac, Stephen Patterson, Fabio Zuccotto, Susan Wyllie
DNDI-6148: A Novel Benzoxaborole Preclinical Candidate for the Treatment of Visceral Leishmaniasis. Journal of medicinal chemistry 64 (21) (2021)
Iva Lukac, Paul G Wyatt, Ian H Gilbert, Fabio Zuccotto
Ligand binding: evaluating the contribution of the water molecules network using the Fragment Molecular Orbital method. Journal of computer-aided molecular design 35 (10) (2021)
Michael G Thomas, Stephen Brand, Manu De Rycker, Fabio Zuccotto, Iva Lukac, Peter G Dodd, Eun-Jung Ko, Sujatha Manthri, Kate McGonagle, Maria Osuna-Cabello, Jennifer Riley, Caterina Pont, Frederick Simeons, Laste Stojanovski, John Thomas, Stephen Thompson, Elisabet Viayna, Jose M Fiandor, J Julio Martin, Paul G Wyatt, Timothy J Miles, Kevin D Read, Maria Marco, Ian H Gilbert
Scaffold-Hopping Strategy on a Series of Proteasome Inhibitors Led to a Preclinical Candidate for the Treatment of Visceral Leishmaniasis. Journal of medicinal chemistry 64 (9) (2021)
Lauren B Arendse, Susan Wyllie, Kelly Chibale, Ian H Gilbert
Plasmodium Kinases as Potential Drug Targets for Malaria: Challenges and Opportunities. ACS infectious diseases 7 (3) (2021)
Marcus Miethke, Marco Pieroni, Tilmann Weber, Mark Brönstrup, Peter Hammann, Ludovic Halby, Paola B Arimondo, Philippe Glaser, Bertrand Aigle, Helge B Bode, Rui Moreira, Yanyan Li, Andriy Luzhetskyy, Marnix H Medema, Jean-Luc Pernodet, Marc Stadler, José Rubén Tormo, Olga Genilloud, Andrew W Truman, Kira J Weissman, Eriko Takano, Stefano Sabatini, Evi Stegmann, Heike Brötz-Oesterhelt, Wolfgang Wohlleben, Myriam Seemann, Martin Empting, Anna K H Hirsch, Brigitta Loretz, Claus-Michael Lehr, Alexander Titz, Jennifer Herrmann, Timo Jaeger, Silke Alt, Thomas Hesterkamp, Mathias Winterhalter, Andrea Schiefer, Kenneth M Pfarr, Achim Hoerauf, Heather Graz, Michael Graz, Mika Lindvall, Savithri Ramurthy, Anders Karlén, Maarten van Dongen, Hrvoje Petkovic, Andreas Keller, Frédéric Peyrane, Stefano Donadio, Laurent Fraisse, Laura J V Piddock, Ian H Gilbert, Heinz E Moser, Daniel Krug
Towards the sustainable discovery and development of new antibiotics. Nature reviews. Chemistry (2021)
Barbara Forte, Sabine Ottilie, Andrew Plater, Brice Campo, Koen J Dechering, Francisco Javier Gamo, Daniel E Goldberg, Eva S Istvan, Marcus Lee, Amanda K Lukens, Case W MacNamara, Jacquin C Niles, John Okombo, Charisse Flerida A Pasaje, Miles G Siegel, Dyann Wirth, Susan Wyllie, David A Fidock, Beatriz Baragaña, Elizabeth A Winzeler, Ian H Gilbert
Prioritization of Molecular Targets for Antimalarial Drug Discovery. ACS infectious diseases 7 (10) (2021)
Karolina Michalska, Robert Jedrzejczak, Jacek Wower, Changsoo Chang, Beatriz Baragaña, Ian H Gilbert, Barbara Forte, Andrzej Joachimiak
Mycobacterium tuberculosis Phe-tRNA synthetase: structural insights into tRNA recognition and aminoacylation. Nucleic acids research 49 (9) (2021)
Michael G Thomas, Manu De Rycker, Richard J Wall, Daniel Spinks, Ola Epemolu, Sujatha Manthri, Suzanne Norval, Maria Osuna-Cabello, Stephen Patterson, Jennifer Riley, Frederick R C Simeons, Laste Stojanovski, John Thomas, Stephen Thompson, Claire Naylor, Jose M Fiandor, Paul G Wyatt, Maria Marco, Susan Wyllie, Kevin D Read, Timothy J Miles, Ian H Gilbert
Identification and Optimization of a Series of 8-Hydroxy Naphthyridines with Potent In Vitro Antileishmanial Activity: Initial SAR and Assessment of In Vivo Activity. Journal of medicinal chemistry 63 (17) (2020)
Leah S Torrie, David A Robinson, Michael G Thomas, Judith V Hobrath, Sharon M Shepherd, John M Post, Eun-Jung Ko, Rafael Alves Ferreira, Claire J Mackenzie, Karolina Wrobel, Darren P Edwards, Ian H Gilbert, David W Gray, Alan H Fairlamb, Manu De Rycker
Discovery of an Allosteric Binding Site in Kinetoplastid Methionyl-tRNA Synthetase. ACS infectious diseases 6 (5) (2020)
Richard J Wall, Sandra Carvalho, Rachel Milne, Juan A Bueren-Calabuig, Sonia Moniz, Juan Cantizani-Perez, Lorna MacLean, Albane Kessler, Ignacio Cotillo, Lalitha Sastry, Sujatha Manthri, Stephen Patterson, Fabio Zuccotto, Stephen Thompson, Julio Martin, Maria Marco, Timothy J Miles, Manu De Rycker, Michael G Thomas, Alan H Fairlamb, Ian H Gilbert, Susan Wyllie
The Qi Site of Cytochrome b is a Promiscuous Drug Target in Trypanosoma cruzi and Leishmania donovani. ACS infectious diseases 6 (3) (2020)
Justin R Harrison, Sandipan Sarkar, Shahienaz E Hampton, Jennifer Riley, Laste Stojanovski, Christer Sahlberg, Pia Appelqvist, Jessey Erath, Vinodhini Mathan, Ana Rodriguez, Marcel Kaiser, Dolores Gonzalez Pacanowska, Kevin D Read, Nils Gunnar Johansson, Ian H Gilbert
Discovery and Optimization of a Compound Series Active against Trypanosoma cruzi, the Causative Agent of Chagas Disease. Journal of medicinal chemistry 63 (6) (2020)
Beatriz Baragaña, Barbara Forte, Ryan Choi, Stephen Nakazawa Hewitt, Juan A Bueren-Calabuig, João Pedro Pisco, Caroline Peet, David M Dranow, David A Robinson, Chimed Jansen, Neil R Norcross, Sumiti Vinayak, Mark Anderson, Carrie F Brooks, Caitlin A Cooper, Sebastian Damerow, Michael Delves, Karen Dowers, James Duffy, Thomas E Edwards, Irene Hallyburton, Benjamin G Horst, Matthew A Hulverson, Liam Ferguson, María Belén Jiménez-Díaz, Rajiv S Jumani, Donald D Lorimer, Melissa S Love, Steven Maher, Holly Matthews, Case W McNamara, Peter Miller, Sandra O'Neill, Kayode K Ojo, Maria Osuna-Cabello, Erika Pinto, John Post, Jennifer Riley, Matthias Rottmann, Laura M Sanz, Paul Scullion, Arvind Sharma, Sharon M Shepherd, Yoko Shishikura, Frederick R C Simeons, Erin E Stebbins, Laste Stojanovski, Ursula Straschil, Fabio K Tamaki, Jevgenia Tamjar, Leah S Torrie, Amélie Vantaux, Benoît Witkowski, Sergio Wittlin, Manickam Yogavel, Fabio Zuccotto, Iñigo Angulo-Barturen, Robert Sinden, Jake Baum, Francisco-Javier Gamo, Pascal Mäser, Dennis E Kyle, Elizabeth A Winzeler, Peter J Myler, Paul G Wyatt, David Floyd, David Matthews, Amit Sharma, Boris Striepen, Christopher D Huston, David W Gray, Alan H Fairlamb, Andrei V Pisliakov, Chris Walpole, Kevin D Read, Wesley C Van Voorhis, Ian H Gilbert
Lysyl-tRNA synthetase as a drug target in malaria and cryptosporidiosis. Proceedings of the National Academy of Sciences of the United States of America 116 (14) (2019)
Susan Wyllie, Stephen Brand, Michael Thomas, Manu De Rycker, Chun-Wa Chung, Imanol Pena, Ryan P Bingham, Juan A Bueren-Calabuig, Juan Cantizani, David Cebrian, Peter D Craggs, Liam Ferguson, Panchali Goswami, Judith Hobrath, Jonathan Howe, Laura Jeacock, Eun-Jung Ko, Justyna Korczynska, Lorna MacLean, Sujatha Manthri, Maria S Martinez, Lydia Mata-Cantero, Sonia Moniz, Andrea Nühs, Maria Osuna-Cabello, Erika Pinto, Jennifer Riley, Sharon Robinson, Paul Rowland, Frederick R C Simeons, Yoko Shishikura, Daniel Spinks, Laste Stojanovski, John Thomas, Stephen Thompson, Elisabet Viayna Gaza, Richard J Wall, Fabio Zuccotto, David Horn, Michael A J Ferguson, Alan H Fairlamb, Jose M Fiandor, Julio Martin, David W Gray, Timothy J Miles, Ian H Gilbert, Kevin D Read, Maria Marco, Paul G Wyatt
Preclinical candidate for the treatment of visceral leishmaniasis that acts through proteasome inhibition. Proceedings of the National Academy of Sciences of the United States of America 116 (19) (2019)
Manu De Rycker, David Horn, Bree Aldridge, Richard K Amewu, Clifton E Barry, Frederick S Buckner, Sarah Cook, Michael A J Ferguson, Nathalie Gobeau, Jennifer Herrmann, Paul Herrling, William Hope, Jennifer Keiser, Maria Jose Lafuente-Monasterio, Paul D Leeson, Didier Leroy, Ujjini H Manjunatha, James McCarthy, Timothy J Miles, Valerie Mizrahi, Olena Moshynets, Jacquin Niles, John P Overington, John Pottage, Srinivasa P S Rao, Kevin D Read, Isabela Ribeiro, Lynn L Silver, Jen Southern, Thomas Spangenberg, Shyam Sundar, Caitlin Taylor, Wes Van Voorhis, Nicholas J White, Susan Wyllie, Paul G Wyatt, Ian H Gilbert
Setting Our Sights on Infectious Diseases. ACS infectious diseases 6 (1) (2019)
Neil R Norcross, Caroline Wilson, Beatriz Baragaña, Irene Hallyburton, Maria Osuna-Cabello, Suzanne Norval, Jennifer Riley, Daniel Fletcher, Robert Sinden, Michael Delves, Andrea Ruecker, Sandra Duffy, Stephan Meister, Yevgeniya Antonova-Koch, Benigno Crespo, Cristina de Cózar, Laura M Sanz, Francisco Javier Gamo, Vicky M Avery, Julie A Frearson, David W Gray, Alan H Fairlamb, Elizabeth A Winzeler, David Waterson, Simon F Campbell, Paul A Willis, Kevin D Read, Ian H Gilbert
Substituted Aminoacetamides as Novel Leads for Malaria Treatment. ChemMedChem 14 (14) (2019)
Victoriano Corpas-Lopez, Sonia Moniz, Michael Thomas, Richard J Wall, Leah S Torrie, Dorothea Zander-Dinse, Michele Tinti, Stephen Brand, Laste Stojanovski, Sujatha Manthri, Irene Hallyburton, Fabio Zuccotto, Paul G Wyatt, Manu De Rycker, David Horn, Michael A J Ferguson, Joachim Clos, Kevin D Read, Alan H Fairlamb, Ian H Gilbert, Susan Wyllie
Pharmacological Validation of N-Myristoyltransferase as a Drug Target in Leishmania donovani. ACS infectious diseases 5 (1) (2018)
Lauren A Webster, Michael Thomas, Michael D Urbaniak, Susan Wyllie, Han Ong, Michele Tinti, Alan H Fairlamb, Markus Boesche, Sonja Ghidelli-Disse, Gerard Drewes, Ian H Gilbert
Development of Chemical Proteomics for the Folateome and Analysis of the Kinetoplastid Folateome. ACS infectious diseases 4 (10) (2018)
Justin R Harrison, Stephen Brand, Victoria Smith, David A Robinson, Stephen Thompson, Alasdair Smith, Kenneth Davies, Ngai Yi Mok, Leah S Torrie, Iain Collie, Irene Hallyburton, Suzanne Norval, Frederick R C Simeons, Laste Stojanovski, Julie A Frearson, Ruth Brenk, Paul G Wyatt, Ian H Gilbert, Kevin D Read
A Molecular Hybridization Approach for the Design of Potent, Highly Selective, and Brain-Penetrant N-Myristoyltransferase Inhibitors. Journal of medicinal chemistry 61 (18) (2018)
Michael G Thomas, Manu De Rycker, Myriam Ajakane, Sébastian Albrecht, Ana Isabel Álvarez-Pedraglio, Markus Boesche, Stephen Brand, Lorna Campbell, Juan Cantizani-Perez, Laura A T Cleghorn, Royston C B Copley, Sabrinia D Crouch, Alain Daugan, Gerard Drewes, Santiago Ferrer, Sonja Ghidelli-Disse, Silvia Gonzalez, Stephanie L Gresham, Alan P Hill, Sean J Hindley, Rhiannon M Lowe, Claire J MacKenzie, Lorna MacLean, Sujatha Manthri, Franck Martin, Juan Miguel-Siles, Van Loc Nguyen, Suzanne Norval, Maria Osuna-Cabello, Andrew Woodland, Stephen Patterson, Imanol Pena, Maria Teresa Quesada-Campos, Iain H Reid, Charlotte Revill, Jennifer Riley, Jose Ramon Ruiz-Gomez, Yoko Shishikura, Frederick R C Simeons, Alasdair Smith, Victoria C Smith, Daniel Spinks, Laste Stojanovski, John Thomas, Stephen Thompson, Tim Underwood, David W Gray, Jose M Fiandor, Ian H Gilbert, Paul G Wyatt, Kevin D Read, Timothy J Miles
Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis. Journal of medicinal chemistry 62 (3) (2018)
Irene Hallyburton, Raffaella Grimaldi, Andrew Woodland, Beatriz Baragaña, Torsten Luksch, Daniel Spinks, Daniel James, Didier Leroy, David Waterson, Alan H Fairlamb, Paul G Wyatt, Ian H Gilbert, Julie A Frearson
Screening a protein kinase inhibitor library against Plasmodium falciparum. Malaria journal 16 (1) (2017)
Tracy Bayliss, David A Robinson, Victoria C Smith, Stephen Brand, Stuart P McElroy, Leah S Torrie, Chido Mpamhanga, Suzanne Norval, Laste Stojanovski, Ruth Brenk, Julie A Frearson, Kevin D Read, Ian H Gilbert, Paul G Wyatt
Design and Synthesis of Brain Penetrant Trypanocidal N-Myristoyltransferase Inhibitors. Journal of medicinal chemistry 60 (23) (2017)
Kathrin Heikamp, Fabio Zuccotto, Michael Kiczun, Peter Ray, Ian H Gilbert
Exhaustive sampling of the fragment space associated to a molecule leading to the generation of conserved fragments. Chemical biology & drug design 91 (3) (2017)
Stephen Brand, Eun Jung Ko, Elisabet Viayna, Stephen Thompson, Daniel Spinks, Michael Thomas, Lars Sandberg, Amanda F Francisco, Shiromani Jayawardhana, Victoria C Smith, Chimed Jansen, Manu De Rycker, John Thomas, Lorna MacLean, Maria Osuna-Cabello, Jennifer Riley, Paul Scullion, Laste Stojanovski, Frederick R C Simeons, Ola Epemolu, Yoko Shishikura, Sabrinia D Crouch, Tania S Bakshi, Christopher J Nixon, Iain H Reid, Alan P Hill, Tim Z Underwood, Sean J Hindley, Sharon A Robinson, John M Kelly, Jose M Fiandor, Paul G Wyatt, Maria Marco, Timothy J Miles, Kevin D Read, Ian H Gilbert
Discovery and Optimization of 5-Amino-1,2,3-triazole-4-carboxamide Series against Trypanosoma cruzi. Journal of medicinal chemistry 60 (17) (2017)
Leah S Torrie, Stephen Brand, David A Robinson, Eun Jung Ko, Laste Stojanovski, Frederick R C Simeons, Susan Wyllie, John Thomas, Lucy Ellis, Maria Osuna-Cabello, Ola Epemolu, Andrea Nühs, Jennifer Riley, Lorna MacLean, Sujatha Manthri, Kevin D Read, Ian H Gilbert, Alan H Fairlamb, Manu De Rycker
Chemical Validation of Methionyl-tRNA Synthetase as a Druggable Target in Leishmania donovani. ACS infectious diseases 3 (10) (2017)

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Ian H Gilbert